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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-{[(ethylamino)carbonyl]amino}-N-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]nicotinamide 1032569-96-2 C27H34N8O5
6-{[(ethylamino)carbonyl]amino}-N-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]nicotinamide
—— 1-cyclopropyl-3-(2-trifluoromethyl-phenyl)-1,3-diaza-spiro[4.5]decan-2-one 1021391-22-9 C18H21F3N2O
1-cyclopropyl-3-(2-trifluoromethyl-phenyl)-1,3-diaza-spiro[4.5]decan-2-one
—— [3-(3-Fluorophenyl)-1H-pyrazol-4-YL]methanamine 1501527-36-1 C10H10FN3
[3-(3-Fluorophenyl)-1H-pyrazol-4-YL]methanamine
—— 4-[2-(2,3-difluoro-4-hydroxy-phenyl)-6-hydroxy-4-trifluoromethyl-3H-inden-1-yl]-thiophene-3-carbonitrile 1019984-72-5 C21H10F5NO2S
4-[2-(2,3-difluoro-4-hydroxy-phenyl)-6-hydroxy-4-trifluoromethyl-3H-inden-1-yl]-thiophene-3-carbonitrile
—— N-(2-hydroxyethyl)-2'-methylspiro[cyclopentane-1,9'-thioxanthene]-3'-sulfonamide 10',10'-dioxide 1027347-28-9 C20H23NO5S2
N-(2-hydroxyethyl)-2'-methylspiro[cyclopentane-1,9'-thioxanthene]-3'-sulfonamide 10',10'-dioxide
—— methyl (1R,9R,10R,12R,20R)-12-ethyl-10-hydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.7.1.01,9.02,7.016,20]icosa-2(7),3,5,13-tetraene-10-carboxylate 1417782-81-0 C24H32N2O4
methyl (1R,9R,10R,12R,20R)-12-ethyl-10-hydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.7.1.01,9.02,7.016,20]icosa-2(7),3,5,13-tetraene-10-carboxylate
—— 5-[6-(7-fluoro-1H-indol-2-yl)pyrazin-2-yl]-2-(4-fluorophenyl)-N-methyl-6-[methyl(methylsulfonyl)amino]-1-benzofuran-3-carboxamide 1426940-98-8 C30H23F2N5O4S
5-[6-(7-fluoro-1H-indol-2-yl)pyrazin-2-yl]-2-(4-fluorophenyl)-N-methyl-6-[methyl(methylsulfonyl)amino]-1-benzofuran-3-carboxamide
—— (1-((2-chloro-6,7-dihydrothieno[3,2-d]pyrimidin-4-yl)amino)cyclobutyl)methanol 1423719-34-9 C11H14ClN3OS
(1-((2-chloro-6,7-dihydrothieno[3,2-d]pyrimidin-4-yl)amino)cyclobutyl)methanol
—— 4-fluoro-4-(2-nitro-1-phenylethyl)-3-phenylisoxazol-5(4H)-one 1416132-94-9 C17H13FN2O4
4-fluoro-4-(2-nitro-1-phenylethyl)-3-phenylisoxazol-5(4H)-one
—— 3-{[(2S)-2-{[(4-bromophenyl)carbamoyl]amino}-3-phenylpropanoyl]amino}propanoic acid 1431754-11-8 C19H20BrN3O4
3-{[(2S)-2-{[(4-bromophenyl)carbamoyl]amino}-3-phenylpropanoyl]amino}propanoic acid
—— 2-(3-fluoro-4-(methylsulfonamidomethyl)phenyl)-N-((2-(2-methoxy-5-methylphenyl)-6-(trifluoromethyl)pyridin-3-yl)methyl)propanamide 1428764-60-6 C26H27F4N3O4S
2-(3-fluoro-4-(methylsulfonamidomethyl)phenyl)-N-((2-(2-methoxy-5-methylphenyl)-6-(trifluoromethyl)pyridin-3-yl)methyl)propanamide
—— 7-methyl-8-(2-(pyridin-2-yl)ethylamino)-10-((2S,3S,4R)-2,3,4,5-tetrahydroxypentyl)benzo[g]pteridine-2,4(3H,10H)-dione 1207985-55-4 C23H26N6O6
7-methyl-8-(2-(pyridin-2-yl)ethylamino)-10-((2S,3S,4R)-2,3,4,5-tetrahydroxypentyl)benzo[g]pteridine-2,4(3H,10H)-dione
—— 2-(3-fluoro-4-(methylsulfonamidomethyl)phenyl)-N-((2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)propanamide 1428789-58-5 C22H26F4N4O3S
2-(3-fluoro-4-(methylsulfonamidomethyl)phenyl)-N-((2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)propanamide
—— 1-(4-isopropylphenyl)-2-(3-methoxyphenyl)-1-quinuclidin-3-yl-ethanol 1428339-57-4 C25H33NO2
1-(4-isopropylphenyl)-2-(3-methoxyphenyl)-1-quinuclidin-3-yl-ethanol
—— (4-pyrrolidin-1-ylphenyl)-quinuclidin-3-yl-methanone 1428324-00-8 C18H24N2O
(4-pyrrolidin-1-ylphenyl)-quinuclidin-3-yl-methanone
—— N-((2-(3-ethoxyphenyl)-6-(trifluoromethyl)pyridin-3-yl)methyl)-2-(3-fluoro-4-(methylsulfonamidomethyl)phenyl)propanamide 1428764-79-7 C26H27F4N3O4S
N-((2-(3-ethoxyphenyl)-6-(trifluoromethyl)pyridin-3-yl)methyl)-2-(3-fluoro-4-(methylsulfonamidomethyl)phenyl)propanamide
—— —— 1034424-48-0 C22H23N3O3
—— —— 1071832-03-5 C25H26F2N2O
—— (10S,15S)-10-(4-bromophenyl)-13-ethyl-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione 1415726-19-0 C21H18BrN3O2
(10S,15S)-10-(4-bromophenyl)-13-ethyl-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
—— N-[6-[4-[(2-fluoro-5-methyl-phenyl)sulfonylamino]phenyl]-1H-pyrazolo[3,4-b]pyrazin-3-yl]thiophene-3-carboxamide 1426215-05-5 C23H17FN6O3S2
N-[6-[4-[(2-fluoro-5-methyl-phenyl)sulfonylamino]phenyl]-1H-pyrazolo[3,4-b]pyrazin-3-yl]thiophene-3-carboxamide
—— 5-(1-imidazol-1-ylpropyl)-2-(1-methyl-1H-pyrazol-4-yl)thiazole 1429097-54-0 C13H15N5S
5-(1-imidazol-1-ylpropyl)-2-(1-methyl-1H-pyrazol-4-yl)thiazole
—— methyl 2-[[(2S)-2-[(2-amino-4,5-dichlorobenzoyl)amino]-3-cyclohexylpropanoyl]amino]-1,3-thiazole-5-carboxylate 1416811-33-0 C21H24Cl2N4O4S
methyl 2-[[(2S)-2-[(2-amino-4,5-dichlorobenzoyl)amino]-3-cyclohexylpropanoyl]amino]-1,3-thiazole-5-carboxylate
—— 7-{(3S,4S)-3-amino-4-methylpyrrolidin-1-yl}-6-fluoro-1-(isoxazol-3-yl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid, acetic acid salt 167073-46-3 C2H4O2*C18H17FN4O4
7-{(3S,4S)-3-amino-4-methylpyrrolidin-1-yl}-6-fluoro-1-(isoxazol-3-yl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid, acetic acid salt
—— —— 1217241-21-8 C28H23BrN4O2
—— —— 1254587-09-1 C31H28N4O5S
—— —— 1254586-92-9 C32H32N4O3S
—— 3,5-diamino-6-[2-(1,4-dimethoxynaphthyl)]-1,2,4-triazine 1174185-24-0 C15H15N5O2
3,5-diamino-6-[2-(1,4-dimethoxynaphthyl)]-1,2,4-triazine
—— cis-6-({4-[(1RS)-1-amino-2-(3-fluoro-6-methoxy-[1,5]naphthyridin-4-yl)-ethyl]-cyclohexylamino}-methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one 1037123-67-3 C25H29FN6O2S
cis-6-({4-[(1RS)-1-amino-2-(3-fluoro-6-methoxy-[1,5]naphthyridin-4-yl)-ethyl]-cyclohexylamino}-methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one
—— 2-[((2S)-1-{[5-(4-fluorophenyl)-2-methyl-1,3-thiazol-4-yl]carbonyl}-2-piperidinyl)methyl]-8-(trifluoromethyl)imidazo[1,2-a]pyridine hydrochloride 1097265-23-0 C25H22F4N4OS*ClH
2-[((2S)-1-{[5-(4-fluorophenyl)-2-methyl-1,3-thiazol-4-yl]carbonyl}-2-piperidinyl)methyl]-8-(trifluoromethyl)imidazo[1,2-a]pyridine hydrochloride
—— —— 1118628-28-6 C26H20Cl2F3N3O2
—— N-(4-((S)-1-(4-((S)-4-isopropyl-2-oxooxazolidin-3-yl)pyrimidin-2-ylamino)ethyl)phenyl)cyclohexanecarboxamide 1429176-54-4 C25H33N5O3
N-(4-((S)-1-(4-((S)-4-isopropyl-2-oxooxazolidin-3-yl)pyrimidin-2-ylamino)ethyl)phenyl)cyclohexanecarboxamide
—— N-((5S)-2'-amino-1-fluoro-3-(5-fluoro-3-pyridinyl)-5',6'-dihydrospiro[chromeno[2,3-c]pyridine-5,4'-[1,3]thiazin]-7-yl)-5-methoxy-2-pyridinecarboxamide 1428633-39-9 C27H20F2N6O3S
N-((5S)-2'-amino-1-fluoro-3-(5-fluoro-3-pyridinyl)-5',6'-dihydrospiro[chromeno[2,3-c]pyridine-5,4'-[1,3]thiazin]-7-yl)-5-methoxy-2-pyridinecarboxamide
—— 1-[2-(4-Methylphenoxy)ethyl]-3-(m-tolylmethyl)pyrimidine-2,4-dione 1424798-80-0 C21H22N2O3
1-[2-(4-Methylphenoxy)ethyl]-3-(m-tolylmethyl)pyrimidine-2,4-dione
—— (3-chloro-4-fluorophenyl)[(7S,8aS)-7-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl]methanone 1429294-98-3 C19H18ClF4N5O
(3-chloro-4-fluorophenyl)[(7S,8aS)-7-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl]methanone
—— 5-(7-fluoro-7,8-dihydro-6H-benzo[2,3][1,5]oxazocino[5,4-a]indol-2-yl)-2-(4 luorophenyl)-N-methyl-6-(N-methylmethylsulfonamido)benzofuran-3-carboxamide 1427033-08-6 C35H29F2N3O5S
5-(7-fluoro-7,8-dihydro-6H-benzo[2,3][1,5]oxazocino[5,4-a]indol-2-yl)-2-(4 luorophenyl)-N-methyl-6-(N-methylmethylsulfonamido)benzofuran-3-carboxamide
—— pyrazine-2-carboxylic acid [5-(3-fluorophenylethynyl)bicyclo[3.2.1]oct-1-yl]amide 1427704-03-7 C21H20FN3O
pyrazine-2-carboxylic acid [5-(3-fluorophenylethynyl)bicyclo[3.2.1]oct-1-yl]amide
—— 3,4,5-trimethoxyphenyl 4-(2-oxo-3-pentylimidazolidin-1-yl)benzenesulfonate 1422527-87-4 C23H30N2O7S
3,4,5-trimethoxyphenyl 4-(2-oxo-3-pentylimidazolidin-1-yl)benzenesulfonate
—— 4-{3-[2-(2-fluoro-4-cyanophenylamino)benzyl]-4,4-dimethyl-2,5-dioxoimidazolidin-1-yl}-2-trifluoromethylbenzonitrile 1006896-24-7 C27H19F4N5O2
4-{3-[2-(2-fluoro-4-cyanophenylamino)benzyl]-4,4-dimethyl-2,5-dioxoimidazolidin-1-yl}-2-trifluoromethylbenzonitrile
—— N-(3-(4-(3,4-dimethoxybenzyl)-6-methoxy-3,5-dioxo-4,5-dihydro-1,2,4-triazin-2(3H)-yl)phenyl)acetamide 1207438-72-9 C21H22N4O6
N-(3-(4-(3,4-dimethoxybenzyl)-6-methoxy-3,5-dioxo-4,5-dihydro-1,2,4-triazin-2(3H)-yl)phenyl)acetamide
—— —— 1187519-21-6 C20H15Cl3F3N3O2
—— 6-((trans-4-aminocyclohexyl)amino)-N-(3-fluoro-4-pyridinyl)-8-((4-(2-hydroxyethoxy)phenyl)amino)imidazo[1,2-b]pyridazine-3-carboxamide 1177415-05-2 C26H29FN8O3
6-((trans-4-aminocyclohexyl)amino)-N-(3-fluoro-4-pyridinyl)-8-((4-(2-hydroxyethoxy)phenyl)amino)imidazo[1,2-b]pyridazine-3-carboxamide
—— 2,5-dimethyl-oxazole-5-carboxylic acid [3-((S)-2-amino-1,4-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyrimidin-4-yl)phenyl]amide hydrochloride 1254196-74-1 C18H21N5O3*ClH
2,5-dimethyl-oxazole-5-carboxylic acid [3-((S)-2-amino-1,4-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyrimidin-4-yl)phenyl]amide hydrochloride
—— —— 1326224-59-2 C30H32FN3O7
—— 2-[3-({6-[2-(2-benzylpiperidin-1-yl)-2-oxoethyl]-5-oxo-1-phenyl-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-4-yl}methyl)-1H-indazol-1-yl]-Nmethyl-N-propylacetamide 1228934-71-1 C44H46N8O3
2-[3-({6-[2-(2-benzylpiperidin-1-yl)-2-oxoethyl]-5-oxo-1-phenyl-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-4-yl}methyl)-1H-indazol-1-yl]-Nmethyl-N-propylacetamide
—— —— 1254313-20-6 C25H14BrCl2F9N2O3
—— 6-(3-fluoro-5-(trifluoromethyl)phenyl)-3-hydroxy1-methyl-2-oxo-N-(3-(2-oxopyrrolidin-1-yl)propyl)-1,2-dihydropyridine-4-carboxamide 1429202-37-8 C21H21F4N3O4
6-(3-fluoro-5-(trifluoromethyl)phenyl)-3-hydroxy1-methyl-2-oxo-N-(3-(2-oxopyrrolidin-1-yl)propyl)-1,2-dihydropyridine-4-carboxamide
—— 1-(deca-5,6-dien-5-yl)-2,3,4,5,6-pentafluorobenzene 1374748-33-0 C16H17F5
1-(deca-5,6-dien-5-yl)-2,3,4,5,6-pentafluorobenzene
—— 8-amino-9-fluoro-10-(3-(furan-2-carboxamido)propylamino)-7-oxo-2,7-dihydrospiro[[1,4]oxazino[2,3,4-ij]quinoline-3,1'-cyclopentane]-6-carboxylic acid 1132813-04-7 C24H25FN4O6
8-amino-9-fluoro-10-(3-(furan-2-carboxamido)propylamino)-7-oxo-2,7-dihydrospiro[[1,4]oxazino[2,3,4-ij]quinoline-3,1'-cyclopentane]-6-carboxylic acid
—— 5-methyl-(3a<i>r</i>,6a<i>c</i>)-hexahydro-thieno[3,4-<i>c</i>]pyrrole 112950-86-4 C7H13NS
5-methyl-(3a<i>r</i>,6a<i>c</i>)-hexahydro-thieno[3,4-<i>c</i>]pyrrole
—— (Pt(4,4'-(CONEt2)2-2,2'-bipyridine))2(3,3',4,4'-tetrahydroxybiphenyl(-4H)) 1253693-99-0 C52H58N8O8Pt2
(Pt(4,4'-(CONEt2)2-2,2'-bipyridine))2(3,3',4,4'-tetrahydroxybiphenyl(-4H))