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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-{(S)-4-carboxy-2-[(4-{2-[(S)-2-(cyclopropylmethyl-carbamoyl)-pyrrolidin-1-yl]-2-oxo-ethoxy}-7-methyl-quinoline-2-carbonyl)-amino]-butyryl}-piperazine-1-carboxylic acid ethyl ester 1073445-81-4 C34H44N6O9
4-{(S)-4-carboxy-2-[(4-{2-[(S)-2-(cyclopropylmethyl-carbamoyl)-pyrrolidin-1-yl]-2-oxo-ethoxy}-7-methyl-quinoline-2-carbonyl)-amino]-butyryl}-piperazine-1-carboxylic acid ethyl ester
—— 1-benzyl-4-(3-methylamino-pyrrolidin-1-yl)-1H-indole-2-carboxylic acid amide hydrochloride 1024028-12-3 C21H24N4O*ClH
1-benzyl-4-(3-methylamino-pyrrolidin-1-yl)-1H-indole-2-carboxylic acid amide hydrochloride
—— 1-(1-ethyl-1H-pyrazol-4-ylmethyl)-4-[3-(4-fluoro-phenyl)-pyridin-2-yl]-piperazine hydrochloride 1082061-42-4 C21H24FN5*ClH
1-(1-ethyl-1H-pyrazol-4-ylmethyl)-4-[3-(4-fluoro-phenyl)-pyridin-2-yl]-piperazine hydrochloride
—— 2-[2-Oxo-6-[3-(trifluoromethyl)phenyl]-3,4-dihydroquinolin-1-yl]acetic acid 1224927-64-3 C18H14F3NO3
2-[2-Oxo-6-[3-(trifluoromethyl)phenyl]-3,4-dihydroquinolin-1-yl]acetic acid
—— 4-[4-(6-cyano-1-ethoxycarbonylmethyl-2-methylindolizin-3-ylsulfanyl)benzenesulfonyl]piperazine-1-carboxylic acid tert-butyl ester 1036714-00-7 C29H34N4O6S2
4-[4-(6-cyano-1-ethoxycarbonylmethyl-2-methylindolizin-3-ylsulfanyl)benzenesulfonyl]piperazine-1-carboxylic acid tert-butyl ester
—— 4-(1,3-dimethyl-1H-pyrazol-4-ylmethyl)-3'-(2-trifluoromethoxy-phenyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride 1082062-38-1 C21H23F3N6O*ClH
4-(1,3-dimethyl-1H-pyrazol-4-ylmethyl)-3'-(2-trifluoromethoxy-phenyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride
—— 2,4-Difluoro-6-methylbenzenesulfonyl chloride 1806332-55-7 C7H5ClF2O2S
2,4-Difluoro-6-methylbenzenesulfonyl chloride
—— 5-[N-(4-aminosulfonylphenyl)-N-methylaminocarbonyl]-3-(3-methylbenzyl)-6-hydroxy-1H-indazole 1001193-47-0 C23H22N4O4S
5-[N-(4-aminosulfonylphenyl)-N-methylaminocarbonyl]-3-(3-methylbenzyl)-6-hydroxy-1H-indazole
—— 1-Methyl-4-phenylpiperidine-2-carboxylic acid hydrochloride 18714-20-0 C13H18ClNO2
1-Methyl-4-phenylpiperidine-2-carboxylic acid hydrochloride
—— 1-(6-Fluoropyridin-3-yl)piperazine dihydrochloride 1909316-98-8 C9H14Cl2FN3
1-(6-Fluoropyridin-3-yl)piperazine dihydrochloride
—— 5-[N-(4-acetamidophenyl)-N-methylaminocarbonyl]-3-(3-methylbenzyl)-6-hydroxy-1H-indazole 1001193-43-6 C25H24N4O3
5-[N-(4-acetamidophenyl)-N-methylaminocarbonyl]-3-(3-methylbenzyl)-6-hydroxy-1H-indazole
—— 5-{N-[4-(4-methylpiperazin-1-yl)phenyl]-N-methylaminocarbonyl}-3-propyl-6-hydroxy-1H-indazole 1001195-31-8 C23H29N5O2
5-{N-[4-(4-methylpiperazin-1-yl)phenyl]-N-methylaminocarbonyl}-3-propyl-6-hydroxy-1H-indazole
—— Methyl2-amino-2-(3-bromo-5-chlorophenyl)acetatehydrochloride 1822450-73-6 C9H10BrCl2NO2
Methyl2-amino-2-(3-bromo-5-chlorophenyl)acetatehydrochloride
—— azetidin-3-yl-(3-pyridin-4-yl-[2,6]naphthyridin-1-yl)amine 1071016-76-6 C16H15N5
azetidin-3-yl-(3-pyridin-4-yl-[2,6]naphthyridin-1-yl)amine
—— N-(2-chloro-5-trifluoromethylphenyl)-2-[(4-methoxybenzyl)amino]-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]-pyrimidine-6(4H)-carboxamide 1016972-16-9 C29H25ClF3N5O3
N-(2-chloro-5-trifluoromethylphenyl)-2-[(4-methoxybenzyl)amino]-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]-pyrimidine-6(4H)-carboxamide
—— 1,3,4-triallylimidazolidin-2-one 1398414-44-2 C12H18N2O
1,3,4-triallylimidazolidin-2-one
—— tert-butyl 9-cyclohexyl-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate 1055880-68-6 C20H29NO3
tert-butyl 9-cyclohexyl-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate
—— 3-{[4-(3-trifluoromethylbenzyl)piperazin-1-yl]methylcarboxamido}methyl-5-isobutyl-1-phenyl-1H-pyrazole 1220347-32-9 C28H34F3N5O
3-{[4-(3-trifluoromethylbenzyl)piperazin-1-yl]methylcarboxamido}methyl-5-isobutyl-1-phenyl-1H-pyrazole
—— 4-[4-(7-chloro-6-cyano-1-ethoxycarbonylmethyl-2-methylindolizin-3-ylsulfanyl)benzenesulfonyl]piperazine-1-carboxylic acid tert-butyl ester 1036714-01-8 C29H33ClN4O6S2
4-[4-(7-chloro-6-cyano-1-ethoxycarbonylmethyl-2-methylindolizin-3-ylsulfanyl)benzenesulfonyl]piperazine-1-carboxylic acid tert-butyl ester
—— 1-{3-[7-(3-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl}-3-(2,2,2-trifluoro-ethyl)-urea hydrochloride 1036984-44-7 C22H16F4N4O*ClH
1-{3-[7-(3-fluoro-phenyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl}-3-(2,2,2-trifluoro-ethyl)-urea hydrochloride
—— N-(3,4-difluorophenyl)-3-(2-fluorophenyl)-2-[(4-methoxybenzyl)amino]-4-oxo-3,5,7,8-tetrahydropyrido[4,3-d]-pyrimidine-6(4H)-carboxamide 1016972-71-6 C28H24F3N5O3
N-(3,4-difluorophenyl)-3-(2-fluorophenyl)-2-[(4-methoxybenzyl)amino]-4-oxo-3,5,7,8-tetrahydropyrido[4,3-d]-pyrimidine-6(4H)-carboxamide
—— (4-cyclopropanecarbonyl-piperazin-1-yl)-[1-isopropyl-5-(1-isopropyl-piperidin-4-yloxy)-6-methyl-1H-indol-2-yl]-methanone 1044760-97-5 C29H42N4O3
(4-cyclopropanecarbonyl-piperazin-1-yl)-[1-isopropyl-5-(1-isopropyl-piperidin-4-yloxy)-6-methyl-1H-indol-2-yl]-methanone
—— (1E,6E)-1-(4-hydroxy-3-methoxyphenyl)-7-(1-methyl-1H-pyrazol-4-yl)hepta-1,6-diene-3,5-dione 1030859-98-3 C18H18N2O4
(1E,6E)-1-(4-hydroxy-3-methoxyphenyl)-7-(1-methyl-1H-pyrazol-4-yl)hepta-1,6-diene-3,5-dione
—— 9-[2-(trifluoromethoxy)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine hydrochloride 1055878-86-8 C16H14F3NO2*ClH
9-[2-(trifluoromethoxy)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine hydrochloride
—— 2-phenethyl-6-(1H-pyrazol-4-yl)benzo[d]thiazole 1213261-37-0 C18H15N3S
2-phenethyl-6-(1H-pyrazol-4-yl)benzo[d]thiazole
—— [1-Methyl-1-(1-methyl-6-oxo-1,6-dihydro-[4,4']bipyrimidinyl-2-yl)-ethyl]-carbamic acid benzyl ester 1083009-93-1 C20H21N5O3
[1-Methyl-1-(1-methyl-6-oxo-1,6-dihydro-[4,4']bipyrimidinyl-2-yl)-ethyl]-carbamic acid benzyl ester
—— 6-Fluoroisoquinoline-8-carboxylic acid 1909335-83-6 C10H6FNO2
6-Fluoroisoquinoline-8-carboxylic acid
—— 1-(2-chloro-5-fluorophenyl)-8-fluoro-6-methoxy-3-methylimidazo[5,1-c][1,2,4]benzotriazine 1226804-29-0 C17H11ClF2N4O
1-(2-chloro-5-fluorophenyl)-8-fluoro-6-methoxy-3-methylimidazo[5,1-c][1,2,4]benzotriazine
—— (2R)-1-[3-[4-[(5-chloro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenoxy]azetidin-1-yl]-2-hydroxy-propan-1-one 1224704-10-2 C24H23ClN6O4
(2R)-1-[3-[4-[(5-chloro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenoxy]azetidin-1-yl]-2-hydroxy-propan-1-one
—— 4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclopentylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073448-38-0 C35H46N6O9
4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclopentylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 5H,6H,7H-pyrrolo[1,2-c]imidazol-6-amine dihydrochloride 1864052-43-6 C6H11Cl2N3
5H,6H,7H-pyrrolo[1,2-c]imidazol-6-amine dihydrochloride
—— N-(4-(3-(pyrimidin-5-yl)pyridin-2-yloxy)phenyl)pyridin-2-amine 2,2,2-trifluoroacetate 1231922-43-2 C2HF3O2*C20H15N5O
N-(4-(3-(pyrimidin-5-yl)pyridin-2-yloxy)phenyl)pyridin-2-amine 2,2,2-trifluoroacetate
—— 4-[(S)-4-carboxy-2-({4-[2-oxo-2-((S)-2-phenyl-pyrrolidin-1-yl)-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073452-97-7 C34H39N5O8
4-[(S)-4-carboxy-2-({4-[2-oxo-2-((S)-2-phenyl-pyrrolidin-1-yl)-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— methyl 4-(benzyloxycarbonylamino)-1-(2-(7-(2-methoxyethoxy)imidazo[1,2-a]pyridin-3-yl)quinolin-8-yl)piperidine-4-carboxylate 1067914-76-4 C34H35N5O6
methyl 4-(benzyloxycarbonylamino)-1-(2-(7-(2-methoxyethoxy)imidazo[1,2-a]pyridin-3-yl)quinolin-8-yl)piperidine-4-carboxylate
—— 1-(1,3-dimethyl-1H-pyrazol-4-ylmethyl)-4-[3-(4-fluoro-phenyl)-pyridin-2-yl]-piperazine hydrochloride 1082061-44-6 C21H24FN5*ClH
1-(1,3-dimethyl-1H-pyrazol-4-ylmethyl)-4-[3-(4-fluoro-phenyl)-pyridin-2-yl]-piperazine hydrochloride
—— (R)-2-amino-5-[2-chloro-4-(3-ethylphenylthio)phenyl]-2-methylpentan-1-ol hydrochloride 1006727-15-6 C20H26ClNOS*ClH
(R)-2-amino-5-[2-chloro-4-(3-ethylphenylthio)phenyl]-2-methylpentan-1-ol hydrochloride
—— (4R)-2-(fluoromethyl)-2-methyl-7-(trifluoromethyl)chroman-4-amine 1221445-30-2 C12H13F4NO
(4R)-2-(fluoromethyl)-2-methyl-7-(trifluoromethyl)chroman-4-amine
—— 3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[(3-piperidin-1-ylbenzoyl)amino]propanoic acid 1323992-97-7 C34H36FN5O6
3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[(3-piperidin-1-ylbenzoyl)amino]propanoic acid
—— 3-bromo-4-chloro-N-(3-fluoro-2-methoxy-phenyl)-N-methyl-benzamide 1070892-11-3 C15H12BrClFNO2
3-bromo-4-chloro-N-(3-fluoro-2-methoxy-phenyl)-N-methyl-benzamide
—— 2-Amino-1-(1,2-oxazolidin-2-yl)ethan-1-one hydrochloride 1909336-42-0 C5H11ClN2O2
2-Amino-1-(1,2-oxazolidin-2-yl)ethan-1-one hydrochloride
—— (1-methyl-1H-pyrazol-4-yl)(1,2,4-oxadiazol-3-yl)methanamine dihydrochloride 1864015-38-2 C7H11Cl2N5O
(1-methyl-1H-pyrazol-4-yl)(1,2,4-oxadiazol-3-yl)methanamine dihydrochloride
—— 5-[N-(3-methoxyphenyl)-N-methylaminocarbonyl]-3-cyclopentylmethyl-6-hydroxy-1H-indazole 1001194-39-3 C22H25N3O3
5-[N-(3-methoxyphenyl)-N-methylaminocarbonyl]-3-cyclopentylmethyl-6-hydroxy-1H-indazole
—— 3'-(4-methoxymethyl-phenyl)-4-(1-phenyl-1H-pyrazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride 1082063-17-9 C26H28N6O*ClH
3'-(4-methoxymethyl-phenyl)-4-(1-phenyl-1H-pyrazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride
—— (2S)-2-[[5-(4-fluoro-3-methylphenyl)furan-2-carbonyl]amino]-3-[3-fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid 1323992-74-0 C34H30F2N4O7
(2S)-2-[[5-(4-fluoro-3-methylphenyl)furan-2-carbonyl]amino]-3-[3-fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid
—— 5-[N-(3,4-dimethoxyphenyl)-N-methylaminocarbonyl]-3-isobutyl-6-hydroxy-1H-indazole 1001193-80-1 C21H25N3O4
5-[N-(3,4-dimethoxyphenyl)-N-methylaminocarbonyl]-3-isobutyl-6-hydroxy-1H-indazole
—— 1-(1-(3,4-dichlorobenzyl)-5-(4-trifluoromethylphenyl)-1H-pyrazol-3-yl) methanol 1086835-85-9 C18H13Cl2F3N2O
1-(1-(3,4-dichlorobenzyl)-5-(4-trifluoromethylphenyl)-1H-pyrazol-3-yl) methanol
—— 1-(diphenylmethyl)-7-fluoro-3-hydroxy-3-(6-hydroxy-2,3-dihydro-1-benzofuran-5-yl)-1,3-dihydro-2H-indol-2-one 1222555-36-3 C29H22FNO4
1-(diphenylmethyl)-7-fluoro-3-hydroxy-3-(6-hydroxy-2,3-dihydro-1-benzofuran-5-yl)-1,3-dihydro-2H-indol-2-one
—— (R)-8-fluoro-2,2-dipropylchroman-4-amine 1221443-81-7 C15H22FNO
(R)-8-fluoro-2,2-dipropylchroman-4-amine
—— 2-(3-ethoxycarbonylpropyl)-1-phenoxycarbonyl-1,2,5,6-tetrahydropyridine 121507-73-1 C18H23NO4
2-(3-ethoxycarbonylpropyl)-1-phenoxycarbonyl-1,2,5,6-tetrahydropyridine
—— 2-[3-Benzyloxy-2-(4-methoxy-phenyl)-4-oxo-4H-chromen-6-yl]-propionic acid methyl ester 141070-57-7 C27H24O6
2-[3-Benzyloxy-2-(4-methoxy-phenyl)-4-oxo-4H-chromen-6-yl]-propionic acid methyl ester