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—— 3-methoxy-4-[[4-[(2-methyl-3-oxo-1H-isoindol-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-N-(oxan-4-yl)benzamide 1227949-56-5 C27H26F3N5O5
3-methoxy-4-[[4-[(2-methyl-3-oxo-1H-isoindol-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-N-(oxan-4-yl)benzamide
—— 4-[5-(5-Chloropyridin-2-yl)-2-ethylphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one 1033759-43-1 C22H24ClNO3
4-[5-(5-Chloropyridin-2-yl)-2-ethylphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one
—— 2-fluoro-4-(3-(quinolin-6-ylmethyl)-3H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)-N-(thiazol-2-yl)benzamide 1350427-39-2 C25H16FN7OS
2-fluoro-4-(3-(quinolin-6-ylmethyl)-3H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)-N-(thiazol-2-yl)benzamide
—— Tert-butyl 2-[[5-[2-(dimethylamino)ethoxy]-2-hydroxybenzoyl]amino]-4-phenylbenzoate 1237519-93-5 C28H32N2O5
Tert-butyl 2-[[5-[2-(dimethylamino)ethoxy]-2-hydroxybenzoyl]amino]-4-phenylbenzoate
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-[(1-cyclopropylcyclopropyl)carbamoyl]-6-methylphenyl]-5-[[4-(trifluoromethyl)triazol-2-yl]methyl]pyrazole-3-carboxamide 1339951-16-4 C28H23ClF3N9O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-[(1-cyclopropylcyclopropyl)carbamoyl]-6-methylphenyl]-5-[[4-(trifluoromethyl)triazol-2-yl]methyl]pyrazole-3-carboxamide
—— trans-2R-[3-acetoxy-2-(6-fluoro-1H-indol-3-ylmethyl)]pyrrolidine-1-carboxylic acid tert-butyl ester 1003961-24-7 C20H25FN2O4
trans-2R-[3-acetoxy-2-(6-fluoro-1H-indol-3-ylmethyl)]pyrrolidine-1-carboxylic acid tert-butyl ester
—— 4-[5-(3,5-Difluorophenyl)-2-methylphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one 1033758-30-3 C22H22F2O3
4-[5-(3,5-Difluorophenyl)-2-methylphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one
—— 5-(sec-butyl)-3-(4-((4-fluorophenyl)ethynyl)phenyl)-1,2,4-oxadiazole 1415142-16-3 C20H17FN2O
5-(sec-butyl)-3-(4-((4-fluorophenyl)ethynyl)phenyl)-1,2,4-oxadiazole
—— 1-{4-[5-(difluoromethyl)-3-phenyl-1,6-naphthyridin-2-yl]phenyl}cyclobutanamine 1238320-04-1 C25H21F2N3
1-{4-[5-(difluoromethyl)-3-phenyl-1,6-naphthyridin-2-yl]phenyl}cyclobutanamine
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(1-cyclopropylethylcarbamoyl)-6-methylphenyl]-5-[[4-(trifluoromethyl)triazol-1-yl]methyl]pyrazole-3-carboxamide 1339949-96-0 C27H23ClF3N9O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(1-cyclopropylethylcarbamoyl)-6-methylphenyl]-5-[[4-(trifluoromethyl)triazol-1-yl]methyl]pyrazole-3-carboxamide
—— 6-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-N,N-dimethylquinolin-2-amine 1207349-49-2 C23H21N7
6-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-N,N-dimethylquinolin-2-amine
—— 4-(5-cyclohexyl-1-methyl-1H-1,2,4-triazol-3-yl)benzonitrile 1218817-40-3 C16H18N4
4-(5-cyclohexyl-1-methyl-1H-1,2,4-triazol-3-yl)benzonitrile
—— [4-(azepane-1-carbonyl)-2-nitro-phenyl]-(6-fluoro-imidazo[1,2-a]pyridin-3-yl)-methanone 1235991-88-4 C21H19FN4O4
[4-(azepane-1-carbonyl)-2-nitro-phenyl]-(6-fluoro-imidazo[1,2-a]pyridin-3-yl)-methanone
—— 2-chloro-N-(1-(4-fluorophenyl)-2-methylpropan-2-yl)quinazolin-4-amine 1095657-73-0 C18H17ClFN3
2-chloro-N-(1-(4-fluorophenyl)-2-methylpropan-2-yl)quinazolin-4-amine
—— 4-(1-(2-methyl-prop-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl)-4-oxo-N-[[3-(trifluoromethyl)phenyl]methyl]butyric acid amide 1229515-31-4 C25H29F3N2O2
4-(1-(2-methyl-prop-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl)-4-oxo-N-[[3-(trifluoromethyl)phenyl]methyl]butyric acid amide
—— (2-Methylbenzaldehyd)-2,4,6-trimethylanil 17432-48-3 C17H19N
(2-Methylbenzaldehyd)-2,4,6-trimethylanil
—— methyl 3-(2-bromoethyl)-2-methyl-benzofuran-7-yloxyacetate 181052-95-9 C14H15BrO4
methyl 3-(2-bromoethyl)-2-methyl-benzofuran-7-yloxyacetate
—— 2-Chloro-2-nitro-pentanedioic acid 1-ethyl ester 5-methyl ester 164795-38-4 C8H12ClNO6
2-Chloro-2-nitro-pentanedioic acid 1-ethyl ester 5-methyl ester
—— methyl (E)-3-(naphthalen-1'-yl)-2-phenylsulfinylpropenoate 154276-53-6 C20H16O3S
methyl (E)-3-(naphthalen-1'-yl)-2-phenylsulfinylpropenoate
—— tert-butyl N-[(2S)-1-[(2S,3S,4R)-4-[4-(4-cyclohexyl-1,3-thiazol-2-yl)-1-propan-2-ylbenzimidazol-2-yl]oxy-2-[[(1R,2S)-2-ethenyl-1-[(1-methylcyclopropyl)sulfonylcarbamoyl]cyclopropyl]carbamoyl]-3-methylpyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate 1367555-86-9 C46H65N7O8S2
tert-butyl N-[(2S)-1-[(2S,3S,4R)-4-[4-(4-cyclohexyl-1,3-thiazol-2-yl)-1-propan-2-ylbenzimidazol-2-yl]oxy-2-[[(1R,2S)-2-ethenyl-1-[(1-methylcyclopropyl)sulfonylcarbamoyl]cyclopropyl]carbamoyl]-3-methylpyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate
—— methyl (3-(2-(3-phenylpropyloxy)ethyl)benzofuran-7-yloxy)acetate 181051-52-5 C22H24O5
methyl (3-(2-(3-phenylpropyloxy)ethyl)benzofuran-7-yloxy)acetate
—— 1-tert-Butyldimethylsiloxy-2,2-dimethyl-3,4-octadiene 141081-35-8 C16H32OSi
1-tert-Butyldimethylsiloxy-2,2-dimethyl-3,4-octadiene
—— 2,3-bis(isopropylthio)naphth<1,8-bc>azepine 132497-11-1 C19H21NS2
2,3-bis(isopropylthio)naphth<1,8-bc>azepine
—— 2-(2-hydroxy-5-amidinophenoxy)-6-(3-(1-methylimidazolin-2-yl)phenoxy)-8-ethyl-9-ethylpurine 1099490-54-6 C26H28N8O3
2-(2-hydroxy-5-amidinophenoxy)-6-(3-(1-methylimidazolin-2-yl)phenoxy)-8-ethyl-9-ethylpurine
—— 5-fluoro-3-[2-(1-isobutyl-4-methyl-2-oxo-1,2-dihydro-pyridin-3-yl)-butyrylamino]-4-oxo-pentanoic acid tert-butyl ester 1025080-20-9 C23H35FN2O5
5-fluoro-3-[2-(1-isobutyl-4-methyl-2-oxo-1,2-dihydro-pyridin-3-yl)-butyrylamino]-4-oxo-pentanoic acid tert-butyl ester
—— N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[(4,5,6-trichlorobenzotriazol-1-yl)methyl]pyrazole-3-carboxamide 1339949-25-5 C29H23Cl4N9O2
N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[(4,5,6-trichlorobenzotriazol-1-yl)methyl]pyrazole-3-carboxamide
—— 1-(3-Chloro-4-piperazin-1-ylphenyl)-9-quinolin-3-ylbenzo[h][1,6]naphthyridin-2-one 1223002-25-2 C31H24ClN5O
1-(3-Chloro-4-piperazin-1-ylphenyl)-9-quinolin-3-ylbenzo[h][1,6]naphthyridin-2-one
—— 3-methoxy-N-(3-methoxypropyl)-4-[[4-[(2-methyl-3-oxo-1H-isoindol-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide 1227950-07-3 C26H26F3N5O5
3-methoxy-N-(3-methoxypropyl)-4-[[4-[(2-methyl-3-oxo-1H-isoindol-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide
—— 5-(2-methoxy-4-phenylmethoxyphenyl)-2-propan-2-yl-1H-imidazole 1239260-13-9 C20H22N2O2
5-(2-methoxy-4-phenylmethoxyphenyl)-2-propan-2-yl-1H-imidazole
—— ethyl 2-(4-chloro-2-{[2-methyl-5-(propylsulfonyl)phenyl]ethynyl}phenoxy)-4-methylpentanoate 1240289-09-1 C26H31ClO5S
ethyl 2-(4-chloro-2-{[2-methyl-5-(propylsulfonyl)phenyl]ethynyl}phenoxy)-4-methylpentanoate
—— 1-[4-(tert-butyldiphenylsilyloxymethyl)-1-isopropyl-1H-imidazol-2-yl]ethanone 1331755-39-5 C25H32N2O2Si
1-[4-(tert-butyldiphenylsilyloxymethyl)-1-isopropyl-1H-imidazol-2-yl]ethanone
—— 6-((5-(pyridin-3-yl)-3H-[1,2,3]triazolo[4,5-b]pyridin-3-yl)methyl)quinoline 1350427-94-9 C20H14N6
6-((5-(pyridin-3-yl)-3H-[1,2,3]triazolo[4,5-b]pyridin-3-yl)methyl)quinoline
—— N-[4-chloro-2-methyl-6-(propan-2-ylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[4-(trifluoromethyl)triazol-2-yl]methyl]pyrazole-3-carboxamide 1339949-57-3 C24H21Cl2F3N8O2
N-[4-chloro-2-methyl-6-(propan-2-ylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[4-(trifluoromethyl)triazol-2-yl]methyl]pyrazole-3-carboxamide
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(1-cyclopropylethylcarbamoyl)-6-methylphenyl]-5-[[4-(trifluoromethyl)triazol-2-yl]methyl]pyrazole-3-carboxamide 1339949-43-7 C27H23ClF3N9O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(1-cyclopropylethylcarbamoyl)-6-methylphenyl]-5-[[4-(trifluoromethyl)triazol-2-yl]methyl]pyrazole-3-carboxamide
—— N-methoxy-3-methyl-4-[[4-[(2-methyl-3-oxo-1H-isoindol-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide 1227950-05-1 C23H20F3N5O4
N-methoxy-3-methyl-4-[[4-[(2-methyl-3-oxo-1H-isoindol-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide
—— tert-butyl {2-oxo-2-[8-((R)-1-[1,2,4]triazolo-[1,5-a]pyrimidin-7-ylpyrrolidin-2-ylmethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]ethyl}carbamate 1235964-23-4 C26H33N7O4
tert-butyl {2-oxo-2-[8-((R)-1-[1,2,4]triazolo-[1,5-a]pyrimidin-7-ylpyrrolidin-2-ylmethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]ethyl}carbamate
—— (1S,3'R,4'S,5'S,6'R)-5-chloro-6-[(4-chlorophenyl)methyl]-3',4',5',6'-tetrahydro-6'-(hydroxymethyl)-spiro[isobenzofuran-1(3H),2'-[2H]pyran]-3',4',5'-triol 1005141-96-7 C20H20Cl2O6
(1S,3'R,4'S,5'S,6'R)-5-chloro-6-[(4-chlorophenyl)methyl]-3',4',5',6'-tetrahydro-6'-(hydroxymethyl)-spiro[isobenzofuran-1(3H),2'-[2H]pyran]-3',4',5'-triol
—— 4-Butoxy-3-[ethyl-[4-(2-methoxyphenyl)-5-oxotetrazole-1-carbonyl]amino]benzoic acid 1346563-30-1 C22H25N5O6
4-Butoxy-3-[ethyl-[4-(2-methoxyphenyl)-5-oxotetrazole-1-carbonyl]amino]benzoic acid
—— 4-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-2-fluoro-N-methyl-N-(1-methylpiperidin-4-yl)benzamide 1207349-90-3 C26H28FN7O
4-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-2-fluoro-N-methyl-N-(1-methylpiperidin-4-yl)benzamide
—— 5-[(4-tert-butyltriazol-1-yl)methyl]-2-(3-chloropyridin-2-yl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]pyrazole-3-carboxamide 1339948-45-6 C26H26ClN9O2
5-[(4-tert-butyltriazol-1-yl)methyl]-2-(3-chloropyridin-2-yl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]pyrazole-3-carboxamide
—— 4-(Furan-3-yl)-2-(naphthalen-1-ylmethoxy)benzoic acid 1221890-44-3 C22H16O4
4-(Furan-3-yl)-2-(naphthalen-1-ylmethoxy)benzoic acid
—— N-(4-chloro-1-((3-hydroxyoxetan-3-yl)methyl)-1H-indol-3-yl)-2-cyclohexylacetamide 1415461-11-8 C20H25ClN2O3
N-(4-chloro-1-((3-hydroxyoxetan-3-yl)methyl)-1H-indol-3-yl)-2-cyclohexylacetamide
—— 2-{1-oxo-6-[4-({[2-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1,2,3,4-tetrahydronaphthalen-2-yl}acetic acid 1414795-69-9 C26H21F3N2O4
2-{1-oxo-6-[4-({[2-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1,2,3,4-tetrahydronaphthalen-2-yl}acetic acid
—— tert-butyl [{5-[(4-chloropyridin-2-ylcarbonyl)amino]naphthalen-1-yl}-(3,5-dichlorophenylsulphonyl)amino]acetate 1192208-36-8 C28H24Cl3N3O5S
tert-butyl [{5-[(4-chloropyridin-2-ylcarbonyl)amino]naphthalen-1-yl}-(3,5-dichlorophenylsulphonyl)amino]acetate
—— 2-fluoro-N-(3-oxo-3-(piperidin-1-yl)propyl)-4-(3-(quinolin-6-ylmethyl)-3H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)benzamide 1350427-46-1 C30H28FN7O2
2-fluoro-N-(3-oxo-3-(piperidin-1-yl)propyl)-4-(3-(quinolin-6-ylmethyl)-3H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)benzamide
—— 2,4,6-trichloro-N-{3-(2-cyano-1H-pyrrol-1-yl)-1-[(4-methylpiperidin-1-yl)carbonyl]propyl}benzenesulfonamide 1191031-93-2 C21H23Cl3N4O3S
2,4,6-trichloro-N-{3-(2-cyano-1H-pyrrol-1-yl)-1-[(4-methylpiperidin-1-yl)carbonyl]propyl}benzenesulfonamide
—— N-[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]-5-[3-({[(4,5-dimethylthiophen-2-yl)carbonyl]amino}methyl)phenyl]furan-2-carboxamide 1227191-75-4 C28H33N3O4S
N-[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]-5-[3-({[(4,5-dimethylthiophen-2-yl)carbonyl]amino}methyl)phenyl]furan-2-carboxamide
—— 4-(N-[4-(2-methoxyphenyl)-5-oxotetrazole-1-carbonyl]anilino)benzoic acid 1346563-23-2 C22H17N5O5
4-(N-[4-(2-methoxyphenyl)-5-oxotetrazole-1-carbonyl]anilino)benzoic acid
—— 4-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-2-fluoro-N,N-dimethylbenzamide 1207349-77-6 C21H19FN6O
4-[2-amino-5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]-2-fluoro-N,N-dimethylbenzamide
—— Benzyl 4-[[4-(2,6-dichlorophenyl)-5-oxotetrazole-1-carbonyl]-(2-pyridin-3-ylethyl)amino]benzoate 1346564-95-1 C29H22Cl2N6O4
Benzyl 4-[[4-(2,6-dichlorophenyl)-5-oxotetrazole-1-carbonyl]-(2-pyridin-3-ylethyl)amino]benzoate