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—— (E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C22H21N3O2
(E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C23H21N5O
(E)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide —— C20H22FN3OS
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide
—— (E)-N-[(R)-cyclopropyl-(4-methylphenyl)methyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C23H27NO4
(E)-N-[(R)-cyclopropyl-(4-methylphenyl)methyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-[(S)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide —— C25H24FN3O2S
(E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-[(S)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide
—— (E)-3-(2,4-dimethylphenyl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C22H23N3O
(E)-3-(2,4-dimethylphenyl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-4-(N,N-diallylsulfamoyl)-N-(4-methoxy-3-methylbenzo[d]thiazol-2(3H)-ylidene)benzamide —— C22H23N3O4S2
(E)-4-(N,N-diallylsulfamoyl)-N-(4-methoxy-3-methylbenzo[d]thiazol-2(3H)-ylidene)benzamide
—— Ethyl 2-(2-{[4-(3-chlorophenyl)-5-{[(thiophen-2-YL)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}acetamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H26ClN5O4S3
Ethyl 2-(2-{[4-(3-chlorophenyl)-5-{[(thiophen-2-YL)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}acetamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-amino-7-(4-methoxyphenyl)-2',5-dioxo-1',2',5,6,7,8-hexahydrospiro[chromene-4,3'-indole]-3-carboxylate —— C26H24N2O6
Ethyl 2-amino-7-(4-methoxyphenyl)-2',5-dioxo-1',2',5,6,7,8-hexahydrospiro[chromene-4,3'-indole]-3-carboxylate
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C21H21N5OS
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide —— C20H20FNO3
(E)-3-(1,3-benzodioxol-5-yl)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide
—— (E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(1R)-2-methyl-1-phenylpropyl]prop-2-enamide —— C21H23NO2
(E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(1R)-2-methyl-1-phenylpropyl]prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(S)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide —— C25H25N3O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(S)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide
—— ethyl N-[2-cyano-3-(3-nitroanilino)prop-2-enoyl]carbamate —— C13H12N4O5
ethyl N-[2-cyano-3-(3-nitroanilino)prop-2-enoyl]carbamate
—— (E)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide —— C23H18F2N4OS
(E)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C25H24ClN3O4
(E)-3-(6-chloro-2H-chromen-3-yl)-N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C26H26ClN5O
(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)prop-2-enamide —— C23H25N5O3S
(E)-N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)prop-2-enamide
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C23H20ClN3O2
(E)-3-(6-chloro-2H-chromen-3-yl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— Ethyl 2-[[2-(4-benzyl-2,5-dioxoimidazolidin-1-yl)acetyl]amino]-4-phenylthiophene-3-carboxylate —— C25H23N3O5S
Ethyl 2-[[2-(4-benzyl-2,5-dioxoimidazolidin-1-yl)acetyl]amino]-4-phenylthiophene-3-carboxylate
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[(S)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide —— C22H22N2O2
(E)-3-[4-(cyanomethoxy)phenyl]-N-[(S)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(S)-(4-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C22H20ClN3O4
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(S)-(4-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C22H20N4O5
(E)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— (E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C22H21N3O2
(E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1R)-2-methyl-1-phenylpropyl]prop-2-enamide —— C20H23N3OS
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1R)-2-methyl-1-phenylpropyl]prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide —— C24H24FN3O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide
—— (E)-N-[(1S)-2-methyl-1-phenylpropyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C22H23N3O
(E)-N-[(1S)-2-methyl-1-phenylpropyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[(R)-(4-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C25H27N5O3
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[(R)-(4-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(R)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide —— C25H25N3O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(R)-cyclopropyl-(4-methylphenyl)methyl]prop-2-enamide
—— (E)-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide —— C23H18F2N4OS
(E)-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide
—— (E)-3-[2,5-dimethyl-1-(2-propan-2-ylpyrazol-3-yl)pyrrol-3-yl]-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C26H29FN6O
(E)-3-[2,5-dimethyl-1-(2-propan-2-ylpyrazol-3-yl)pyrrol-3-yl]-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C23H19FN4OS
(E)-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C21H20FN5OS
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-(2,4-dimethylphenyl)-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C22H22FN3O
(E)-3-(2,4-dimethylphenyl)-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— ethyl 5-(2,4-dichlorophenyl)-1-[4-[[(1R)-2,3-dihydro-1H-inden-1-yl]carbamoyl]phenyl]pyrazole-3-carboxylate —— C28H23Cl2N3O3
ethyl 5-(2,4-dichlorophenyl)-1-[4-[[(1R)-2,3-dihydro-1H-inden-1-yl]carbamoyl]phenyl]pyrazole-3-carboxylate
—— (E)-3-(2,4-dimethylphenyl)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C22H23N3O
(E)-3-(2,4-dimethylphenyl)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-3-(2,4-dimethylphenyl)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C22H22FN3O
(E)-3-(2,4-dimethylphenyl)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C23H19ClFN3O2
(E)-3-(6-chloro-2H-chromen-3-yl)-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C22H20N4O5
(E)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C23H19ClFN3O2
(E)-3-(6-chloro-2H-chromen-3-yl)-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enamide —— C29H33N5O3
(E)-N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enamide
—— (E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide —— C24H24FN3O2S
(E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C21H21N5OS
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— ethyl 5-(2,4-dichlorophenyl)-1-[4-[[(1S)-2,3-dihydro-1H-inden-1-yl]carbamoyl]phenyl]pyrazole-3-carboxylate —— C28H23Cl2N3O3
ethyl 5-(2,4-dichlorophenyl)-1-[4-[[(1S)-2,3-dihydro-1H-inden-1-yl]carbamoyl]phenyl]pyrazole-3-carboxylate
—— (E)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C21H21FN2O5
(E)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— (E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide —— C27H29N5O
(E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1S)-2-methyl-1-phenylpropyl]prop-2-enamide —— C20H23N3OS
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1S)-2-methyl-1-phenylpropyl]prop-2-enamide
—— (E)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C22H26FNO4
(E)-N-[(1S)-1-(4-fluorophenyl)-2-methylpropyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[(R)-cyclopropyl-(4-methylphenyl)methyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C22H22N2O5
(E)-N-[(R)-cyclopropyl-(4-methylphenyl)methyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— ethyl 1-benzyl-3-[[(3R)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]amino]-4-(4-methoxyphenyl)pyrrole-2-carboxylate —— C30H28N2O6
ethyl 1-benzyl-3-[[(3R)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]amino]-4-(4-methoxyphenyl)pyrrole-2-carboxylate