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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-{4,5-dichloro-2-[(2-thienylsulfonyl)amino]phenyl}-1-benzofuran-5-sulfonamide 1381970-43-9 C18H12Cl2N2O5S3
N-{4,5-dichloro-2-[(2-thienylsulfonyl)amino]phenyl}-1-benzofuran-5-sulfonamide
—— cyclo-(CPFVFLM)-SH 1366272-69-6 C42H59N7O7S2
cyclo-(CPFVFLM)-SH
—— 5-fluoro-2-(4-{[(3S)-3-(4-fluorophenyl)pyrrolidin-1-yl]carbonyl}-5-{1-[(4-methanesulfonylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-1-yl)pyrimidine 1381979-91-4 C31H32F2N6O3S
5-fluoro-2-(4-{[(3S)-3-(4-fluorophenyl)pyrrolidin-1-yl]carbonyl}-5-{1-[(4-methanesulfonylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-1-yl)pyrimidine
—— N-ethyl-4-fluoro-N-{2-[3-(5-fluoropyridin-2-yl)-1H-pyrazol-1-yl]ethyl}-2-(2H-1,2,3-triazol-2-yl)benzamide 1381971-49-8 C21H19F2N7O
N-ethyl-4-fluoro-N-{2-[3-(5-fluoropyridin-2-yl)-1H-pyrazol-1-yl]ethyl}-2-(2H-1,2,3-triazol-2-yl)benzamide
—— 2-(1-((5-chloro-3-fluoropyridin-2-yl)methyl)-2,5-dimethyl-1H-indol-3-yl)-N-(2-methoxypyridin-4-yl)-2-oxoacetamide 1383923-52-1 C24H20ClFN4O3
2-(1-((5-chloro-3-fluoropyridin-2-yl)methyl)-2,5-dimethyl-1H-indol-3-yl)-N-(2-methoxypyridin-4-yl)-2-oxoacetamide
—— N-[4-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-yl)butyl]-7-quinolinesulfonamide 1350978-09-4 C20H23N3O2S2
N-[4-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-yl)butyl]-7-quinolinesulfonamide
—— 3-[3-[[[[3-[(aminoiminomethyl)amino]phenyl]-carbonyl]amino]methyl]phenyl]-2-propenoic acid 198192-53-9 C18H18N4O3
3-[3-[[[[3-[(aminoiminomethyl)amino]phenyl]-carbonyl]amino]methyl]phenyl]-2-propenoic acid
—— 2-[4-[4-(Butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenyl]sulfanylphenyl]acetic acid 1357346-67-8 C25H24Cl2N2O5S2
2-[4-[4-(Butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenyl]sulfanylphenyl]acetic acid
—— (R)-N-{1-(phenethylamino)propan-2-yl}isoquinoline-6-sulfonamide 1383725-17-4 C20H23N3O2S
(R)-N-{1-(phenethylamino)propan-2-yl}isoquinoline-6-sulfonamide
—— N,N-dimethyl-2-(2-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)ethyl)-4-phenyl-1H-imidazole-1-sulfonamide 1351515-77-9 C21H20N4O4S
N,N-dimethyl-2-(2-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)ethyl)-4-phenyl-1H-imidazole-1-sulfonamide
—— 3-[4-[[[3-[(5,6-dihydro-4H-1,3-thiazin-2-yl)amino]phenyl]carbonyl]amino]3,5-dimethylphenyl]propenoic acid 198193-76-9 C22H23N3O3S
3-[4-[[[3-[(5,6-dihydro-4H-1,3-thiazin-2-yl)amino]phenyl]carbonyl]amino]3,5-dimethylphenyl]propenoic acid
—— N-[1-(3',5,5'-trichloro-2-methoxy-6-methylbiphenyl-3-yl)ethyl]-9H-purin-6-amine 1382993-29-4 C21H18Cl3N5O
N-[1-(3',5,5'-trichloro-2-methoxy-6-methylbiphenyl-3-yl)ethyl]-9H-purin-6-amine
—— 2-chloro-N-cyclopropyl-4-(6-[4-(dimethylamino)phenyl]-8-{[(1-methyl-1H-pyrazol-5-yl)methyl]amino}imidazo[1,2-a]pyrazin-3-yl)benzamide 1382478-77-4 C29H29ClN8O
2-chloro-N-cyclopropyl-4-(6-[4-(dimethylamino)phenyl]-8-{[(1-methyl-1H-pyrazol-5-yl)methyl]amino}imidazo[1,2-a]pyrazin-3-yl)benzamide
—— (13E,15E)-(3S,6S,9R,10R,11s,12S,21s)-3-(3-hydroxy-benzyl)-6-isopropyl-10,12-dimethoxy-9,11-dimethyl-1,4,7,19,25-pentaaza-bicyclo[19.3.1]pentacosa-13,15-diene-2,5,8,20-tetraone 1381808-35-0 C34H51N5O7
(13E,15E)-(3S,6S,9R,10R,11s,12S,21s)-3-(3-hydroxy-benzyl)-6-isopropyl-10,12-dimethoxy-9,11-dimethyl-1,4,7,19,25-pentaaza-bicyclo[19.3.1]pentacosa-13,15-diene-2,5,8,20-tetraone
—— 4-[3-ethoxy-4-oxo-2-[[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]amino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carbonyl]benzonitrile 1256548-76-1 C26H24F3N5O3
4-[3-ethoxy-4-oxo-2-[[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]amino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carbonyl]benzonitrile
—— Methyl 6-trifluoromethyl-2-(4,5,6-trimethoxy1H-indol-2-ylcarbonyl)-1,2,8,8a-tetrahydrocyclopropa[c]pyrrolo[3,2-e]indol-4 (5H)-one-7-carboxylate 157822-78-1 C26H22F3N3O7
Methyl 6-trifluoromethyl-2-(4,5,6-trimethoxy1H-indol-2-ylcarbonyl)-1,2,8,8a-tetrahydrocyclopropa[c]pyrrolo[3,2-e]indol-4 (5H)-one-7-carboxylate
—— [(2R,3R,4S,5S,6R)-4-(dimethylamino)-2-[[(4R,5S,6S,7R,9R,11E,13E,15R,16R)-16-ethyl-4-hydroxy-15-[[(2R,3R,4R,5R,6R)-5-hydroxy-3,4-dimethoxy-6-methyloxan-2-yl]oxymethyl]-5,9,13-trimethyl-2,10-dioxo-7-(2-oxoethyl)-1-oxacyclohexadeca-11,13-dien-6-yl]oxy]-6-methyl-5-(2-phenylethylcarbamoyloxy)oxan-3-yl] acetate 1054614-15-1 C50H76N2O16
[(2R,3R,4S,5S,6R)-4-(dimethylamino)-2-[[(4R,5S,6S,7R,9R,11E,13E,15R,16R)-16-ethyl-4-hydroxy-15-[[(2R,3R,4R,5R,6R)-5-hydroxy-3,4-dimethoxy-6-methyloxan-2-yl]oxymethyl]-5,9,13-trimethyl-2,10-dioxo-7-(2-oxoethyl)-1-oxacyclohexadeca-11,13-dien-6-yl]oxy]-6-methyl-5-(2-phenylethylcarbamoyloxy)oxan-3-yl] acetate
—— Benzyl 2-[[2-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylpropanoyl]amino]acetate 1382489-13-5 C19H19F3N2O5S
Benzyl 2-[[2-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylpropanoyl]amino]acetate
—— N-[N'-tert-butyl-N-[5-(3-chloro-5-fluorophenyl)-1H-pyrazol-3-yl]carbamimidoyl]-3,4-difluorobenzamide 1381825-71-3 C21H19ClF3N5O
N-[N'-tert-butyl-N-[5-(3-chloro-5-fluorophenyl)-1H-pyrazol-3-yl]carbamimidoyl]-3,4-difluorobenzamide
—— N-{2-[4-(4-fluorophenyl)-1H-pyrazol-1-yl]ethyl}-N,5-dimethyl-2-(2H-1,2,3-triazol-2-yl)benzamide 1381970-67-7 C22H21FN6O
N-{2-[4-(4-fluorophenyl)-1H-pyrazol-1-yl]ethyl}-N,5-dimethyl-2-(2H-1,2,3-triazol-2-yl)benzamide
—— Dimethyl 1'-benzyl-7,7-dimethyl-1-(4-methylphenyl)-2',5-dioxospiro[6,8-dihydroquinoline-2,3'-indole]-3,4-dicarboxylate 1374747-71-3 C36H34N2O6
Dimethyl 1'-benzyl-7,7-dimethyl-1-(4-methylphenyl)-2',5-dioxospiro[6,8-dihydroquinoline-2,3'-indole]-3,4-dicarboxylate
—— N-[2-(5-hydroxy-4-methylpent-3-en-1-yl)benzyl]-p-toluenesulfonamide 1403502-62-4 C20H25NO3S
N-[2-(5-hydroxy-4-methylpent-3-en-1-yl)benzyl]-p-toluenesulfonamide
—— 3-dimethylamino-N-[9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl]-butyramide 1208611-32-8 C27H32N2O8
3-dimethylamino-N-[9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl]-butyramide
—— (S)-N-((1R, 3S)-3-((2-(5-chloro-1H-pyrazolo[3,4-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl)amino)cyclohexyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide 1383446-99-8 C22H26ClFN8O2
(S)-N-((1R, 3S)-3-((2-(5-chloro-1H-pyrazolo[3,4-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl)amino)cyclohexyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
—— N-cyclopropyl-4-{6-[4-(2-methylpropoxy)phenyl]-8-[(2-methylpropyl)amino]imidazo[1,2a]pyrazin-3-yl}benzamide 1263421-84-6 C21H25N5O
N-cyclopropyl-4-{6-[4-(2-methylpropoxy)phenyl]-8-[(2-methylpropyl)amino]imidazo[1,2a]pyrazin-3-yl}benzamide
—— —— 1412895-22-7 C17H21BrO4
—— N-(benzyloxy)-N-(6-(3,4-dioxo-2-(pyridin-4-ylamino)cyclobut-1-enylamino)hexyl)methanesulfonamide 1258219-62-3 C23H28N4O5S
N-(benzyloxy)-N-(6-(3,4-dioxo-2-(pyridin-4-ylamino)cyclobut-1-enylamino)hexyl)methanesulfonamide
—— (1-{4'-[4-(1-hydroxy-4-phenylbutyl)thiophen-3-yl]biphenyl-4-yl}cyclopropyl)acetic acid 1380587-63-2 C31H30O3S
(1-{4'-[4-(1-hydroxy-4-phenylbutyl)thiophen-3-yl]biphenyl-4-yl}cyclopropyl)acetic acid
—— (S)-7-(2-(3,4-dimethylpiperazin-1-yl)ethoxy)-N-(1-((4,6-dimethylpyridin-2-yl)methyl)-3-methyl-1H-indazol-4-yl)imidazo[1,2-a]pyridine-3-carboxamide 1383471-72-4 C32H38N8O2
(S)-7-(2-(3,4-dimethylpiperazin-1-yl)ethoxy)-N-(1-((4,6-dimethylpyridin-2-yl)methyl)-3-methyl-1H-indazol-4-yl)imidazo[1,2-a]pyridine-3-carboxamide
—— N-(5-ethoxymethyl-pyrazin-2-yl)-3-(4-fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-propionamide 1380645-98-6 C23H24FN3O4S
N-(5-ethoxymethyl-pyrazin-2-yl)-3-(4-fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-propionamide
—— (1R,5R,6S)-[6-(2-(5-hydroxypyridin-3-yl)phenoxy)]-3-azabicyclo[3.2.1]octane hydrochloride 1244772-61-9 C18H20N2O2*ClH
(1R,5R,6S)-[6-(2-(5-hydroxypyridin-3-yl)phenoxy)]-3-azabicyclo[3.2.1]octane hydrochloride
—— (2-(4-(2-(5-amino-8-methylbenzo[f][1,7]naphthyridin-2-yl)ethyl)-3-methylphenoxy)ethyl)phosphonic acid 1258595-32-2 C24H26N3O4P
(2-(4-(2-(5-amino-8-methylbenzo[f][1,7]naphthyridin-2-yl)ethyl)-3-methylphenoxy)ethyl)phosphonic acid
—— (2S)-2-amino-3-cyclobutyl-1-[2-(4-fluorophenyl)-3-[(4-fluorophenyl)amino]-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl]propan-1-one 1261114-51-5 C25H27F2N5O
(2S)-2-amino-3-cyclobutyl-1-[2-(4-fluorophenyl)-3-[(4-fluorophenyl)amino]-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl]propan-1-one
—— pyrrolidin-1-yl(2-(m-tolylamino)-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl)methanone 1383776-56-4 C19H23N5O
pyrrolidin-1-yl(2-(m-tolylamino)-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl)methanone
—— 3-(2,2,2-trifluoro-acetylamino)-oxetane-3-carboxylic acid {(R)-1-[5'-chloro-3,3'-difluoro-2'-(2-methyl-2H-tetrazol-5-yl)-biphenyl-4-yl]-ethyl}-amide 1384171-14-5 C22H18ClF5N6O3
3-(2,2,2-trifluoro-acetylamino)-oxetane-3-carboxylic acid {(R)-1-[5'-chloro-3,3'-difluoro-2'-(2-methyl-2H-tetrazol-5-yl)-biphenyl-4-yl]-ethyl}-amide
—— 4-(5-(3,5-dichloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl)-N-(1,1‑oxythiophen-3-yl)-2-methylbenzamide 1424280-19-2 C21H16Cl2F4N2O4S
4-(5-(3,5-dichloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl)-N-(1,1‑oxythiophen-3-yl)-2-methylbenzamide
—— 1-{4'-[2-(1-hydroxy-4-phenylbutyl)thiophen-3-yl]biphenyl-4-yl}cyclopropanecarboxylic acid 1380587-42-7 C30H28O3S
1-{4'-[2-(1-hydroxy-4-phenylbutyl)thiophen-3-yl]biphenyl-4-yl}cyclopropanecarboxylic acid
—— 4-chloro-N-[N'-[[3-(trifluoromethyl)phenyl]methyl]-N-[5-(trifluoromethyl)-1H-pyrazol-3-yl]carbamimidoyl]benzamide 1381804-62-1 C20H14ClF6N5O
4-chloro-N-[N'-[[3-(trifluoromethyl)phenyl]methyl]-N-[5-(trifluoromethyl)-1H-pyrazol-3-yl]carbamimidoyl]benzamide
—— N-{1-[5-chloro-3-(6-fluoropyridin-3-yl)-2-methoxy-4-methylphenyl]ethyl}-9H-purin-6-amine 1382993-33-0 C20H18ClFN6O
N-{1-[5-chloro-3-(6-fluoropyridin-3-yl)-2-methoxy-4-methylphenyl]ethyl}-9H-purin-6-amine
—— N-(6-chloro-3-methylimidazo[1,2-a]pyridin-2-yl)-4-pyrazol-1-yl-N-[[4-(trifluoromethoxy)phenyl]methyl]benzenesulfonamide 1381785-15-4 C25H19ClF3N5O3S
N-(6-chloro-3-methylimidazo[1,2-a]pyridin-2-yl)-4-pyrazol-1-yl-N-[[4-(trifluoromethoxy)phenyl]methyl]benzenesulfonamide
—— 8-(4-methyl-piperazin-1-ylmethyl)-2,9-dihydro-1,2,7,9-tetraaza-phenalen-3-one 1140964-83-5 C15H18N6O
8-(4-methyl-piperazin-1-ylmethyl)-2,9-dihydro-1,2,7,9-tetraaza-phenalen-3-one
—— ((R)-2-benzylpiperazin-1-yl)(3-(2-chlorophenyl)-5-cyclopropylisoxazol-4-yl)methanone 1144508-38-2 C24H24ClN3O2
((R)-2-benzylpiperazin-1-yl)(3-(2-chlorophenyl)-5-cyclopropylisoxazol-4-yl)methanone
—— (4S,5R)-2-(6-tert-butyl-4-ethoxy-pyridin-3-yl)-4,5-bis-(4-chloro-phenyl)-4,5-dimethyl-4,5-dihydro-imidazole-1-carboxylic acid dimethylamide 1143520-34-6 C31H36Cl2N4O2
(4S,5R)-2-(6-tert-butyl-4-ethoxy-pyridin-3-yl)-4,5-bis-(4-chloro-phenyl)-4,5-dimethyl-4,5-dihydro-imidazole-1-carboxylic acid dimethylamide
—— (S)-N-[1-(3-methoxy-phenyl)-pyrrolidin-3-yl]-2,2-dimethyl-propionamide 1146970-77-5 C16H24N2O2
(S)-N-[1-(3-methoxy-phenyl)-pyrrolidin-3-yl]-2,2-dimethyl-propionamide
—— (1R,3aS,3bS,10aR,10bS,11S,12aS)-1-{[(cyanomethyl)thio]carbonyl}-7-(4-fluorophenyl)-11-hydroxy-10a,12a-dimethyl-1,2,3,3a,3b,4,5,7,10,10a,10b,11,12,12a-tetradecahydro-cyclopenta[5,6]naphtho[1,2-f]indazol-1-yl isoxazole-5-carboxylate 1138811-46-7 C33H33FN4O5S
(1R,3aS,3bS,10aR,10bS,11S,12aS)-1-{[(cyanomethyl)thio]carbonyl}-7-(4-fluorophenyl)-11-hydroxy-10a,12a-dimethyl-1,2,3,3a,3b,4,5,7,10,10a,10b,11,12,12a-tetradecahydro-cyclopenta[5,6]naphtho[1,2-f]indazol-1-yl isoxazole-5-carboxylate
—— N-(2-amino-2-oxoethyl)-4-(4-{[4-[5-fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)benzamide 1142952-32-6 C31H33F4N5O4
N-(2-amino-2-oxoethyl)-4-(4-{[4-[5-fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)benzamide
—— (1R)-1-(naphthyl)-N-{[1-(phenylsulfonyl)-1H-pyrrol-2-yl]methyl}ethanamine 1143520-14-2 C23H22N2O2S
(1R)-1-(naphthyl)-N-{[1-(phenylsulfonyl)-1H-pyrrol-2-yl]methyl}ethanamine
—— 8-Amino-7-fluoro-10-oxo-6-[2-(pyridine-2-carbonylamino)ethylamino]spiro[4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-2,1'-cyclopentane]-11-carboxylic acid 1132813-66-1 C24H24FN5O5
8-Amino-7-fluoro-10-oxo-6-[2-(pyridine-2-carbonylamino)ethylamino]spiro[4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-2,1'-cyclopentane]-11-carboxylic acid
—— 5-(3-chloro-4-fluorophenyl)-1-(1H-imidazol-4-yl)-3-methyl-3-(pyrimidin-5-ylmethyl)-1,3-dihydro-2H-indol-2-one 1141080-26-3 C23H17ClFN5O
5-(3-chloro-4-fluorophenyl)-1-(1H-imidazol-4-yl)-3-methyl-3-(pyrimidin-5-ylmethyl)-1,3-dihydro-2H-indol-2-one
—— (R) 2-[5-(3,5-bis-trifluoromethyl-benzylamino)-4'-trifluoromethyl-biphenyl-3-yl]-4-methyl-pentanoic acid 1145691-93-5 C28H24F9NO2
(R) 2-[5-(3,5-bis-trifluoromethyl-benzylamino)-4'-trifluoromethyl-biphenyl-3-yl]-4-methyl-pentanoic acid