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中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl (1S,2R)-1-[benzyl-[(1R)-1-phenylethyl]amino]-6-fluoro-2,3-dihydro-1H-indene-2-carboxylate —— C26H26FNO2
methyl (1S,2R)-1-[benzyl-[(1R)-1-phenylethyl]amino]-6-fluoro-2,3-dihydro-1H-indene-2-carboxylate
—— methyl 5-ethyl-2-[[(5S)-4-oxo-3-phenyl-2-phenylimino-1,3-thiazolidine-5-carbonyl]amino]thiophene-3-carboxylate —— C24H21N3O4S2
methyl 5-ethyl-2-[[(5S)-4-oxo-3-phenyl-2-phenylimino-1,3-thiazolidine-5-carbonyl]amino]thiophene-3-carboxylate
—— methyl 4-[[(2S)-5-chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]carbamoylamino]benzoate —— C17H12ClF3N2O5
methyl 4-[[(2S)-5-chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]carbamoylamino]benzoate
—— methyl 6-[(3S)-3-methylpiperidin-1-yl]pyridine-2-carboxylate —— C13H18N2O2
methyl 6-[(3S)-3-methylpiperidin-1-yl]pyridine-2-carboxylate
—— Methyl 3-[4-carbamoyl-5-[(2,3-dimethylbenzoyl)carbamothioylamino]pyrazol-1-yl]benzoate —— C22H21N5O4S
Methyl 3-[4-carbamoyl-5-[(2,3-dimethylbenzoyl)carbamothioylamino]pyrazol-1-yl]benzoate
—— methyl 2-[(3R)-4-[(3S)-7-[[4-[[(3S,5S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-5-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidin-3-yl]carbamoyl]benzoyl]amino]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-2-yl]-2-methyl-3-[[(2S)-2-(methylamino)propanoyl]amino]-4-oxobutan-2-yl]sulfanylacetate —— C65H84N10O10S
methyl 2-[(3R)-4-[(3S)-7-[[4-[[(3S,5S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-5-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidin-3-yl]carbamoyl]benzoyl]amino]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-2-yl]-2-methyl-3-[[(2S)-2-(methylamino)propanoyl]amino]-4-oxobutan-2-yl]sulfanylacetate
—— methyl 2-[[2-(4-aminoquinazolin-2-yl)sulfanylacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C19H18N4O3S2
methyl 2-[[2-(4-aminoquinazolin-2-yl)sulfanylacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— methyl 6-[(3S)-3-aminopiperidin-1-yl]pyridine-2-carboxylate —— C12H17N3O2
methyl 6-[(3S)-3-aminopiperidin-1-yl]pyridine-2-carboxylate
—— methyl 2-[[(3S)-2-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinoline-7-carbonyl]amino]-1,3-benzothiazole-5-carboxylate —— C40H46N6O6S
methyl 2-[[(3S)-2-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinoline-7-carbonyl]amino]-1,3-benzothiazole-5-carboxylate
—— Methyl 4-(((S)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate —— C29H29N3O4
Methyl 4-(((S)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate
—— Methyl 4-((N-((S)-2-((S)-2-((S)-2-((tert-butoxycarbonyl)(methyl)amino) propanamido)-3,3-dimethylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)acetamido)methyl)benzoate —— C46H59N5O8
Methyl 4-((N-((S)-2-((S)-2-((S)-2-((tert-butoxycarbonyl)(methyl)amino) propanamido)-3,3-dimethylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)acetamido)methyl)benzoate
—— methyl 1-[[(3S,5S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoyl]amino]butanoyl]-5-[[(1R,3Z,5Z)-7-methylidenecyclodeca-3,5-dien-1-yl]carbamoyl]pyrrolidin-3-yl]carbamoyl]indole-5-carboxylate —— C42H58N6O8
methyl 1-[[(3S,5S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoyl]amino]butanoyl]-5-[[(1R,3Z,5Z)-7-methylidenecyclodeca-3,5-dien-1-yl]carbamoyl]pyrrolidin-3-yl]carbamoyl]indole-5-carboxylate
—— Methyl 4-(((S)-2-((R)-2-amino-3-methyl-3-(methylthio)butanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate —— C35H40N4O5S
Methyl 4-(((S)-2-((R)-2-amino-3-methyl-3-(methylthio)butanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate
—— Methyl 4-[2-(propanoylamino)ethyl]benzoate —— C13H17NO3
Methyl 4-[2-(propanoylamino)ethyl]benzoate
—— Methyl 4-(((S)-2-((R)-2-((tert-butoxycarbonyl)amino)-3-methyl-3-(methylthio)butanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate —— C40H48N4O7S
Methyl 4-(((S)-2-((R)-2-((tert-butoxycarbonyl)amino)-3-methyl-3-(methylthio)butanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate
—— methyl 4-[[(3S,5S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-5-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidin-3-yl]amino]-4-oxobutanoate —— C30H45N5O6
methyl 4-[[(3S,5S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-5-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidin-3-yl]amino]-4-oxobutanoate
—— methyl 4-[[(3S)-2-[(2R)-3-methyl-2-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoyl]amino]-3-methylsulfanylbutanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-7-yl]carbamoyl]benzoate —— C44H55N5O8S
methyl 4-[[(3S)-2-[(2R)-3-methyl-2-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoyl]amino]-3-methylsulfanylbutanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-7-yl]carbamoyl]benzoate
—— methyl 3-[2-(2-aminoethoxy)-5-tert-butylphenyl]-3-(4-methoxyphenyl)-2-oxo-1H-indole-7-carboxylate —— C29H32N2O5
methyl 3-[2-(2-aminoethoxy)-5-tert-butylphenyl]-3-(4-methoxyphenyl)-2-oxo-1H-indole-7-carboxylate
—— methyl 4-[[(E)-3-(4-methylphenyl)prop-2-enoyl]oxymethyl]benzoate —— C19H18O4
methyl 4-[[(E)-3-(4-methylphenyl)prop-2-enoyl]oxymethyl]benzoate
—— methyl 4-[[(3S)-2-[(2S)-2-amino-3,3-dimethylbutanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]benzoate —— C35H41N3O5
methyl 4-[[(3S)-2-[(2S)-2-amino-3,3-dimethylbutanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]benzoate
—— methyl 4-((((S)-2-((S)-2-((S)-2-((tert-butoxycarbonyl)(methyl)amino)propanamido)-3,3-dimethylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)oxy)methyl)benzoate —— C44H56N4O8
methyl 4-((((S)-2-((S)-2-((S)-2-((tert-butoxycarbonyl)(methyl)amino)propanamido)-3,3-dimethylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)oxy)methyl)benzoate
—— Methyl 2-[2-[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]ethyl-[[6-[[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]methyl]-4-[2-[4-(2-chloro-2-oxoethoxy)phenyl]ethynyl]pyridin-2-yl]methyl]amino]acetate —— C46H65ClN4O12
Methyl 2-[2-[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]ethyl-[[6-[[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]methyl]-4-[2-[4-(2-chloro-2-oxoethoxy)phenyl]ethynyl]pyridin-2-yl]methyl]amino]acetate
—— methyl 4-[[(2S,4R)-1-[(2S)-2-amino-3,3-dimethylbutanoyl]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]piperidin-4-yl]oxymethyl]benzoate —— C31H41N3O5
methyl 4-[[(2S,4R)-1-[(2S)-2-amino-3,3-dimethylbutanoyl]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]piperidin-4-yl]oxymethyl]benzoate
—— Methyl 2-(4-fluorophenyl)-7-(methylamino)-4-methylidenecycloheptane-1-carboxylate —— C17H22FNO2
Methyl 2-(4-fluorophenyl)-7-(methylamino)-4-methylidenecycloheptane-1-carboxylate
—— Methyl [(4,5-dioxo-1,3,4,2-dioxasilaborolan-2-yl)oxy-oxosilyl]formate —— C3H3BO8Si2
Methyl [(4,5-dioxo-1,3,4,2-dioxasilaborolan-2-yl)oxy-oxosilyl]formate
—— methyl 4-[[(3S)-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl]oxymethyl]benzoate —— C29H30N2O4
methyl 4-[[(3S)-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl]oxymethyl]benzoate
—— Methyl 1-(6-azaspiro[3.4]octan-2-yl)-4-fluoropiperidine-4-carboxylate —— C14H23FN2O2
Methyl 1-(6-azaspiro[3.4]octan-2-yl)-4-fluoropiperidine-4-carboxylate
—— Methyl 4-((((2S,4R)-2-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)piperidin-4-yl)oxy)methyl)benzoate —— C25H30N2O4
Methyl 4-((((2S,4R)-2-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)piperidin-4-yl)oxy)methyl)benzoate
—— Methyl 4-((((S)-2-((S)-2-((S)-2-((tert-butoxycarbonyl)(methyl)amino) propanamido)-3,3-dimethylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)amino)methyl)benzoate —— C44H57N5O7
Methyl 4-((((S)-2-((S)-2-((S)-2-((tert-butoxycarbonyl)(methyl)amino) propanamido)-3,3-dimethylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)amino)methyl)benzoate
—— methyl 2-[(2S)-1-[2-[[5-(4-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-3-oxopiperazin-2-yl]acetate —— C18H21N5O5S2
methyl 2-[(2S)-1-[2-[[5-(4-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-3-oxopiperazin-2-yl]acetate
—— methyl 4-[3-[(6aS)-3-[3-[[(6aS)-2-methoxy-8-[4-(4-methylpiperazin-1-yl)phenyl]-11-oxo-6a,7-dihydropyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxy]propoxy]-2-methoxy-11-oxo-5,6,6a,7-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-8-yl]-N-methylanilino]-4-oxobutanoate —— C52H57N7O9
methyl 4-[3-[(6aS)-3-[3-[[(6aS)-2-methoxy-8-[4-(4-methylpiperazin-1-yl)phenyl]-11-oxo-6a,7-dihydropyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxy]propoxy]-2-methoxy-11-oxo-5,6,6a,7-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-8-yl]-N-methylanilino]-4-oxobutanoate
—— methyl 2-[(2R)-1-[2-[[5-(4-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-3-oxopiperazin-2-yl]acetate —— C18H21N5O5S2
methyl 2-[(2R)-1-[2-[[5-(4-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-3-oxopiperazin-2-yl]acetate
—— Methyl 4-(((S)-2-((R)-2-((tert-butoxycarbonyl)amino)-3-mercapto-3-methylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate —— C39H46N4O7S
Methyl 4-(((S)-2-((R)-2-((tert-butoxycarbonyl)amino)-3-mercapto-3-methylbutanoyl)-3-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)carbamoyl)benzoate
—— methyl 4-[[(3S)-2-[(2S)-3,3-dimethyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]benzoate —— C40H49N3O7
methyl 4-[[(3S)-2-[(2S)-3,3-dimethyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]benzoate
—— Methyl 4-[4-carbamoyl-5-[(3,4,5-trimethoxybenzoyl)carbamothioylamino]pyrazol-1-yl]benzoate —— C23H23N5O7S
Methyl 4-[4-carbamoyl-5-[(3,4,5-trimethoxybenzoyl)carbamothioylamino]pyrazol-1-yl]benzoate
—— methyl (4E)-2-methyl-4-[(4-methylsulfanylphenyl)methylidene]-5-oxo-1-propylpyrrole-3-carboxylate —— C18H21NO3S
methyl (4E)-2-methyl-4-[(4-methylsulfanylphenyl)methylidene]-5-oxo-1-propylpyrrole-3-carboxylate
—— Methyl 5-[[(2-fluorophenyl)sulfonyl-(furan-2-ylmethyl)amino]methyl]furan-2-carboxylate —— C18H16FNO6S
Methyl 5-[[(2-fluorophenyl)sulfonyl-(furan-2-ylmethyl)amino]methyl]furan-2-carboxylate
—— methyl (4Z)-1-butyl-4-[(3-ethoxy-2-hydroxyphenyl)methylidene]-2-methyl-5-oxopyrrole-3-carboxylate —— C20H25NO5
methyl (4Z)-1-butyl-4-[(3-ethoxy-2-hydroxyphenyl)methylidene]-2-methyl-5-oxopyrrole-3-carboxylate
—— methyl 1-[2-[2-(1H-indol-3-yl)acetyl]oxyacetyl]piperidine-4-carboxylate —— C19H22N2O5
methyl 1-[2-[2-(1H-indol-3-yl)acetyl]oxyacetyl]piperidine-4-carboxylate
—— Methyl 1-[2-(2,5-dimethyl-1-phenylpyrrole-3-carbonyl)oxyacetyl]piperidine-4-carboxylate —— C22H26N2O5
Methyl 1-[2-(2,5-dimethyl-1-phenylpyrrole-3-carbonyl)oxyacetyl]piperidine-4-carboxylate
—— Methyl 4-[2,5-dimethyl-3-[2-[2-(trifluoromethyl)anilino]-1,3-thiazol-4-yl]pyrrol-1-yl]benzoate —— C24H20F3N3O2S
Methyl 4-[2,5-dimethyl-3-[2-[2-(trifluoromethyl)anilino]-1,3-thiazol-4-yl]pyrrol-1-yl]benzoate
—— methyl (4E)-1-butyl-4-[(4-methoxycarbonylphenyl)methylidene]-2-methyl-5-oxopyrrole-3-carboxylate —— C20H23NO5
methyl (4E)-1-butyl-4-[(4-methoxycarbonylphenyl)methylidene]-2-methyl-5-oxopyrrole-3-carboxylate
—— Methyl [(4,5-dioxo-1,3,2-dioxaborolan-2-yl)oxy-oxosilyl]formate —— C4H3BO8Si
Methyl [(4,5-dioxo-1,3,2-dioxaborolan-2-yl)oxy-oxosilyl]formate
—— methyl-[(1Z)-2-methylbuta-1,3-dienyl]diazene —— C6H10N2
methyl-[(1Z)-2-methylbuta-1,3-dienyl]diazene
—— methyl 1-[2-[(E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enoyl]oxyacetyl]piperidine-4-carboxylate —— C19H23NO7
methyl 1-[2-[(E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enoyl]oxyacetyl]piperidine-4-carboxylate
—— methyl (4Z)-4-[(2-ethoxyphenyl)methylidene]-2-methyl-5-oxo-1-propylpyrrole-3-carboxylate —— C19H23NO4
methyl (4Z)-4-[(2-ethoxyphenyl)methylidene]-2-methyl-5-oxo-1-propylpyrrole-3-carboxylate
—— methyl (4E)-4-[(2,3-dimethoxyphenyl)methylidene]-2-methyl-5-oxo-1-propylpyrrole-3-carboxylate —— C19H23NO5
methyl (4E)-4-[(2,3-dimethoxyphenyl)methylidene]-2-methyl-5-oxo-1-propylpyrrole-3-carboxylate
—— methyl (4Z)-1-butyl-4-[(4-methoxycarbonylphenyl)methylidene]-2-methyl-5-oxopyrrole-3-carboxylate —— C20H23NO5
methyl (4Z)-1-butyl-4-[(4-methoxycarbonylphenyl)methylidene]-2-methyl-5-oxopyrrole-3-carboxylate
—— Methyl 5-[[5-[(4-ethylphenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-methylfuran-3-carboxylate —— C22H25N3O4S
Methyl 5-[[5-[(4-ethylphenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-methylfuran-3-carboxylate
—— Methyl 2-[2-[bis(2-methoxy-2-oxoethyl)amino]ethyl-[[6-[[2-[bis(2-methoxy-2-oxoethyl)amino]ethyl-(2-methoxy-2-oxoethyl)amino]methyl]-4-[2-[4-[4-[chloro(2-cyanoethoxy)phosphanyl]oxybutoxy]phenyl]ethynyl]pyridin-2-yl]methyl]amino]acetate —— C44H60ClN6O15P
Methyl 2-[2-[bis(2-methoxy-2-oxoethyl)amino]ethyl-[[6-[[2-[bis(2-methoxy-2-oxoethyl)amino]ethyl-(2-methoxy-2-oxoethyl)amino]methyl]-4-[2-[4-[4-[chloro(2-cyanoethoxy)phosphanyl]oxybutoxy]phenyl]ethynyl]pyridin-2-yl]methyl]amino]acetate