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—— ethyl (4R)-4-ethyl-6-[[4-(2-nitrophenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H27N5O5
ethyl (4R)-4-ethyl-6-[[4-(2-nitrophenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(6-nitro-1,3-benzodioxol-5-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C26H28N2O8
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(6-nitro-1,3-benzodioxol-5-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-2-cyano-3-(5-cyano-1,2-dimethylpyrrol-3-yl)-N-phenylprop-2-enamide —— C17H14N4O
(E)-2-cyano-3-(5-cyano-1,2-dimethylpyrrol-3-yl)-N-phenylprop-2-enamide
—— (E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C27H31NO5
(E)-3-(2,3-dihydro-1-benzofuran-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C25H31N3O6
(E)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C26H31N3O4S
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(6-nitro-1,3-benzodioxol-5-yl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C26H28N2O8
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(6-nitro-1,3-benzodioxol-5-yl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C26H31N3O4S
(E)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl 2-[({7-[chloro(difluoro)methyl]-5-(furan-2-yl)pyrazolo[1,5-a]pyrimidin-2-yl}carbonyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C24H21ClF2N4O4S
ethyl 2-[({7-[chloro(difluoro)methyl]-5-(furan-2-yl)pyrazolo[1,5-a]pyrimidin-2-yl}carbonyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— ethyl 3-[(3-methoxy-4-prop-2-enoxyphenyl)methyl-[[(2S)-oxolan-2-yl]methyl]carbamoyl]-5-nitrobenzoate —— C26H30N2O8
ethyl 3-[(3-methoxy-4-prop-2-enoxyphenyl)methyl-[[(2S)-oxolan-2-yl]methyl]carbamoyl]-5-nitrobenzoate
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C26H28ClNO6
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C28H31N3O4
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C26H30FNO5
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C28H31N3O4
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(1-methylpyrazol-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C23H29N3O4
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(1-methylpyrazol-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(4-ethoxy-3-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C28H35NO6
(E)-3-(4-ethoxy-3-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C28H35NO7
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C28H35NO7
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(1-methylpyrazol-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C23H29N3O4
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(1-methylpyrazol-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(1-benzyltriazol-4-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C28H32N4O4
(E)-3-(1-benzyltriazol-4-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C26H30FNO5
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C28H33NO7
(E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(4-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C26H31NO5
(E)-3-(4-methoxyphenyl)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-N-(3-(2-ethoxyethyl)-4,6-difluorobenzo[d]thiazol-2(3H)-ylidene)-4-oxo-4H-chromene-2-carboxamide —— C21H16F2N2O4S
(E)-N-(3-(2-ethoxyethyl)-4,6-difluorobenzo[d]thiazol-2(3H)-ylidene)-4-oxo-4H-chromene-2-carboxamide
—— ethyl (4S)-4-(5-methylfuran-2-yl)-2-oxo-6-[[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H22N6O4S2
ethyl (4S)-4-(5-methylfuran-2-yl)-2-oxo-6-[[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(5-methylfuran-2-yl)-6-[[5-(3-methylphenyl)-4-propyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H29N5O4S
ethyl (4R)-4-(5-methylfuran-2-yl)-6-[[5-(3-methylphenyl)-4-propyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(2-nitrophenyl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C25H28N2O6
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(2-nitrophenyl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl (4R)-6-[(5-butylsulfanyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N4O4S3
ethyl (4R)-6-[(5-butylsulfanyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(5-methylfuran-2-yl)-2-oxo-6-[[5-[(E)-2-thiophen-2-ylethenyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21N5O4S2
ethyl (4S)-4-(5-methylfuran-2-yl)-2-oxo-6-[[5-[(E)-2-thiophen-2-ylethenyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— Ethyl 4-(2-oxo-3-prop-2-enylimidazolidin-1-yl)benzoate —— C15H18N2O3
Ethyl 4-(2-oxo-3-prop-2-enylimidazolidin-1-yl)benzoate
—— Ethyl {[5-(2-amino-4-hydroxy-6-methyl-5-pyrimidinyl)pentanoyl]amino}acetate —— C14H22N4O4
Ethyl {[5-(2-amino-4-hydroxy-6-methyl-5-pyrimidinyl)pentanoyl]amino}acetate
—— ethyl 5-[2-[3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C25H22FN3O4S
ethyl 5-[2-[3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (4R)-6-[[5-[acetyl(cyclopropyl)amino]-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H23N5O5S2
ethyl (4R)-6-[[5-[acetyl(cyclopropyl)amino]-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-(1-benzothiophene-3-carbonyloxymethyl)-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H20N2O6S
ethyl (4S)-6-(1-benzothiophene-3-carbonyloxymethyl)-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(4-benzyl-5-oxo-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H23N5O5S
ethyl (4S)-6-[(4-benzyl-5-oxo-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(5-butylsulfanyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N4O4S3
ethyl (4S)-6-[(5-butylsulfanyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(5-methylfuran-2-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C24H29NO5
(E)-N-[(3-methoxy-4-prop-2-enoxyphenyl)methyl]-3-(5-methylfuran-2-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-5-methoxy-2-nitrophenyl]-N-[3-[(1S)-1-phenylethoxy]propyl]prop-2-enamide —— C22H24F2N2O6
(E)-3-[4-(difluoromethoxy)-5-methoxy-2-nitrophenyl]-N-[3-[(1S)-1-phenylethoxy]propyl]prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[3-[(1R)-1-phenylethoxy]propyl]prop-2-enamide —— C21H22ClNO4
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[3-[(1R)-1-phenylethoxy]propyl]prop-2-enamide
—— ethyl (4S)-6-[[5-(cyclopentylmethyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H27N5O4S
ethyl (4S)-6-[[5-(cyclopentylmethyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(1-benzyltetrazol-5-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H22N6O4S
ethyl (4R)-6-[(1-benzyltetrazol-5-yl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(3,4-difluorophenyl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H18F2N2O4S
ethyl (4R)-6-[(3,4-difluorophenyl)sulfanylmethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-(furan-3-ylmethylidene)-5-(4-hydroxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H18N2O5S
ethyl 2-(furan-3-ylmethylidene)-5-(4-hydroxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (4R)-4-(5-methylfuran-2-yl)-2-oxo-6-[[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H22N6O4S2
ethyl (4R)-4-(5-methylfuran-2-yl)-2-oxo-6-[[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[3-[(1S)-1-phenylethoxy]propyl]prop-2-enamide —— C24H29N3O3
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[3-[(1S)-1-phenylethoxy]propyl]prop-2-enamide
—— ethyl 2-[[2-[1-[2-(naphthalene-2-carbonylamino)ethyl]indol-3-yl]sulfanylacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C33H31N3O4S2
ethyl 2-[[2-[1-[2-(naphthalene-2-carbonylamino)ethyl]indol-3-yl]sulfanylacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl (4S)-4-(5-methylfuran-2-yl)-6-[[5-(3-methylphenyl)-4-propyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H29N5O4S
ethyl (4S)-4-(5-methylfuran-2-yl)-6-[[5-(3-methylphenyl)-4-propyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(5-methylfuran-2-yl)-2-oxo-6-[[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H26N6O4S
ethyl (4R)-4-(5-methylfuran-2-yl)-2-oxo-6-[[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(5-methylfuran-2-yl)-6-[(4-methyl-6-phenylpyrimidin-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H24N4O4S
ethyl (4R)-4-(5-methylfuran-2-yl)-6-[(4-methyl-6-phenylpyrimidin-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— Ethyl 2-({4-[(4-bromophenoxy)methyl]benzoyl}amino)-5-(1-phenylethyl)-3-thiophenecarboxylate —— C29H26BrNO4S
Ethyl 2-({4-[(4-bromophenoxy)methyl]benzoyl}amino)-5-(1-phenylethyl)-3-thiophenecarboxylate