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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3'-(4-fluorophenyl)-4-(1H-pyrazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride 1082061-81-1 C18H19FN6*ClH
3'-(4-fluorophenyl)-4-(1H-pyrazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride
—— 4-{(S)-4-ethoxycarbonyl-2-[(6-fluoro-7-methyl-4-{2-oxo-2-[(S)-2-(pyrrolidine-1-carbonyl)-pyrrolidin-1-yl]-ethoxy}-quinoline-2-carbonyl)-amino]-butyryl}-piperazine-1-carboxylic acid ethyl ester 1073449-75-8 C36H47FN6O9
4-{(S)-4-ethoxycarbonyl-2-[(6-fluoro-7-methyl-4-{2-oxo-2-[(S)-2-(pyrrolidine-1-carbonyl)-pyrrolidin-1-yl]-ethoxy}-quinoline-2-carbonyl)-amino]-butyryl}-piperazine-1-carboxylic acid ethyl ester
—— 4-[(S)-4-carboxy-2-({4-[2-((S)-2-ethylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methoxy-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073448-85-7 C32H42N6O10
4-[(S)-4-carboxy-2-({4-[2-((S)-2-ethylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methoxy-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 5-[N-(3-morpholin-4-ylphenyl)-N-methylaminocarbonyl]-3-butyl-6-hydroxy-1H-indazole 1001195-27-2 C23H28N4O3
5-[N-(3-morpholin-4-ylphenyl)-N-methylaminocarbonyl]-3-butyl-6-hydroxy-1H-indazole
—— 1-[4-(3-pyridin-4-yl-[2,6]naphthyridin-1-yl)piperazin-1-yl]ethanone 1071015-93-4 C19H19N5O
1-[4-(3-pyridin-4-yl-[2,6]naphthyridin-1-yl)piperazin-1-yl]ethanone
—— N-(3,4-difluorophenyl)-4-oxo-3-phenyl-2-phenylamino-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide 1016974-98-3 C26H21F2N5O2
N-(3,4-difluorophenyl)-4-oxo-3-phenyl-2-phenylamino-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide
—— Butyl 4-[(2S)-2-amino-3-cyclobutyl-1-oxopropyl]-1-piperazinecarboxylate 1073556-08-7 C16H29N3O3
Butyl 4-[(2S)-2-amino-3-cyclobutyl-1-oxopropyl]-1-piperazinecarboxylate
—— N-{(1S,2R)-1-benzyl-2-hydroxy-3-({(1R)-1-[3-(trifluoromethyl)phenyl]ethyl}amino)propyl}-1-ethyl-5-[(2-propylpiperidin-1-yl)carbonyl]-1H-pyrazole-3-carboxamide 1106668-84-1 C34H44F3N5O3
N-{(1S,2R)-1-benzyl-2-hydroxy-3-({(1R)-1-[3-(trifluoromethyl)phenyl]ethyl}amino)propyl}-1-ethyl-5-[(2-propylpiperidin-1-yl)carbonyl]-1H-pyrazole-3-carboxamide
—— (+/-)-8-benzyl-9,10-dimethoxy-5,8,13,13a-tetrahydro-6H-[1,3]dioxolo[4,5-g]isoquino[3,2-a]isoquinoline hydrochloride 1099738-77-8 C27H27NO4*ClH
(+/-)-8-benzyl-9,10-dimethoxy-5,8,13,13a-tetrahydro-6H-[1,3]dioxolo[4,5-g]isoquino[3,2-a]isoquinoline hydrochloride
—— 5-[3-(3-methoxy-phenyl)-prop-2-ynyl]-pyrazolo[1,5-a]pyrimidine 1228353-33-0 C16H13N3O
5-[3-(3-methoxy-phenyl)-prop-2-ynyl]-pyrazolo[1,5-a]pyrimidine
—— (2R,3R)-2-hydroxy-4-phenyl-3-({5-propyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-1H-[1,2,4]triazole-3-carbonyl}amino)butyric acid 1206696-62-9 C30H30N8O4
(2R,3R)-2-hydroxy-4-phenyl-3-({5-propyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmethyl]-1H-[1,2,4]triazole-3-carbonyl}amino)butyric acid
—— tert-butyl 9-(1-methylethyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate 1055880-92-6 C17H25NO3
tert-butyl 9-(1-methylethyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxylate
—— 3-(2-methoxy-naphthalen-6-yl)-1H-pyrrolo[2,3-b]pyridine 1027786-60-2 C18H14N2O
3-(2-methoxy-naphthalen-6-yl)-1H-pyrrolo[2,3-b]pyridine
—— 4-(1-Chloroethyl)-1,2,3-thiadiazole 1416331-47-9 C4H5ClN2S
4-(1-Chloroethyl)-1,2,3-thiadiazole
—— {1-[Amino(oxan-4-yl)methyl]cyclobutyl}methanol hydrochloride 1909306-02-0 C11H22ClNO2
{1-[Amino(oxan-4-yl)methyl]cyclobutyl}methanol hydrochloride
—— 2-[(3-Bromophenyl)methyl]pyrrolidine hydrochloride 1909309-28-9 C11H15BrClN
2-[(3-Bromophenyl)methyl]pyrrolidine hydrochloride
—— 6-amino-7-fluoro-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one 1909347-79-0 C7H6FN3O2
6-amino-7-fluoro-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
—— 6-(Aminomethyl)-1,2-benzoxazol-3-amine dihydrochloride 1860893-14-6 C8H11Cl2N3O
6-(Aminomethyl)-1,2-benzoxazol-3-amine dihydrochloride
—— tert-butyl 1-(piperidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxylate 1909305-30-1 C15H24N4O2
tert-butyl 1-(piperidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxylate
—— [3-(Difluoromethyl)-1,2,4-oxadiazol-5-yl]methanamine hydrochloride 1909325-73-0 C4H6ClF2N3O
[3-(Difluoromethyl)-1,2,4-oxadiazol-5-yl]methanamine hydrochloride
—— 5-methyl-5H,6H,7H,8H-imidazo[1,2-a]pyridine-2-sulfonyl chloride 1909318-73-5 C8H11ClN2O2S
5-methyl-5H,6H,7H,8H-imidazo[1,2-a]pyridine-2-sulfonyl chloride
—— 5-[N-(4-aminocarbonylphenyl)-N-methylaminocarbonyl]-3-(3-methylbenzyl)-6-hydroxy-1H-indazole 1001193-41-4 C24H22N4O3
5-[N-(4-aminocarbonylphenyl)-N-methylaminocarbonyl]-3-(3-methylbenzyl)-6-hydroxy-1H-indazole
—— 4-benzyl-9-bromo-6-fluoro-2,3,4,5-tetrahydrobenzo[f][1,4]oxazepine 1055881-11-2 C16H15BrFNO
4-benzyl-9-bromo-6-fluoro-2,3,4,5-tetrahydrobenzo[f][1,4]oxazepine
—— 9-(morpholin-4-ylcarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine hydrobromide 1055879-23-6 BrH*C14H18N2O3
9-(morpholin-4-ylcarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine hydrobromide
—— 4-[(S)-4-carboxy-2-({4-[2-(4-carboxy-piperidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073447-28-5 C30H37N5O10
4-[(S)-4-carboxy-2-({4-[2-(4-carboxy-piperidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 7-methoxymethyl-6-methyl-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine 1065066-32-1 C10H15NOS
7-methoxymethyl-6-methyl-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine
—— (5-methyl-furan-2-ylmethyl)-(6-phenylaminomethyl-quinolin-2-yl)-amine 1136479-69-0 C22H21N3O
(5-methyl-furan-2-ylmethyl)-(6-phenylaminomethyl-quinolin-2-yl)-amine
—— (3R)-1-[4-[(5-fluoro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenyl]pyrrolidin-3-ol 1224704-75-9 C22H21FN6O2
(3R)-1-[4-[(5-fluoro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenyl]pyrrolidin-3-ol
—— [7-cyano-1-(6-fluoroquinolin-2-ylmethyl)-2-methylindolizin-3-yl]acetic acid ethyl ester 1062559-21-0 C24H20FN3O2
[7-cyano-1-(6-fluoroquinolin-2-ylmethyl)-2-methylindolizin-3-yl]acetic acid ethyl ester
—— 4-[4-carboxy-(2S)-({4-[2-oxo-2-(2-pyrimidin-4-yl-pyrrolidin-1-yl)-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073453-19-6 C32H37N7O8
4-[4-carboxy-(2S)-({4-[2-oxo-2-(2-pyrimidin-4-yl-pyrrolidin-1-yl)-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 4-(1,5-dimethyl-1H-pyrazol-4-ylmethyl)-3'-phenyl-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl hydrochloride 1082061-84-4 C20H24N6*ClH
4-(1,5-dimethyl-1H-pyrazol-4-ylmethyl)-3'-phenyl-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl hydrochloride
—— N2-(2-methoxy-benzyl)-N6-(3-methyl-3H-imidazol-4-ylmethyl)-quinoline-2,6-diamine 1136479-23-6 C22H23N5O
N2-(2-methoxy-benzyl)-N6-(3-methyl-3H-imidazol-4-ylmethyl)-quinoline-2,6-diamine
—— 4-(5-methyl-1-phenyl-1H-pyrazol-4-ylmethyl)-3'-(4-fluorophenyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride 1082060-42-1 C25H25FN6*ClH
4-(5-methyl-1-phenyl-1H-pyrazol-4-ylmethyl)-3'-(4-fluorophenyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride
—— N-(3,4-difluorophenyl)-2-cyclohexylamino-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide 1016975-01-1 C26H27F2N5O2
N-(3,4-difluorophenyl)-2-cyclohexylamino-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide
—— 2-{4-[4-(2,6-difluoro-phenyl)-5-oxo-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H-[1,2,4]triazol-3-ylmethoxy]-2-methyl-phenoxy}-2-methyl-propionic acid 1050441-07-0 C27H22F5N3O5
2-{4-[4-(2,6-difluoro-phenyl)-5-oxo-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H-[1,2,4]triazol-3-ylmethoxy]-2-methyl-phenoxy}-2-methyl-propionic acid
—— 3-(trifluoromethyl)piperidine hydrochloride 1124199-60-5 C6H10F3N*ClH
3-(trifluoromethyl)piperidine hydrochloride
—— 2,2,2-trifluoroethyl 4-({6-[5-(isobutylsulfonyl)indolin-1-yl]pyrimidin-4-yl}oxy)piperidine-1-carboxylate 1145658-01-0 C24H29F3N4O5S
2,2,2-trifluoroethyl 4-({6-[5-(isobutylsulfonyl)indolin-1-yl]pyrimidin-4-yl}oxy)piperidine-1-carboxylate
—— 5-[5-(2-fluoromethyl-thiazol-4-ylethynyl)-thiophen-2-yl]-pyrazolo[1,5-a]pyrimidine 1228353-82-9 C16H9FN4S2
5-[5-(2-fluoromethyl-thiazol-4-ylethynyl)-thiophen-2-yl]-pyrazolo[1,5-a]pyrimidine
—— N-cyclopentyl-4-(4-methoxyphenyl)-N-methyl-1H-imidazole-1-carboxamide 1233855-09-8 C17H21N3O2
N-cyclopentyl-4-(4-methoxyphenyl)-N-methyl-1H-imidazole-1-carboxamide
—— N-(6-(4-fluorophenoxy)pyridin-3-yl)-6-(4-(4-(4-methylpiperazin-1-yl)benzoyl)piperidine-1-carbonyl)nicotinamide 1356627-48-9 C35H35FN6O4
N-(6-(4-fluorophenoxy)pyridin-3-yl)-6-(4-(4-(4-methylpiperazin-1-yl)benzoyl)piperidine-1-carbonyl)nicotinamide
—— 2-(2-(3,4-dichloro-N-methylphenylsulfonamido)cyclohexyloxy)-N-(2-(4-((dimethylamino)(thiophen-2-yl)methyl)cyclohexyl)ethyl)acetamide 1073597-44-0 C30H43Cl2N3O4S2
2-(2-(3,4-dichloro-N-methylphenylsulfonamido)cyclohexyloxy)-N-(2-(4-((dimethylamino)(thiophen-2-yl)methyl)cyclohexyl)ethyl)acetamide
—— N-(1-benzylpiperidin-4-yl)-N-methyl-4-(4-nitrophenyl)-1H-imidazole-1-carboxamide 1356960-41-2 C23H25N5O3
N-(1-benzylpiperidin-4-yl)-N-methyl-4-(4-nitrophenyl)-1H-imidazole-1-carboxamide
—— (6-bromo-4-chloroquinolin-3-yl)(cyclopropyl)methanone 1356953-24-6 C13H9BrClNO
(6-bromo-4-chloroquinolin-3-yl)(cyclopropyl)methanone
—— 3-azido-1-methyl-5-nitro-1H-[1,2,4]triazole 1021187-20-1 C3H3N7O2
3-azido-1-methyl-5-nitro-1H-[1,2,4]triazole
—— 2,3-dihydro-benzo[1,4]dioxine-5-carboxylic acid [3-(2-methyl-5-m-tolyl-thiazole-4-carbonyl)-oxazolidin-2-ylmethyl]-amide 1220347-01-2 C25H25N3O5S
2,3-dihydro-benzo[1,4]dioxine-5-carboxylic acid [3-(2-methyl-5-m-tolyl-thiazole-4-carbonyl)-oxazolidin-2-ylmethyl]-amide
—— (R)-2-amino-3-(4-octylphenylamino)propan-1-ol 1200143-97-0 C17H30N2O
(R)-2-amino-3-(4-octylphenylamino)propan-1-ol
—— (2S,3S)-N-(4-(5-(2-cyclohexylethyl)-1,2,4-oxadiazol-3-yl)benzyl)-3-hydroxypyrrolidine-2-carboxamide 1218816-65-9 C22H30N4O3
(2S,3S)-N-(4-(5-(2-cyclohexylethyl)-1,2,4-oxadiazol-3-yl)benzyl)-3-hydroxypyrrolidine-2-carboxamide
—— phenyl 2,3,4-tri-O-acetyl-α-L-rhamnopyranosyl-(1->2)-4,6-O-benzylidene-1-deoxy-1-thio-β-D-glucopyranoside 1394170-32-1 C31H36O12S
phenyl 2,3,4-tri-O-acetyl-α-L-rhamnopyranosyl-(1->2)-4,6-O-benzylidene-1-deoxy-1-thio-β-D-glucopyranoside
—— 1-((tert-butyldimethylsilyl)oxy)-2-(4-methoxyphenoxy)-N,N-dimethylethen-1-amine 1136235-87-4 C17H29NO3Si
1-((tert-butyldimethylsilyl)oxy)-2-(4-methoxyphenoxy)-N,N-dimethylethen-1-amine
—— 3,6,9,12,15,18-hexa-oxa-henicos-20-enyl 2,3,6-tri-O-acetyl-4-O-(2,3,4,6-tetra-O-acetyl-β-D-galactopyranosyl)-β-D-glucopyranoside 1065697-77-9 C41H64O24
3,6,9,12,15,18-hexa-oxa-henicos-20-enyl 2,3,6-tri-O-acetyl-4-O-(2,3,4,6-tetra-O-acetyl-β-D-galactopyranosyl)-β-D-glucopyranoside