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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-{9-Isobutyl-8-[4-(methylsulfonyl)-1,4-diazepan-1-yl]-6-morpholin-4-yl-9H-purin-2-yl}pyrimidin-2-amine 1222104-26-8 C23H34N10O3S
5-{9-Isobutyl-8-[4-(methylsulfonyl)-1,4-diazepan-1-yl]-6-morpholin-4-yl-9H-purin-2-yl}pyrimidin-2-amine
—— 5-[4-(cyclopropylsulfonyl)phenyl]-1-[5-(1,2-dihydroxy-2-methylpropyl)-1,3-thiazol-2-yl]-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080060-83-8 C27H35NO7S2
5-[4-(cyclopropylsulfonyl)phenyl]-1-[5-(1,2-dihydroxy-2-methylpropyl)-1,3-thiazol-2-yl]-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-methyl-5-[5-(methylsulfanyl)pyridin-2-yl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080061-36-4 C23H28N2O3S
5-methyl-5-[5-(methylsulfanyl)pyridin-2-yl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[3-fluoro-4-(methylsulfanyl)phenyl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080061-15-9 C23H26FNO3S
5-[3-fluoro-4-(methylsulfanyl)phenyl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[3-chloro-4-(methylsulfonyl)phenyl]-1-[5-(1,3-dioxolan-2-yl)pyridin-2-yl]-6-[(2R,3R,7R)-2,3-diphenyl-1,4-dioxaspiro[4.4]non-7-yl]hexane-1,4-dione 1080061-06-8 C40H40ClNO8S
5-[3-chloro-4-(methylsulfonyl)phenyl]-1-[5-(1,3-dioxolan-2-yl)pyridin-2-yl]-6-[(2R,3R,7R)-2,3-diphenyl-1,4-dioxaspiro[4.4]non-7-yl]hexane-1,4-dione
—— 5-[4-(cyclopropylsulfonyl)phenyl]-6-(tetrahydro-2H-pyran-4-yl)-1-{5-[(tetrahydro-2H-pyran-2-yloxy)methyl]-1,3-thiazol-2-yl}hexane-1,4-dione 1080060-58-7 C29H37NO7S2
5-[4-(cyclopropylsulfonyl)phenyl]-6-(tetrahydro-2H-pyran-4-yl)-1-{5-[(tetrahydro-2H-pyran-2-yloxy)methyl]-1,3-thiazol-2-yl}hexane-1,4-dione
—— 5-(2,2,2-trifluoro-1-hydroxyethyl)-1,3-thiazole-2-carbaldehyde 1080060-76-9 C6H4F3NO2S
5-(2,2,2-trifluoro-1-hydroxyethyl)-1,3-thiazole-2-carbaldehyde
—— 5-[5-(methylsulfanyl)pyridin-2-yl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080061-12-6 C22H26N2O3S
5-[5-(methylsulfanyl)pyridin-2-yl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-(2-methyl-5-[1,4]oxazepan-4-yl-pentanoylamino)-3-(6-methyl-pyridin-3-yl)-pyrazole-1-carboxylic acid tert-butyl ester 1205531-98-1 C25H37N5O4
5-(2-methyl-5-[1,4]oxazepan-4-yl-pentanoylamino)-3-(6-methyl-pyridin-3-yl)-pyrazole-1-carboxylic acid tert-butyl ester
—— 5-[4-(methylsulfonyl)phenyl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080060-01-0 C23H27NO5S
5-[4-(methylsulfonyl)phenyl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[3-chloro-4-(methylsulfonyl)phenyl]-6-[(2R,3R,7R)-2,3-diphenyl-1,4-dioxaspiro[4.4]non-7-yl]-1-(pyridin-2-yl)hexane-1,4-dione 1080060-99-6 C37H36ClNO6S
5-[3-chloro-4-(methylsulfonyl)phenyl]-6-[(2R,3R,7R)-2,3-diphenyl-1,4-dioxaspiro[4.4]non-7-yl]-1-(pyridin-2-yl)hexane-1,4-dione
—— 5-(2-(azetidin-1-yl)-2-oxoethyl)-2-(5-{1-[4-(cyclopropylsulfonyl)phenyl]-2-(tetrahydro-2H-pyran-4-yl)ethyl}-1H-pyrrol-2-yl)pyridine 1080062-78-7 C30H35N3O4S
5-(2-(azetidin-1-yl)-2-oxoethyl)-2-(5-{1-[4-(cyclopropylsulfonyl)phenyl]-2-(tetrahydro-2H-pyran-4-yl)ethyl}-1H-pyrrol-2-yl)pyridine
—— [5-({[tert-butyl(diphenyl)silyl]oxy}methyl)-1,3,4-thiadiazol-2-yl]methanol 1080061-25-1 C20H24N2O2SSi
[5-({[tert-butyl(diphenyl)silyl]oxy}methyl)-1,3,4-thiadiazol-2-yl]methanol
—— 5-(1-{[tert-butyl(dimethyl)silyl]oxy}ethyl)-2-(5-{1-[4-(cyclopropylsulfonyl)phenyl]-2-(tetrahydro-2H-pyran-4-yl)ethyl}-3-methyl-1H-pyrrol-2-yl)pyridine 1080062-41-4 C34H48N2O4SSi
5-(1-{[tert-butyl(dimethyl)silyl]oxy}ethyl)-2-(5-{1-[4-(cyclopropylsulfonyl)phenyl]-2-(tetrahydro-2H-pyran-4-yl)ethyl}-3-methyl-1H-pyrrol-2-yl)pyridine
—— 5-(4-Chlorophenyl)-2-({[4-(3-thienylmethoxy)phenyl]acetyl}amino)indan-2-carboxylic acid 907947-75-5 C29H24ClNO4S
5-(4-Chlorophenyl)-2-({[4-(3-thienylmethoxy)phenyl]acetyl}amino)indan-2-carboxylic acid
—— 5-[(tetrahydro-2H-pyran-2-yloxy)methyl]-1,3-thiazole-2-carbaldehyde 1080060-57-6 C10H13NO3S
5-[(tetrahydro-2H-pyran-2-yloxy)methyl]-1,3-thiazole-2-carbaldehyde
—— 5-methyl-2,3,5,6-tetrahydropyrido[2,3-b][1,5]diazocin-4(1H)-one 1003023-91-3 C10H13N3O
5-methyl-2,3,5,6-tetrahydropyrido[2,3-b][1,5]diazocin-4(1H)-one
—— 5-(4-Fluoro-3-hydroxyphenyl)-4,4-dimethyl-2,4-dihydropyrazol-3-one 1010801-09-8 C11H11FN2O2
5-(4-Fluoro-3-hydroxyphenyl)-4,4-dimethyl-2,4-dihydropyrazol-3-one
—— 5-[(4-fluoro-1-methylpiperidin-4-yl)carbonyl]-N-(3-fluoro-6-methylpyridin-2-yl)-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-amine 1046787-26-1 C20H26F2N6O
5-[(4-fluoro-1-methylpiperidin-4-yl)carbonyl]-N-(3-fluoro-6-methylpyridin-2-yl)-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-amine
—— 5-[3-chloro-4-(methylsulfonyl)phenyl]-6-(tetrahydro-2H-pyran-4-yl)-1-{5-[(tetrahydro-2H-pyran-2-yloxy)methyl]-1,3-thiazol-2-yl}hexane-1,4-dione 1080061-04-6 C27H34ClNO7S2
5-[3-chloro-4-(methylsulfonyl)phenyl]-6-(tetrahydro-2H-pyran-4-yl)-1-{5-[(tetrahydro-2H-pyran-2-yloxy)methyl]-1,3-thiazol-2-yl}hexane-1,4-dione
—— 5-[3-chloro-4-(methylsulfonyl)phenyl]-1-[5-(2,2-dimethyl-1,3-dioxolan-4-yl)pyridin-2-yl]-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080060-18-9 C28H34ClNO7S
5-[3-chloro-4-(methylsulfonyl)phenyl]-1-[5-(2,2-dimethyl-1,3-dioxolan-4-yl)pyridin-2-yl]-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[4-(cyclopropylsulfonyl)phenyl]-1-{5-[2-methoxy-1-(tetrahydro-2H-pyran-2-yloxy)ethyl]pyridin-2-yl}-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080060-90-7 C33H43NO8S
5-[4-(cyclopropylsulfonyl)phenyl]-1-{5-[2-methoxy-1-(tetrahydro-2H-pyran-2-yloxy)ethyl]pyridin-2-yl}-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[4-(cyclopropylsulfonyl)phenyl]-1-[5-(1-hydroxy-2-methoxyethyl)-1,3-thiazol-2-yl]-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080060-67-8 C26H33NO7S2
5-[4-(cyclopropylsulfonyl)phenyl]-1-[5-(1-hydroxy-2-methoxyethyl)-1,3-thiazol-2-yl]-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[(2-methoxyethoxy)methyl]-1,3-thiazole-2-carbaldehyde 1080060-70-3 C8H11NO3S
5-[(2-methoxyethoxy)methyl]-1,3-thiazole-2-carbaldehyde
—— 5-(1,2-dihydroxy-2-methylpropyl)-1,3-thiazole-2-carbaldehyde 1080060-82-7 C8H11NO3S
5-(1,2-dihydroxy-2-methylpropyl)-1,3-thiazole-2-carbaldehyde
—— 5-[3-chloro-4-(methylsulfonyl)phenyl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione 1080061-03-5 C23H26ClNO5S
5-[3-chloro-4-(methylsulfonyl)phenyl]-1-(pyridin-2-yl)-6-(tetrahydro-2H-pyran-4-yl)hexane-1,4-dione
—— 5-[9-(Cyclopropylmethyl)-6,8-dimorpholin-4-yl-9H-purin-2-yl]pyrimidin-2-amine 1222103-98-1 C21H27N9O2
5-[9-(Cyclopropylmethyl)-6,8-dimorpholin-4-yl-9H-purin-2-yl]pyrimidin-2-amine
—— 5-[4-(cyclopropylsulfonyl)phenyl]-6-(tetrahydro-2H-pyran-4-yl)-1-[5-(2,2,2-trifluoro-1-hydroxyethyl)-1,3-thiazol-2-yl]hexane-1,4-dione 1080060-77-0 C25H28F3NO6S2
5-[4-(cyclopropylsulfonyl)phenyl]-6-(tetrahydro-2H-pyran-4-yl)-1-[5-(2,2,2-trifluoro-1-hydroxyethyl)-1,3-thiazol-2-yl]hexane-1,4-dione
—— 5-[9-(cyclopropylmethyl)-6-morpholin-4-yl-9H-purin-2-yl]-N-methylpyrimidin-2-amine 1222105-72-7 C18H22N8O
5-[9-(cyclopropylmethyl)-6-morpholin-4-yl-9H-purin-2-yl]-N-methylpyrimidin-2-amine
—— 5-[6,8-dimorpholin-4-yl-9-(tetrahydrofuran-3-ylmethyl)-9H-purin-2-yl]pyrimidin-2-amine 1222104-01-9 C22H29N9O3
5-[6,8-dimorpholin-4-yl-9-(tetrahydrofuran-3-ylmethyl)-9H-purin-2-yl]pyrimidin-2-amine
—— 5-[3-(acetylamino)phenyl]-1-benzothiophene-2-carboxylic acid 907945-23-7 C17H13NO3S
5-[3-(acetylamino)phenyl]-1-benzothiophene-2-carboxylic acid
—— 5-[8-(4-acetylpiperazin-1-yl)-6-morpholin-4-yl-9-(2,2,2-trifluoroethyl)-9H-purin-2-yl]-N-methylpyrimidin-2-amine 1222105-19-2 C22H27F3N10O2
5-[8-(4-acetylpiperazin-1-yl)-6-morpholin-4-yl-9-(2,2,2-trifluoroethyl)-9H-purin-2-yl]-N-methylpyrimidin-2-amine
—— 5-methyl-N-[3-[(1S)-1-[(6-morpholin-4-ylpyrazin-2-yl)amino]ethyl]phenyl]pyridine-3-carboxamide 1027254-01-8 C23H26N6O2
5-methyl-N-[3-[(1S)-1-[(6-morpholin-4-ylpyrazin-2-yl)amino]ethyl]phenyl]pyridine-3-carboxamide
—— 5-[9-(cyclopropylmethyl)-6-morpholin-4-yl-8-piperazin-1-ylpurin-2-yl]-N,4-dimethylpyrimidin-2-amine 1222106-08-2 C23H32N10O
5-[9-(cyclopropylmethyl)-6-morpholin-4-yl-8-piperazin-1-ylpurin-2-yl]-N,4-dimethylpyrimidin-2-amine
—— 5-amino-3-(6-methoxy-pyridin-3-yl)-pyrazole-1-carboxylic acid tert-butyl ester 1205531-55-0 C14H18N4O3
5-amino-3-(6-methoxy-pyridin-3-yl)-pyrazole-1-carboxylic acid tert-butyl ester
—— 5-[6-Morpholin-4-yl-9-(tetrahydrofuran-3-ylmethyl)-9H-purin-2-yl]pyrimidin-2-amine 1222105-39-6 C18H22N8O2
5-[6-Morpholin-4-yl-9-(tetrahydrofuran-3-ylmethyl)-9H-purin-2-yl]pyrimidin-2-amine
—— 5-[6,8-dimorpholin-4-yl-9-(tetrahydrofuran-3-ylmethyl)-9H-purin-2-yl]-N-methylpyrimidin-2-amine 1222104-02-0 C23H31N9O3
5-[6,8-dimorpholin-4-yl-9-(tetrahydrofuran-3-ylmethyl)-9H-purin-2-yl]-N-methylpyrimidin-2-amine
—— 5-amino-3-(6-methyl-pyridin-3-yl)-pyrazole-1-carboxylic acid tert-butyl ester 1205531-60-7 C14H18N4O2
5-amino-3-(6-methyl-pyridin-3-yl)-pyrazole-1-carboxylic acid tert-butyl ester
—— 5-[8-(4,7-Diazaspiro[2.5]oct-7-yl)-6-morpholin-4-yl-9-(2,2,2-trifluoroethyl)-9H-purin-2-yl]pyrimidin-2-amine 1222105-03-4 C21H25F3N10O
5-[8-(4,7-Diazaspiro[2.5]oct-7-yl)-6-morpholin-4-yl-9-(2,2,2-trifluoroethyl)-9H-purin-2-yl]pyrimidin-2-amine
—— 5-[9-(cyclopropylmethyl)-6,8-dimorpholin-4-yl-9H-purin-2-yl]-N-methylpyrimidin-2-amine 1222104-17-7 C22H29N9O2
5-[9-(cyclopropylmethyl)-6,8-dimorpholin-4-yl-9H-purin-2-yl]-N-methylpyrimidin-2-amine
—— 5-{9-(cyclopropylmethyl)-8-[4-(methylsulfonyl)piperazin-1-yl]-6-morpholin-4-yl-9H-purin-2-yl}-N,N,4-trimethylpyrimidin-2-amine 1222104-22-4 C25H36N10O3S
5-{9-(cyclopropylmethyl)-8-[4-(methylsulfonyl)piperazin-1-yl]-6-morpholin-4-yl-9H-purin-2-yl}-N,N,4-trimethylpyrimidin-2-amine
—— 5-{9-(Cyclopropylmethyl)-6-morpholin-4-yl-8-[3-(phenylsulfonyl)pyrrolidin-1-yl]-9H-purin-2-yl}pyrimidin-2-amine 1222104-09-7 C27H31N9O3S
5-{9-(Cyclopropylmethyl)-6-morpholin-4-yl-8-[3-(phenylsulfonyl)pyrrolidin-1-yl]-9H-purin-2-yl}pyrimidin-2-amine
—— 5-[8-(4-acetyl-4,7-diazaspiro[2.5]oct-7-yl)-6-morpholin-4-yl-9-(2,2,2-trifluoroethyl)-9H-purin-2-yl]pyrimidin-2-amine 1222105-04-5 C23H27F3N10O2
5-[8-(4-acetyl-4,7-diazaspiro[2.5]oct-7-yl)-6-morpholin-4-yl-9-(2,2,2-trifluoroethyl)-9H-purin-2-yl]pyrimidin-2-amine
—— 5-(3-Methoxy-4-methoxymethyloxyphenyl)-4,4-dimethyl-2,4-dihydropyrazol-3-one 1093857-86-3 C14H18N2O4
5-(3-Methoxy-4-methoxymethyloxyphenyl)-4,4-dimethyl-2,4-dihydropyrazol-3-one
—— 5-(trifluoromethyl)-1H-benzo[d][1,2,3]triazole-7-carbaldehyde 1100215-68-6 C8H4F3N3O
5-(trifluoromethyl)-1H-benzo[d][1,2,3]triazole-7-carbaldehyde
—— 5-[4-(dimethylamino)phenyl]-1-benzothiophene-2-carboxylic acid 907945-28-2 C17H15NO2S
5-[4-(dimethylamino)phenyl]-1-benzothiophene-2-carboxylic acid
—— 5-(6-{2-[N-(tert-butoxycarbonyl)-N-methylamino]ethoxy}-2,3-difluorobenzyloxy)-2-fluoroaniline 1075700-86-5 C21H25F3N2O4
5-(6-{2-[N-(tert-butoxycarbonyl)-N-methylamino]ethoxy}-2,3-difluorobenzyloxy)-2-fluoroaniline
—— 5-(4-Chlorophenyl)-2-{[(4-fluorobenzyl)sulfonyl]amino}indan-2-carboxylic acid 907947-38-0 C23H19ClFNO4S
5-(4-Chlorophenyl)-2-{[(4-fluorobenzyl)sulfonyl]amino}indan-2-carboxylic acid
—— 5-(2-Fluoro-3-hydroxyphenyl)-4,4-dimethyl-2,4-dihydropyrazol-3-one 1010801-12-3 C11H11FN2O2
5-(2-Fluoro-3-hydroxyphenyl)-4,4-dimethyl-2,4-dihydropyrazol-3-one
—— 5,5'-([1,1'-Biphenyl]-4,4'-diyl)bis(8-phenyl-5H-pyrido[4,3-b]indole) 869799-62-2 C46H30N4
5,5'-([1,1'-Biphenyl]-4,4'-diyl)bis(8-phenyl-5H-pyrido[4,3-b]indole)