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中文名称 英文名称 CAS号 化学式 结构式图片
—— CH2CHCH2-NHC(CO)SC6H4-p-Br 1262963-23-4 C10H10BrNOS
CH2CHCH2-NHC(CO)SC6H4-p-Br
—— 3-methylbut-2-enyl 2,4,5-trichlorophenyl ether 102222-99-1 C11H11Cl3O
3-methylbut-2-enyl 2,4,5-trichlorophenyl ether
—— (S)-5-(biphenyl-4-ylmethyl)-11-phenyl-2,4,7,10-tetraoxaundecane 1608463-86-0 C26H30O4
(S)-5-(biphenyl-4-ylmethyl)-11-phenyl-2,4,7,10-tetraoxaundecane
—— 3-((5-chloro-2-(trifluoromethyl)phenyl)ethynyl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine 1613332-96-9 C24H19ClF3N5
3-((5-chloro-2-(trifluoromethyl)phenyl)ethynyl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine
—— (+-)-1-methyl-(4ar,8ac)-decahydro-naphthalene-1t,2t-dicarboxylic acid dimethyl ester 101262-85-5 C15H24O4
(+-)-1-methyl-(4ar,8ac)-decahydro-naphthalene-1t,2t-dicarboxylic acid dimethyl ester
—— (Z)-5-chloro-2-(isopropoxydimethylsilyl)-1-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pent-1-ene 1023756-92-4 C16H32BClO3Si
(Z)-5-chloro-2-(isopropoxydimethylsilyl)-1-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pent-1-ene
—— 1-Diethyl-3-imino-3H-1λ<sup>6</sup>,2,6-thiadiazin-4,5-dicarbonitril 108675-30-5 C9H11N5S
1-Diethyl-3-imino-3H-1λ<sup>6</sup>,2,6-thiadiazin-4,5-dicarbonitril
—— N-[1-(β-acetoxy-phenethyl)-1H-[2]pyridyliden]-acetamide 101574-95-2 C17H18N2O3
N-[1-(β-acetoxy-phenethyl)-1H-[2]pyridyliden]-acetamide
—— [κ<sup>2</sup>-(anisyl)<sub>2</sub>P,O]Pd(Et)(PPh<sub>3</sub>) 1412440-86-8 C40H38O5P2PdS
[κ<sup>2</sup>-(anisyl)<sub>2</sub>P,O]Pd(Et)(PPh<sub>3</sub>)
—— 4-[(2E)-2-methylhex-2-en-1-yl]morpholine 1414942-64-5 C11H21NO
4-[(2E)-2-methylhex-2-en-1-yl]morpholine
—— 3-(Methoxycarbonyloxy)-5-methyl-2-methylene-N,N-dimethylhexanamide 141331-32-0 C12H21NO4
3-(Methoxycarbonyloxy)-5-methyl-2-methylene-N,N-dimethylhexanamide
—— N-(3-azidopropyl)-2,4-difluorobenzenesulfonamide 1160749-96-1 C9H10F2N4O2S
N-(3-azidopropyl)-2,4-difluorobenzenesulfonamide
—— (3-fluoro-4-trifluoromethyl-phenyl)-(3H-imidazol-4-ylmethyl)-isopropyl-amine 1020815-45-5 C14H15F4N3
(3-fluoro-4-trifluoromethyl-phenyl)-(3H-imidazol-4-ylmethyl)-isopropyl-amine
—— 4-[6-[4-(4-Amino-5-fluoropyrimidin-2-yl)oxypiperidin-1-yl]-5-fluoropyrimidin-4-yl]oxy-3-methoxybenzaldehyde 1033840-37-7 C21H20F2N6O4
4-[6-[4-(4-Amino-5-fluoropyrimidin-2-yl)oxypiperidin-1-yl]-5-fluoropyrimidin-4-yl]oxy-3-methoxybenzaldehyde
—— 4-chloro-3-hydroxysulfamoylbenzoic acid 1135370-43-2 C7H6ClNO5S
4-chloro-3-hydroxysulfamoylbenzoic acid
—— 1-[4-(3,5-bis-trifluoromethyl-phenoxy)-phenyl]carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan] 1159093-25-0 C28H24F6N2O3
1-[4-(3,5-bis-trifluoromethyl-phenoxy)-phenyl]carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan]
—— 4-(4-(2,6-dimethyl-4-(pyrimidin-4-yl)phenoxy)-5-methyl-5H-pyrrolo[3,2-d]pyrimidin-2-ylamino)benzonitrile 1164099-53-9 C26H21N7O
4-(4-(2,6-dimethyl-4-(pyrimidin-4-yl)phenoxy)-5-methyl-5H-pyrrolo[3,2-d]pyrimidin-2-ylamino)benzonitrile
—— 2-fluoro-5-(5-isopropyl-tetrazol-1-yl)-N-(5-methyl-pyrazin-2-ylmethyl)-3-(5-methyl-pyridin-2-yl)-benzamide 1161859-21-7 C23H23FN8O
2-fluoro-5-(5-isopropyl-tetrazol-1-yl)-N-(5-methyl-pyrazin-2-ylmethyl)-3-(5-methyl-pyridin-2-yl)-benzamide
—— 2-((1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)piperidin-2-yl)methoxy)-1-(4-(1-methylpiperidin-4-yl)piperazin-1-yl)ethanone 1018821-62-9 C23H35ClN6O4S2
2-((1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)piperidin-2-yl)methoxy)-1-(4-(1-methylpiperidin-4-yl)piperazin-1-yl)ethanone
—— dichloro-(2,3,4,6-tetrachloro-phenoxy)-[1,3,5]triazine 109047-34-9 C9HCl6N3O
dichloro-(2,3,4,6-tetrachloro-phenoxy)-[1,3,5]triazine
—— (3'R,4'S)-N-(5-methoxyoxazolo[5,4-b]pyridin-2-yl)-4H-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octan]-2-amine 1346215-71-1 C16H19N5O3
(3'R,4'S)-N-(5-methoxyoxazolo[5,4-b]pyridin-2-yl)-4H-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octan]-2-amine
—— 4-(3-(6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)phenylsulfonamido)benzylphosphonic acid 1234363-93-9 C23H23Cl2N2O5PS
4-(3-(6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)phenylsulfonamido)benzylphosphonic acid
—— 3-[4-(4-nitorobenzyloxy)-4'-(trifluoromethoxy)biphenyl-3-yl]propanoic acid 1018959-23-3 C23H18F3NO6
3-[4-(4-nitorobenzyloxy)-4'-(trifluoromethoxy)biphenyl-3-yl]propanoic acid
—— (1S,5S)-3-(3,3,3-trifluoropropanoyl)-3,6-diazabicyclo[3.2.1]octane 1215170-46-9 C9H13F3N2O
(1S,5S)-3-(3,3,3-trifluoropropanoyl)-3,6-diazabicyclo[3.2.1]octane
—— 1-ethyl-3-[6-(6-fluoro-pyridin-3-yl)-8-methyl-isoquinolin-3-yl]-urea 1338255-68-7 C18H17FN4O
1-ethyl-3-[6-(6-fluoro-pyridin-3-yl)-8-methyl-isoquinolin-3-yl]-urea
—— [2,3-dimethoxy-6-(1-oxo-3H-isobenzofuran-4-yl)phenyl]-3-methylsulfanylpropanoate 1345881-11-9 C20H20O6S
[2,3-dimethoxy-6-(1-oxo-3H-isobenzofuran-4-yl)phenyl]-3-methylsulfanylpropanoate
—— 3-methyl-N-(4-pyridin-3-yl-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2,4,6,12,14-hexaen-13-yl)pyridine-4-carboxamide 1017588-86-1 C25H21N5O
3-methyl-N-(4-pyridin-3-yl-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2,4,6,12,14-hexaen-13-yl)pyridine-4-carboxamide
—— US10202379, Reference Example 515 1370242-47-9 C27H29N3O4
US10202379, Reference Example 515
—— [(R)-3-(6-chloro-benzooxazol-2-ylamino)-pyrrolidin-1-yl]-[2-(1H-imidazol-2-yl)-phenyl]-methanone 1163121-54-7 C21H18ClN5O2
[(R)-3-(6-chloro-benzooxazol-2-ylamino)-pyrrolidin-1-yl]-[2-(1H-imidazol-2-yl)-phenyl]-methanone
—— 4-[4-(2,3-difluorophenyl)pyrimidin-2-yl]-N-pyridin-3-ylpiperazine-1-carboxamide 1143578-83-9 C20H18F2N6O
4-[4-(2,3-difluorophenyl)pyrimidin-2-yl]-N-pyridin-3-ylpiperazine-1-carboxamide
—— [1,1'-biphenyl]-4-yl(3-(2-(2,4-difluorophenyl)thiazol-4-yl)-8-methyl-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)methanone 1338372-94-3 C28H21F2N5OS
[1,1'-biphenyl]-4-yl(3-(2-(2,4-difluorophenyl)thiazol-4-yl)-8-methyl-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)methanone
—— N-(4-cyano-phenyl)-N'-(2-methanesulphonyloxyethyl)-N'-[4-(2-methoxycarbonyl-ethyl)-2-methyl-phenyl]-urea 1097299-31-4 C22H25N3O6S
N-(4-cyano-phenyl)-N'-(2-methanesulphonyloxyethyl)-N'-[4-(2-methoxycarbonyl-ethyl)-2-methyl-phenyl]-urea
—— 1-(2-Chlorophenyl)-1-(4-methyl-5-thiazolyl)methanol 162099-44-7 C11H10ClNOS
1-(2-Chlorophenyl)-1-(4-methyl-5-thiazolyl)methanol
—— (2S)-1-cyclopentyl-5-oxopyrrolidine-2-carboxylic acid 1164113-48-7 C10H15NO3
(2S)-1-cyclopentyl-5-oxopyrrolidine-2-carboxylic acid
—— 5-chloro-2-(4-methylsulfanyl-phenoxy)-benzaldehyde 1160655-64-0 C14H11ClO2S
5-chloro-2-(4-methylsulfanyl-phenoxy)-benzaldehyde
—— 2-methyl-4H-chromeno[4,3-c]pyrazole-3-carboxylic acid 1354408-27-7 C12H10N2O3
2-methyl-4H-chromeno[4,3-c]pyrazole-3-carboxylic acid
—— 5-(3-(difluoromethyl)phenyl)-1-isopropyl-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxylic acid ((5-methanesulfonylthiophen-2-yl)methyl)amide 1569648-75-4 C23H24F2N2O4S2
5-(3-(difluoromethyl)phenyl)-1-isopropyl-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxylic acid ((5-methanesulfonylthiophen-2-yl)methyl)amide
—— 4-oxo-4H,5H,6H,7H,8H-thieno[3,2-c]azepine-2-carboxylicacid 1501177-75-8 C9H9NO3S
4-oxo-4H,5H,6H,7H,8H-thieno[3,2-c]azepine-2-carboxylicacid
—— N-(3-azidopropyl)-4-methoxybenzenesulfonamide 1160750-04-8 C10H14N4O3S
N-(3-azidopropyl)-4-methoxybenzenesulfonamide
—— 2-(4-methoxy-2-oxopyridin-1(2H)-yl)-4-methylthiazole-5-carboxylic acid 1105690-73-0 C11H10N2O4S
2-(4-methoxy-2-oxopyridin-1(2H)-yl)-4-methylthiazole-5-carboxylic acid
—— ethyl 1-[(1S)-1-(1-hydroxycyclohexyl)ethyl]-5-phenyl-1H-imidazole-4-carboxylate 1084793-51-0 C20H26N2O3
ethyl 1-[(1S)-1-(1-hydroxycyclohexyl)ethyl]-5-phenyl-1H-imidazole-4-carboxylate
—— (S)-N'-cyano-N-(3-(N-isopropylsulfamoyl)phenyl)-2-methyl-4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazine-1-carboximidamide 1116570-37-6 C23H29N9O2S
(S)-N'-cyano-N-(3-(N-isopropylsulfamoyl)phenyl)-2-methyl-4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazine-1-carboximidamide
—— benzyl ((S)-1-((2-(((S)-1-((2-(2,6-dioxocyclohexyl)-2-oxoethyl)amino)-4-methyl-1-oxo-pentan-2-yl)amino)-2-oxoethyl)amino)-1-oxo-3-phenylpropan-2-yl)carbamate 1384584-19-3 C33H40N4O8
benzyl ((S)-1-((2-(((S)-1-((2-(2,6-dioxocyclohexyl)-2-oxoethyl)amino)-4-methyl-1-oxo-pentan-2-yl)amino)-2-oxoethyl)amino)-1-oxo-3-phenylpropan-2-yl)carbamate
—— 4-bromo-2,2,5,5-tetramethyl-3-[(phenylamino)carbonyl]-2,5-dihydro-1H-pyrrol-1-oxyl 1422058-64-7 C15H20BrN2O2
4-bromo-2,2,5,5-tetramethyl-3-[(phenylamino)carbonyl]-2,5-dihydro-1H-pyrrol-1-oxyl
—— benzyl 2-fluoro-3-(1-(6-(2-methoxyethoxy)-1H-indol-3-yl)-2-nitroethyl)phenylcarbamate 1352835-78-9 C27H26FN3O6
benzyl 2-fluoro-3-(1-(6-(2-methoxyethoxy)-1H-indol-3-yl)-2-nitroethyl)phenylcarbamate
—— trans-2-Acetoxy-3,5-dimethyl-2,3-dihydronaphtho<2,3-b>furan-4,9-dione 133700-96-6 C16H14O5
trans-2-Acetoxy-3,5-dimethyl-2,3-dihydronaphtho<2,3-b>furan-4,9-dione
—— (Z)-3-(3,6-Dichloro-pyridazin-4-yl)-3-hydroxy-2-(1-methyl-1H-benzoimidazol-2-yl)-acrylonitrile 120776-45-6 C15H9Cl2N5O
(Z)-3-(3,6-Dichloro-pyridazin-4-yl)-3-hydroxy-2-(1-methyl-1H-benzoimidazol-2-yl)-acrylonitrile
—— [(C4H6N2(Bu-t)2)(CH2)4OB(pentafluorophenyl)3] 1313574-33-2 C34H32BF15N2O
[(C4H6N2(Bu-t)2)(CH2)4OB(pentafluorophenyl)3]
—— ethyl 1-methyl-4,5-bis(4-methylphenyl)-1H-pyrrole-2-carboxylate 1399297-40-5 C22H23NO2
ethyl 1-methyl-4,5-bis(4-methylphenyl)-1H-pyrrole-2-carboxylate
—— 9-butyl-2,2,4,4-tetrachloro-9-ethyl-7,11-dioxa-1,3,5-triaza-2l5,4l5,6l5-triphosphaspiro[5.5]undeca-1(6),2,4-triene 1257063-63-0 C9H18Cl4N3O2P3
9-butyl-2,2,4,4-tetrachloro-9-ethyl-7,11-dioxa-1,3,5-triaza-2l5,4l5,6l5-triphosphaspiro[5.5]undeca-1(6),2,4-triene