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—— [(6S,7R)-6-(4-chlorophenyl)-3-cyclopropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone —— C21H17ClF2N4O2S
[(6S,7R)-6-(4-chlorophenyl)-3-cyclopropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone
—— 6-[[(8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[e][1,3]oxazin-6-yl]methyl]-3,4-dihydro-2H-1,3-benzoxazine —— C17H24N2O2
6-[[(8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[e][1,3]oxazin-6-yl]methyl]-3,4-dihydro-2H-1,3-benzoxazine
—— 6-[[(8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[e][1,3]oxazin-6-yl]methyl]-3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[e][1,3]oxazine —— C17H30N2O2
6-[[(8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[e][1,3]oxazin-6-yl]methyl]-3,4,4a,5,6,7,8,8a-octahydro-2H-benzo[e][1,3]oxazine
—— [(6R,7S)-6-(4-chlorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-(4-methylpiperidin-1-yl)methanone —— C18H22ClN5OS
[(6R,7S)-6-(4-chlorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-(4-methylpiperidin-1-yl)methanone
—— [(6R,7R)-6-(4-chlorophenyl)-3-cyclopropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone —— C21H17ClF2N4O2S
[(6R,7R)-6-(4-chlorophenyl)-3-cyclopropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone
—— [(6S,7S)-6-(4-chlorophenyl)-3-cyclohexyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone —— C24H23ClF2N4O2S
[(6S,7S)-6-(4-chlorophenyl)-3-cyclohexyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone
—— [(6R,7R)-6-(4-chlorophenyl)-3-cyclohexyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone —— C24H23ClF2N4O2S
[(6R,7R)-6-(4-chlorophenyl)-3-cyclohexyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone
—— 6-Bromo-2-ethyl-3-thionitrosoimidazo[1,2-a]pyridine —— C9H8BrN3S
6-Bromo-2-ethyl-3-thionitrosoimidazo[1,2-a]pyridine
—— [(6S,7S)-6-(4-chlorophenyl)-3-cyclopropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone —— C21H17ClF2N4O2S
[(6S,7S)-6-(4-chlorophenyl)-3-cyclopropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone
—— [(6S,7R)-6-(4-chlorophenyl)-3-cyclohexyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone —— C24H23ClF2N4O2S
[(6S,7R)-6-(4-chlorophenyl)-3-cyclohexyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[4-(difluoromethoxy)phenyl]methanone
—— 6-O-tert-butyl 7-O-methyl (7S)-4-hydroxy-1-methyl-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine-6,7-dicarboxylate —— C14H21N3O5
6-O-tert-butyl 7-O-methyl (7S)-4-hydroxy-1-methyl-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine-6,7-dicarboxylate
—— [[(6S)-6-[(2-amino-2-cyclopropylethoxy)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C14H24N4O8S
[[(6S)-6-[(2-amino-2-cyclopropylethoxy)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— (6S)-6-methyl-2-[[2-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H22N4O2S3
(6S)-6-methyl-2-[[2-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6-bromo-2-ethyl-imidazo[1,2-a]pyridin-3-yl)-[3-(4-chloro-phenyl)-[1,2,4]thiadiazol-5-yl]-methyl-amine —— C18H15BrClN5S
(6-bromo-2-ethyl-imidazo[1,2-a]pyridin-3-yl)-[3-(4-chloro-phenyl)-[1,2,4]thiadiazol-5-yl]-methyl-amine
—— (6-bromo-2-ethyl-imidazo[1,2-a]pyridin-3-yl)-[3-(4-fluoro-phenyl)-[1,2,4]thiadiazol-5-yl]-methyl-amine —— C18H15BrFN5S
(6-bromo-2-ethyl-imidazo[1,2-a]pyridin-3-yl)-[3-(4-fluoro-phenyl)-[1,2,4]thiadiazol-5-yl]-methyl-amine
—— 6-O-tert-butyl 7-O-methyl (7S)-4-(butoxyamino)-1-methyl-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine-6,7-dicarboxylate —— C18H30N4O5
6-O-tert-butyl 7-O-methyl (7S)-4-(butoxyamino)-1-methyl-5,7-dihydro-4H-pyrazolo[3,4-c]pyridine-6,7-dicarboxylate
—— 6-N-(6-methylsulfonylquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine —— C16H17N5O2S2
6-N-(6-methylsulfonylquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine
—— 6-chloro-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinazolin-4-amine —— C15H14ClN5
6-chloro-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinazolin-4-amine
—— 6-bromo-2-(2,2,2-trifluoro-ethyl)-imidazo[1,2-a]pyridin-3-amine —— C9H7BrF3N3
6-bromo-2-(2,2,2-trifluoro-ethyl)-imidazo[1,2-a]pyridin-3-amine
—— 6-N-(6-fluoroquinazolin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,6-diamine —— C16H15FN6
6-N-(6-fluoroquinazolin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,6-diamine
—— [[(6S)-6-[(2-amino-2-phenylethoxy)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C17H24N4O8S
[[(6S)-6-[(2-amino-2-phenylethoxy)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— (6R)-6-methyl-2-[[2-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H22N4O2S3
(6R)-6-methyl-2-[[2-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— [6-(1-ethenesulfonyl-piperidin-4-yl)-2-ethyl-imidazo[1,2-a]pyridin-3-yl]-[4-(4-fluoro-phenyl)-thiazol-2-yl]-methyl-amine —— C26H28FN5O2S2
[6-(1-ethenesulfonyl-piperidin-4-yl)-2-ethyl-imidazo[1,2-a]pyridin-3-yl]-[4-(4-fluoro-phenyl)-thiazol-2-yl]-methyl-amine
—— 6-fluoro-N-(2-methyl-5,6,7,8-tetrahydroquinazolin-6-yl)quinazolin-4-amine —— C17H16FN5
6-fluoro-N-(2-methyl-5,6,7,8-tetrahydroquinazolin-6-yl)quinazolin-4-amine
—— (6-bromo-2-cyclopropyl-imidazo[1,2-a]pyridin-3-yl)-methyl-amine —— C11H12BrN3
(6-bromo-2-cyclopropyl-imidazo[1,2-a]pyridin-3-yl)-methyl-amine
—— 6-bromo-2-ethyl-7-fluoro-N-(2,4,4-trimethylpentan-2-yl)imidazo[1,2-a]pyridin-3-amine —— C17H25BrFN3
6-bromo-2-ethyl-7-fluoro-N-(2,4,4-trimethylpentan-2-yl)imidazo[1,2-a]pyridin-3-amine
—— [[(6S)-6-(benzamidocarbamoyl)-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C16H20N4O8S
[[(6S)-6-(benzamidocarbamoyl)-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— [[(6S)-6-[(pyrrolidine-3-carbonylamino)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C14H23N5O8S
[[(6S)-6-[(pyrrolidine-3-carbonylamino)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— 6-N-(6-chloroquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine —— C15H14ClN5S
6-N-(6-chloroquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine
—— (6-bromo-2-ethyl-7-fluoro-imidazo[1,2-a]pyridin-3-yl)-methyl-amine —— C10H11BrFN3
(6-bromo-2-ethyl-7-fluoro-imidazo[1,2-a]pyridin-3-yl)-methyl-amine
—— 6-ethyl-2,2-dimethyl-3a,7a-dihydro-3H-1-benzofuran —— C12H18O
6-ethyl-2,2-dimethyl-3a,7a-dihydro-3H-1-benzofuran
—— 6-Methyl-2,3-dihydro-1,2-benzoxazole —— C8H9NO
6-Methyl-2,3-dihydro-1,2-benzoxazole
—— 6-methylsulfonyl-N-[5-(2-morpholin-4-ylethoxy)-2,3-dihydro-1H-inden-1-yl]quinazolin-4-amine —— C24H28N4O4S
6-methylsulfonyl-N-[5-(2-morpholin-4-ylethoxy)-2,3-dihydro-1H-inden-1-yl]quinazolin-4-amine
—— (6-bromo-2-ethyl-imidazo[1,2-a]pyridin-3-yl)-[4-(4-chloro-phenyl)-thiazol-2-yl]-methyl-amine —— C19H16BrClN4S
(6-bromo-2-ethyl-imidazo[1,2-a]pyridin-3-yl)-[4-(4-chloro-phenyl)-thiazol-2-yl]-methyl-amine
—— 6-fluoro-N-(4,5,6,7-tetrahydro-2H-isoindol-5-yl)quinazolin-4-amine —— C16H15FN4
6-fluoro-N-(4,5,6,7-tetrahydro-2H-isoindol-5-yl)quinazolin-4-amine
—— 6-Ethoxy-2,2-dimethyl-3,4-dihydrochromene —— C13H18O2
6-Ethoxy-2,2-dimethyl-3,4-dihydrochromene
—— 6-O-butyl 5-O-tert-butyl (6S)-4-oxo-5-azaspiro[2.4]heptane-5,6-dicarboxylate —— C16H25NO5
6-O-butyl 5-O-tert-butyl (6S)-4-oxo-5-azaspiro[2.4]heptane-5,6-dicarboxylate
—— 6-Amino-5-[2-(3-benzyl-4-oxoquinazolin-2-yl)sulfanylacetyl]-1,3-dimethylpyrimidine-2,4-dione —— C23H21N5O4S
6-Amino-5-[2-(3-benzyl-4-oxoquinazolin-2-yl)sulfanylacetyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-fluoro-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinazolin-4-amine —— C15H14FN5
6-fluoro-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinazolin-4-amine
—— [[(6S)-6-[[2-amino-2-(furan-2-yl)ethoxy]carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C15H22N4O9S
[[(6S)-6-[[2-amino-2-(furan-2-yl)ethoxy]carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— 6-Methylbenzo[d][1,3,2]benzodioxaphosphepine 6-oxide —— C13H11O3P
6-Methylbenzo[d][1,3,2]benzodioxaphosphepine 6-oxide
—— [[(6S)-6-[(2-amino-2-thiophen-2-ylethoxy)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C15H22N4O8S2
[[(6S)-6-[(2-amino-2-thiophen-2-ylethoxy)carbamoyl]-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— 6-fluoro-N-[5-(2-morpholin-4-ylethoxy)-2,3-dihydro-1H-inden-1-yl]quinazolin-4-amine —— C23H25FN4O2
6-fluoro-N-[5-(2-morpholin-4-ylethoxy)-2,3-dihydro-1H-inden-1-yl]quinazolin-4-amine
—— 6-N-(7-chloroquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine —— C15H14ClN5S
6-N-(7-chloroquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine
—— 6-N-(6-fluoroquinazolin-4-yl)-6,7-dihydro-5H-cyclopenta[b]pyridine-3,6-diamine —— C16H14FN5
6-N-(6-fluoroquinazolin-4-yl)-6,7-dihydro-5H-cyclopenta[b]pyridine-3,6-diamine
—— [[(6S)-6-(3-aminopropoxycarbamoyl)-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate —— C12H22N4O8S
[[(6S)-6-(3-aminopropoxycarbamoyl)-2-oxa-7-azaspiro[3.5]nonane-7-carbonyl]amino] hydrogen sulfate
—— 6-[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]-2,4,5,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-3-one —— C23H18F2N8O2
6-[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]-2,4,5,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-3-one
—— 6-N-(7-fluoroquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine —— C15H14FN5S
6-N-(7-fluoroquinazolin-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine
—— 6-N-(6-chloroquinazolin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,6-diamine —— C16H15ClN6
6-N-(6-chloroquinazolin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,6-diamine
—— (6-bromo-2-ethyl-7-fluoro-imidazo[1,2-a]pyridin-3-yl)-[4-(4-fluoro-phenyl)-thiazol-2-yl]-methyl-amine —— C19H15BrF2N4S
(6-bromo-2-ethyl-7-fluoro-imidazo[1,2-a]pyridin-3-yl)-[4-(4-fluoro-phenyl)-thiazol-2-yl]-methyl-amine