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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl (1S,6R)-3-(pyridin-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C18H27N3O2
tert-butyl (1S,6R)-3-(pyridin-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl N-methyl-N-[2-[(2R)-2-(methylcarbamoyl)piperidin-1-yl]-2-oxoethyl]carbamate —— C15H27N3O4
tert-butyl N-methyl-N-[2-[(2R)-2-(methylcarbamoyl)piperidin-1-yl]-2-oxoethyl]carbamate
—— tert-butyl (1R,6S)-3-(2-pyrazol-1-ylethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C17H28N4O2
tert-butyl (1R,6S)-3-(2-pyrazol-1-ylethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (3S)-3-[3-[3-(cyclopropylmethoxymethyl)anilino]-3-oxopropyl]pyrrolidine-1-carboxylate —— C23H34N2O4
tert-butyl (3S)-3-[3-[3-(cyclopropylmethoxymethyl)anilino]-3-oxopropyl]pyrrolidine-1-carboxylate
—— tert-butyl (2R)-2-[(2R)-1-[[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate —— C22H36N4O4
tert-butyl (2R)-2-[(2R)-1-[[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl (3R)-3-[(1-methylimidazole-2-carbonyl)amino]azepane-1-carboxylate —— C16H26N4O3
tert-butyl (3R)-3-[(1-methylimidazole-2-carbonyl)amino]azepane-1-carboxylate
—— tert-butyl (2R)-2-[(2S)-1-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate —— C23H31ClN4O3
tert-butyl (2R)-2-[(2S)-1-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl (3R)-3-[(2-fluorophenyl)carbamoylamino]azepane-1-carboxylate —— C18H26FN3O3
tert-butyl (3R)-3-[(2-fluorophenyl)carbamoylamino]azepane-1-carboxylate
—— tert-butyl (2R)-2-[(2S)-1-[[5-(trifluoromethyl)-1,3-benzoxazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate —— C23H30F3N3O3
tert-butyl (2R)-2-[(2S)-1-[[5-(trifluoromethyl)-1,3-benzoxazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl (2S)-2-[(2R)-1-[[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate —— C22H36N4O4
tert-butyl (2S)-2-[(2R)-1-[[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl (3R)-3-[[(1R,2S)-2-(4-chlorophenyl)cyclopropanecarbonyl]sulfamoyl]pyrrolidine-1-carboxylate —— C19H25ClN2O5S
tert-butyl (3R)-3-[[(1R,2S)-2-(4-chlorophenyl)cyclopropanecarbonyl]sulfamoyl]pyrrolidine-1-carboxylate
—— tert-butyl (3S)-3-[(2-methyl-1,2,4-triazol-3-yl)methylamino]pyrrolidine-1-carboxylate —— C13H23N5O2
tert-butyl (3S)-3-[(2-methyl-1,2,4-triazol-3-yl)methylamino]pyrrolidine-1-carboxylate
—— tert-butyl (1S,6R)-3-[2-(1,2,4-triazol-1-yl)ethyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C16H27N5O2
tert-butyl (1S,6R)-3-[2-(1,2,4-triazol-1-yl)ethyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (1R,5S)-3-(cyclopropanecarbonylamino)-8-azabicyclo[3.2.1]octane-8-carboxylate —— C16H26N2O3
tert-butyl (1R,5S)-3-(cyclopropanecarbonylamino)-8-azabicyclo[3.2.1]octane-8-carboxylate
—— tert-butyl (1S,6R)-3-[3-(1-methylpyrazol-4-yl)propyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C19H32N4O2
tert-butyl (1S,6R)-3-[3-(1-methylpyrazol-4-yl)propyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl 4-[2-[[(2S)-4-hydroxy-3,3-dimethyl-2-phenylbutyl]amino]-2-oxoethyl]piperidine-1-carboxylate —— C24H38N2O4
tert-butyl 4-[2-[[(2S)-4-hydroxy-3,3-dimethyl-2-phenylbutyl]amino]-2-oxoethyl]piperidine-1-carboxylate
—— tert-butyl (1S,5R)-3-(3-methylsulfonylpropylamino)-8-azabicyclo[3.2.1]octane-8-carboxylate —— C16H30N2O4S
tert-butyl (1S,5R)-3-(3-methylsulfonylpropylamino)-8-azabicyclo[3.2.1]octane-8-carboxylate
—— tert-butyl (2S)-2-[(2R)-1-[[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate —— C24H31N5O3
tert-butyl (2S)-2-[(2R)-1-[[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl (1R,6S)-3-[(1-methylimidazol-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C17H28N4O2
tert-butyl (1R,6S)-3-[(1-methylimidazol-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (1R,6S)-3-(7-methyl-4-oxo-1H-1,8-naphthyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C22H28N4O4
tert-butyl (1R,6S)-3-(7-methyl-4-oxo-1H-1,8-naphthyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (3S,4S)-3-[(2-chloro-4-fluorobenzoyl)amino]-4-methoxypyrrolidine-1-carboxylate —— C17H22ClFN2O4
tert-butyl (3S,4S)-3-[(2-chloro-4-fluorobenzoyl)amino]-4-methoxypyrrolidine-1-carboxylate
—— tert-butyl (3S)-3-[[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]amino]pyrrolidine-1-carboxylate —— C16H26N2O3S
tert-butyl (3S)-3-[[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]amino]pyrrolidine-1-carboxylate
—— tert-butyl (2R)-2-[(2S)-1-[[5-(3-chlorophenyl)-1,3-oxazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate —— C24H32ClN3O3
tert-butyl (2R)-2-[(2S)-1-[[5-(3-chlorophenyl)-1,3-oxazol-2-yl]methyl]piperidin-2-yl]pyrrolidine-1-carboxylate
—— tert-butyl (1R,5S)-3-[methyl-[2-[2-oxo-3-(trifluoromethyl)pyridin-1-yl]acetyl]amino]-8-azabicyclo[3.2.1]octane-8-carboxylate —— C21H28F3N3O4
tert-butyl (1R,5S)-3-[methyl-[2-[2-oxo-3-(trifluoromethyl)pyridin-1-yl]acetyl]amino]-8-azabicyclo[3.2.1]octane-8-carboxylate
—— tert-butyl (3R)-3-[[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]carbamoylamino]azepane-1-carboxylate —— C21H30N4O5
tert-butyl (3R)-3-[[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]carbamoylamino]azepane-1-carboxylate
—— tert-butyl (2R)-2-[[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]methylcarbamoyl]pyrrolidine-1-carboxylate —— C21H31N3O4S
tert-butyl (2R)-2-[[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]methylcarbamoyl]pyrrolidine-1-carboxylate
—— tert-butyl (1R,6S)-3-(pyridin-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C18H27N3O2
tert-butyl (1R,6S)-3-(pyridin-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (1R,6S)-3-[2-(1,2,4-triazol-1-yl)ethyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C16H27N5O2
tert-butyl (1R,6S)-3-[2-(1,2,4-triazol-1-yl)ethyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (1S,6R)-3-(1,3-thiazol-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C16H25N3O2S
tert-butyl (1S,6R)-3-(1,3-thiazol-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (3R,4S)-3-[[2-(2-fluorophenyl)acetyl]amino]-4-methoxypyrrolidine-1-carboxylate —— C18H25FN2O4
tert-butyl (3R,4S)-3-[[2-(2-fluorophenyl)acetyl]amino]-4-methoxypyrrolidine-1-carboxylate
—— tert-butyl (1S,5R)-3-[methyl-(5-methylthiophene-2-carbonyl)amino]-8-azabicyclo[3.2.1]octane-8-carboxylate —— C19H28N2O3S
tert-butyl (1S,5R)-3-[methyl-(5-methylthiophene-2-carbonyl)amino]-8-azabicyclo[3.2.1]octane-8-carboxylate
—— tert-butyl (1S,6R)-3-(7-methyl-4-oxo-1H-1,8-naphthyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate —— C22H28N4O4
tert-butyl (1S,6R)-3-(7-methyl-4-oxo-1H-1,8-naphthyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— tert-butyl (3S)-3-[(2S)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate —— C19H28N2O4
tert-butyl (3S)-3-[(2S)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate
—— tert-butyl (3S)-3-[(2R)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate —— C19H28N2O4
tert-butyl (3S)-3-[(2R)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate
—— tert-butyl (3R)-3-[(2R)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate —— C19H28N2O4
tert-butyl (3R)-3-[(2R)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate
—— tert-butyl (3R)-3-[(2S)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate —— C19H28N2O4
tert-butyl (3R)-3-[(2S)-2-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]pyrrolidine-1-carboxylate
—— tert-butyl (3S,4S)-3-methoxy-4-[[2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]acetyl]amino]pyrrolidine-1-carboxylate —— C22H29N3O4S
tert-butyl (3S,4S)-3-methoxy-4-[[2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]acetyl]amino]pyrrolidine-1-carboxylate
—— tert-butyl N-[(2R)-2-methyl-3-[[2-[2-(4-methylanilino)-2-oxoethyl]sulfanylacetyl]amino]propyl]carbamate —— C20H31N3O4S
tert-butyl N-[(2R)-2-methyl-3-[[2-[2-(4-methylanilino)-2-oxoethyl]sulfanylacetyl]amino]propyl]carbamate
—— tert-butyl (3S,4R)-3-methoxy-4-[[2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]acetyl]amino]pyrrolidine-1-carboxylate —— C22H29N3O4S
tert-butyl (3S,4R)-3-methoxy-4-[[2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]acetyl]amino]pyrrolidine-1-carboxylate
—— tert-butyl N-[(2S)-2-methyl-3-[[2-[2-(4-methylanilino)-2-oxoethyl]sulfanylacetyl]amino]propyl]carbamate —— C20H31N3O4S
tert-butyl N-[(2S)-2-methyl-3-[[2-[2-(4-methylanilino)-2-oxoethyl]sulfanylacetyl]amino]propyl]carbamate
—— tert-butyl N-[(2S)-1-[[4-[4-(hydroxymethyl)piperidin-1-yl]phenyl]methylamino]-3,3-dimethyl-1-oxobutan-2-yl]carbamate —— C24H39N3O4
tert-butyl N-[(2S)-1-[[4-[4-(hydroxymethyl)piperidin-1-yl]phenyl]methylamino]-3,3-dimethyl-1-oxobutan-2-yl]carbamate
—— tert-butyl N-[(2R)-1-[[4-[4-(hydroxymethyl)piperidin-1-yl]phenyl]methylamino]-3,3-dimethyl-1-oxobutan-2-yl]carbamate —— C24H39N3O4
tert-butyl N-[(2R)-1-[[4-[4-(hydroxymethyl)piperidin-1-yl]phenyl]methylamino]-3,3-dimethyl-1-oxobutan-2-yl]carbamate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C42H56N4O11
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[3-(dimethylamino)-3-oxoprop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C44H55N3O12
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[3-[2-(2-hydroxyethoxy)ethenyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C46H57N3O11
tert-butyl (4S)-4-[[(2R)-1-[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-11-[[4-[3-(2-hydroxyphenyl)prop-1-enyl]phenyl]methyl]-9-oxo-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[2-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate —— C57H67N3O16
tert-butyl (4S)-5-hydroxy-4-[[(2R)-2-[methyl-[(1S,2S,6S,7R,10R,13S)-9-oxo-4,4-diphenyl-11-[[2-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-3-phenylpropanoyl]amino]pentanoate
—— tert-butyl (4S)-4-[[(2R)-1-[(3aR,7R,7aS)-7-hydroxy-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate —— C22H34N2O8
tert-butyl (4S)-4-[[(2R)-1-[(3aR,7R,7aS)-7-hydroxy-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carbonyl]pyrrolidine-2-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(3aR,7R,7aS)-7-hydroxy-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carbonyl]amino]-5-hydroxypentanoate —— C17H27NO7
tert-butyl (4S)-4-[[(3aR,7R,7aS)-7-hydroxy-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate —— C41H56N2O15
tert-butyl (4S)-4-[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]-5-hydroxypentanoate
—— tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate —— C49H63N3O16
tert-butyl (4S)-4-[[3-[[[(1S,2S,6S,7R,10R,13S)-4,4-dicyclopropyl-9-oxo-11-[[3-[3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyprop-1-enyl]phenyl]methyl]-3,5,8,12-tetraoxa-11-azatetracyclo[5.5.2.02,6.010,13]tetradecane-13-carbonyl]amino]methyl]benzoyl]amino]-5-hydroxypentanoate