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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(5-{[6-(1H-indazol-6-yl)imidazo[1,2-a]pyrazin-8-yl]amino}pyridin-2-yl)-2-methylpropan-1-ol 1228795-65-0 C22H21N7O
2-(5-{[6-(1H-indazol-6-yl)imidazo[1,2-a]pyrazin-8-yl]amino}pyridin-2-yl)-2-methylpropan-1-ol
—— (R)-3-(cyclopentylmethyl)-4-(cyclopropyl(4-(2-(6-(2-oxopyrrolidin-1-yl)pyridin-3-yl)phenyl)thiazol-2-yl)amino)-4-oxobutanoic acid 1229364-35-5 C31H34N4O4S
(R)-3-(cyclopentylmethyl)-4-(cyclopropyl(4-(2-(6-(2-oxopyrrolidin-1-yl)pyridin-3-yl)phenyl)thiazol-2-yl)amino)-4-oxobutanoic acid
—— [(3S,4R)-1-(5'-carbamoyl-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-4-carbonyl)-4-(4-chloro-phenyl)-pyrrolidin-3-yl]-ethyl-carbamic acid 4-fluoro-phenyl ester 1312667-55-2 C31H33ClFN5O4
[(3S,4R)-1-(5'-carbamoyl-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-4-carbonyl)-4-(4-chloro-phenyl)-pyrrolidin-3-yl]-ethyl-carbamic acid 4-fluoro-phenyl ester
—— (2S,5S,6S,5'S)-5'-hydroxy-2'-oxospiropent-3'-ene-5,6-dimethoxy-5,6-dimethyl-[1,4]dioxane 1042925-87-0 C12H18O6
(2S,5S,6S,5'S)-5'-hydroxy-2'-oxospiropent-3'-ene-5,6-dimethoxy-5,6-dimethyl-[1,4]dioxane
—— (3'aS,11'aS)-11'a-(2-hydroxyethyl)-3'a-methylspiro[1,3-dioxolane-2,3'-4,5-dihydro-2H-indeno[4,5-b]chromene]-8'-ol 1092526-75-4 C21H24O5
(3'aS,11'aS)-11'a-(2-hydroxyethyl)-3'a-methylspiro[1,3-dioxolane-2,3'-4,5-dihydro-2H-indeno[4,5-b]chromene]-8'-ol
—— 2,5-Difluoro-4-(methylsulfanyl)phenol 1879026-13-7 C7H6F2OS
2,5-Difluoro-4-(methylsulfanyl)phenol
—— [(7-ethynyl-4-hydroxy-3-methyl-isothiazolo[5,4-c]pyridine-5-carbonyl)-amino]-acetic acid 1172590-56-5 C12H9N3O4S
[(7-ethynyl-4-hydroxy-3-methyl-isothiazolo[5,4-c]pyridine-5-carbonyl)-amino]-acetic acid
—— 1-Ethyl-6-fluoro-4-oxo-5-piperazin-1-yl-1,4-dihydroquinoline-3-carboxylic acid 106847-42-1 C16H18FN3O3
1-Ethyl-6-fluoro-4-oxo-5-piperazin-1-yl-1,4-dihydroquinoline-3-carboxylic acid
—— [3-methyl-4-(2',3',4',6'-tetra-O-acetyl-β-D-glucopyranosylthio)-1H-thieno[3,4-c]pyrazol-6-yl](phenyl)methanone 1064665-79-7 C27H28N2O10S2
[3-methyl-4-(2',3',4',6'-tetra-O-acetyl-β-D-glucopyranosylthio)-1H-thieno[3,4-c]pyrazol-6-yl](phenyl)methanone
—— 1,2-bis(methoxycarbonyl)-3-(1-diphenylphosphinoylhexyl)phenanthrene 1078710-60-7 C36H35O5P
1,2-bis(methoxycarbonyl)-3-(1-diphenylphosphinoylhexyl)phenanthrene
—— [8-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[1,5-a]pyrazin-2-yl]-(3-morpholin-4-yl-phenyl)amine 1451386-18-7 C19H20N8O
[8-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[1,5-a]pyrazin-2-yl]-(3-morpholin-4-yl-phenyl)amine
—— 2,3-dihydro-furo[2,3-b]pyridine-3-carboxylic acid [2-(4,4-difluoro-piperidin-1-yl)-2-(2-trifluoromethyl-pyrimidin-5-yl)-ethyl]-amide 1448335-70-3 C20H20F5N5O2
2,3-dihydro-furo[2,3-b]pyridine-3-carboxylic acid [2-(4,4-difluoro-piperidin-1-yl)-2-(2-trifluoromethyl-pyrimidin-5-yl)-ethyl]-amide
—— (3aR,4S,7aR)-4,7a-dimethyl-3,3a,4,7-tetrahydro-2H-1-benzofuran 1064682-74-1 C10H16O
(3aR,4S,7aR)-4,7a-dimethyl-3,3a,4,7-tetrahydro-2H-1-benzofuran
—— 5-(4-methoxyphenyl)-6-oxo-N-(4-tolylsulfonylmethyl)-4,5,6,7-tetrahydro-3,5,7a-triazacyclohepta[jk]fluorene-4-carboxamide 1290047-21-0 C30H26N4O5S
5-(4-methoxyphenyl)-6-oxo-N-(4-tolylsulfonylmethyl)-4,5,6,7-tetrahydro-3,5,7a-triazacyclohepta[jk]fluorene-4-carboxamide
—— (E)-6-chloro-1-phenylseleno-1-hexene 1454270-78-0 C12H15ClSe
(E)-6-chloro-1-phenylseleno-1-hexene
—— N-(pyridin-2-yl)-3-(3-methyl-1H-pyrazol-4-yl)-1,2,4-thiadiazol-5-ylamine 1105038-80-9 C11H10N6S
N-(pyridin-2-yl)-3-(3-methyl-1H-pyrazol-4-yl)-1,2,4-thiadiazol-5-ylamine
—— 4-[[3-(3-Fluorophenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenol 1124320-38-2 C18H13FN4O
4-[[3-(3-Fluorophenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenol
—— 4-(6-ethoxy-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-3-yl)phenol 1228282-72-1 C12H12N4O2S
4-(6-ethoxy-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-3-yl)phenol
—— dimethyl (E)-2-(1-(4-chlorophenyl)-3-(prop-2-ynyloxy)prop-1-en-2-yl)malonate 1263816-49-4 C17H17ClO5
dimethyl (E)-2-(1-(4-chlorophenyl)-3-(prop-2-ynyloxy)prop-1-en-2-yl)malonate
—— (1R,5S,6R)-6-bromo-6-fluoro-1-phenylbicyclo[3.1.0]hexane 1201786-43-7 C12H12BrF
(1R,5S,6R)-6-bromo-6-fluoro-1-phenylbicyclo[3.1.0]hexane
—— (4aR,7aS)-N-{3-[1-(2-chloro-4-fluoro-benzyl)-4-hydroxy-2-oxo-2,4-a,5,6,7,7a-hexahydro-1H-[1]pyrindin-3-yl]-1,1-dioxo-1,4-dihydro-1λ6-thieno[2,3-e][1,2,4]thiadiazin-7-ylmethyl}-methanesulfonamide 1198470-11-9 C22H22ClFN4O6S3
(4aR,7aS)-N-{3-[1-(2-chloro-4-fluoro-benzyl)-4-hydroxy-2-oxo-2,4-a,5,6,7,7a-hexahydro-1H-[1]pyrindin-3-yl]-1,1-dioxo-1,4-dihydro-1λ6-thieno[2,3-e][1,2,4]thiadiazin-7-ylmethyl}-methanesulfonamide
—— 4-[({1-methyl-5-[2-(3-methyl-1,2,4-oxadiazol-5-yl)-1H-indol-5-yl]-1H-pyrazole-3-carbonyl}-amino)-methyl]-benzoic acid 1222173-30-9 C24H20N6O4
4-[({1-methyl-5-[2-(3-methyl-1,2,4-oxadiazol-5-yl)-1H-indol-5-yl]-1H-pyrazole-3-carbonyl}-amino)-methyl]-benzoic acid
—— N-{2-[1,3-dihydro-2H-isoindol-2-yl(methyl)amino]-2-oxoethyl}-N-[2-methyl-5-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)phenyl]glycine 1190894-33-7 C22H23N5O5
N-{2-[1,3-dihydro-2H-isoindol-2-yl(methyl)amino]-2-oxoethyl}-N-[2-methyl-5-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)phenyl]glycine
—— (S)-3-{[4-(5-cyclopropylmethoxy-benzo[1,3]dioxol-4-yl)-5H-pyrrolo[3,2-d]pyrimidine-7-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester 1185837-53-9 C28H33N5O6
(S)-3-{[4-(5-cyclopropylmethoxy-benzo[1,3]dioxol-4-yl)-5H-pyrrolo[3,2-d]pyrimidine-7-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester
—— 3-({1-[bis(4-chlorophenyl)methyl]azetidin-3-yl}(methanesulphonyl)amino)-5-cyanobenzoic acid methyl ester 1186130-33-5 C26H23Cl2N3O4S
3-({1-[bis(4-chlorophenyl)methyl]azetidin-3-yl}(methanesulphonyl)amino)-5-cyanobenzoic acid methyl ester
—— ethyl 7-(methylsulfonyl)chromane-2-carboxylate 1193709-61-3 C13H16O5S
ethyl 7-(methylsulfonyl)chromane-2-carboxylate
—— benzothiazole-7-carboxylic acid {(1R,3R,4S)-2-[5-(3-chloro-phenyl)-2-(ethyl-methyl-amino)-thiazole-4-carbonyl]-2-aza-bicyclo[2.2.1]hept-3-ylmethyl}-amide 1181572-01-9 C28H28ClN5O2S2
benzothiazole-7-carboxylic acid {(1R,3R,4S)-2-[5-(3-chloro-phenyl)-2-(ethyl-methyl-amino)-thiazole-4-carbonyl]-2-aza-bicyclo[2.2.1]hept-3-ylmethyl}-amide
—— prop-2-ynyl-bAla-N(prop-2-ynyl)bAla-N(prop-2-ynyl)bAla-N(prop-2-ynyl)bAla-OtBu 1013635-53-4 C28H38N4O5
prop-2-ynyl-bAla-N(prop-2-ynyl)bAla-N(prop-2-ynyl)bAla-N(prop-2-ynyl)bAla-OtBu
—— 5-[(4S,6R)-8-hydroxy-2,6-dimethyloct-2-en-4-yl]-2-methoxy-3-methylcyclohexa-2,5-diene-1,4-dione 1266245-89-9 C18H26O4
5-[(4S,6R)-8-hydroxy-2,6-dimethyloct-2-en-4-yl]-2-methoxy-3-methylcyclohexa-2,5-diene-1,4-dione
—— naphthalen-1-yl (E)-4-(2-bromovinyl)benzoate 1132093-98-1 C19H13BrO2
naphthalen-1-yl (E)-4-(2-bromovinyl)benzoate
—— 3-{N-[2-(N-trimethylsilylamino)ethyl]amino}-1,1-diphenyl-1,2-dihydropentalene 1044197-06-9 C26H32N2Si
3-{N-[2-(N-trimethylsilylamino)ethyl]amino}-1,1-diphenyl-1,2-dihydropentalene
—— (E)-1-(5-(2-methyloxiran-2-yl)pent-2-enoyl)pyrrolidin-2-one 1203791-98-3 C12H17NO3
(E)-1-(5-(2-methyloxiran-2-yl)pent-2-enoyl)pyrrolidin-2-one
—— N-(4-bromophenyl)-2-[2-[2-[(4-bromophenyl)carbamoylamino]-2-oxoethyl]cyclohexen-1-yl]-2-cyanoacetamide 1188547-41-2 C24H22Br2N4O3
N-(4-bromophenyl)-2-[2-[2-[(4-bromophenyl)carbamoylamino]-2-oxoethyl]cyclohexen-1-yl]-2-cyanoacetamide
—— (4-(2,4,6-trifluoro-3,5-diiodostyryl)pyridine 1-oxide) 1029608-35-2 C13H6F3I2NO
(4-(2,4,6-trifluoro-3,5-diiodostyryl)pyridine 1-oxide)
—— 2-amino-1-{3-[(3-chloro-4-fluorophenyl)amino]-2-(4-fluorophenyl)-8,8-dimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}ethan-1-one 1261114-07-1 C22H22ClF2N5O
2-amino-1-{3-[(3-chloro-4-fluorophenyl)amino]-2-(4-fluorophenyl)-8,8-dimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}ethan-1-one
—— 3-{[(3R)-3-hydroxypiperidin-1-yl]sulfonyl}-N-(2-methoxyphenyl)benzamide 1192231-96-1 C19H22N2O5S
3-{[(3R)-3-hydroxypiperidin-1-yl]sulfonyl}-N-(2-methoxyphenyl)benzamide
—— tert-butyl 3-hydroxy-3-((4-((S)-1-((S)-6-(2-hydroxy-2-methylpropyl)-2-oxo-6-phenyl-1,3-oxazinan-3-yl)ethyl)phenyl)ethynyl)azetidine-1-carboxylate 1259034-62-2 C32H40N2O6
tert-butyl 3-hydroxy-3-((4-((S)-1-((S)-6-(2-hydroxy-2-methylpropyl)-2-oxo-6-phenyl-1,3-oxazinan-3-yl)ethyl)phenyl)ethynyl)azetidine-1-carboxylate
—— 1-(3-chloro-benzyl)-5-fluoro-1H-indazol-3-ylamine 1021388-75-9 C14H11ClFN3
1-(3-chloro-benzyl)-5-fluoro-1H-indazol-3-ylamine
—— 4-[5-(5-chloro-1H-indol-1-yl)-1,3-dimethyl-1H-pyrazol-4-yl]-N-[(pentylamino)sulfonyl]butanamide 1048020-22-9 C22H30ClN5O3S
4-[5-(5-chloro-1H-indol-1-yl)-1,3-dimethyl-1H-pyrazol-4-yl]-N-[(pentylamino)sulfonyl]butanamide
—— 2-((3S,5S)-3,5-dimethylmorpholino)-N-(quinuclidine-8-yl)benzoxazole-4-carboxamide hydrochloride 1007111-73-0 C21H28N4O3*ClH
2-((3S,5S)-3,5-dimethylmorpholino)-N-(quinuclidine-8-yl)benzoxazole-4-carboxamide hydrochloride
—— 6-(pyridin-2-ylmethylamino)-2-phenyl-N-(2-(thiazolo[5,4-c]pyridin-2-yl)phenyl)pyrimidine-4-carboxamide hydrochloride 1152095-52-7 C29H21N7OS*ClH
6-(pyridin-2-ylmethylamino)-2-phenyl-N-(2-(thiazolo[5,4-c]pyridin-2-yl)phenyl)pyrimidine-4-carboxamide hydrochloride
—— 8-(2-phenoxy-ethoxy)-octanoic acid 1192596-61-4 C16H24O4
8-(2-phenoxy-ethoxy)-octanoic acid
—— 10-(2,3-difluoro-phenyl)-dec-9-enoic acid 1192177-46-0 C16H20F2O2
10-(2,3-difluoro-phenyl)-dec-9-enoic acid
—— (E)-3-(3-hydroxy-4-methoxyphenyl)-1-(5-hydroxybenzo[d][1,3]oxathiol-6-yl)prop-2-en-1-one 1262430-14-7 C17H14O5S
(E)-3-(3-hydroxy-4-methoxyphenyl)-1-(5-hydroxybenzo[d][1,3]oxathiol-6-yl)prop-2-en-1-one
—— 4-(8-(4-isopropylphenylamino)imidazo[1,2-a]pyrazin-3-yl)phenol 1124320-24-6 C21H20N4O
4-(8-(4-isopropylphenylamino)imidazo[1,2-a]pyrazin-3-yl)phenol
—— 4-(3-{[(5-oxo-4,5-dihydropyrazolo[1,5-a]quinazolin-2-yl)carbonyl]amino}propyl)morpholin-4-ium trifluoroacetate 1041467-01-9 C2HF3O2*C18H21N5O3
4-(3-{[(5-oxo-4,5-dihydropyrazolo[1,5-a]quinazolin-2-yl)carbonyl]amino}propyl)morpholin-4-ium trifluoroacetate
—— 3-[3,4-dimethyl-8-(trifluoromethoxy)imidazo[1,5-a]quinoxalin-1-yl]benzamide 1159794-91-8 C20H15F3N4O2
3-[3,4-dimethyl-8-(trifluoromethoxy)imidazo[1,5-a]quinoxalin-1-yl]benzamide
—— N-(4-isopropoxyphenyl)-3-(1H-pyrazol-4-ylsulfonyl)benzamide 1192232-86-2 C19H19N3O4S
N-(4-isopropoxyphenyl)-3-(1H-pyrazol-4-ylsulfonyl)benzamide
—— (2E)-3-[1,3-dimethyl-5-(1-methyl-1H-indol-3-yl)-1H-pyrazol-4-yl]-N-(pentylsulfonyl)acrylamide 1048021-07-3 C22H28N4O3S
(2E)-3-[1,3-dimethyl-5-(1-methyl-1H-indol-3-yl)-1H-pyrazol-4-yl]-N-(pentylsulfonyl)acrylamide
—— (4-(1-azepanyl)-6-{[(1,2-dimethyl-1H-imidazol-4-yl)thio]methyl}-2-pyridinyl)(2,2,2-trifluoroethyl)carbamic acid tert-butyl ester 1186690-04-9 C24H34F3N5O2S
(4-(1-azepanyl)-6-{[(1,2-dimethyl-1H-imidazol-4-yl)thio]methyl}-2-pyridinyl)(2,2,2-trifluoroethyl)carbamic acid tert-butyl ester