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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[(S)-3-carboxy-2-({4-[2-((S)-2-cyclopentylcarbamoyl-azetidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-propionyl]-piperazine-1-carboxylic acid ethyl ester 1073448-77-7 C32H40N6O9
4-[(S)-3-carboxy-2-({4-[2-((S)-2-cyclopentylcarbamoyl-azetidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-propionyl]-piperazine-1-carboxylic acid ethyl ester
—— 3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[[6-(4-methylphenyl)pyridin-3-yl]carbamoylamino]propanoic acid 1323992-01-3 C35H33FN6O6
3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[[6-(4-methylphenyl)pyridin-3-yl]carbamoylamino]propanoic acid
—— 4,7-bis-(3-bromophenyl)-2,9-diphenyl-1,10-phenanthroline 1215007-71-8 C36H22Br2N2
4,7-bis-(3-bromophenyl)-2,9-diphenyl-1,10-phenanthroline
—— 4-Pyridin-4-ylmethyl-piperidine-4-carbonitrile 1229830-92-5 C12H15N3
4-Pyridin-4-ylmethyl-piperidine-4-carbonitrile
—— (Z)-3-{3-butoxy-4-[2-(3-fluoro-4-pentyloxy-phenyl)-ethoxy]-phenyl}-2-ethoxy-acrylic acid 1092167-05-9 C28H37FO6
(Z)-3-{3-butoxy-4-[2-(3-fluoro-4-pentyloxy-phenyl)-ethoxy]-phenyl}-2-ethoxy-acrylic acid
—— [4-(Methoxymethyl)oxan-4-yl]methanol 1564571-67-0 C8H16O3
[4-(Methoxymethyl)oxan-4-yl]methanol
—— 2-[[2-(4-fluoro-3-methylphenyl)-1H-imidazole-5-carbonyl]amino]-3-[3-fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid 1323991-53-2 C33H30F2N6O6
2-[[2-(4-fluoro-3-methylphenyl)-1H-imidazole-5-carbonyl]amino]-3-[3-fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid
—— (3R)-1-(4-phenylbutyl)-3-{[(2S)-2-phenyl-2-piperidin-1-ylpropanoyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide 1034916-61-4 Br*C31H43N2O2
(3R)-1-(4-phenylbutyl)-3-{[(2S)-2-phenyl-2-piperidin-1-ylpropanoyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
—— 4-[(S)-4-carboxy-2-({7-methyl-4-[2-oxo-2-(5-oxo-[1,4]diazepan-1-yl)-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073445-29-0 C30H38N6O9
4-[(S)-4-carboxy-2-({7-methyl-4-[2-oxo-2-(5-oxo-[1,4]diazepan-1-yl)-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 3-(2-{[4-chloro-3-(4-cyano-6-trifluoromethyl-pyridin-3-yl)-benzoyl]-methyl-amino}-phenoxy)-propionic acid 1-isopropoxycarbonyloxy-ethyl ester 1070891-24-5 C30H27ClF3N3O7
3-(2-{[4-chloro-3-(4-cyano-6-trifluoromethyl-pyridin-3-yl)-benzoyl]-methyl-amino}-phenoxy)-propionic acid 1-isopropoxycarbonyloxy-ethyl ester
—— 4-Isobutyl-piperidine-4-carboxylic acid ethyl ester hydrochloride 1227170-02-6 C12H23NO2*ClH
4-Isobutyl-piperidine-4-carboxylic acid ethyl ester hydrochloride
—— N-{(1S,2R)-1-benzyl-2-hydroxy-3-({(1S)-1-[3-methoxyphenyl]propyl}amino)propyl}-1-ethyl-5-[(2-propylpiperidin-1-yl)carbonyl]-1H-pyrazole-3-carboxamide 1106668-88-5 C35H49N5O4
N-{(1S,2R)-1-benzyl-2-hydroxy-3-({(1S)-1-[3-methoxyphenyl]propyl}amino)propyl}-1-ethyl-5-[(2-propylpiperidin-1-yl)carbonyl]-1H-pyrazole-3-carboxamide
—— 4-[(S)-4-carboxy-2-({4-[2-((R)-2-cyclopropylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073445-93-8 C33H42N6O9
4-[(S)-4-carboxy-2-({4-[2-((R)-2-cyclopropylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— (2R,3R)-2-(2,4-difluorophenyl)-3-(4-((thiophen-2-yl)methyl)piperazin-1-yl)-1-(1H-1,2,4-triazol-1-yl)butan-2-ol 1092849-20-1 C21H25F2N5OS
(2R,3R)-2-(2,4-difluorophenyl)-3-(4-((thiophen-2-yl)methyl)piperazin-1-yl)-1-(1H-1,2,4-triazol-1-yl)butan-2-ol
—— (2R)-2-({4-[([1,3]oxathiolo[5,4-c]pyridin-6-ylmethyl)amino]-1-piperidinyl}methyl)-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione hydrochloride 1075234-91-1 C22H24N6O3S*ClH
(2R)-2-({4-[([1,3]oxathiolo[5,4-c]pyridin-6-ylmethyl)amino]-1-piperidinyl}methyl)-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione hydrochloride
—— 5-[3-(2-fluoro-phenyl)-prop-2-ynyloxy]-pyrazolo[1,5-a]pyrimidine 1228354-54-8 C15H10FN3O
5-[3-(2-fluoro-phenyl)-prop-2-ynyloxy]-pyrazolo[1,5-a]pyrimidine
—— N-(3,4-difluorophenyl)-2-[(4-methoxybenzyl)amino]-3-(3-methoxyphenyl)-4-oxo-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide 1016972-65-8 C29H27F2N5O4
N-(3,4-difluorophenyl)-2-[(4-methoxybenzyl)amino]-3-(3-methoxyphenyl)-4-oxo-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide
—— 4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclobutylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-5-fluoro-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073449-88-3 C34H43FN6O9
4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclobutylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-5-fluoro-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— (4-{1-[2-(3,4-dimethoxy-phenyl)-acetyl]-4,5-dihydro-1H-pyrazol-3-yl}-phenyl)-carbamic acid 4-nitro-phenyl ester 1076690-78-2 C26H24N4O7
(4-{1-[2-(3,4-dimethoxy-phenyl)-acetyl]-4,5-dihydro-1H-pyrazol-3-yl}-phenyl)-carbamic acid 4-nitro-phenyl ester
—— 8-fluoro-6-methoxy-1-(5-methoxypyridin-3-yl)-3-methylimidazo[5,1-c][1,2,4]benzotriazine 1226804-38-1 C17H14FN5O2
8-fluoro-6-methoxy-1-(5-methoxypyridin-3-yl)-3-methylimidazo[5,1-c][1,2,4]benzotriazine
—— (2S)-1-[4-[4-[(5-chloro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenyl]-1-piperidyl]-2-methoxy-propan-1-one 1224704-13-5 C27H29ClN6O3
(2S)-1-[4-[4-[(5-chloro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenyl]-1-piperidyl]-2-methoxy-propan-1-one
—— N-(2,4-dichlorophenyl)-2-[(4-methoxybenzoyl)amino]-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]-pyrimidine-6(4H)-carboxamide 1016975-25-9 C28H23Cl2N5O4
N-(2,4-dichlorophenyl)-2-[(4-methoxybenzoyl)amino]-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]-pyrimidine-6(4H)-carboxamide
—— 1-{3-[7-(3,4-dimethoxy-phenyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl}-3-(2,2,2-trifluoro-ethyl)-urea formate 1036987-45-7 CH2O2*C24H21F3N4O3
1-{3-[7-(3,4-dimethoxy-phenyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl}-3-(2,2,2-trifluoro-ethyl)-urea formate
—— 3-hydroxy-3-(7-hydroxy-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-[(2R)-tetrahydrofuran-2-ylmethyl]-1,3-dihydro-2H-indol-2-one 1222555-57-8 C22H24N2O5
3-hydroxy-3-(7-hydroxy-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-[(2R)-tetrahydrofuran-2-ylmethyl]-1,3-dihydro-2H-indol-2-one
—— tert-butyl N-(1-phenyl-1H-imidazol-5-yl)carbamate 1864014-56-1 C14H17N3O2
tert-butyl N-(1-phenyl-1H-imidazol-5-yl)carbamate
—— 5-Bromo-3-hydroxy-8-methoxy-1,2-dihydroquinolin-2-one 1824277-24-8 C10H8BrNO3
5-Bromo-3-hydroxy-8-methoxy-1,2-dihydroquinolin-2-one
—— 5-[N-(2-methoxyethyl)-N-methylaminocarbonyl]-3-(2-methylbenzyl)-6-hydroxy-1H-indazole 1001191-89-4 C20H23N3O3
5-[N-(2-methoxyethyl)-N-methylaminocarbonyl]-3-(2-methylbenzyl)-6-hydroxy-1H-indazole
—— 5-{N-[4-(3-oxomorpholin-4-yl)phenyl]-N-methylaminocarbonyl}-3-(3-methylbutyl)-6-hydroxy-1H-indazole 1001195-56-7 C24H28N4O4
5-{N-[4-(3-oxomorpholin-4-yl)phenyl]-N-methylaminocarbonyl}-3-(3-methylbutyl)-6-hydroxy-1H-indazole
—— 5-(N-phenyl-N-methylaminocarbonyl)-3-butyl-6-hydroxy-1H-indazole 1001193-09-4 C19H21N3O2
5-(N-phenyl-N-methylaminocarbonyl)-3-butyl-6-hydroxy-1H-indazole
—— 5-{N-[4-(3-oxomorpholin-4-yl)phenyl]-N-methylaminocarbonyl}-3-butyl-6-hydroxy-1H-indazole 1001195-17-0 C23H26N4O4
5-{N-[4-(3-oxomorpholin-4-yl)phenyl]-N-methylaminocarbonyl}-3-butyl-6-hydroxy-1H-indazole
—— 1-(diphenylmethyl)-3-(8-hydroxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1,3-dihydro-2H-indol-2-one 1222555-19-2 C30H25NO4
1-(diphenylmethyl)-3-(8-hydroxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1,3-dihydro-2H-indol-2-one
—— (R)-N-(5-(3-(2,2-dimethyl-7-fluorochroman-4-yl)ureido)isoquinolin-3-yl)acetamide 1221444-66-1 C23H23FN4O3
(R)-N-(5-(3-(2,2-dimethyl-7-fluorochroman-4-yl)ureido)isoquinolin-3-yl)acetamide
—— 4-[(S)-4-carboxy-2-({4-[2-((2S,4R)-2-ethoxycarbonyl-4-hydroxy-pyrrolidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073446-16-8 C31H39N5O11
4-[(S)-4-carboxy-2-({4-[2-((2S,4R)-2-ethoxycarbonyl-4-hydroxy-pyrrolidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 5-[3-(1-methyl-1H-pyrazol-3-yl)-prop-2-ynyloxy]-pyrazolo[1,5-a]pyrimidine 1228354-41-3 C13H11N5O
5-[3-(1-methyl-1H-pyrazol-3-yl)-prop-2-ynyloxy]-pyrazolo[1,5-a]pyrimidine
—— {4-[4-(1-phenyl-1H-pyrazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl-3'-yl]-phenyl}-methanol hydrochloride 1082063-15-7 C25H26N6O*ClH
{4-[4-(1-phenyl-1H-pyrazol-4-ylmethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazinyl-3'-yl]-phenyl}-methanol hydrochloride
—— 4-[(S)-2-({4-[2-((S)-2-cyclopentylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-4-ethoxycarbonyl-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073449-92-9 C37H50N6O9
4-[(S)-2-({4-[2-((S)-2-cyclopentylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-7-methyl-quinoline-2-carbonyl}-amino)-4-ethoxycarbonyl-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 1-[9-(4-benzoyl-phenyl)-9H-carbazol-3-yl]-4-(benzothiazol-2-ylsulfanyl)-butan-1-one 1082065-54-0 C36H26N2O2S2
1-[9-(4-benzoyl-phenyl)-9H-carbazol-3-yl]-4-(benzothiazol-2-ylsulfanyl)-butan-1-one
—— (S)-ethyl 2-tert-butoxy-2-(5-cyclohexenyl-2-(hydroxymethyl)-7-methylquinolin-6-yl)acetate 1354188-94-5 C25H33NO4
(S)-ethyl 2-tert-butoxy-2-(5-cyclohexenyl-2-(hydroxymethyl)-7-methylquinolin-6-yl)acetate
—— (R)-2,2-diethyl-8-fluorochroman-4-amine 1144501-83-6 C13H18FNO
(R)-2,2-diethyl-8-fluorochroman-4-amine
—— 3-(2-ethyl-4-{5-[2-(ethyl-methyl-amino)-6-methyl-pyridin-4-yl]-[1,2,4]oxadiazol-3-yl}-6-methyl-phenyl)-propionic acid tert-butyl ester 1062669-81-1 C27H36N4O3
3-(2-ethyl-4-{5-[2-(ethyl-methyl-amino)-6-methyl-pyridin-4-yl]-[1,2,4]oxadiazol-3-yl}-6-methyl-phenyl)-propionic acid tert-butyl ester
—— 4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclopropylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-8-fluoro-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073448-10-8 C32H39FN6O9
4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclopropylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-8-fluoro-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 4-[1-(2-ethanesulfonyl-ethyl)-pyrazol-4-ylmethyl]-3'-(4-fluoro-phenyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride 1082062-88-1 C22H27FN6O2S*ClH
4-[1-(2-ethanesulfonyl-ethyl)-pyrazol-4-ylmethyl]-3'-(4-fluoro-phenyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyrazine hydrochloride
—— 4-[4-[(5-fluoro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenyl]-N,N-dimethyl-piperazine-1-sulfonamide 1224704-64-6 C24H27FN8O3S
4-[4-[(5-fluoro-4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-yl)amino]-3-methoxy-phenyl]-N,N-dimethyl-piperazine-1-sulfonamide
—— 1-(2-chloro-5-ethoxyphenyl)-8-fluoro-6-methoxy-3-methylimidazo[5,1-c][1,2,4]benzotriazine 1226804-13-2 C19H16ClFN4O2
1-(2-chloro-5-ethoxyphenyl)-8-fluoro-6-methoxy-3-methylimidazo[5,1-c][1,2,4]benzotriazine
—— 1-[4-[4-[[5-chloro-4-(7-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino]-3-methoxy-phenyl]piperazin-1-yl]-2-hydroxy-ethanone 1224706-58-4 C25H26ClN7O3
1-[4-[4-[[5-chloro-4-(7-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino]-3-methoxy-phenyl]piperazin-1-yl]-2-hydroxy-ethanone
—— 5-iodo-1-(4-oxazol-5-yl-benzenesulfonyl)-1H-indole 1063993-01-0 C17H11IN2O3S
5-iodo-1-(4-oxazol-5-yl-benzenesulfonyl)-1H-indole
—— N-(3,4-difluorophenyl)-2-[(3-fluorobenzyl)-amino]-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide 1016974-86-9 C27H22F3N5O2
N-(3,4-difluorophenyl)-2-[(3-fluorobenzyl)-amino]-4-oxo-3-phenyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidine-6(4H)-carboxamide
—— N-(8-bromo-[1,2,4]triazolo[1,5-a]pyridin-2-yl)-benzene-1,4-diamine 1206640-57-4 C12H10BrN5
N-(8-bromo-[1,2,4]triazolo[1,5-a]pyridin-2-yl)-benzene-1,4-diamine
—— 3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[[5-(2-fluorophenyl)pyridin-2-yl]carbamoylamino]propanoic acid 1323992-15-9 C34H30F2N6O6
3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[[5-(2-fluorophenyl)pyridin-2-yl]carbamoylamino]propanoic acid
—— (7-chloro-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-6-yl)methanol 1075238-30-0 C8H9ClN2O2
(7-chloro-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-6-yl)methanol