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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1,1-dimethylethyl (3S)-3-[(3-chloro-4-cyanophenyl)amino]-4-[[(2-nitrophenyl)sulfonyl](2-propen-1-yl)amino]butanoate 1006036-49-2 C24H27ClN4O6S
1,1-dimethylethyl (3S)-3-[(3-chloro-4-cyanophenyl)amino]-4-[[(2-nitrophenyl)sulfonyl](2-propen-1-yl)amino]butanoate
—— 3-[1-[3-(4-fluorobenzoyl)-5-isopropylbenzyl]-5-((S)-2-methylaminopropionylamino)-6-oxo-1,6-dihydropyrimidin-2-yl]-2,N-dimethylbenzamide 1033000-01-9 C34H36FN5O4
3-[1-[3-(4-fluorobenzoyl)-5-isopropylbenzyl]-5-((S)-2-methylaminopropionylamino)-6-oxo-1,6-dihydropyrimidin-2-yl]-2,N-dimethylbenzamide
—— N-(6-(5-fluoro-2-methoxyphenyl)pyrimidin-4-yl)-2-(pyridin-3-yl)acetamide 1142002-75-2 C18H15FN4O2
N-(6-(5-fluoro-2-methoxyphenyl)pyrimidin-4-yl)-2-(pyridin-3-yl)acetamide
—— N-((1R,2R)-1-(2,3-dihydrobenzo[β][1,4]dioxin-6-yl)-1-hydroxy-3-(pyrrolidin-1-yl)propan-2-yl)-2-o-tolylacetamide 1092465-60-5 C24H30N2O4
N-((1R,2R)-1-(2,3-dihydrobenzo[β][1,4]dioxin-6-yl)-1-hydroxy-3-(pyrrolidin-1-yl)propan-2-yl)-2-o-tolylacetamide
—— benzyl N-[(1R,2R)-1-(2,2-difluoro-1,3-benzodioxol-5-yl)-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]carbamate 1092469-51-6 C22H24F2N2O5
benzyl N-[(1R,2R)-1-(2,2-difluoro-1,3-benzodioxol-5-yl)-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]carbamate
—— 2,2,2-trichloroethyl 3-ethyl-1-(quinolin-6-yl)-1H-pyrazol-5-ylcarbamate 1020173-51-6 C17H15Cl3N4O2
2,2,2-trichloroethyl 3-ethyl-1-(quinolin-6-yl)-1H-pyrazol-5-ylcarbamate
—— N-[(2R,4R)-2-(1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]chromane-6-carboxamide hydrochloride 1095173-68-4 C23H26N4O2*ClH
N-[(2R,4R)-2-(1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]chromane-6-carboxamide hydrochloride
—— tert-butyl 5-(5-amino-3-ethyl-pyrazol-1-yl)-indazole-1-carboxylate 1020173-66-3 C17H21N5O2
tert-butyl 5-(5-amino-3-ethyl-pyrazol-1-yl)-indazole-1-carboxylate
—— (1S,1aS,6aR)-4-[[5-[2,6-dimethyl-4-[(3-methyloxetan-3-yl)methoxy]phenyl]-2-fluorophenyl]methoxy]-1,1a,6,6a-tetrahydrocyclopropa[a]indene-1-carboxylic acid 1149378-89-1 C31H31FO5
(1S,1aS,6aR)-4-[[5-[2,6-dimethyl-4-[(3-methyloxetan-3-yl)methoxy]phenyl]-2-fluorophenyl]methoxy]-1,1a,6,6a-tetrahydrocyclopropa[a]indene-1-carboxylic acid
—— N-[2-(4-{6-amino-5-[(2,4-difluorophenyl)carbonyl]-2-oxopyridin-1(2H)-yl}phenyl)ethyl]-L-isoleucine 1151805-12-7 C26H27F2N3O4
N-[2-(4-{6-amino-5-[(2,4-difluorophenyl)carbonyl]-2-oxopyridin-1(2H)-yl}phenyl)ethyl]-L-isoleucine
—— 3-(5-(4-hydroxyphenyl)-1-phenyl-4,5-dihydro-1H-pyrazol-3-yl)chromen-2-one 1148141-49-4 C24H18N2O3
3-(5-(4-hydroxyphenyl)-1-phenyl-4,5-dihydro-1H-pyrazol-3-yl)chromen-2-one
—— 1-[(2R,4R)-2-(1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]-3-(6-methoxypyridin-3-yl)urea hydrochloride 1095174-71-2 C20H24N6O2*ClH
1-[(2R,4R)-2-(1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]-3-(6-methoxypyridin-3-yl)urea hydrochloride
—— 3-(4-chloro-phenyl)-2-propyl-4,5,7,8-tetrahydro-2H-1,2,6-triaza-azulene-6-carboxylic acid tert-butyl ester 1018453-08-1 C21H28ClN3O2
3-(4-chloro-phenyl)-2-propyl-4,5,7,8-tetrahydro-2H-1,2,6-triaza-azulene-6-carboxylic acid tert-butyl ester
—— methyl 2-(2-tert-butyl-7-p-tolyl-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)-6,6,6-trifluorohexanoate 1313376-92-9 C25H30F3N3O2
methyl 2-(2-tert-butyl-7-p-tolyl-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)-6,6,6-trifluorohexanoate
—— 1-(4-cyanophenyl)-3-[(2R,4R)-2-(5,6-dimethyl-1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]urea hydrochloride 1095174-06-3 C23H26N6O*ClH
1-(4-cyanophenyl)-3-[(2R,4R)-2-(5,6-dimethyl-1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]urea hydrochloride
—— 4-[4-[(2,5-dimethoxyphenyl)sulfonyl]-1,4-diazepan-1-yl]-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]butanenitrile 1270979-77-5 C26H30N8O4S
4-[4-[(2,5-dimethoxyphenyl)sulfonyl]-1,4-diazepan-1-yl]-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]butanenitrile
—— 1-[(2R,4R)-2-(5,6-dimethyl-1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]-3-(6-methoxypyridin-3-yl)urea hydrochloride 1095175-79-3 C22H28N6O2*ClH
1-[(2R,4R)-2-(5,6-dimethyl-1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]-3-(6-methoxypyridin-3-yl)urea hydrochloride
—— 4-[5-bromo-3-(5-chloro-2-thienyl)-1H-pyrazol-4-yl]pyridine 1313380-28-7 C12H7BrClN3S
4-[5-bromo-3-(5-chloro-2-thienyl)-1H-pyrazol-4-yl]pyridine
—— N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)piperidin-4-yl]-6-(3-fluorophenyl)nicotinamide 1033840-05-9 C27H28FN3O3
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)piperidin-4-yl]-6-(3-fluorophenyl)nicotinamide
—— 2-(2-tert-butyl-7-(2-fluoro-4-methoxyphenyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)pentanoic acid 1313377-63-7 C23H28FN3O3
2-(2-tert-butyl-7-(2-fluoro-4-methoxyphenyl)-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)pentanoic acid
—— N-(3-[2-(1-hydroxycyclobutyl)-1,3-thiazol-5-yl]-5-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)butanamide 1312497-60-1 C22H22F3N5O2S
N-(3-[2-(1-hydroxycyclobutyl)-1,3-thiazol-5-yl]-5-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)butanamide
—— N-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-6-(3-fluorophenyl)nicotinamide 1033840-44-6 C24H28FN3O
N-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-6-(3-fluorophenyl)nicotinamide
—— dibenzyl[3-(5-piperid-4-yl[1,2,4]oxadiazol-3-yl)phenyl]amine hydrochloride 1001468-35-4 C27H28N4O*ClH
dibenzyl[3-(5-piperid-4-yl[1,2,4]oxadiazol-3-yl)phenyl]amine hydrochloride
—— 1-Phenyl-5-[[6-(trifluoromethyl)-2,3-dihydro-1,4-benzoxazin-4-yl]methyl]pyrazol-3-amine 1152721-11-3 C19H17F3N4O
1-Phenyl-5-[[6-(trifluoromethyl)-2,3-dihydro-1,4-benzoxazin-4-yl]methyl]pyrazol-3-amine
—— [(Pd2Cl2(1,4-[(9,10-(C8H16O5)C6H3)NCH]2C6H2-C2,C5,N,N'))2(μ-bis(diphenylphosphino)methane)2] 1263817-11-3 C122H128Cl4N4O20P4Pd4
[(Pd2Cl2(1,4-[(9,10-(C8H16O5)C6H3)NCH]2C6H2-C2,C5,N,N'))2(μ-bis(diphenylphosphino)methane)2]
—— 4-trifluoromethylpyridine-2-carboxylic acid (4-methyl-3-{2-[4-(4-methyl-piperazin-1-carbonyl)-phenylamino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl}-phenyl)-amide 1332329-15-3 C33H33F3N8O2
4-trifluoromethylpyridine-2-carboxylic acid (4-methyl-3-{2-[4-(4-methyl-piperazin-1-carbonyl)-phenylamino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl}-phenyl)-amide
—— Boc-­L-γ-­Ach-D-γ-<sup>Me</sup>N-Acp-D-γ-(Ac)<sub>3</sub>Aga-D-γ-<sup>Me</sup>N-Acp-OAll 1409957-09-0 C41H62N4O14
Boc-­L-γ-­Ach-D-γ-<sup>Me</sup>N-Acp-D-γ-(Ac)<sub>3</sub>Aga-D-γ-<sup>Me</sup>N-Acp-OAll
—— [Cu(2-amino-3-hydroxypyridine(-1H))(histamine)]Cl 1318251-67-0 C5H5N2O*C5H9N3*Cl*Cu
[Cu(2-amino-3-hydroxypyridine(-1H))(histamine)]Cl
—— tert-butyl (2-(5-butoxy-1H-indol-3-yl)ethyl)carbamate 1432473-05-6 C19H28N2O3
tert-butyl (2-(5-butoxy-1H-indol-3-yl)ethyl)carbamate
—— (+/-)-1-(4-hydroxybenzyl)-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroisoquinoline hydrochloride 17934-80-4 C17H19NO3*ClH
(+/-)-1-(4-hydroxybenzyl)-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroisoquinoline hydrochloride
—— (2E,4E,6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcyclohex-1-en-1-yl)nona-2,4,6,8-tetraen-1-yl 2-hydroxy-3-methoxybenzoate 1121716-12-8 C28H36O4
(2E,4E,6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcyclohex-1-en-1-yl)nona-2,4,6,8-tetraen-1-yl 2-hydroxy-3-methoxybenzoate
—— methyl 3-(3'-hydroxy-5'hydroxymethyl-2'-methyl-4'-pyridyl)-2-azabicyclo(3.3.0)octane-2-carboxylate 127949-71-7 C16H22N2O4
methyl 3-(3'-hydroxy-5'hydroxymethyl-2'-methyl-4'-pyridyl)-2-azabicyclo(3.3.0)octane-2-carboxylate
—— 2-(tert-butoxy)-2-(1-(2,5-difluorobenzyl)-6-methyl-4-(p-tolyl)-1H-pyrrolo[2,3-b]pyridin-5-yl)acetic acid 1418712-83-0 C28H28F2N2O3
2-(tert-butoxy)-2-(1-(2,5-difluorobenzyl)-6-methyl-4-(p-tolyl)-1H-pyrrolo[2,3-b]pyridin-5-yl)acetic acid
—— {5-cyclopropyl-3-[2-{[(cyclopropylcarbonyl)(ethyl)amino]methyl}-4-(trifluoromethyl)phenyl]-1H-pyrrolo[3,2-b]pyridin-1-yl}acetic acid 1420071-04-0 C26H26F3N3O3
{5-cyclopropyl-3-[2-{[(cyclopropylcarbonyl)(ethyl)amino]methyl}-4-(trifluoromethyl)phenyl]-1H-pyrrolo[3,2-b]pyridin-1-yl}acetic acid
—— 1-(4-Cyanobenzylidenamino)-4-(9-xanthenyl)-piperazin 13055-99-7 C25H22N4O
1-(4-Cyanobenzylidenamino)-4-(9-xanthenyl)-piperazin
—— 5-(5-((5-p-tolyl-1,3,4-oxadiazol-2-yl)methylthio)-4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl)pyrimidin-2-amine 1257542-72-5 C22H17ClN8OS
5-(5-((5-p-tolyl-1,3,4-oxadiazol-2-yl)methylthio)-4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl)pyrimidin-2-amine
—— (R)-6-bromo-1-(3-methylmorpholino)phthalazine 1067904-82-8 C13H14BrN3O
(R)-6-bromo-1-(3-methylmorpholino)phthalazine
—— 2,4-dichloro-3-(4-methoxyphenyl)-1,5-diphenylpent-2-ene-1,5-dione 139183-06-5 C24H18Cl2O3
2,4-dichloro-3-(4-methoxyphenyl)-1,5-diphenylpent-2-ene-1,5-dione
—— 2,2,2-trifluoro-1-(2-methyl-6a-phenyl-4,5,6,6a-tetrahydro-3aH-cyclopenta[b]furan-3-yl)ethanone 1330122-13-8 C16H15F3O2
2,2,2-trifluoro-1-(2-methyl-6a-phenyl-4,5,6,6a-tetrahydro-3aH-cyclopenta[b]furan-3-yl)ethanone
—— (E)-1-methyl-3-(3-(naphthalen-1-yl)-1-phenylallyl)-1H-indole 1393743-44-6 C28H23N
(E)-1-methyl-3-(3-(naphthalen-1-yl)-1-phenylallyl)-1H-indole
—— N'-<1-<(ethoxycarbonyl)amino>-2-oxo-2-phenylethylidene>-N-formyl-N-methyl-1,2-benzenediamine 130090-75-4 C19H19N3O4
N'-<1-<(ethoxycarbonyl)amino>-2-oxo-2-phenylethylidene>-N-formyl-N-methyl-1,2-benzenediamine
—— (3-chroman-6-yl-4,5-dihydropyrazol-1-yl)methanone 1417708-86-1 C19H17FN2O2
(3-chroman-6-yl-4,5-dihydropyrazol-1-yl)methanone
—— (8S,15S,19S)-8-amino-2,9,17-trioxo-1-(4,7,10-tris(carboxymethyl)-1,4,7,10-tetraazacyclododecan-1-yl)-3,10,16,18-tetraazahenicosane-15,19,21-tricarboxylic acid 1422158-81-3 C34H59N9O15
(8S,15S,19S)-8-amino-2,9,17-trioxo-1-(4,7,10-tris(carboxymethyl)-1,4,7,10-tetraazacyclododecan-1-yl)-3,10,16,18-tetraazahenicosane-15,19,21-tricarboxylic acid
—— (R)-tert-butyl 3-(2-(5-chloro-2-methoxypyridin-3-ylamino)-5-methylpyrimidin-4-ylamino)piperidine-1-carboxylate 1421757-73-4 C21H29ClN6O3
(R)-tert-butyl 3-(2-(5-chloro-2-methoxypyridin-3-ylamino)-5-methylpyrimidin-4-ylamino)piperidine-1-carboxylate
—— 4-(3,3-dimethylpiperidin-1-yl)-6-(5-isopropyl-2-methylphenyl)-2-(2-(trifluoromethoxy)phenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine 1421250-04-5 C31H37F3N4O
4-(3,3-dimethylpiperidin-1-yl)-6-(5-isopropyl-2-methylphenyl)-2-(2-(trifluoromethoxy)phenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— 4-(8-amino-3-(3-(morpholine-4-carbonyl)piperidin-1-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide 1419216-39-9 C28H30N8O3
4-(8-amino-3-(3-(morpholine-4-carbonyl)piperidin-1-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide
—— 2-amino-(2-bromo-benzenesulfonylamino)propanoic acid methyl ester 1422027-89-1 C10H13BrN2O4S
2-amino-(2-bromo-benzenesulfonylamino)propanoic acid methyl ester
—— [1-(3-chloropyridin-2-yl)-5-(trichloromethyl)-1H-pyrazol-3-yl]methyl acetate 1262281-62-8 C12H9Cl4N3O2
[1-(3-chloropyridin-2-yl)-5-(trichloromethyl)-1H-pyrazol-3-yl]methyl acetate
—— (2S,5R)-5-(2-chlorophenyl)-1-(2',3,6'-trimethoxy-[2,3'-bipyridine]-5-carbonyl)pyrrolidine-2-carboxylic acid 1312802-54-2 C25H24ClN3O6
(2S,5R)-5-(2-chlorophenyl)-1-(2',3,6'-trimethoxy-[2,3'-bipyridine]-5-carbonyl)pyrrolidine-2-carboxylic acid
—— 7-fluoro-3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-tosyl-1H-indole 1421254-72-9 C22H25BFNO4S
7-fluoro-3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-tosyl-1H-indole