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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-bromo-2-trifluoromethyl-1H-pyrrolo[2,3-b]pyridine 1354759-15-1 C8H4BrF3N2
5-bromo-2-trifluoromethyl-1H-pyrrolo[2,3-b]pyridine
—— 5-Hydroxy-1H-benzimidazole-6-carboxylic acid 92222-06-5 C8H6N2O3
5-Hydroxy-1H-benzimidazole-6-carboxylic acid
—— 5-[(5-cyclopropyl-3-methylcarbamoyl-2-p-tolyl-furo[2,3-b]pyridin-6-yl)-methanesulfonyl-amino]-pent-2-enoic acid methyl ester 1345184-07-7 C26H29N3O6S
5-[(5-cyclopropyl-3-methylcarbamoyl-2-p-tolyl-furo[2,3-b]pyridin-6-yl)-methanesulfonyl-amino]-pent-2-enoic acid methyl ester
—— 5-{2-[4-(1-tert-butoxycarbonylamino-cyclobutyl)-phenyl]-3-phenyl-imidazo[1,2-a]pyridin-6-yl}-3-methyl-pyrazole-1-carboxylic acid tert-butyl ester 1356001-98-3 C37H41N5O4
5-{2-[4-(1-tert-butoxycarbonylamino-cyclobutyl)-phenyl]-3-phenyl-imidazo[1,2-a]pyridin-6-yl}-3-methyl-pyrazole-1-carboxylic acid tert-butyl ester
—— 5-amino-2-(2,6-difluorophenyl)pyrimidine-4-carboxylic acid 1052714-32-5 C11H7F2N3O2
5-amino-2-(2,6-difluorophenyl)pyrimidine-4-carboxylic acid
—— 5-But-2-ynyloxy-3-methyl-pyrazine-2-carboxylic acid 1262860-65-0 C10H10N2O3
5-But-2-ynyloxy-3-methyl-pyrazine-2-carboxylic acid
—— 5-ethyl-6-fluoro-3-(2-oxo-1,2-dihydro-pyridin-3-yl)-1H-indole-2-carboxylic acid methyl ester 1126423-59-3 C17H15FN2O3
5-ethyl-6-fluoro-3-(2-oxo-1,2-dihydro-pyridin-3-yl)-1H-indole-2-carboxylic acid methyl ester
—— 5-[({1-[3-(1-Methylethyl)-1,2,4-thiadiazol-5-yl]-4-piperidinyl}methyl)oxy]-2-[4-(methylsulfonyl)phenyl]pyridine trifluoroacetate 1032824-69-3 C2HF3O2*C23H28N4O3S2
5-[({1-[3-(1-Methylethyl)-1,2,4-thiadiazol-5-yl]-4-piperidinyl}methyl)oxy]-2-[4-(methylsulfonyl)phenyl]pyridine trifluoroacetate
—— 5-(3-[(1S)-2-hydroxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyridin-2-sulfonamide 1177419-95-2 C23H26N4O6S
5-(3-[(1S)-2-hydroxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyridin-2-sulfonamide
—— [5-(5-amino-2-fluoro-phenyl)-5-difluoromethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-3-yl]-carbamic acid tert-butyl ester 1262860-07-0 C17H22F3N3O3
[5-(5-amino-2-fluoro-phenyl)-5-difluoromethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-3-yl]-carbamic acid tert-butyl ester
—— 5-[(2-chloro-4-fluorophenyl)acetyl]-1-(2,6-dichlorophenyl)pyridin-2(1H)-one 887307-14-4 C19H11Cl3FNO2
5-[(2-chloro-4-fluorophenyl)acetyl]-1-(2,6-dichlorophenyl)pyridin-2(1H)-one
—— 5-hydroxy-1-[1-(S)-phenylethyl]-4-ethyl-1,5-dihydropyrrol-2-one 1355169-48-0 C14H17NO2
5-hydroxy-1-[1-(S)-phenylethyl]-4-ethyl-1,5-dihydropyrrol-2-one
—— (5-{5-[(5-Bromo-pyridine-2-carbonyl)-amino]-2-fluoro-phenyl}-5-difluoromethyl-2-methyl-5,6-dihydro-2H-[1,4]oxazin-3-yl)-carbamic acid tert-butyl ester 1262859-82-4 C23H24BrF3N4O4
(5-{5-[(5-Bromo-pyridine-2-carbonyl)-amino]-2-fluoro-phenyl}-5-difluoromethyl-2-methyl-5,6-dihydro-2H-[1,4]oxazin-3-yl)-carbamic acid tert-butyl ester
—— 5-(3-Bromo-phenyl)-5-trifluoromethyl-morpholin-3-one 1262859-14-2 C11H9BrF3NO2
5-(3-Bromo-phenyl)-5-trifluoromethyl-morpholin-3-one
—— 5-bromo-2-chloro-6-nitro-1,3-benzothiazole 1355241-08-5 C7H2BrClN2O2S
5-bromo-2-chloro-6-nitro-1,3-benzothiazole
—— 5-chloro-6-isobutylpyridin-3-ol 1355067-49-0 C9H12ClNO
5-chloro-6-isobutylpyridin-3-ol
—— 5-bromo-8-(3-methoxy-benzyl)-5,6,7,8-tetrahydro-2H-1,2,8-triaza-azulen-4-one 1355994-69-2 C15H16BrN3O2
5-bromo-8-(3-methoxy-benzyl)-5,6,7,8-tetrahydro-2H-1,2,8-triaza-azulen-4-one
—— 5-chloro-6-(3,3,3-trifluoropropoxy)pyridin-3-ol 1355067-70-7 C8H7ClF3NO2
5-chloro-6-(3,3,3-trifluoropropoxy)pyridin-3-ol
—— 5-bromo-pyridine-2-carboxylic acid[3-((S)-3-amino-5-difluoromethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-5-yl)-4-fluoro-phenyl]-amide hydrochloride 1262856-22-3 C18H16BrF3N4O2*ClH
5-bromo-pyridine-2-carboxylic acid[3-((S)-3-amino-5-difluoromethyl-2,5,6,7-tetrahydro-[1,4]oxazepin-5-yl)-4-fluoro-phenyl]-amide hydrochloride
—— 5-[(S)-3-(4-Bromo-phenyl)-3-o-tolyl-propionyl]-1-methyl-1H-pyridin-2-one 1354817-59-6 C22H20BrNO2
5-[(S)-3-(4-Bromo-phenyl)-3-o-tolyl-propionyl]-1-methyl-1H-pyridin-2-one
—— 5-(2-methoxy-ethoxy)-3-methyl-pyrazine-2-carboxylic acid 1262860-64-9 C9H12N2O4
5-(2-methoxy-ethoxy)-3-methyl-pyrazine-2-carboxylic acid
—— 5-((E)-3-dimethylamino-acryloyl)-1-methyl-1H-pyrrole-3-carboxylic acid ethyl ester 1246752-93-1 C13H18N2O3
5-((E)-3-dimethylamino-acryloyl)-1-methyl-1H-pyrrole-3-carboxylic acid ethyl ester
—— 5,7-dimethoxy-2-(4-(3-(methylamino)pyrrolidin-1-yl)phenyl)quinazolin-4(3H)-one 1246249-87-5 C21H24N4O3
5,7-dimethoxy-2-(4-(3-(methylamino)pyrrolidin-1-yl)phenyl)quinazolin-4(3H)-one
—— 5-bromo-2-(4-bromo-2-fluorophenylamino)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester 853109-50-9 C14H11Br2FN2O3
5-bromo-2-(4-bromo-2-fluorophenylamino)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester
—— 5-ethyl-6-fluoro-3-(2-methoxy-pyridin-3-yl)-1H-indole-2-carboxylic acid methyl ester 1126423-57-1 C18H17FN2O3
5-ethyl-6-fluoro-3-(2-methoxy-pyridin-3-yl)-1H-indole-2-carboxylic acid methyl ester
—— 5,7-dimethoxy-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)quinazolin-4(3H)-one 1246250-53-2 C22H25N3O4
5,7-dimethoxy-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)quinazolin-4(3H)-one
—— 5-{2-[4-(4-methyl-piperazin-1-yl)-2-trifluoromethoxy-phenylamino]-pyrimidin-4-yl}-1H-pyrrole-3-carboxylic acid ethyl ester 1246752-94-2 C23H25F3N6O3
5-{2-[4-(4-methyl-piperazin-1-yl)-2-trifluoromethoxy-phenylamino]-pyrimidin-4-yl}-1H-pyrrole-3-carboxylic acid ethyl ester
—— 5-bromo-3-trifluoromethyl-1,5,6,7-tetrahydro-indazol-4-one 1246307-19-6 C8H6BrF3N2O
5-bromo-3-trifluoromethyl-1,5,6,7-tetrahydro-indazol-4-one
—— 5-{2-[2-methoxy-4-(4-methyl-piperazin-1-yl)-phenylamino]-pyrimidin-4-yl}-1H-pyrrole-3-carboxylic acid ethyl ester 1246752-96-4 C23H28N6O3
5-{2-[2-methoxy-4-(4-methyl-piperazin-1-yl)-phenylamino]-pyrimidin-4-yl}-1H-pyrrole-3-carboxylic acid ethyl ester
—— 5-ethyl-6-fluoro-3-(2-oxo-1,2-dihydro-pyridin-3-yl)-1H-indole-2-carboxylic acid 1126423-61-7 C16H13FN2O3
5-ethyl-6-fluoro-3-(2-oxo-1,2-dihydro-pyridin-3-yl)-1H-indole-2-carboxylic acid
—— 5-[({1-[3-(1-methylethyl)-1,2,4-oxadiazol-5-yl]-4-piperidinyl}methyl)oxy]-2-[2-methyl-4-(methylthio)phenyl]pyridine 1032825-88-9 C24H30N4O2S
5-[({1-[3-(1-methylethyl)-1,2,4-oxadiazol-5-yl]-4-piperidinyl}methyl)oxy]-2-[2-methyl-4-(methylthio)phenyl]pyridine
—— 5-Hydroxy-2-(2-methylpropyl)-1,3-dioxane 896447-14-6 C8H16O3
5-Hydroxy-2-(2-methylpropyl)-1,3-dioxane
—— 5-(3-{5-[(4R)-4-Ethyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}-5-[(1S)-2-methoxy-1-methylethoxy]phenoxy)-2-(methylsulfonyl)pyridine 1177420-93-7 C25H29N3O6S
5-(3-{5-[(4R)-4-Ethyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}-5-[(1S)-2-methoxy-1-methylethoxy]phenoxy)-2-(methylsulfonyl)pyridine
—— (5S)-2-(5-{3-[(1S)-2-Methoxy-1-methylethoxy]-5-[(triisopropylsilyl)oxy]phenyl}-1H-pyrrol-2-yl)-5-methyl-4,5-dihydro-1,3-oxazole 1177421-76-9 C27H42N2O4Si
(5S)-2-(5-{3-[(1S)-2-Methoxy-1-methylethoxy]-5-[(triisopropylsilyl)oxy]phenyl}-1H-pyrrol-2-yl)-5-methyl-4,5-dihydro-1,3-oxazole
—— 5-methyl-2-[1-(triisopropylsilyl)-1H-pyrrol-2-yl]-1,3-thiazole 1177420-14-2 C17H28N2SSi
5-methyl-2-[1-(triisopropylsilyl)-1H-pyrrol-2-yl]-1,3-thiazole
—— 5-(3-[(1S)-2-hydroxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyrazine-2-carboxamide 1177419-97-4 C23H25N5O5
5-(3-[(1S)-2-hydroxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyrazine-2-carboxamide
—— 5-(4-chloro-3-methylphenyl)-6-(2,2,2-trifluoroethoxy)nicotinic acid 1364678-18-1 C15H11ClF3NO3
5-(4-chloro-3-methylphenyl)-6-(2,2,2-trifluoroethoxy)nicotinic acid
—— 5-methyl-2-(1H-pyrrol-2-yl)-1,3-thiazole 1177420-15-3 C8H8N2S
5-methyl-2-(1H-pyrrol-2-yl)-1,3-thiazole
—— 5-fluoro-2-{[4-(6-methoxy-2,3-dihydro-1H-indol-1-yl)-4-oxobutyl]thio}benzoic acid 1229952-40-2 C20H20FNO4S
5-fluoro-2-{[4-(6-methoxy-2,3-dihydro-1H-indol-1-yl)-4-oxobutyl]thio}benzoic acid
—— 5-chloro-2-({[3-(cyclohex-1-en-1-yl)phenyl]carbonyl}amino)benzoic acid 1247823-78-4 C20H18ClNO3
5-chloro-2-({[3-(cyclohex-1-en-1-yl)phenyl]carbonyl}amino)benzoic acid
—— 5-(3-[(1S)-2-methoxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyridine-2-sulfonamide 1177419-94-1 C24H28N4O6S
5-(3-[(1S)-2-methoxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyridine-2-sulfonamide
—— 5-(3-[(1S)-2-methoxy-1-methylethoxy]-5-{5-[(4R,5S)-5-methyl-4-{[(triisopropylsilyl)oxy]methyl}-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-2-(methylsulfonyl)pyridine 1177421-22-5 C34H49N3O7SSi
5-(3-[(1S)-2-methoxy-1-methylethoxy]-5-{5-[(4R,5S)-5-methyl-4-{[(triisopropylsilyl)oxy]methyl}-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-2-(methylsulfonyl)pyridine
—— 5-(3-{5-[(4R,5S)-4,5-dimethyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}-5-[(1S)-2-methoxy-1-methylethoxy]phenoxy)-2-(methylsulfonyl)pyridine 1177420-99-3 C25H29N3O6S
5-(3-{5-[(4R,5S)-4,5-dimethyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}-5-[(1S)-2-methoxy-1-methylethoxy]phenoxy)-2-(methylsulfonyl)pyridine
—— (5S)-2-(5-{3-[(1S)-2-methoxy-1-methylethoxy]-5-[4-(methylsulfonyl)phenoxy]phenyl}-1H-pyrrol-2-yl)-5-{[(triisopropylsilyl)oxy]methyl}-4,5-dihydro-1,3-oxazole 1177420-48-2 C34H48N2O7SSi
(5S)-2-(5-{3-[(1S)-2-methoxy-1-methylethoxy]-5-[4-(methylsulfonyl)phenoxy]phenyl}-1H-pyrrol-2-yl)-5-{[(triisopropylsilyl)oxy]methyl}-4,5-dihydro-1,3-oxazole
—— 5-(5-bromopyridin-2-yl)-2-chloro-4-methyloxazole 1146696-22-1 C9H6BrClN2O
5-(5-bromopyridin-2-yl)-2-chloro-4-methyloxazole
—— 5-(3-[(1S)-2-hydroxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyridine-2-carboxamide 1177419-96-3 C24H26N4O5
5-(3-[(1S)-2-hydroxy-1-methylethoxy]-5-{5-[(5S)-5-methyl-4,5-dihydro-1,3-oxazol-2-yl]-1H-pyrrol-2-yl}phenoxy)-N-methylpyridine-2-carboxamide
—— 5-[2-(2-chloro-4-methoxy-phenyl)-acetyl]-1,3-dimethyl-1,3-dihydro-benzoimidazol-2-one 1246685-15-3 C18H17ClN2O3
5-[2-(2-chloro-4-methoxy-phenyl)-acetyl]-1,3-dimethyl-1,3-dihydro-benzoimidazol-2-one
—— 5-(1-tert-butoxycarbonyl-2-propyl-pyrrolidine-2-carbonyl)-indole-1-carboxylic acid tert-butyl ester 1033820-24-4 C26H36N2O5
5-(1-tert-butoxycarbonyl-2-propyl-pyrrolidine-2-carbonyl)-indole-1-carboxylic acid tert-butyl ester
—— 5-(4-fluoro-4-piperidinyl)quinoline 876922-61-1 C14H15FN2
5-(4-fluoro-4-piperidinyl)quinoline
—— 5-benzofuran-2-yl-methyl-3-methoxy-2-(2,4,6-trimethylphenyl)cyclopent-2-enone 1229581-30-9 C24H24O3
5-benzofuran-2-yl-methyl-3-methoxy-2-(2,4,6-trimethylphenyl)cyclopent-2-enone