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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(3-cyanophenyl)-6-[3-(hydroxymethyl)phenyl]imidazo[1,2-a]pyridine-2-carboxamide 1167055-16-4 C22H16N4O2
N-(3-cyanophenyl)-6-[3-(hydroxymethyl)phenyl]imidazo[1,2-a]pyridine-2-carboxamide
—— (S)-1-[2-(1,1-dioxo-tetrahydro-1λ6-thiophen-3-yl)-acetyl]-piperidine-2-carboxylic acid (5-tert-butyl-isoxazol-3-yl)-amide 1240058-63-2 C19H29N3O5S
(S)-1-[2-(1,1-dioxo-tetrahydro-1λ6-thiophen-3-yl)-acetyl]-piperidine-2-carboxylic acid (5-tert-butyl-isoxazol-3-yl)-amide
—— N-[(1R)-2-(1-azabicyclo[2.2.2]oct-3-ylamino)-2-oxo-1-{[(phenylmethyl)oxy]methyl}ethyl]-2-{[2-chloro-4-(trifluoromethyl)phenyl]oxy}-pyridine-3-carboxamide 1239355-27-1 C30H30ClF3N4O4
N-[(1R)-2-(1-azabicyclo[2.2.2]oct-3-ylamino)-2-oxo-1-{[(phenylmethyl)oxy]methyl}ethyl]-2-{[2-chloro-4-(trifluoromethyl)phenyl]oxy}-pyridine-3-carboxamide
—— N-[2-cyano-4-(2-{[6-(hydroxymethyl)pyridin-3-yl]amino}pyrimidin-4-yl)phenyl]cyclopropanecarboxamide 1403248-27-0 C21H18N6O2
N-[2-cyano-4-(2-{[6-(hydroxymethyl)pyridin-3-yl]amino}pyrimidin-4-yl)phenyl]cyclopropanecarboxamide
—— 2-Chloro-4-hex-5-enyl-1-propan-2-ylbenzimidazole 1365749-54-7 C16H21ClN2
2-Chloro-4-hex-5-enyl-1-propan-2-ylbenzimidazole
—— US8653087, III-297 1213245-84-1 C26H24F4N8O
US8653087, III-297
—— 8-cyclopentyl-N-[6-(3-methoxypyrrolidin-1-yl)pyridazin-3-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-amine 1169693-69-9 C23H26N8O
8-cyclopentyl-N-[6-(3-methoxypyrrolidin-1-yl)pyridazin-3-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-amine
—— 2-(9-phenanthrenyl)-1-iso-butylbenzimidazole 1192255-53-0 C25H22N2
2-(9-phenanthrenyl)-1-iso-butylbenzimidazole
—— 2-(xanthen-9-yliden-ethylidene)-indolin-3-one 114947-35-2 C23H15NO2
2-(xanthen-9-yliden-ethylidene)-indolin-3-one
—— tert-butyl N-[(2S)-1-(5-bromopyridin-3-yl)oxy-3-(3-fluorophenyl)propan-2-yl]carbamate 1026911-26-1 C19H22BrFN2O3
tert-butyl N-[(2S)-1-(5-bromopyridin-3-yl)oxy-3-(3-fluorophenyl)propan-2-yl]carbamate
—— —— 1450912-37-4 C49H60F6O8
—— 3-benzothiazol-2-yl-2,2,3,3-tetrafluoro-propionamide 15208-41-0 C10H6F4N2OS
3-benzothiazol-2-yl-2,2,3,3-tetrafluoro-propionamide
—— S<sup>6</sup>-(N-propyl-N-methoxycarbonyl)aminomethyl-6-mercaptopurine 126616-99-7 C11H15N5O2S
S<sup>6</sup>-(N-propyl-N-methoxycarbonyl)aminomethyl-6-mercaptopurine
—— (2S)-2-[[(3β,15α,16α,23R,24S)-16,23-epoxy-15-(triethylsilyl)oxy-24,25-dihydroxy-9,19-cyclolanostan-3-yl]-oxy]-4-[1-(tert-butoxycarbonyl)azetidin-3-yl]morpholine 1426230-19-4 C48H84N2O8Si
(2S)-2-[[(3β,15α,16α,23R,24S)-16,23-epoxy-15-(triethylsilyl)oxy-24,25-dihydroxy-9,19-cyclolanostan-3-yl]-oxy]-4-[1-(tert-butoxycarbonyl)azetidin-3-yl]morpholine
—— 2-{4-[7-amino-8-ethyl-5-oxo-6-(1-{[2-(trimethylsilyl)ethoxy]methyl}-1H-imidazol-2-yl)-5,8-dihydro-1,8-naphthyridin-2-yl]phenyl}-N-[(4-cyclopropylmorpholin-3-yl)methyl]acetamide 1308917-80-7 C35H47N7O4Si
2-{4-[7-amino-8-ethyl-5-oxo-6-(1-{[2-(trimethylsilyl)ethoxy]methyl}-1H-imidazol-2-yl)-5,8-dihydro-1,8-naphthyridin-2-yl]phenyl}-N-[(4-cyclopropylmorpholin-3-yl)methyl]acetamide
—— (S)-Phenyl-((1R,2S)-2-vinyl-cyclopentyl)-methanol 137502-40-0 C14H18O
(S)-Phenyl-((1R,2S)-2-vinyl-cyclopentyl)-methanol
—— 1-(2-deoxy-3-O-methanesulfonyl-5-O-triphenylmethyl-β-D-erythro-pentofuranosyl)-6-methyluracil 130745-15-2 C30H30N2O7S
1-(2-deoxy-3-O-methanesulfonyl-5-O-triphenylmethyl-β-D-erythro-pentofuranosyl)-6-methyluracil
—— 2-[2-(2-methoxyanilino)-6H-1,3,4-thiadiazin-5-yl]benzo[f]chromen-3-one 129574-00-1 C23H17N3O3S
2-[2-(2-methoxyanilino)-6H-1,3,4-thiadiazin-5-yl]benzo[f]chromen-3-one
—— ethyl 5-aminopent-2-enoate 1352280-55-7 C7H13NO2
ethyl 5-aminopent-2-enoate
—— methyl [(2S)-1-{(2S)-2-[5-(3-fluoro-7-{2-[(2S)-1-{(2S)-2-[(methoxycarbonyl)amino]-3-methylbutanoyl}pyrrolidin-2-yl]-1H-imidazol-5-yl}oxanthren-2-yl)-1H-imidazol-2-yl]pyrrolidin-1-yl}-3-methyl-1-oxobutan-2-yl]carbamate 1354655-63-2 C40H47FN8O8
methyl [(2S)-1-{(2S)-2-[5-(3-fluoro-7-{2-[(2S)-1-{(2S)-2-[(methoxycarbonyl)amino]-3-methylbutanoyl}pyrrolidin-2-yl]-1H-imidazol-5-yl}oxanthren-2-yl)-1H-imidazol-2-yl]pyrrolidin-1-yl}-3-methyl-1-oxobutan-2-yl]carbamate
—— 4-[8-[[3,5-Diethoxy-4-[4-(trifluoromethoxy)phenyl]phenyl]methyl]-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzoic acid 1254731-25-3 C33H35F3N2O6
4-[8-[[3,5-Diethoxy-4-[4-(trifluoromethoxy)phenyl]phenyl]methyl]-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzoic acid
—— 2-[[(2R)-1-[1-[(4-chloro-3-methylphenyl)methyl]piperidin-4-yl]-5-oxopyrrolidine-2-carbonyl]amino]-N,N-dimethyl-6-propan-2-ylpyridine-4-carboxamide 1251528-70-7 C29H38ClN5O3
2-[[(2R)-1-[1-[(4-chloro-3-methylphenyl)methyl]piperidin-4-yl]-5-oxopyrrolidine-2-carbonyl]amino]-N,N-dimethyl-6-propan-2-ylpyridine-4-carboxamide
—— (2S,3R)-2-[4-(3,3-difluorocyclobutyl)phenyl]-4,4,4-trifluoro-3-methylbutanoic acid 1297553-08-2 C15H15F5O2
(2S,3R)-2-[4-(3,3-difluorocyclobutyl)phenyl]-4,4,4-trifluoro-3-methylbutanoic acid
—— (4-methoxybenzyl)-[5-(3-trifluoromethoxyphenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]amine 1206203-16-8 C19H15F3N4O2S
(4-methoxybenzyl)-[5-(3-trifluoromethoxyphenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]amine
—— [(3S,4R)-4-(4-chloro-phenyl)-1-(3'-chloro-5'-trifluoromethyl-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-4-carbonyl)-pyrrolidin-3-yl]-methyl-carbamic acid 4-fluoro-phenyl ester 1310820-51-9 C30H28Cl2F4N4O3
[(3S,4R)-4-(4-chloro-phenyl)-1-(3'-chloro-5'-trifluoromethyl-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-4-carbonyl)-pyrrolidin-3-yl]-methyl-carbamic acid 4-fluoro-phenyl ester
—— (R)-phenyl-[2-[phenyl-[[2-(trifluoromethyl)phenyl]methyl]phosphanyl]ethyl]-[[2-(trifluoromethyl)phenyl]methyl]phosphane 1064689-13-9 C30H26F6P2
(R)-phenyl-[2-[phenyl-[[2-(trifluoromethyl)phenyl]methyl]phosphanyl]ethyl]-[[2-(trifluoromethyl)phenyl]methyl]phosphane
—— —— 134262-84-3 C23H44N2O9S
—— (E)-4-(5-cinnamamido-1,3,4-thiadiazol-2-yl)benzoic acid 1361230-12-7 C18H13N3O3S
(E)-4-(5-cinnamamido-1,3,4-thiadiazol-2-yl)benzoic acid
—— 5-azido-2,2-dimethoxypentane 157825-85-9 C7H15N3O2
5-azido-2,2-dimethoxypentane
—— 6,7-dichloro-3-(3,4,5-trimethoxybenzyl)quinoxalin-2(1H)-one 1327165-37-6 C18H16Cl2N2O4
6,7-dichloro-3-(3,4,5-trimethoxybenzyl)quinoxalin-2(1H)-one
—— 6-amino-3,7-dichloro-1,1-dioxo-1,2-dihydro-1λ<sup>6</sup>-naphtho[1,8-<i>cd</i>]isothiazole-5-sulfonic acid 14366-28-0 C10H6Cl2N2O5S2
6-amino-3,7-dichloro-1,1-dioxo-1,2-dihydro-1λ<sup>6</sup>-naphtho[1,8-<i>cd</i>]isothiazole-5-sulfonic acid
—— —— 1430835-63-4 C42H38N4O4
—— (S)-4,5-dihydro-3-<(2-methyl-1,3-dioxolan-2-yl)methyl>-5-isoxazolemethanol 128358-18-9 C9H15NO4
(S)-4,5-dihydro-3-<(2-methyl-1,3-dioxolan-2-yl)methyl>-5-isoxazolemethanol
—— 3-(4-bromophenyl)-2-cyano-3-(2-hydroxy-4,4-dimethyl-6-oxocyclohexen-1-yl)propanethioamide;morpholine 131270-69-4 C4H9NO*C18H19BrN2O2S
3-(4-bromophenyl)-2-cyano-3-(2-hydroxy-4,4-dimethyl-6-oxocyclohexen-1-yl)propanethioamide;morpholine
—— 1-(3-(1-hydroxy-2-(5H-imidazo[5,1-α]isoindol-5-yl)ethyl)azetidin-1-yl)-2-phenylethanone 1402837-56-2 C23H23N3O2
1-(3-(1-hydroxy-2-(5H-imidazo[5,1-α]isoindol-5-yl)ethyl)azetidin-1-yl)-2-phenylethanone
—— (S)-4-(2-(3-(isopropyl(methyl)amino)pyrrolidin-1-yl)benzo[d]thiazol-6-yl)benzonitrile 1161730-74-0 C22H24N4S
(S)-4-(2-(3-(isopropyl(methyl)amino)pyrrolidin-1-yl)benzo[d]thiazol-6-yl)benzonitrile
—— 3-(4-Methoxy-benzenesulfonylmethyl)-furan 129759-59-7 C12H12O4S
3-(4-Methoxy-benzenesulfonylmethyl)-furan
—— [(2R,3R,4R,5R)-3,4-diacetyloxy-5-[6-[14-[[9-[(2R,3R,4R,5R)-3,4-diacetyloxy-5-(acetyloxymethyl)oxolan-2-yl]purin-6-yl]amino]tetradecylamino]purin-9-yl]oxolan-2-yl]methyl acetate 129789-48-6 C46H64N10O14
[(2R,3R,4R,5R)-3,4-diacetyloxy-5-[6-[14-[[9-[(2R,3R,4R,5R)-3,4-diacetyloxy-5-(acetyloxymethyl)oxolan-2-yl]purin-6-yl]amino]tetradecylamino]purin-9-yl]oxolan-2-yl]methyl acetate
—— 2-(4,5-Difluoro-1H-indol-3-yl)acetic acid 126030-75-9 C10H7F2NO2
2-(4,5-Difluoro-1H-indol-3-yl)acetic acid
—— (1R,2R)-3,4-bis(hydroxymethyl)-2-[(E)-2-methoxyethenyl]cyclopent-3-en-1-ol 129715-16-8 C10H16O4
(1R,2R)-3,4-bis(hydroxymethyl)-2-[(E)-2-methoxyethenyl]cyclopent-3-en-1-ol
—— (Z)-(R)-Dec-2-en-4-ol 137764-94-4 C10H20O
(Z)-(R)-Dec-2-en-4-ol
—— 3-(2-chloro-3,6-difluorophenyl)-4-hydroxy-1-methaneyl-1,5-naphthyridine-2(1H)-one 1173014-82-8 C15H9ClF2N2O2
3-(2-chloro-3,6-difluorophenyl)-4-hydroxy-1-methaneyl-1,5-naphthyridine-2(1H)-one
—— N-(6-(3-tert-butyl-5-(2,4-di-tert-butoxypyrimidin-5-yl)-2-methoxyphenyl)naphthalen-2-yl)methanesulfonamide 1245899-22-2 C34H43N3O5S
N-(6-(3-tert-butyl-5-(2,4-di-tert-butoxypyrimidin-5-yl)-2-methoxyphenyl)naphthalen-2-yl)methanesulfonamide
—— N-((4-((dimethylamino)(3-fluorophenyl)methyl)cyclohexyl)methyl)-2-((1-(4-methoxyphenylsulfonyl)pyrrolidin-2-yl)methoxy)acetamide 1073598-40-9 C30H42FN3O5S
N-((4-((dimethylamino)(3-fluorophenyl)methyl)cyclohexyl)methyl)-2-((1-(4-methoxyphenylsulfonyl)pyrrolidin-2-yl)methoxy)acetamide
—— ethyl N-[3-(aminoiminomethyl)phenyl]-N-[4-(4-aminophenyl)butyl]glycine mono(trifluoroacetate) 195717-38-5 C2HF3O2*C21H28N4O2
ethyl N-[3-(aminoiminomethyl)phenyl]-N-[4-(4-aminophenyl)butyl]glycine mono(trifluoroacetate)
—— 1-[4-methyl-3-[3-[[1-methyl-1-[2-[2-(methylamino)ethoxy]phenyl]ethyl]amino]-2-oxo-1(2H)-pyrazinyl]benzoyl]-azetidine 1095004-38-8 C27H33N5O3
1-[4-methyl-3-[3-[[1-methyl-1-[2-[2-(methylamino)ethoxy]phenyl]ethyl]amino]-2-oxo-1(2H)-pyrazinyl]benzoyl]-azetidine
—— 5,6-dichloro-2-(5-methoxypyridin-3-yl)-1-methyl-1H-benzimidazole 1356481-19-0 C14H11Cl2N3O
5,6-dichloro-2-(5-methoxypyridin-3-yl)-1-methyl-1H-benzimidazole
—— (4-Propoxy-4,4-diphenylbutyl)-dimethylamin 16856-91-0 C21H29NO
(4-Propoxy-4,4-diphenylbutyl)-dimethylamin
—— 6-(3,4-Methylendioxy-trans-styryl)-3,5-dioxo-2,3,4,5-tetrahydro-1,2,4-triazin 16943-46-7 C12H9N3O4
6-(3,4-Methylendioxy-trans-styryl)-3,5-dioxo-2,3,4,5-tetrahydro-1,2,4-triazin
—— tert-butyl 1-(cyclobutylmethyl)-2-oxo-3-(pyridin-3-yl)-1,2,7,8-tetrahydro-1,6-naphthyridine-6(5H)-carboxylate 1036381-59-5 C23H29N3O3
tert-butyl 1-(cyclobutylmethyl)-2-oxo-3-(pyridin-3-yl)-1,2,7,8-tetrahydro-1,6-naphthyridine-6(5H)-carboxylate