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—— (E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(2-methoxy-5-methylphenyl)prop-2-enamide —— C26H34N2O5
(E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(2-methoxy-5-methylphenyl)prop-2-enamide
—— (E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(4-ethylphenyl)prop-2-enamide —— C26H34N2O4
(E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(4-ethylphenyl)prop-2-enamide
—— (E)-3-(2-bromophenyl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide —— C24H29BrN2O4
(E)-3-(2-bromophenyl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide
—— (E)-3-(2-chloro-6-fluorophenyl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide —— C24H28ClFN2O4
(E)-3-(2-chloro-6-fluorophenyl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide
—— (E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(3-fluoro-4-methoxyphenyl)prop-2-enamide —— C25H31FN2O5
(E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(3-fluoro-4-methoxyphenyl)prop-2-enamide
—— (E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(4-ethoxyphenyl)prop-2-enamide —— C26H34N2O5
(E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(4-ethoxyphenyl)prop-2-enamide
—— (E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C27H34N2O7
(E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— (E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-[4-(trifluoromethoxy)phenyl]prop-2-enamide —— C25H29F3N2O5
(E)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-[4-(trifluoromethoxy)phenyl]prop-2-enamide
—— (E)-3-(5-bromothiophen-2-yl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide —— C22H27BrN2O4S
(E)-3-(5-bromothiophen-2-yl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide
—— (E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(3-methylthiophen-2-yl)prop-2-enamide —— C23H30N2O4S
(E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(3-methylthiophen-2-yl)prop-2-enamide
—— (E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(2-methoxy-5-methylphenyl)prop-2-enamide —— C26H34N2O5
(E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(2-methoxy-5-methylphenyl)prop-2-enamide
—— (E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(2-ethoxyphenyl)prop-2-enamide —— C26H34N2O5
(E)-N-[(2R)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]-3-(2-ethoxyphenyl)prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide —— C25H29ClN2O6
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-2-morpholin-4-ylethyl]prop-2-enamide
—— (E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C23H22FN3O4
(E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— ethyl 2-[[2-[[3-(4-ethoxyphenyl)-4-oxo-5H-pyrimido[5,4-b]indol-2-yl]sulfanyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C30H28N4O5S2
ethyl 2-[[2-[[3-(4-ethoxyphenyl)-4-oxo-5H-pyrimido[5,4-b]indol-2-yl]sulfanyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— (E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide —— C23H18F2N4OS
(E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide
—— ethyl 3-[[(1R)-1-(3-benzamidophenyl)ethyl]-methylcarbamoyl]-5-nitrobenzoate —— C26H25N3O6
ethyl 3-[[(1R)-1-(3-benzamidophenyl)ethyl]-methylcarbamoyl]-5-nitrobenzoate
—— (E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide —— C25H22FN3O2
(E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide
—— (E)-2,3-dihydro-1,4-benzodioxin-6-yl{2-(2,3-dimethoxyphenyl)-1-[3-(1H-imidazol-3-ium-1-yl)propyl]-4,5-dioxopyrrolidin-3-ylidene}methanolate —— C27H27N3O7
(E)-2,3-dihydro-1,4-benzodioxin-6-yl{2-(2,3-dimethoxyphenyl)-1-[3-(1H-imidazol-3-ium-1-yl)propyl]-4,5-dioxopyrrolidin-3-ylidene}methanolate
—— (E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C22H19FN4O5
(E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— (E)-3-(2,4-dimethylphenyl)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C22H22FN3O
(E)-3-(2,4-dimethylphenyl)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C23H20FN5O
(E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— Ethyl 3-acetyl-4-(3,4-dimethoxyphenyl)-6-methyl-2-oxo-1,4-dihydropyrimidine-5-carboxylate —— C18H22N2O6
Ethyl 3-acetyl-4-(3,4-dimethoxyphenyl)-6-methyl-2-oxo-1,4-dihydropyrimidine-5-carboxylate
—— (E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide —— C25H22FN3O2
(E)-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide
—— (E)-3-[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]-N-[2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]prop-2-enamide —— C19H20N4O2
(E)-3-[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]-N-[2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]prop-2-enamide
—— ethyl (2R)-2-(4-chlorophenyl)-2-[4-(4-cyano-2-methyl-5-pyrrol-1-ylfuran-3-carbonyl)piperazin-1-yl]acetate —— C25H25ClN4O4
ethyl (2R)-2-(4-chlorophenyl)-2-[4-(4-cyano-2-methyl-5-pyrrol-1-ylfuran-3-carbonyl)piperazin-1-yl]acetate
—— (E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide —— C23H18F2N4OS
(E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-[2-(4-fluorophenyl)-1,3-thiazol-4-yl]prop-2-enamide
—— ethyl 5-[[3-(3,4-dihydro-2H-pyrrol-5-ylsulfamoyl)phenyl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C20H24N4O5S
ethyl 5-[[3-(3,4-dihydro-2H-pyrrol-5-ylsulfamoyl)phenyl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]-N-[2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]prop-2-enamide —— C19H20N4O2
(E)-3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]-N-[2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]prop-2-enamide
—— (E)-3-(2,4-dimethylphenyl)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C22H22FN3O
(E)-3-(2,4-dimethylphenyl)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C23H22FN3O4
(E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— (E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-(dimethylamino)ethyl]-3-(2-nitrophenyl)prop-2-enamide —— C19H19ClFN3O3
(E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-(dimethylamino)ethyl]-3-(2-nitrophenyl)prop-2-enamide
—— Ethyl 6-amino-4-(2-hydroxy-5-nitrophenyl)-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carboxylate —— C16H16N4O6
Ethyl 6-amino-4-(2-hydroxy-5-nitrophenyl)-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carboxylate
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C24H24FN5O2
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— ethyl 5-(methoxymethyl)-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C17H20N4O3S
ethyl 5-(methoxymethyl)-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 2-(4-chloroanilino)-5-[(4-ethylphenyl)methylidene]-4-oxothiophene-3-carboxylate —— C22H20ClNO3S
ethyl 2-(4-chloroanilino)-5-[(4-ethylphenyl)methylidene]-4-oxothiophene-3-carboxylate
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C21H19F2N3O2
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— (E)-1-[(2S)-2-(1-methylpyrrol-2-yl)azepan-1-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one —— C22H25N3O5
(E)-1-[(2S)-2-(1-methylpyrrol-2-yl)azepan-1-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one
—— (E)-N-[(2S)-2-(2-chloro-6-fluorophenyl)-2-(dimethylamino)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C22H22ClFN4O
(E)-N-[(2S)-2-(2-chloro-6-fluorophenyl)-2-(dimethylamino)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C26H25ClFN5O
(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(R)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— Ethyl 4-(2-oxo-2-{[4-(trifluoromethoxy)phenyl]amino}ethyl)piperazine-1-carboxylate —— C16H20F3N3O4
Ethyl 4-(2-oxo-2-{[4-(trifluoromethoxy)phenyl]amino}ethyl)piperazine-1-carboxylate
—— (E)-N-[(2S)-2-(2-chloro-6-fluorophenyl)-2-(dimethylamino)ethyl]-3-(2-nitrophenyl)prop-2-enamide —— C19H19ClFN3O3
(E)-N-[(2S)-2-(2-chloro-6-fluorophenyl)-2-(dimethylamino)ethyl]-3-(2-nitrophenyl)prop-2-enamide
—— (E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C22H19FN4O5
(E)-N-[(S)-(2-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— (E)-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one —— C20H18N2O5
(E)-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one
—— ethyl 3-[[(1S)-1-(3-benzamidophenyl)ethyl]-methylcarbamoyl]-5-nitrobenzoate —— C26H25N3O6
ethyl 3-[[(1S)-1-(3-benzamidophenyl)ethyl]-methylcarbamoyl]-5-nitrobenzoate
—— (E)-1-[(2S)-2-(1-methylpyrrol-2-yl)azepan-1-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-en-1-one —— C18H23N3OS
(E)-1-[(2S)-2-(1-methylpyrrol-2-yl)azepan-1-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-en-1-one
—— (E)-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]-N-[2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]prop-2-enamide —— C19H20N4O2
(E)-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]-N-[2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]prop-2-enamide
—— (E)-3-(3-methoxy-4-prop-2-enoxyphenyl)-1-[(2R)-2-(1-methylpyrrol-2-yl)azepan-1-yl]prop-2-en-1-one —— C24H30N2O3
(E)-3-(3-methoxy-4-prop-2-enoxyphenyl)-1-[(2R)-2-(1-methylpyrrol-2-yl)azepan-1-yl]prop-2-en-1-one
—— (E)-1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one —— C18H22N2O5
(E)-1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one
—— (E)-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one —— C17H20N2O6
(E)-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-en-1-one