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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C46H59N3O14
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[2-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C41H55N3O12
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[2-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate —— C50H63N3O11
tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C48H59N3O11
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C46H52N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C45H56N4O11
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C47H50N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C49H57N3O11
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[4-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C49H63N3O16
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[4-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C45H59N3O11
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C44H55N3O12
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate —— C47H60N4O11
tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C42H52F3N3O12
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]pentanoate —— C55H57N3O11
tert-butyl (4S)-5-hydroxy-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate —— C47H52N2O13
tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate —— C53H60N4O11
tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C52H59N3O14
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C46H63N3O16
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C46H52N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C55H71N3O11
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[2-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C45H56N4O11
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[2-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate —— C47H56F3N3O12
tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[2-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C52H71N3O11
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[2-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate —— C53H56F3N3O12
tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate —— C43H49N3O10
tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[3-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C53H64N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[3-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]pentanoate —— C48H52F3N3O12
tert-butyl (4S)-5-hydroxy-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate —— C57H63N3O14
tert-butyl (4S)-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]pentanoate —— C48H52F3N3O12
tert-butyl (4S)-5-hydroxy-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate —— C47H52N2O13
tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C47H50N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate —— C43H49N3O10
tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]pentanoate —— C55H57N3O11
tert-butyl (4S)-5-hydroxy-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-11-[[3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate —— C56H63N3O11
tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-11-[[3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C43H45F3N2O11
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]pentanoate —— C52H57N3O11
tert-butyl (4S)-5-hydroxy-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[2-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C55H71N3O11
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[2-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[4-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C53H64N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[4-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]pentanoate —— C57H61N3O11
tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]-methylamino]-3-phenylpropanoyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C34H44N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C42H48N2O11
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate —— C53H56F3N3O12
tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C52H59N3O14
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[4-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]pentanoate —— C61H71N3O11
tert-butyl (4S)-5-hydroxy-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[4-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C42H48N2O11
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[2-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[2-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C47H56N2O15
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[2-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[2-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C41H56N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[2-[[(1R,4R,10S)-4,12,12-trimethyl-5-oxatricyclo[8.2.0.04,6]dodecan-9-ylidene]methyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C46H52N2O10
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-11-[[3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate —— C47H52N2O13
tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-11-[[4-[3-[(3R)-4,4-dimethyl-2-oxooxolan-3-yl]oxy-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate —— C43H45F3N2O11
tert-butyl (4S)-5-hydroxy-4-[[(1S,2S,6S,7R,10R,13S)-9-oxo-11-[[4-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]phenyl]methyl]-4,4-diphenyl-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]pentanoate