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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-((4-(4-((naphthalen-2-yloxy)methyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonyl)-1,2,3,4-tetrahydroisoquinoline 1615201-23-4 C28H24N4O3S
2-((4-(4-((naphthalen-2-yloxy)methyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonyl)-1,2,3,4-tetrahydroisoquinoline
—— 1-(2-hydroxy-2-(4-(5-(5-phenyl-4-propylisoxazol-3-yl)-1,2,4-oxadiazol-3-yl)phenyl)ethyl)pyrrolidine-3-carboxylic acid 1265321-67-2 C27H28N4O5
1-(2-hydroxy-2-(4-(5-(5-phenyl-4-propylisoxazol-3-yl)-1,2,4-oxadiazol-3-yl)phenyl)ethyl)pyrrolidine-3-carboxylic acid
—— 2-(2-chloroethyl)-2,5,6,7-tetrahydro-3H-pyrrolo[2,1-c]-1,2,4-triazol-3-one 133365-54-5 C7H10ClN3O
2-(2-chloroethyl)-2,5,6,7-tetrahydro-3H-pyrrolo[2,1-c]-1,2,4-triazol-3-one
—— 6,7-dimethoxy-2-((4-(4-((naphthalen-2-yloxy)methyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonyl)-1,2,3,4-tetrahydroisoquinoline 1615201-33-6 C30H28N4O5S
6,7-dimethoxy-2-((4-(4-((naphthalen-2-yloxy)methyl)-1H-1,2,3-triazol-1-yl)phenyl)sulfonyl)-1,2,3,4-tetrahydroisoquinoline
—— 5-[2-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-oxazole 1146694-93-0 C11H7F4NO
5-[2-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-oxazole
—— 3-(4-(oxiran-2-yl)phenyl)-5-(5-phenyl-4-propylisoxazol-3-yl)-1,2,4-oxadiazole 1265323-45-2 C22H19N3O3
3-(4-(oxiran-2-yl)phenyl)-5-(5-phenyl-4-propylisoxazol-3-yl)-1,2,4-oxadiazole
—— 2-(1-(2-hydroxy-2-(4-(5-(5-phenyl-4-propylisoxazol-3-yl)-1,2,4-oxadiazol-3-yl)phenyl)ethyl)piperidin-3-yl)acetic acid 1265322-06-2 C29H32N4O5
2-(1-(2-hydroxy-2-(4-(5-(5-phenyl-4-propylisoxazol-3-yl)-1,2,4-oxadiazol-3-yl)phenyl)ethyl)piperidin-3-yl)acetic acid
—— 2-methyl-4-(5-methyl-2-thienyl)-1,3-thiazole 1450665-80-1 C9H9NS2
2-methyl-4-(5-methyl-2-thienyl)-1,3-thiazole
—— 5-(5-phenyl-4-propylisoxazol-3-yl)-3-(4-vinylphenyl)-1,2,4-oxadiazole 1265323-43-0 C22H19N3O2
5-(5-phenyl-4-propylisoxazol-3-yl)-3-(4-vinylphenyl)-1,2,4-oxadiazole
—— N-{3-[1-(1-acetylpiperidin-4-yl)-4-(2-aminopyridin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluorobenzenesulfonamide 1357587-19-9 C27H25F3N6O3S
N-{3-[1-(1-acetylpiperidin-4-yl)-4-(2-aminopyridin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluorobenzenesulfonamide
—— 5-fluoro-1-(3-fluoro-4-hydroxyphenyl)-1H-indazol-4-ol 1056262-30-6 C13H8F2N2O2
5-fluoro-1-(3-fluoro-4-hydroxyphenyl)-1H-indazol-4-ol
—— 4-bromo-5-fluoro-1-{3-fluoro-4-[(phenylmethyl)oxy]phenyl}-1H-indazole 1056264-29-9 C20H13BrF2N2O
4-bromo-5-fluoro-1-{3-fluoro-4-[(phenylmethyl)oxy]phenyl}-1H-indazole
—— 1-Imidazol-1-yl-4,4-dimethyl-2-phenylpentan-3-one 95546-24-0 C16H20N2O
1-Imidazol-1-yl-4,4-dimethyl-2-phenylpentan-3-one
—— 5-amino-4-carboxamido-3-methyl-1-phenylfuro[2,3-c]pyrazole 112036-75-6 C13H12N4O2
5-amino-4-carboxamido-3-methyl-1-phenylfuro[2,3-c]pyrazole
—— 5-amino-3-methyl-1-phenyl-1H-pyrazolo[4,5-d][1,3]oxazole 252937-67-0 C11H10N4O
5-amino-3-methyl-1-phenyl-1H-pyrazolo[4,5-d][1,3]oxazole
—— 5-amino-3-methyl-1-phenyl-1H-pyrazolo[4,5-d][1,3]thiazole 252937-68-1 C11H10N4S
5-amino-3-methyl-1-phenyl-1H-pyrazolo[4,5-d][1,3]thiazole
—— 4-[3-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl]pyridine-2-carboxamide 1357587-40-6 C27H25F3N6O3S
4-[3-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl]pyridine-2-carboxamide
—— 2-Amino-3-cyano-4-methyl-6-phenylfuro<2,3-c>pyrazole 112036-72-3 C13H10N4O
2-Amino-3-cyano-4-methyl-6-phenylfuro<2,3-c>pyrazole
—— 2-(3-methoxypiperidin-1-yl)-4-trifluoromethyloxazole-5-carboxylic acid 1227934-94-2 C11H13F3N2O4
2-(3-methoxypiperidin-1-yl)-4-trifluoromethyloxazole-5-carboxylic acid
—— 1-phenyl-3-methyl-4-nitroso-2-pyrazolin-5-thione 66479-47-8 C10H9N3OS
1-phenyl-3-methyl-4-nitroso-2-pyrazolin-5-thione
—— 3-methyl-1-phenylpyrazolo[3,4-d][1,3]thiazol-5-amine 297158-57-7 C11H10N4S
3-methyl-1-phenylpyrazolo[3,4-d][1,3]thiazol-5-amine
—— 1H-Pyrazole-3-carboxamide, 5-(4-methylphenyl)-N-2-thiazolyl- 130421-53-3 C14H12N4OS
1H-Pyrazole-3-carboxamide, 5-(4-methylphenyl)-N-2-thiazolyl-
—— N'-(4-methoxybenzoyl)-5-(4-methylphenyl)-1-phenylpyrazole-3-carbohydrazide 124928-40-1 C25H22N4O3
N'-(4-methoxybenzoyl)-5-(4-methylphenyl)-1-phenylpyrazole-3-carbohydrazide
—— N-{3-[4-(2-aminopyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluorobenzenesulfonamide 1357587-06-4 C26H25F3N6O2S
N-{3-[4-(2-aminopyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluorobenzenesulfonamide
—— (R)-4-(8-amino-3-(1-(3-methyloxetane-3-carbonyl)piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419214-33-7 C29H28F3N7O3
(R)-4-(8-amino-3-(1-(3-methyloxetane-3-carbonyl)piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— 4-(4-(2-cyanopyridin-4-yl)-3-{3-[(2,5-difluorobenzenesulfonyl)methoxymethylamino]-2-fluorophenyl}pyrazol-1-yl)piperidine-1-carboxylic acid tert-butyl ester 1357588-20-5 C33H33F3N6O5S
4-(4-(2-cyanopyridin-4-yl)-3-{3-[(2,5-difluorobenzenesulfonyl)methoxymethylamino]-2-fluorophenyl}pyrazol-1-yl)piperidine-1-carboxylic acid tert-butyl ester
—— N-{3-[4-(2-tert-butylaminopyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide 1357587-99-5 C32H37F3N6O3S
N-{3-[4-(2-tert-butylaminopyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide
—— 4-(3-{3-[(2,5-difluorobenzenesulfonyl)methoxymethylamino]-2-fluorophenyl}-4-pyridin-4-ylpyrazol-1-yl)piperidine-1-carboxylic acid tert-butyl ester 1357587-67-7 C32H34F3N5O5S
4-(3-{3-[(2,5-difluorobenzenesulfonyl)methoxymethylamino]-2-fluorophenyl}-4-pyridin-4-ylpyrazol-1-yl)piperidine-1-carboxylic acid tert-butyl ester
—— (R)-benzyl 3-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)piperidine-1-carboxylate 1419214-71-3 C32H28F3N7O3
(R)-benzyl 3-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)piperidine-1-carboxylate
—— N-{3-[1-(1-acetylpiperidin-4-yl)-4-(2-tert-butylaminopyridin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide 1357588-00-1 C33H37F3N6O4S
N-{3-[1-(1-acetylpiperidin-4-yl)-4-(2-tert-butylaminopyridin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide
—— tert-butyl 1-(4-(2-phenyl-3H-imidazo[4,5-b]pyridin-3-yl)phenyl)cyclobutylcarbamate 1439394-18-9 C27H28N4O2
tert-butyl 1-(4-(2-phenyl-3H-imidazo[4,5-b]pyridin-3-yl)phenyl)cyclobutylcarbamate
—— N-{3-[4-(2-cyanopyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide 1357588-21-6 C29H27F3N6O3S
N-{3-[4-(2-cyanopyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide
—— (R)-4-(8-amino-3-(piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419214-70-2 C24H22F3N7O
(R)-4-(8-amino-3-(piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— N-{3-[4-(2-tert-butylaminopyridin-4-yl)-1-piperidin-4-yl-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide 1357587-98-4 C31H35F3N6O3S
N-{3-[4-(2-tert-butylaminopyridin-4-yl)-1-piperidin-4-yl-1H-pyrazol-3-yl]-2-fluorophenyl}-2,5-difluoro-N-methoxymethylbenzenesulfonamide
—— 2,5-difluoro-N-[2-fluoro-3-(2H-pyrazol-3-yl)-phenyl]-N-methoxymethylbenzenesulfonamide 1357587-48-4 C17H14F3N3O3S
2,5-difluoro-N-[2-fluoro-3-(2H-pyrazol-3-yl)-phenyl]-N-methoxymethylbenzenesulfonamide
—— 4-(1-(4-(perfluoroethoxy)phenyl)-1H-1,2,4-triazol-3-yl)aniline 1181214-79-8 C16H11F5N4O
4-(1-(4-(perfluoroethoxy)phenyl)-1H-1,2,4-triazol-3-yl)aniline
—— 2,5-difluoro-N-{2-fluoro-3-[1-(1-methylpiperidin-4-yl)-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}benzenesulfonamide 1357587-25-7 C28H25F3N6O2S
2,5-difluoro-N-{2-fluoro-3-[1-(1-methylpiperidin-4-yl)-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}benzenesulfonamide
—— 4-[3-{3-[(2,5-difluorobenzenesulfonyl)methoxymethylamino]-2-fluorophenyl}-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazol-1-yl]piperidine-1-carboxylic acid tert-butyl ester 1357588-08-9 C34H35F3N6O5S
4-[3-{3-[(2,5-difluorobenzenesulfonyl)methoxymethylamino]-2-fluorophenyl}-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazol-1-yl]piperidine-1-carboxylic acid tert-butyl ester
—— 5-methyl-2-(4-propoxy-phenyl)-benzooxazole 62725-23-9 C17H17NO2
5-methyl-2-(4-propoxy-phenyl)-benzooxazole
—— 1-(4-Methylsulfonylphenyl)-5-(4-propoxyphenyl)imidazole(60 % yield) 265113-67-5 C19H20N2O3S
1-(4-Methylsulfonylphenyl)-5-(4-propoxyphenyl)imidazole(60 % yield)
—— (E,3S,4S)-4-methoxy-3-methyl-6-[2-(2-propan-2-yl-1,3-thiazol-4-yl)-1,3-thiazol-4-yl]hex-5-en-2-ol 501012-95-9 C17H24N2O2S2
(E,3S,4S)-4-methoxy-3-methyl-6-[2-(2-propan-2-yl-1,3-thiazol-4-yl)-1,3-thiazol-4-yl]hex-5-en-2-ol
—— (+)-cystothiazole A 207399-36-8 C20H26N2O4S2
(+)-cystothiazole A
—— tert-butyl [(1S,3S)-(4-benzyl-1,3-oxazol-2-yl)cyclopentyl]carbamate 875898-18-3 C20H26N2O3
tert-butyl [(1S,3S)-(4-benzyl-1,3-oxazol-2-yl)cyclopentyl]carbamate
—— 1H-Pyrazolo[3,4-d]thiazol-5-amine, 1,3-diphenyl- 662109-76-4 C16H12N4S
1H-Pyrazolo[3,4-d]thiazol-5-amine, 1,3-diphenyl-
—— N'-[(3,4-difluorophenyl)acetyl]-3-methoxy-4-(2-methyl-1,3-oxazol-5-yl)benzohydrazide 1363144-11-9 C20H17F2N3O4
N'-[(3,4-difluorophenyl)acetyl]-3-methoxy-4-(2-methyl-1,3-oxazol-5-yl)benzohydrazide
—— 2-guanidino-4,6-diphenylpyrazolo[5,4-d]thiazole 753019-03-3 C17H14N6S
2-guanidino-4,6-diphenylpyrazolo[5,4-d]thiazole
—— 2-(3,4-difluorobenzyl)-5-[3-methoxy-4-(2-methyl-1,3-oxazol-5-yl)phenyl]-1,3,4-oxadiazole 1363144-17-5 C20H15F2N3O3
2-(3,4-difluorobenzyl)-5-[3-methoxy-4-(2-methyl-1,3-oxazol-5-yl)phenyl]-1,3,4-oxadiazole
—— (4,5-Dicyan-1-methyl-1H-imidazol-2-yl)diphenyltelluronium-trifluoromethansulfonat 131407-23-3 CF3O3S*C18H13N4Te
(4,5-Dicyan-1-methyl-1H-imidazol-2-yl)diphenyltelluronium-trifluoromethansulfonat
—— (S)-(5-amino-[1,3,4]thiadiazol-2-yl)phenylmethanol 1259552-16-3 C9H9N3OS
(S)-(5-amino-[1,3,4]thiadiazol-2-yl)phenylmethanol
—— (6RS,8SR)-6-{[tert-butyl(dimethyl)silyl]oxy}-8-(3,4-difluorophenyl)-3-[3-methoxy-4-(2-methyl-1,3-oxazol-5-yl)phenyl]-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridine 1363144-23-3 C29H34F2N4O3Si
(6RS,8SR)-6-{[tert-butyl(dimethyl)silyl]oxy}-8-(3,4-difluorophenyl)-3-[3-methoxy-4-(2-methyl-1,3-oxazol-5-yl)phenyl]-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridine