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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S,4S)-1-(2-(1H-1,2,4-triazol-1-yl)acetyl)-4-((5-chloro-2-thienyl)methyl)-N-(4-(4-fluorophenoxy)phenyl)pyrrolidine-2-carboxamide 1221877-98-0 C26H23ClFN5O3S
(2S,4S)-1-(2-(1H-1,2,4-triazol-1-yl)acetyl)-4-((5-chloro-2-thienyl)methyl)-N-(4-(4-fluorophenoxy)phenyl)pyrrolidine-2-carboxamide
—— (S)-4-(3-chloro-4-fluorophenyl)-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one 1269650-27-2 C29H29ClFN7O3Si
(S)-4-(3-chloro-4-fluorophenyl)-3-(3-(4-(1-((2-(trimethylsilyl)ethoxy)methyl)-1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)oxazolidin-2-one
—— 1-{3-[2-isobutylaminopyridin-4-yl]-[2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid isobutylamide 1071133-58-8 C27H36N6O
1-{3-[2-isobutylaminopyridin-4-yl]-[2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid isobutylamide
—— 4,6-dihydroxy-2-[(4-hydroxy-1-methyl-1H-indol-3-yl)methylene]-1-benzofuran-3(2H)-one 1200532-57-5 C18H13NO5
4,6-dihydroxy-2-[(4-hydroxy-1-methyl-1H-indol-3-yl)methylene]-1-benzofuran-3(2H)-one
—— 4-(4-chlorophenyl)-1-(7-(2-methoxyphenylthio)benzo[c][1,2,5]oxadiazol-4-ylsulfonyl)piperidin-4-ol 1062659-00-0 C24H22ClN3O5S2
4-(4-chlorophenyl)-1-(7-(2-methoxyphenylthio)benzo[c][1,2,5]oxadiazol-4-ylsulfonyl)piperidin-4-ol
—— 3-hydroxy-6-phenyl-2-(1-phenylcyclopropyl)-8-(trifluoromethyl)quinoline-4-carboxylic acid 1067187-21-6 C26H18F3NO3
3-hydroxy-6-phenyl-2-(1-phenylcyclopropyl)-8-(trifluoromethyl)quinoline-4-carboxylic acid
—— 5,12,18,25,31,38,44,51-octahexoxy-2,15,28,41,53,54,55,56-octazatridecacyclo[40.10.1.13,14.116,27.129,40.04,13.06,11.017,26.019,24.030,39.032,37.043,52.045,50]hexapentaconta-1,3,5,7,9,11,13,15,17,19,21,23,25,27,29(54),30,32,34,36,38,40,42(53),43,45,47,49,51-heptacosaene 162208-17-5 C96H122N8O8
5,12,18,25,31,38,44,51-octahexoxy-2,15,28,41,53,54,55,56-octazatridecacyclo[40.10.1.13,14.116,27.129,40.04,13.06,11.017,26.019,24.030,39.032,37.043,52.045,50]hexapentaconta-1,3,5,7,9,11,13,15,17,19,21,23,25,27,29(54),30,32,34,36,38,40,42(53),43,45,47,49,51-heptacosaene
—— 1-[6-Deuterio-4-[(2,4-dioxo-3,1-benzoxazin-1-yl)methyl]pyridin-2-yl]-3-methylurea 1228273-83-3 C16H14N4O4
1-[6-Deuterio-4-[(2,4-dioxo-3,1-benzoxazin-1-yl)methyl]pyridin-2-yl]-3-methylurea
—— (1S,2R)-2-(4-{[(2S)-2-(1H-benzimidazol-1-ylmethyl)piperazin-1-yl]carbonyl}-5-phenyl-1H-imidazol-1-yl)-1-(methoxymethyl)cyclohexanol 1083850-05-8 C30H36N6O3
(1S,2R)-2-(4-{[(2S)-2-(1H-benzimidazol-1-ylmethyl)piperazin-1-yl]carbonyl}-5-phenyl-1H-imidazol-1-yl)-1-(methoxymethyl)cyclohexanol
—— [(1S,2S,3S)-2-methyl-2-(4-methylpent-3-enyl)-3-phenylcyclopropyl]methanol 1193729-58-6 C17H24O
[(1S,2S,3S)-2-methyl-2-(4-methylpent-3-enyl)-3-phenylcyclopropyl]methanol
—— 1-[(2Z)-2-{[1-methyl-4-(3-oxa-9-azabicyclo[3.3.1]non-9-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-3-oxo-2,3-dihydro-1-benzofuran-5-yl]-3-pyridin-3-ylurea 1198277-33-6 C30H28N6O4
1-[(2Z)-2-{[1-methyl-4-(3-oxa-9-azabicyclo[3.3.1]non-9-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-3-oxo-2,3-dihydro-1-benzofuran-5-yl]-3-pyridin-3-ylurea
—— 1-chloro-4-[(R)-1-(9H-purin-6-yl)pyrrolidin-2-yl-methoxy]isoquinoline 1201581-35-2 C19H17ClN6O
1-chloro-4-[(R)-1-(9H-purin-6-yl)pyrrolidin-2-yl-methoxy]isoquinoline
—— 2-[4-(4-Carbamoylpiperazin-1-yl)anilino]-4-(3-methylanilino)pyrimidine-5-carboxamide 1198304-17-4 C23H26N8O2
2-[4-(4-Carbamoylpiperazin-1-yl)anilino]-4-(3-methylanilino)pyrimidine-5-carboxamide
—— 2-fluoro-6-({3-[3-methyl-8-(trifluoromethyl)quinolin-4-yl]benzyl}amino)benzoic acid 1127737-21-6 C25H18F4N2O2
2-fluoro-6-({3-[3-methyl-8-(trifluoromethyl)quinolin-4-yl]benzyl}amino)benzoic acid
—— 2-[4-fluoro-2-(trifluoromethyl)phenyl]-N-[6-(pyrrolidin-1-ylmethyl)pyridin-2-yl]imidazo[1,2-a]pyridine-8-carboxamide 1198168-91-0 C25H21F4N5O
2-[4-fluoro-2-(trifluoromethyl)phenyl]-N-[6-(pyrrolidin-1-ylmethyl)pyridin-2-yl]imidazo[1,2-a]pyridine-8-carboxamide
—— 5-(4-chorophenyl)-4-(1-(p-tolylamino)ethylene)-1-(4-hydroxyphenyl)pyrrolidine-2,3-dione 1240245-85-5 C25H21ClN2O3
5-(4-chorophenyl)-4-(1-(p-tolylamino)ethylene)-1-(4-hydroxyphenyl)pyrrolidine-2,3-dione
—— N-((S)-2-((3aS,6S,6aR)-6-methyl-3-oxodihydro-2H-furo[3,2-b]pyrrol-4(5H,6H,6aH)-yl)-1-(1-methylcyclopentyl)-2-oxoethyl)-4-sulfamoylbenzamide 1198092-25-9 C22H29N3O6S
N-((S)-2-((3aS,6S,6aR)-6-methyl-3-oxodihydro-2H-furo[3,2-b]pyrrol-4(5H,6H,6aH)-yl)-1-(1-methylcyclopentyl)-2-oxoethyl)-4-sulfamoylbenzamide
—— 4-(7-bromo-1H-indol-3-yl)-4-[4-(trifluoromethyl)phenyl]butan-1-ol 1202463-08-8 C19H17BrF3NO
4-(7-bromo-1H-indol-3-yl)-4-[4-(trifluoromethyl)phenyl]butan-1-ol
—— [4-chloro-3-(piperidine-1-sulfonyl)-phenyl]-(4aS,8aR)-decahydro-isoquinolin-2-yl-methanone 1046270-85-2 C21H29ClN2O3S
[4-chloro-3-(piperidine-1-sulfonyl)-phenyl]-(4aS,8aR)-decahydro-isoquinolin-2-yl-methanone
—— 2-(3-(4-fluorobenzyl)-2-oxoimidazolidin-1-yl)-N-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)isonicotinamide 1202927-50-1 C20H19FN6O3
2-(3-(4-fluorobenzyl)-2-oxoimidazolidin-1-yl)-N-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)isonicotinamide
—— propynoic acid (cyclohexylcarbamoylmethyl)methylamide 1201220-29-2 C12H18N2O2
propynoic acid (cyclohexylcarbamoylmethyl)methylamide
—— 1-[5-hydroxymethyl-3-(4-methoxybenzyl)-3H-[1,2,3]triazol-4-yl]ethanone 1233012-04-8 C13H15N3O3
1-[5-hydroxymethyl-3-(4-methoxybenzyl)-3H-[1,2,3]triazol-4-yl]ethanone
—— N-(3-(benzyloxy)phenyl)-2-hydroxy-4-(4-(trifluoromethyl)phenyl)butanamide 1033777-22-8 C24H22F3NO3
N-(3-(benzyloxy)phenyl)-2-hydroxy-4-(4-(trifluoromethyl)phenyl)butanamide
—— 2-(3,4-difluorophenoxy)-N-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethyl]-acetamide 1092946-21-8 C20H19F3N2O2
2-(3,4-difluorophenoxy)-N-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethyl]-acetamide
—— 10-methyl-3,6,8,10,11-pentaazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2,7,11-tetraene-7-thiol 1092291-84-3 C8H9N5S
10-methyl-3,6,8,10,11-pentaazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2,7,11-tetraene-7-thiol
—— N-(3,4-dichloro-benzyl)-2-(3,4-dichloro-phenyl)-4-(4-methanesulfonyl-piperazin-1-yl)-2-methylbutyramide 1093078-09-1 C23H27Cl4N3O3S
N-(3,4-dichloro-benzyl)-2-(3,4-dichloro-phenyl)-4-(4-methanesulfonyl-piperazin-1-yl)-2-methylbutyramide
—— 5-(6-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-3-yl)pyrazin-2-ylamine 1084951-81-4 C16H11F3N8
5-(6-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-3-yl)pyrazin-2-ylamine
—— methyl 2-(3-((N-(3-(4-amino-2-(2-methoxyethyl)-1H-imidazo[4,5-c]quinolin-1-yl)propyl)-2-(4-methylpiperazin-1-yl)acetamido)methyl)phenyl)acetate 1080009-61-5 C33H43N7O4
methyl 2-(3-((N-(3-(4-amino-2-(2-methoxyethyl)-1H-imidazo[4,5-c]quinolin-1-yl)propyl)-2-(4-methylpiperazin-1-yl)acetamido)methyl)phenyl)acetate
—— [3-(7-chloro-imidazo[1,2-a]pyridin-3-yl)-phenyl]-[1,3,4]thiadiazol-2-yl-amine 1036761-82-6 C15H10ClN5S
[3-(7-chloro-imidazo[1,2-a]pyridin-3-yl)-phenyl]-[1,3,4]thiadiazol-2-yl-amine
—— 4-(2,4-dichlorophenyl)-6-[(2-fluorophenyl)acetyl]-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-2-amine 1046859-13-5 C20H15Cl2FN4O
4-(2,4-dichlorophenyl)-6-[(2-fluorophenyl)acetyl]-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-2-amine
—— 4-bromo-1-isopropyl-1H-indole 1219741-49-7 C11H12BrN
4-bromo-1-isopropyl-1H-indole
—— (E)-2-cyano-3-(5'-(5''-(p-(di-p-tolylamino)phenyl)thiophen-2''-yl)thiophen-2'-yl)acrylic acid 1219091-37-8 C32H24N2O2S2
(E)-2-cyano-3-(5'-(5''-(p-(di-p-tolylamino)phenyl)thiophen-2''-yl)thiophen-2'-yl)acrylic acid
—— 2-(4-fluorophenyl)-5-[4-(2-hydroxyethylcarbamoyl)phenyl]-N-methyl-1-benzofuran-3-carboxamide 1217335-05-1 C25H21FN2O4
2-(4-fluorophenyl)-5-[4-(2-hydroxyethylcarbamoyl)phenyl]-N-methyl-1-benzofuran-3-carboxamide
—— (2-benzyl-3-oxo-2,3-dihydro-pyridazin-4-yl)-acetic acid ethyl ester 1005750-70-8 C15H16N2O3
(2-benzyl-3-oxo-2,3-dihydro-pyridazin-4-yl)-acetic acid ethyl ester
—— 4-(4-methyl-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-7-yl)-N-(3-methyl-4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)phenyl)pyrimidin-2-amine 1182181-31-2 C25H29N7O
4-(4-methyl-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-7-yl)-N-(3-methyl-4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)phenyl)pyrimidin-2-amine
—— 3-oxo-2-[2-(2-oxopyrrolidin-1-yl)etthyl]-N-[[4-(trifluoromethoxy)phenyl]methyl]-1H-isoindole-1-carboxamide 1198160-20-1 C23H22F3N3O4
3-oxo-2-[2-(2-oxopyrrolidin-1-yl)etthyl]-N-[[4-(trifluoromethoxy)phenyl]methyl]-1H-isoindole-1-carboxamide
—— 2,4-dichloro-N-(4-(4-phenyl-5-(trifluoromethyl)oxazol-2-yl)phenyl)benzamide 1200404-44-9 C23H13Cl2F3N2O2
2,4-dichloro-N-(4-(4-phenyl-5-(trifluoromethyl)oxazol-2-yl)phenyl)benzamide
—— 6-{[6-(3,5-dimethyl-1H-pyrazol-4-yl)-1H-imidazo[4,5-b]pyridin-2-yl]methyl}-3-(2,4,6-trifluorobenzoyl)-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one 1201597-12-7 C26H18F3N7O2
6-{[6-(3,5-dimethyl-1H-pyrazol-4-yl)-1H-imidazo[4,5-b]pyridin-2-yl]methyl}-3-(2,4,6-trifluorobenzoyl)-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one
—— 3-cyclobutyl-1-[4-(2,2-difluoro-1-phenyl-vinyl)-phenyl]-imidazo[1,5-a]pyrazin-8-ylamine 1196388-60-9 C24H20F2N4
3-cyclobutyl-1-[4-(2,2-difluoro-1-phenyl-vinyl)-phenyl]-imidazo[1,5-a]pyrazin-8-ylamine
—— 4-[(3R)-3-aminopyrrolidin-1-yl]-7a,8,9,10,11,11a-hexahydro[1]benzofuro[2,3-h]quinazolin-2-amine 1348366-90-4 C18H23N5O
4-[(3R)-3-aminopyrrolidin-1-yl]-7a,8,9,10,11,11a-hexahydro[1]benzofuro[2,3-h]quinazolin-2-amine
—— 3-ethoxymethyl-2-phenylimino-2H-chromene 1371631-09-2 C18H17NO2
3-ethoxymethyl-2-phenylimino-2H-chromene
—— 3-Fluoro-5-hydroxymethyl-2-(4-isopropoxy benzoyl)phenol 1005488-17-4 C17H17FO4
3-Fluoro-5-hydroxymethyl-2-(4-isopropoxy benzoyl)phenol
—— 2-(2,3-difluorobenzyl)-6,7-dimethoxyisoindolin-1-one 1123214-30-1 C17H15F2NO3
2-(2,3-difluorobenzyl)-6,7-dimethoxyisoindolin-1-one
—— [{1-[5-(2-acetylamino-ethoxy)-pyrazin-2-yl]-1H-indol-5-yl}-(3,5-dichloro-phenylsulphonyl)-amino]-acetic acid 1049029-80-2 C24H21Cl2N5O6S
[{1-[5-(2-acetylamino-ethoxy)-pyrazin-2-yl]-1H-indol-5-yl}-(3,5-dichloro-phenylsulphonyl)-amino]-acetic acid
—— 4-Chloro-3-cyclopropyl-1-phenyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid 1026223-22-2 C16H12ClN3O2
4-Chloro-3-cyclopropyl-1-phenyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
—— 4-[(1R)-1-({[(6R)-6-(5-chloro-2-methoxybenzyl)-7-oxo-3-(phenoxyimino)-1,4-diazepan-1-yl]carbonyl}amino)propyl]-2-fluorobenzoic acid 1312768-82-3 C30H30ClFN4O6
4-[(1R)-1-({[(6R)-6-(5-chloro-2-methoxybenzyl)-7-oxo-3-(phenoxyimino)-1,4-diazepan-1-yl]carbonyl}amino)propyl]-2-fluorobenzoic acid
—— 1-[4-((5R,8S,11R,13S,14S,17S)-5,17-dihydroxy-17-pentafluoroethyl-5',5',13-trimethyl-1,2,3,4,6,7,8,11,12,13,14,15,16,17-tetradecahydrospiro[cyclopenta[a]phenanthrene-3,2'-[1,3]dioxan]-11-yl)benzyl]-3-(3,5-dimethyl isoxazol-4-yl)urea 1262049-66-0 C38H48F5N3O6
1-[4-((5R,8S,11R,13S,14S,17S)-5,17-dihydroxy-17-pentafluoroethyl-5',5',13-trimethyl-1,2,3,4,6,7,8,11,12,13,14,15,16,17-tetradecahydrospiro[cyclopenta[a]phenanthrene-3,2'-[1,3]dioxan]-11-yl)benzyl]-3-(3,5-dimethyl isoxazol-4-yl)urea
—— 2-(2,6-difluorophenyl)-5-(4-(methylsulfonyl)phenyl)oxazole-4-carboxamide 1082440-75-2 C17H12F2N2O4S
2-(2,6-difluorophenyl)-5-(4-(methylsulfonyl)phenyl)oxazole-4-carboxamide
—— 4-(4-methoxy-3-nitrophenyl)-6-(3,4,5-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-2-thione 1073793-03-9 C20H21N3O6S
4-(4-methoxy-3-nitrophenyl)-6-(3,4,5-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-2-thione
—— N-tert-butyl-2-[1-(2-hydroxypropyl)-2-[3-(trifluoromethyl)phenyl]indol-5-yl]-2-methylpropanamide 1076219-77-6 C26H31F3N2O2
N-tert-butyl-2-[1-(2-hydroxypropyl)-2-[3-(trifluoromethyl)phenyl]indol-5-yl]-2-methylpropanamide