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苯和取代衍生物

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-chloro-N-[(dimethylamino)methylene]-3-(trifluoromethyl)benzamide 936220-62-1 C11H10ClF3N2O
2-chloro-N-[(dimethylamino)methylene]-3-(trifluoromethyl)benzamide
—— 2-acetylamino-3,5-dichloro-N-(4-cyclopropyl-benzyl)-N-[2-(3-trifluoromethoxy-phenyl)-ethyl]-benzamide 946117-66-4 C28H25Cl2F3N2O3
2-acetylamino-3,5-dichloro-N-(4-cyclopropyl-benzyl)-N-[2-(3-trifluoromethoxy-phenyl)-ethyl]-benzamide
—— 3-({1-[bis(4-chlorophenyl)methyl]azetidin-3-yl}(methanesulphonyl)amino)-5-fluorobenzoic acid methyl ester 1186130-02-8 C25H23Cl2FN2O4S
3-({1-[bis(4-chlorophenyl)methyl]azetidin-3-yl}(methanesulphonyl)amino)-5-fluorobenzoic acid methyl ester
—— N-(((3S,5S)-1-((R)-1,1-diphenylpropan-2-yl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)-2-naphthamide 1185650-06-9 C36H42N6O2
N-(((3S,5S)-1-((R)-1,1-diphenylpropan-2-yl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)-2-naphthamide
—— {[3'-({(butoxy carbonyl)[2-(butylamino)-2-oxoethyl]amino}methyl)-5-methylbiphenyl-2-yl]oxy} acetic acid 1171884-73-3 C27H36N2O6
{[3'-({(butoxy carbonyl)[2-(butylamino)-2-oxoethyl]amino}methyl)-5-methylbiphenyl-2-yl]oxy} acetic acid
—— 2-(2-(N-benzylphenylsulfonamido)ethoxy)-N-(4-((dimethylamino)(3-fluorophenyl)methyl)cyclohexyl)acetamide 1073597-05-3 C32H40FN3O4S
2-(2-(N-benzylphenylsulfonamido)ethoxy)-N-(4-((dimethylamino)(3-fluorophenyl)methyl)cyclohexyl)acetamide
—— (4-chloro-2-(hydroxymethyl)phenyl)boronic acid 1365244-07-0 C7H8BClO3
(4-chloro-2-(hydroxymethyl)phenyl)boronic acid
—— 4-(5-{[[1-(3,4-dichlorobenzoyl)piperidin-4-yl](methyl)amino]methyl}pyrazin-2-yl)-2-fluoro-N-propylbenzamide 1348760-04-2 C28H30Cl2FN5O2
4-(5-{[[1-(3,4-dichlorobenzoyl)piperidin-4-yl](methyl)amino]methyl}pyrazin-2-yl)-2-fluoro-N-propylbenzamide
—— N-(((3S,5S)-1-(2,2-diphenylethyl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)benzo[b]thiophene-5-carboxamide 1185582-56-2 C33H38N6O2S
N-(((3S,5S)-1-(2,2-diphenylethyl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)benzo[b]thiophene-5-carboxamide
—— 4-tert-butyl-N-(3-{8-[3-(2-hydroxyethyl)ureido]imidazo[1,2-b]pyridazin-6-yl}-2-methylphenyl)benzamide 1161846-60-1 C27H30N6O3
4-tert-butyl-N-(3-{8-[3-(2-hydroxyethyl)ureido]imidazo[1,2-b]pyridazin-6-yl}-2-methylphenyl)benzamide
—— 2-[2-[3-methoxy-4-(2-methyl-thiazol-5-yl)-phenylamino]-6-(4-trifluoromethyl-phenyl)-pyrimidin-4-yl]-propan-2-ol 1185018-22-7 C25H23F3N4O2S
2-[2-[3-methoxy-4-(2-methyl-thiazol-5-yl)-phenylamino]-6-(4-trifluoromethyl-phenyl)-pyrimidin-4-yl]-propan-2-ol
—— 3-(3-benzenesulfonylhydrazono-butyl)-3<i>H</i>-benzothiazol-2-one 69195-21-7 C17H17N3O3S2
3-(3-benzenesulfonylhydrazono-butyl)-3<i>H</i>-benzothiazol-2-one
—— Benzoic acid 4-[(2-indan-1-yl-ethyl)-methyl-amino]-butyl ester 69061-73-0 C23H29NO2
Benzoic acid 4-[(2-indan-1-yl-ethyl)-methyl-amino]-butyl ester
—— 2,2,2-Trichloro-1-(4-fluoro-phenyl)-ethylamine; hydrochloride 70123-03-4 C8H7Cl3FN*ClH
2,2,2-Trichloro-1-(4-fluoro-phenyl)-ethylamine; hydrochloride
—— N-[2-[2-[1-(6-fluoro-1-benzothiophen-3-yl)ethylidene]hydrazinyl]-2-oxoethyl]-3,4-dimethoxybenzamide 1569079-10-2 C21H20FN3O4S
N-[2-[2-[1-(6-fluoro-1-benzothiophen-3-yl)ethylidene]hydrazinyl]-2-oxoethyl]-3,4-dimethoxybenzamide
—— N-[N'-[(2-methoxyphenyl)methyl]-N-[5-(trifluoromethyl)-1H-pyrazol-3-yl]carbamimidoyl]-4-(trifluoromethyl)benzamide 1381836-84-5 C21H17F6N5O2
N-[N'-[(2-methoxyphenyl)methyl]-N-[5-(trifluoromethyl)-1H-pyrazol-3-yl]carbamimidoyl]-4-(trifluoromethyl)benzamide
—— Z-Aib-ONM 1240264-07-6 C18H20N2O8
Z-Aib-ONM
—— (E)-3-(3',4'-Dichloro-biphenyl-2-yl)-acrylic acid ethyl ester 371147-99-8 C17H14Cl2O2
(E)-3-(3',4'-Dichloro-biphenyl-2-yl)-acrylic acid ethyl ester
—— 1-(4-bromo-phenyl)-3-phenyl-2-thioxo-dihydro-pyrimidine-4,5,6-trione 5-[(2-methoxy-phenyl)-hydrazone] 70203-29-1 C23H17BrN4O3S
1-(4-bromo-phenyl)-3-phenyl-2-thioxo-dihydro-pyrimidine-4,5,6-trione 5-[(2-methoxy-phenyl)-hydrazone]
—— [1-(3,4-dimethoxy-phenethyl)-2-oxo-[4]piperidyl]-acetic acid 109156-86-7 C17H23NO5
[1-(3,4-dimethoxy-phenethyl)-2-oxo-[4]piperidyl]-acetic acid
—— phenyl 4-(bis(4-chlorophenyl)methyl)piperazine-1-carboxylate 1028991-81-2 C24H22Cl2N2O2
phenyl 4-(bis(4-chlorophenyl)methyl)piperazine-1-carboxylate
—— 5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-N,2-diphenyl-2H-1,2,3-triazole-4-carboxamide 1144525-60-9 C33H27N5O3
5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-N,2-diphenyl-2H-1,2,3-triazole-4-carboxamide
—— 2-(4-(tert-butyl)phenyl)-2-isothiocyanatoethyl pivalate 1375102-75-2 C18H25NO2S
2-(4-(tert-butyl)phenyl)-2-isothiocyanatoethyl pivalate
—— oxobis(triphenyl-l5-phosphaneyl)osmium(VII) chloride 25398-91-8 C36H30Cl3OOsP2
oxobis(triphenyl-l5-phosphaneyl)osmium(VII) chloride
—— {RuBr2(CS)(triphenylphosphine)3} 133982-77-1 C55H45Br2P3RuS
{RuBr2(CS)(triphenylphosphine)3}
—— 1-(2,6-dichloro-benzoyl)-2,3-dihydro-1<i>H</i>-imidazo[1,2-<i>a</i>]imidazole 67139-10-0 C12H9Cl2N3O
1-(2,6-dichloro-benzoyl)-2,3-dihydro-1<i>H</i>-imidazo[1,2-<i>a</i>]imidazole
—— 3-Buthoxytolyl-sulfochlorid 68978-30-3 C11H15ClO3S
3-Buthoxytolyl-sulfochlorid
—— 4-[5-(4-methoxy-phenyl)-1-<i>p</i>-tolyl-1<i>H</i>-[1,2,4]triazole-3-carbonylamino]-benzoic acid 68766-58-5 C24H20N4O4
4-[5-(4-methoxy-phenyl)-1-<i>p</i>-tolyl-1<i>H</i>-[1,2,4]triazole-3-carbonylamino]-benzoic acid
—— 1-Methyl-3-(2-chlor-1-hydroxy-1-phenyl-ethyl)-2-pyrrolidon 67506-05-2 C13H16ClNO2
1-Methyl-3-(2-chlor-1-hydroxy-1-phenyl-ethyl)-2-pyrrolidon
—— 2-chloro-<i>N</i>-[3-(2,3,5,6-tetrahydro-imidazo[2,1-<i>b</i>]thiazol-6-yl)-phenyl]-acetamide 59549-06-3 C13H14ClN3OS
2-chloro-<i>N</i>-[3-(2,3,5,6-tetrahydro-imidazo[2,1-<i>b</i>]thiazol-6-yl)-phenyl]-acetamide
—— 3-trimethylstannyl-N-diphenylmethylenealanine ethyl ester 224964-15-2 C21H27NO2Sn
3-trimethylstannyl-N-diphenylmethylenealanine ethyl ester
—— (2R<sup>*</sup>,4S<sup>*</sup>)-4-(ethoxycarbonyl)-2-phenyl-1-(phenylsulfonyl)-1,2,3,4-tetrahydropyridine 130146-90-6 C20H21NO4S
(2R<sup>*</sup>,4S<sup>*</sup>)-4-(ethoxycarbonyl)-2-phenyl-1-(phenylsulfonyl)-1,2,3,4-tetrahydropyridine
—— 1,1'-(1,4-phenylene)bis(propane-1,2-dione) 1587661-05-9 C12H10O4
1,1'-(1,4-phenylene)bis(propane-1,2-dione)
—— (E)-N-benzyl-5-amino-1-methoxypent-2-ene 634180-66-8 C13H19NO
(E)-N-benzyl-5-amino-1-methoxypent-2-ene
—— 4-[2-nitro-4-(trifluoromethyl)aniline]cyclohexanol 1012925-47-1 C13H15F3N2O3
4-[2-nitro-4-(trifluoromethyl)aniline]cyclohexanol
—— ethyl 4-[2-(benzofuran-2-ylcarbonylamino)ethoxy]benzoate 1101929-48-9 C20H19NO5
ethyl 4-[2-(benzofuran-2-ylcarbonylamino)ethoxy]benzoate
—— 130774-65-1 C32H27N4OP
—— dimethyl 2-ethyl-2,6,6-trimethyl-3-oxo-5-phenyl-1,7-heptanedioate 1242096-21-4 C20H28O5
dimethyl 2-ethyl-2,6,6-trimethyl-3-oxo-5-phenyl-1,7-heptanedioate
—— (2R)-2-[2-[(4-chlorophenyl)methyl]-1,2,4-triazol-3-yl]-N-[2-chloro-4-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide 1140489-08-2 C21H18Cl2F3N5O
(2R)-2-[2-[(4-chlorophenyl)methyl]-1,2,4-triazol-3-yl]-N-[2-chloro-4-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide
—— N-cyclopropyl-4-{8-[(2-methylpropyl)amino]6-(4-phenoxyphenyl)imidazo[1,2-a]pyrazin-3-yl}benzamide 1382478-21-8 C32H31N5O2
N-cyclopropyl-4-{8-[(2-methylpropyl)amino]6-(4-phenoxyphenyl)imidazo[1,2-a]pyrazin-3-yl}benzamide
—— (2R)-N-[(6S,8S)-3-cyclopropyl-6-(2,3-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-8-yl]-2'-oxospiro[1,3-dihydroindene-2,3'-1H-pyrrolo[2,3-b]pyridine]-5-carboxamide 1383733-31-0 C32H27F2N5O2
(2R)-N-[(6S,8S)-3-cyclopropyl-6-(2,3-difluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-8-yl]-2'-oxospiro[1,3-dihydroindene-2,3'-1H-pyrrolo[2,3-b]pyridine]-5-carboxamide
—— N-(6-chloropyridazin-3-yl)-2-[(3,4-dimethoxyphenyl)oxymethyl]-2-phenylcyclopropanecarboxamide 1383745-68-3 C23H22ClN3O4
N-(6-chloropyridazin-3-yl)-2-[(3,4-dimethoxyphenyl)oxymethyl]-2-phenylcyclopropanecarboxamide
—— (3,5-difluorophenyl)-[2-(phenoxymethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methanone 1380506-62-6 C20H17F2N3O2
(3,5-difluorophenyl)-[2-(phenoxymethyl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methanone
—— N-((1R,5S)-5-((4-aminophenylsulfonyl)(isopropyl)amino)-1-cyclopropyl-6-hydroxyhexyl)-Nα-methoxycarbonyl-β-phenyl-L-phenylalaninamide 1138084-21-5 C35H46N4O6S
N-((1R,5S)-5-((4-aminophenylsulfonyl)(isopropyl)amino)-1-cyclopropyl-6-hydroxyhexyl)-Nα-methoxycarbonyl-β-phenyl-L-phenylalaninamide
—— 3-((3,4-dichlorophenyl)(2-(trifluoromethoxy)phenoxy)methyl)azetidine hydrochloride 1398707-09-9 C17H14Cl2F3NO2*ClH
3-((3,4-dichlorophenyl)(2-(trifluoromethoxy)phenoxy)methyl)azetidine hydrochloride
—— 4-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)-1-[3-(1H-tetrazol-1-yl)benzoyl]piperidine 1138328-32-1 C23H24F3N5O3S
4-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)-1-[3-(1H-tetrazol-1-yl)benzoyl]piperidine
—— (Z)-3-cyclopentyl-5-[(4'-fluorobiphenyl-4-yl)methylene]-2-thioxothiazolidin-4-one 1149337-54-1 C21H18FNOS2
(Z)-3-cyclopentyl-5-[(4'-fluorobiphenyl-4-yl)methylene]-2-thioxothiazolidin-4-one
—— 2-chloro-3-([4-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)piperidin-1-yl]carbonyl)-6-(trifluoromethyl)pyridine 1138329-37-9 C22H21ClF6N2O3S
2-chloro-3-([4-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)piperidin-1-yl]carbonyl)-6-(trifluoromethyl)pyridine
—— 4-chlorobenzyl 4-[2-methyl-3-oxo-3-(2-oxo-2,3-dihydrobenzoxazol-6-yl)propyl]piperazine-1-carboxylate 1144036-92-9 C23H24ClN3O5
4-chlorobenzyl 4-[2-methyl-3-oxo-3-(2-oxo-2,3-dihydrobenzoxazol-6-yl)propyl]piperazine-1-carboxylate
—— 2-[(4-Chlorophenyl)methoxy]-3-methyl-4-(piperidin-4-yl)pyridine 1160872-46-7 C18H21ClN2O
2-[(4-Chlorophenyl)methoxy]-3-methyl-4-(piperidin-4-yl)pyridine