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中文名称 英文名称 CAS号 化学式 结构式图片
—— —— 1361136-95-9 C11H13ClN6O
—— —— 1072437-23-0 C45H63N3O3
—— (S)-3-[(S)-1-(2-chloro-3-fluorophenoxy)-2-isopropylsulfanylethyl]pyrrolidine trifluoroacetate 1262116-06-2 C2HF3O2*C15H21ClFNOS
(S)-3-[(S)-1-(2-chloro-3-fluorophenoxy)-2-isopropylsulfanylethyl]pyrrolidine trifluoroacetate
—— (E)-2-(4-(cyclopropylsulfonyl)phenyl)-3-[(1α,3α,4α)-3,4-difluorocyclopentyl]-N-(6-fluorobenzo[d]thiazol-2-yl)propenoic acid amide 1193394-79-4 C24H21F3N2O3S2
(E)-2-(4-(cyclopropylsulfonyl)phenyl)-3-[(1α,3α,4α)-3,4-difluorocyclopentyl]-N-(6-fluorobenzo[d]thiazol-2-yl)propenoic acid amide
—— methyl 2-[4-[{4-butyl-2-methyl-6-oxo-1-(pyridin-2-yl)-1,6-dihydropyrimidin-5-yl}methyl]-2,6-dipropylphenoxy]-2-(2-chlorophenyl)acetate 1256780-02-5 C36H42ClN3O4
methyl 2-[4-[{4-butyl-2-methyl-6-oxo-1-(pyridin-2-yl)-1,6-dihydropyrimidin-5-yl}methyl]-2,6-dipropylphenoxy]-2-(2-chlorophenyl)acetate
—— 3-[4-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-1-yl)butyl]-5,5-dimethyl-imidazolidine-2,4-dione 1417032-78-0 C26H31N5O2S
3-[4-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-1-yl)butyl]-5,5-dimethyl-imidazolidine-2,4-dione
—— (S)-2-({2-[3-(3-hydroxy-phenyl)propylamino]-4,6-dimethyl-pyrimidine-5-carbonyl}amino)-3-[(3-methyl-thiophene-2-carbonyl)amino]propionic acid 1400704-71-3 C25H29N5O5S
(S)-2-({2-[3-(3-hydroxy-phenyl)propylamino]-4,6-dimethyl-pyrimidine-5-carbonyl}amino)-3-[(3-methyl-thiophene-2-carbonyl)amino]propionic acid
—— 1-(3-(4-(2-aminopyridin-4-yl)-2-methylthiazol-5-yl)phenyl)-3-(4-chlorophenyl)urea 1400214-72-3 C22H18ClN5OS
1-(3-(4-(2-aminopyridin-4-yl)-2-methylthiazol-5-yl)phenyl)-3-(4-chlorophenyl)urea
—— (2S,3S)-2-[({2-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl}methyl)amino]butane-1,3-diol 1401164-26-8 C16H18F3N3O2
(2S,3S)-2-[({2-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl}methyl)amino]butane-1,3-diol
—— tert-butyl cyclopropyl[3-hydroxy-5-(3-methoxypropoxy)benzyl]carbamate 1399849-51-4 C19H29NO5
tert-butyl cyclopropyl[3-hydroxy-5-(3-methoxypropoxy)benzyl]carbamate
—— —— 1448006-44-7 C13H14N2O4
—— —— 1361958-90-8 C20H18ClFN2O5
—— —— 1361138-69-3 C13H16BrN5OS
—— (S)-1-(4-chloro-phenyl)-2-{4-[(S)-1-hydroxy-1-(7-oxa-bicyclo[2.2.1]hept-1-yl)-ethyl]phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416909-48-2 C33H36ClNO5
(S)-1-(4-chloro-phenyl)-2-{4-[(S)-1-hydroxy-1-(7-oxa-bicyclo[2.2.1]hept-1-yl)-ethyl]phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— N(1)Gly-D-hPhe-Bip-D-Phe-Phe(4-CO2H)(1)-OH 1211439-07-4 C46H45N5O7
N(1)Gly-D-hPhe-Bip-D-Phe-Phe(4-CO2H)(1)-OH
—— tert-butyl N-[(4aR,11bR)-10-[(5-chloropyrazine-2-carbonyl)amino]-3,3,6,6,11b-pentamethyl-4,4-dioxo-4a,5-dihydro-[1]-benzoxepino[4,5-b][1,4]thiazin-2-yl]-N-tert-butoxycarbonylcarbamate 1620981-54-5 C32H42ClN5O8S
tert-butyl N-[(4aR,11bR)-10-[(5-chloropyrazine-2-carbonyl)amino]-3,3,6,6,11b-pentamethyl-4,4-dioxo-4a,5-dihydro-[1]-benzoxepino[4,5-b][1,4]thiazin-2-yl]-N-tert-butoxycarbonylcarbamate
—— (3'R,4'aR,8'aR)-N-(cyclopropylmethyl)-1'-methylspiro[1,3-dioxolane-2,6'-2,3,4,4a,5,7,8,8a-octahydroquinoline]-3'-carboxamide 1399447-57-4 C17H28N2O3
(3'R,4'aR,8'aR)-N-(cyclopropylmethyl)-1'-methylspiro[1,3-dioxolane-2,6'-2,3,4,4a,5,7,8,8a-octahydroquinoline]-3'-carboxamide
—— N-(3-amino-2,4-difluorophenyl)-3-fluoro-N-(4-methoxybenzyl)propane-1-sulfonamide 1269421-53-5 C17H19F3N2O3S
N-(3-amino-2,4-difluorophenyl)-3-fluoro-N-(4-methoxybenzyl)propane-1-sulfonamide
—— 1-cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(5-(morpholinomethyl)pyridin-2-yl)-1H-indazole-4-carboxamide 1396772-90-9 C31H36N6O3
1-cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(5-(morpholinomethyl)pyridin-2-yl)-1H-indazole-4-carboxamide
—— —— 1260720-25-9 C15H19N3O4
—— —— 1350805-79-6 C24H22F5N5O2
—— —— 1361340-47-7 C18H18Cl2F2N2O3S
—— —— 1252879-39-2 C23H24ClFN2O5
—— —— 1252879-65-4 C23H24ClFN2O5
—— 6-Fluoro-7-pyridin-4-yl-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417180-59-6 C24H18FN3O
6-Fluoro-7-pyridin-4-yl-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-(pyridin-2-ylmethoxy)pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol 1416860-04-2 C21H16F4N6O2
2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-(pyridin-2-ylmethoxy)pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol
—— 8-bromo-1-(5-chloropyridin-3-yl)-4-methyl[1,2,4]triazolo[4,3-a]quinoxaline 1417410-86-6 C15H9BrClN5
8-bromo-1-(5-chloropyridin-3-yl)-4-methyl[1,2,4]triazolo[4,3-a]quinoxaline
—— 6-chloro-N-[[1-[2-(2,3-dihydro-1,4-benzodioxin-5-yloxy)ethyl]azetidin-3-yl]methyl]naphthalene-2-sulphonamide 1417309-46-6 C24H25ClN2O5S
6-chloro-N-[[1-[2-(2,3-dihydro-1,4-benzodioxin-5-yloxy)ethyl]azetidin-3-yl]methyl]naphthalene-2-sulphonamide
—— 2-(4-chloro-2-fluorophenyl)-1,1-difluoro-1-(5-chloropyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol 1416733-75-9 C15H10Cl2F3N5O
2-(4-chloro-2-fluorophenyl)-1,1-difluoro-1-(5-chloropyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol
—— (8R,11S,14S,17S)-14-(2-methylpropyl)-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211436-40-6 C41H45N5O7S
(8R,11S,14S,17S)-14-(2-methylpropyl)-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— N-(2,6-difluorophenyl)-4-[5-(1-hydroxy-1-methyl-2-{methyl[2-(trifluoromethyl)pyrimidin-4-yl]amino}ethyl)-2-methylpyrimidin-4-yl]piperidine-1-carboxamide 1603905-05-0 C26H28F5N7O2
N-(2,6-difluorophenyl)-4-[5-(1-hydroxy-1-methyl-2-{methyl[2-(trifluoromethyl)pyrimidin-4-yl]amino}ethyl)-2-methylpyrimidin-4-yl]piperidine-1-carboxamide
—— 1-[(1S)-2-methoxy-1-phenylethyl]-3-{3-[(2S)-2-methylmorpholin-4-yl]-1H-pyrazolo[4,3-c]pyridin-6-yl}urea 1589536-42-4 C21H26N6O3
1-[(1S)-2-methoxy-1-phenylethyl]-3-{3-[(2S)-2-methylmorpholin-4-yl]-1H-pyrazolo[4,3-c]pyridin-6-yl}urea
—— 1-[(3-chlorophenyl)methyl]-3-(2,4-dioxo-1H-thieno[3,4-d]pyrimidin-3-yl)-5-(trifluoromethyl)indole-2-carboxylic acid 1154601-16-7 C23H13ClF3N3O4S
1-[(3-chlorophenyl)methyl]-3-(2,4-dioxo-1H-thieno[3,4-d]pyrimidin-3-yl)-5-(trifluoromethyl)indole-2-carboxylic acid
—— 1-(1H-indazol-4-yl)-3-[(1S,3R)-3-(4-methyl-1,3-oxazol-2-yl)cyclopentyl]urea 1401077-86-8 C17H19N5O2
1-(1H-indazol-4-yl)-3-[(1S,3R)-3-(4-methyl-1,3-oxazol-2-yl)cyclopentyl]urea
—— (2R)-2-[({3-fluoro-6-[1-(4-fluorophenyl)ethyl]pyridin-2-yl}methyl)amino]-3-methylbutan-1-ol 1401164-03-1 C19H24F2N2O
(2R)-2-[({3-fluoro-6-[1-(4-fluorophenyl)ethyl]pyridin-2-yl}methyl)amino]-3-methylbutan-1-ol
—— 1-(1-methyl-1H-pyrazol-4-yl)-3-[3-(2-methylpyrimidin-4-yl)benzyl]pyridazin-4(1H)-one 1314380-97-6 C20H18N6O
1-(1-methyl-1H-pyrazol-4-yl)-3-[3-(2-methylpyrimidin-4-yl)benzyl]pyridazin-4(1H)-one
—— (2R)-2-[({3-fluoro-6-[3-(trifluoromethyl)pyrrolidin-1-yl]pyridin-2-yl}methyl)amino]-3-methylbutan-1-ol 1401163-18-5 C16H23F4N3O
(2R)-2-[({3-fluoro-6-[3-(trifluoromethyl)pyrrolidin-1-yl]pyridin-2-yl}methyl)amino]-3-methylbutan-1-ol
—— N-(cyclopropylmethyl)-N-[4-[3-[(2S)-1-hydroxypropan-2-yl]oxy-5-[(1-methylpyrazol-3-yl)carbamoyl]phenoxy]phenyl]oxane-4-carboxamide 1310806-92-8 C30H36N4O6
N-(cyclopropylmethyl)-N-[4-[3-[(2S)-1-hydroxypropan-2-yl]oxy-5-[(1-methylpyrazol-3-yl)carbamoyl]phenoxy]phenyl]oxane-4-carboxamide
—— (S)-methyl 4-(tert-butoxycarbonyl(methyl)amino)-3-(4-chloro-3-fluorophenyl)butanoate 1395078-63-3 C17H23ClFNO4
(S)-methyl 4-(tert-butoxycarbonyl(methyl)amino)-3-(4-chloro-3-fluorophenyl)butanoate
—— 2-amino-6-[[5-(4-chlorophenyl)-1,3-oxazol-4-yl]methylsulfanyl]-4-[4-[(2S)-2,3-dihydroxypropoxy]phenyl]pyridine-3,5-dicarbonitrile 1107662-62-3 C26H20ClN5O4S
2-amino-6-[[5-(4-chlorophenyl)-1,3-oxazol-4-yl]methylsulfanyl]-4-[4-[(2S)-2,3-dihydroxypropoxy]phenyl]pyridine-3,5-dicarbonitrile
—— 2-(4-fluoro-2-methyl-phenylamino)-5,8-dihydro-6H-pyrido[3,4-d]pyrimidine-7-carboxylic acid [(S)-1-(4-chloro-3-fluoro-phenyl)-2-hydroxy-ethyl]-amide 1395076-22-8 C23H22ClF2N5O2
2-(4-fluoro-2-methyl-phenylamino)-5,8-dihydro-6H-pyrido[3,4-d]pyrimidine-7-carboxylic acid [(S)-1-(4-chloro-3-fluoro-phenyl)-2-hydroxy-ethyl]-amide
—— (S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416952-52-7 C35H41ClN2O4
(S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— 2-methyl-8-(4-pyridinyl)-3-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]-imidazo[1,2-a]pyrazine 1334166-40-3 C17H13F3N6
2-methyl-8-(4-pyridinyl)-3-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]-imidazo[1,2-a]pyrazine
—— 6-[2-(6-Chloro-1,3-benzothiazol-2-yl)ethyl]-4-(4-pyridyl)-7H-pyrrolo[3,4-b]pyridin-5-one 1417185-86-4 C21H15ClN4OS
6-[2-(6-Chloro-1,3-benzothiazol-2-yl)ethyl]-4-(4-pyridyl)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (S)-1-(4-chloro-phenyl)-2-[4-(1-hydroxy-1-methyl-propyl)-phenyl]-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416907-73-7 C29H32ClNO4
(S)-1-(4-chloro-phenyl)-2-[4-(1-hydroxy-1-methyl-propyl)-phenyl]-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— —— 1361339-07-2 C17H15Cl2NO3S
—— —— 1263421-41-5 C19H21N5O2
—— —— 1361958-33-9 C21H22N2O6
—— —— 1361340-26-2 C16H11BrClF5N2O4S
—— 3-(4-{[1-(4-methoxyphenyl)ethyl]amino}phenyl)-2-furancarboxylic acid-2-(4-hydroxy-3-nitrobenzoyl)hydrazide hydrochloride 1255148-77-6 C27H24N4O7*ClH
3-(4-{[1-(4-methoxyphenyl)ethyl]amino}phenyl)-2-furancarboxylic acid-2-(4-hydroxy-3-nitrobenzoyl)hydrazide hydrochloride