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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1,8,8-trimethyl-3-aza-bicyclo[3.2.1]octane-2,4-dione 402920-44-9 C21H25N3O3
3-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1,8,8-trimethyl-3-aza-bicyclo[3.2.1]octane-2,4-dione
—— 3-[5-cyclopropanecarbonyl-1-(2,4-difluorobenzyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile 1279839-85-8 C24H20F2N4O
3-[5-cyclopropanecarbonyl-1-(2,4-difluorobenzyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
—— N-(3-(5-(2-((3-methylphenyl)amino)pyrimidin-4-yl)imidazo[2,1-b][1,3]thiazol-6-yl)phenyl)-2-phenylacetamide 1159884-04-4 C30H24N6OS
N-(3-(5-(2-((3-methylphenyl)amino)pyrimidin-4-yl)imidazo[2,1-b][1,3]thiazol-6-yl)phenyl)-2-phenylacetamide
—— 2-(2-chlrophenyl)-1-(4-chlorophenyl)-N-[(2S)-2-(hydroxymethyl)-1-piperidinyl]-1H-imidazole-4-carboxamide 527361-11-1 C22H22Cl2N4O2
2-(2-chlrophenyl)-1-(4-chlorophenyl)-N-[(2S)-2-(hydroxymethyl)-1-piperidinyl]-1H-imidazole-4-carboxamide
—— 3-(2,4-dihydroxy-5-isopropylphenyl)-1-methyl-4-(1-methyl-1H-indol-5-yl)-1H-1,2,4-triazol-5(4H)-one 1207598-28-4 C21H22N4O3
3-(2,4-dihydroxy-5-isopropylphenyl)-1-methyl-4-(1-methyl-1H-indol-5-yl)-1H-1,2,4-triazol-5(4H)-one
—— 1207746-14-2 C23H19ClN2O2S
—— 5-(1-((2-(4,4-dimethylpiperidin-1-yl)pyridin-4-yl)methyl)-5-methyl-1H-1,2,4-triazol-3-yl)-3-(4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazole 1570494-96-0 C25H26F3N7O2
5-(1-((2-(4,4-dimethylpiperidin-1-yl)pyridin-4-yl)methyl)-5-methyl-1H-1,2,4-triazol-3-yl)-3-(4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazole
—— (R)-2-methoxy-N-(6-methoxy-3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-2-phenylacetamide 1338793-79-5 C23H22N4O5S
(R)-2-methoxy-N-(6-methoxy-3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-2-phenylacetamide
—— (4R,5R)-5-ethyl-4-methyl-6-(2-phenyl-benzoxazol-6-yl)-4,5-dihydro-2H-pyridazin-3-one 1346699-92-0 C20H19N3O2
(4R,5R)-5-ethyl-4-methyl-6-(2-phenyl-benzoxazol-6-yl)-4,5-dihydro-2H-pyridazin-3-one
—— (2R,3R)-2,3-dihydroxy-N-methyl-N'-[4-(1H-pyrazol-5-yl)phenyl]butanediamide 905445-74-1 C14H16N4O4
(2R,3R)-2,3-dihydroxy-N-methyl-N'-[4-(1H-pyrazol-5-yl)phenyl]butanediamide
—— (1H-imidazol-4-ylmethyl)-isopropyl-(1-phenyl-1H-pyrazol-3-yl)-amine 1020817-85-9 C16H19N5
(1H-imidazol-4-ylmethyl)-isopropyl-(1-phenyl-1H-pyrazol-3-yl)-amine
—— 5-Chloro-1-methyl-1H-pyrazole-4-carboxylic acid 2-acetylhydrazide 110763-10-5 C7H9ClN4O2
5-Chloro-1-methyl-1H-pyrazole-4-carboxylic acid 2-acetylhydrazide
—— (3-(1-(2-methoxyethyl)-3-phenyl-1H-pyrazol-5-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone 1338374-66-5 C28H26N6O2S
(3-(1-(2-methoxyethyl)-3-phenyl-1H-pyrazol-5-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone
—— 1193351-85-7 C17H12Cl2F2N2O
—— 4-[5-(4-chlorophenyl)-1-phenyl-1H-pyrazol-3-yl]-1-(2-phenylethyl)piperidine 1349861-84-2 C28H28ClN3
4-[5-(4-chlorophenyl)-1-phenyl-1H-pyrazol-3-yl]-1-(2-phenylethyl)piperidine
—— 1393095-73-2 C26H15Cl2F8N7O2
—— 3-[5-(4-fluorophenyl)-2-pyrimidin-2-ylpyrazol-3-yl]-N-(2-propan-2-ylphenyl)piperidine-1-carboxamide 1350880-83-9 C28H29FN6O
3-[5-(4-fluorophenyl)-2-pyrimidin-2-ylpyrazol-3-yl]-N-(2-propan-2-ylphenyl)piperidine-1-carboxamide
—— 1182280-97-2 C19H15F6N3O2S
—— 1577250-55-5 C18H12F6N8Pt
—— 1-(3,5-bis-trifluoromethyl-benzyl)-5-(4-methylsulfanyl-phenyl)-1H-[1,2,3]triazole-4-carboxylic acid methyl ester 823189-61-3 C20H15F6N3O2S
1-(3,5-bis-trifluoromethyl-benzyl)-5-(4-methylsulfanyl-phenyl)-1H-[1,2,3]triazole-4-carboxylic acid methyl ester
—— (S)-N-(3-fluoro-4-(5-methyl-1H-1,2,4-triazol-1-yl)phenyl)-9-(4-(trifluoromethoxy)phenyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[1,5-a]azepin-2-amine 1235495-29-0 C23H21F4N7O
(S)-N-(3-fluoro-4-(5-methyl-1H-1,2,4-triazol-1-yl)phenyl)-9-(4-(trifluoromethoxy)phenyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[1,5-a]azepin-2-amine
—— 2-(2-tert-butyl-2H-1,2,3,4-tetrazol-5-yl)ethan-1-ol 1955541-16-8 C7H14N4O
2-(2-tert-butyl-2H-1,2,3,4-tetrazol-5-yl)ethan-1-ol
—— (S)-N-(3-(1-(4-fluorophenyl)-1H-indazol-5-yl)-2,2-dimethyl-3-phenylpropyl)-4-methylpentanamide 1025766-67-9 C30H34FN3O
(S)-N-(3-(1-(4-fluorophenyl)-1H-indazol-5-yl)-2,2-dimethyl-3-phenylpropyl)-4-methylpentanamide
—— 1-(4-aminophenyl)-5-ethyl-1H-pyrazole-4-carboxamide 1172318-49-8 C12H14N4O
1-(4-aminophenyl)-5-ethyl-1H-pyrazole-4-carboxamide
—— N-[5-Amino-4,6-dicyano-2-phenyl-2H-pyridazin-(3E)-ylidene]-acetamide 123775-50-8 C14H10N6O
N-[5-Amino-4,6-dicyano-2-phenyl-2H-pyridazin-(3E)-ylidene]-acetamide
—— Methyl 2-(aminomethyl)-1,3-oxazole-4-carboxylate hydrochloride 1006619-33-5 C6H9ClN2O3
Methyl 2-(aminomethyl)-1,3-oxazole-4-carboxylate hydrochloride
—— 4-(4-Methoxy-phenylamino)-3-methyl-1-phenyl-1,4,4a,7a-tetrahydro-furo[3',4':5,6]selenino[2,3-c]pyrazole-5,7-dione 109576-89-8 C22H19N3O4Se
4-(4-Methoxy-phenylamino)-3-methyl-1-phenyl-1,4,4a,7a-tetrahydro-furo[3',4':5,6]selenino[2,3-c]pyrazole-5,7-dione
—— 5-{3,5-dimethyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl}-3-{(1R)-1-[5-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]ethoxy}pyridin-2-amine 1346816-31-6 C22H24FN7O3S
5-{3,5-dimethyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl}-3-{(1R)-1-[5-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]ethoxy}pyridin-2-amine
—— bis(2-propyl)-4-amino-6-bromo-5-cyano-1-(2-phosphonomethoxyethyl)pyrrolo<2,3-d>pyrimidine 151965-52-5 C16H23BrN5O4P
bis(2-propyl)-4-amino-6-bromo-5-cyano-1-(2-phosphonomethoxyethyl)pyrrolo<2,3-d>pyrimidine
—— ethyl 2-(2-((4-chlorophenyl)(diethoxyphosphoryl)methylamino)thiazol-4-yl)-2-(methoxyimino)acetate 1456776-36-5 C19H25ClN3O6PS
ethyl 2-(2-((4-chlorophenyl)(diethoxyphosphoryl)methylamino)thiazol-4-yl)-2-(methoxyimino)acetate
—— 4-((3,5-Dibromo-2-hydroxybenzylidene)amino)-3-(2-methoxyphenyl)-1H-1,2,4-triazole-5(4H)-thione 478257-38-4 C16H12Br2N4O2S
4-((3,5-Dibromo-2-hydroxybenzylidene)amino)-3-(2-methoxyphenyl)-1H-1,2,4-triazole-5(4H)-thione
—— N-(cyclohexylmethyl)-3-(3-sulfamoylphenyl)-1H-indazole-5-carboxamide 1338794-34-5 C21H24N4O3S
N-(cyclohexylmethyl)-3-(3-sulfamoylphenyl)-1H-indazole-5-carboxamide
—— (S)-N-(4-methylbenzyl)-1-(2-(4-(oxazol-5-yl)phenylamino)pyrimidin-4-yl)piperidine-3-carboxamide 1347757-91-8 C27H28N6O2
(S)-N-(4-methylbenzyl)-1-(2-(4-(oxazol-5-yl)phenylamino)pyrimidin-4-yl)piperidine-3-carboxamide
—— 3-(2,5-dichlorophenyl)-5-[3-(3-cyclopentyloxy-4-methoxyphenyl)-5-methyl-4,5-dihydro-isoxazol-5-yl]-[1,2,4]oxadiazole 853582-23-7 C24H23Cl2N3O4
3-(2,5-dichlorophenyl)-5-[3-(3-cyclopentyloxy-4-methoxyphenyl)-5-methyl-4,5-dihydro-isoxazol-5-yl]-[1,2,4]oxadiazole
—— 1154098-42-6 C21H20FN5O3
—— 1199801-15-4 C22H15ClN4OS
—— 1199801-12-1 C23H15ClN4O2S
—— (5-methyl-1-phenyl-1H-1,2,3-triazol-4-yl)(5-methyl-3-phenyl-1H-pyrazol-1-yl)methanone 1333229-33-6 C20H17N5O
(5-methyl-1-phenyl-1H-1,2,3-triazol-4-yl)(5-methyl-3-phenyl-1H-pyrazol-1-yl)methanone
—— [3-(4-Chloro-phenyl)-1-(3-trifluoromethyl-phenyl)-1H-pyrazol-4-yl]-acetyl chloride 1026189-85-4 C18H11Cl2F3N2O
[3-(4-Chloro-phenyl)-1-(3-trifluoromethyl-phenyl)-1H-pyrazol-4-yl]-acetyl chloride
—— US10138229, Example 112 1558037-43-6 C22H25N5O3
US10138229, Example 112
—— 8-(2,6-dichlorophenyl)-9-[[(3R)-piperidin-3-yl]methyl]-N-[(5-pyridin-2-ylthiophen-2-yl)methyl]purin-2-amine 1021696-63-8 C27H25Cl2N7S
8-(2,6-dichlorophenyl)-9-[[(3R)-piperidin-3-yl]methyl]-N-[(5-pyridin-2-ylthiophen-2-yl)methyl]purin-2-amine
—— N,4,5-Trimethyl-I+/--3-thienyl-2-thiazolemethanamine 1249298-71-2 C11H14N2S2
N,4,5-Trimethyl-I+/--3-thienyl-2-thiazolemethanamine
—— 1-(4-chlorophenyl)-3,5-diphenyl-1H-pyrazole 53187-39-6 C21H15ClN2
1-(4-chlorophenyl)-3,5-diphenyl-1H-pyrazole
—— (1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (1-morpholin-4-yl-cyclopentylmethyl)-amide 1268877-34-4 C24H28F2N4O2
(1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (1-morpholin-4-yl-cyclopentylmethyl)-amide
—— 5-methyl-6-(5-{4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 1286750-87-5 C21H23N3O2*ClH
5-methyl-6-(5-{4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydroisoquinoline hydrochloride
—— 5-(2-Methylpropanoylamino)-3-(3-oxo-2-isopropyl-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridine 403492-97-7 C24H25N5O2
5-(2-Methylpropanoylamino)-3-(3-oxo-2-isopropyl-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridine
—— N-(2-Hydroxyethyl)-3-(3-oxo-2-isopropyl-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridine-5-carboxamide 403491-53-2 C23H23N5O3
N-(2-Hydroxyethyl)-3-(3-oxo-2-isopropyl-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridine-5-carboxamide
—— 4-[1-(4-fluorophenyl)-4-trifluoromethyl-1H-imidazol-2-yl]benzenesulfonamide 189297-20-9 C16H11F4N3O2S
4-[1-(4-fluorophenyl)-4-trifluoromethyl-1H-imidazol-2-yl]benzenesulfonamide
—— (3S)-N-[[2-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-5-(2,6-dimethyl-4-pyridinyl)-4-thiazolyl]methyl]tetrahydro-3-furancarboxamide 1309442-07-6 C22H30N4O3S
(3S)-N-[[2-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-5-(2,6-dimethyl-4-pyridinyl)-4-thiazolyl]methyl]tetrahydro-3-furancarboxamide
—— 3-[3-Aminophenyl]-5-[2-[(3,4,5-trimethoxyphenyl)amino]-4-amino-5-thiazolyl]-1,2,4-oxadiazole 312762-59-7 C20H20N6O4S
3-[3-Aminophenyl]-5-[2-[(3,4,5-trimethoxyphenyl)amino]-4-amino-5-thiazolyl]-1,2,4-oxadiazole