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—— Methyl 5-[4-cyano-2-[(3,4-dihydroxy-1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C28H28F3N6O5+
Methyl 5-[4-cyano-2-[(3,4-dihydroxy-1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[3-(2-methylpyridin-1-ium-1-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C32H29F3N6O5
Methyl 5-[4-cyano-2-[3-(2-methylpyridin-1-ium-1-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[4-cyano-2-(3-hydroxypropyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C25H22F3N5O4
Methyl 5-[4-cyano-2-(3-hydroxypropyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-[4-cyano-2-[2-[1-(2-formyloxyethyl)pyrrolidin-1-ium-1-yl]ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C31H32F3N6O5+
methyl (5R)-5-[4-cyano-2-[2-[1-(2-formyloxyethyl)pyrrolidin-1-ium-1-yl]ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-(2-trimethylsilylethynyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C27H24F3N5O3Si
Methyl 5-[4-cyano-2-(2-trimethylsilylethynyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl 7-[(1R,4S,5R)-4-[tert-butyl(dimethyl)silyl]oxy-5-[(E)-3-[tert-butyl(dimethyl)silyl]oxy-5-(3-chloro-1-benzothiophen-2-yl)pent-4-enyl]-3,3-dimethyl-2-oxocyclopentyl]hept-5-ynoate —— C40H61ClO5SSi2
methyl 7-[(1R,4S,5R)-4-[tert-butyl(dimethyl)silyl]oxy-5-[(E)-3-[tert-butyl(dimethyl)silyl]oxy-5-(3-chloro-1-benzothiophen-2-yl)pent-4-enyl]-3,3-dimethyl-2-oxocyclopentyl]hept-5-ynoate
—— methyl (5Z)-2-anilino-5-[(3-hydroxyphenyl)methylidene]-4-oxothiophene-3-carboxylate —— C19H15NO4S
methyl (5Z)-2-anilino-5-[(3-hydroxyphenyl)methylidene]-4-oxothiophene-3-carboxylate
—— Methyl 5-[2-[4-(1-azoniabicyclo[2.2.2]octan-1-yl)butyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C34H37F3N6O5
Methyl 5-[2-[4-(1-azoniabicyclo[2.2.2]octan-1-yl)butyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl 2-{[({1-[4-(propoxycarbonyl)phenyl]-1H-tetrazol-5-yl}sulfanyl)acetyl]amino}benzoate —— C21H21N5O5S
methyl 2-{[({1-[4-(propoxycarbonyl)phenyl]-1H-tetrazol-5-yl}sulfanyl)acetyl]amino}benzoate
—— Methyl 5-[2-(5-bromopentyl)-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C27H25BrF3N5O3
Methyl 5-[2-(5-bromopentyl)-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[(4-methyl-1,4-oxazepan-4-ium-4-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C30H31F3N6O6
Methyl 5-[4-cyano-2-[(4-methyl-1,4-oxazepan-4-ium-4-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[4-cyano-2-[2-[1-(2-hydroxyethyl)pyrrolidin-1-ium-1-yl]ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C30H32F3N6O4+
Methyl 5-[4-cyano-2-[2-[1-(2-hydroxyethyl)pyrrolidin-1-ium-1-yl]ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-(2-methoxy-2-oxoethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C25H20F3N5O5
Methyl 5-[4-cyano-2-(2-methoxy-2-oxoethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[3-(2-methylpyridin-1-ium-1-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C31H28F3N6O3+
Methyl 5-[4-cyano-2-[3-(2-methylpyridin-1-ium-1-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl (5E)-2-anilino-5-[(3-nitrophenyl)methylidene]-4-oxothiophene-3-carboxylate —— C19H14N2O5S
methyl (5E)-2-anilino-5-[(3-nitrophenyl)methylidene]-4-oxothiophene-3-carboxylate
—— Methyl 5-[4-cyano-2-(pyridin-1-ium-1-ylmethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C29H23F3N6O5
Methyl 5-[4-cyano-2-(pyridin-1-ium-1-ylmethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl (5R)-5-[4-cyano-2-[(4-methyl-1,4-oxazepan-4-ium-4-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C29H30F3N6O4+
methyl (5R)-5-[4-cyano-2-[(4-methyl-1,4-oxazepan-4-ium-4-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[2-(4-methylmorpholin-4-ium-4-yl)ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C30H31F3N6O6
Methyl 5-[4-cyano-2-[2-(4-methylmorpholin-4-ium-4-yl)ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl (E)-2-[[4-(2-methylpropoxy)benzoyl]amino]-3-phenylprop-2-enoate —— C21H23NO4
methyl (E)-2-[[4-(2-methylpropoxy)benzoyl]amino]-3-phenylprop-2-enoate
—— Methyl 5-[4-cyano-2-[(3,4-dihydroxy-1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C29H29F3N6O7
Methyl 5-[4-cyano-2-[(3,4-dihydroxy-1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[4-cyano-2-[(4-methyl-1,4-oxazepan-4-ium-4-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C29H30F3N6O4+
Methyl 5-[4-cyano-2-[(4-methyl-1,4-oxazepan-4-ium-4-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[2-[3-(4-aza-1-azoniabicyclo[2.2.2]octan-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C31H33F3N7O3+
Methyl 5-[2-[3-(4-aza-1-azoniabicyclo[2.2.2]octan-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[2-[(3-chloropyridin-1-ium-1-yl)methyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C28H21ClF3N6O3+
Methyl 5-[2-[(3-chloropyridin-1-ium-1-yl)methyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[2-(4-methylmorpholin-4-ium-4-yl)ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C29H30F3N6O4+
Methyl 5-[4-cyano-2-[2-(4-methylmorpholin-4-ium-4-yl)ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-(3-pyridin-1-ium-1-ylpropyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;chloride —— C30H26ClF3N6O3
Methyl 5-[4-cyano-2-(3-pyridin-1-ium-1-ylpropyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;chloride
—— methyl (5R)-5-[4-cyano-2-[2-(4-formyloxy-1-methylpiperidin-1-ium-1-yl)ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C31H32F3N6O5+
methyl (5R)-5-[4-cyano-2-[2-(4-formyloxy-1-methylpiperidin-1-ium-1-yl)ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-[4-cyano-2-(2-piperidin-1-ium-1-ylethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C30H31F3N6O5
methyl (5R)-5-[4-cyano-2-(2-piperidin-1-ium-1-ylethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl (5R)-5-[4-cyano-2-[[3-(formyloxymethyl)pyridin-1-ium-1-yl]methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C30H24F3N6O5+
methyl (5R)-5-[4-cyano-2-[[3-(formyloxymethyl)pyridin-1-ium-1-yl]methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[(1,4-dimethylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C30H32F3N7O5
Methyl 5-[4-cyano-2-[(1,4-dimethylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[4-cyano-2-[(1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C28H28F3N6O3+
Methyl 5-[4-cyano-2-[(1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[2-[4-(1-azoniabicyclo[2.2.2]octan-1-yl)butyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C33H36F3N6O3+
Methyl 5-[2-[4-(1-azoniabicyclo[2.2.2]octan-1-yl)butyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[(1-methyl-4-methylsulfonylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C29H31F3N7O5S+
Methyl 5-[4-cyano-2-[(1-methyl-4-methylsulfonylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[(1-methyl-4-methylsulfonylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C30H32F3N7O7S
Methyl 5-[4-cyano-2-[(1-methyl-4-methylsulfonylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[2-[(3-chloropyridin-1-ium-1-yl)methyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C29H22ClF3N6O5
Methyl 5-[2-[(3-chloropyridin-1-ium-1-yl)methyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[4-cyano-2-(3-pyridin-1-ium-1-ylpropyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;bromide —— C30H26BrF3N6O3
Methyl 5-[4-cyano-2-(3-pyridin-1-ium-1-ylpropyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;bromide
—— Methyl 5-[2-[3-(3-chloropyridin-1-ium-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C31H26ClF3N6O5
Methyl 5-[2-[3-(3-chloropyridin-1-ium-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl (5R)-5-[4-cyano-2-(2-piperidin-1-ylethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C29H29F3N6O3
methyl (5R)-5-[4-cyano-2-(2-piperidin-1-ylethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[3-(4-methylmorpholin-4-ium-4-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C30H32F3N6O4+
Methyl 5-[4-cyano-2-[3-(4-methylmorpholin-4-ium-4-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-[4-cyano-2-[(1-methyl-4-methylsulfonylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C29H31F3N7O5S+
methyl (5R)-5-[4-cyano-2-[(1-methyl-4-methylsulfonylpiperazin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-[4-cyano-2-[2-[4-(dimethylamino)oxan-3-yl]ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C31H33F3N6O4
methyl (5R)-5-[4-cyano-2-[2-[4-(dimethylamino)oxan-3-yl]ethyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[2-[3-(3-chloropyridin-1-ium-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C30H25ClF3N6O3+
Methyl 5-[2-[3-(3-chloropyridin-1-ium-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[(1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C29H29F3N6O5
Methyl 5-[4-cyano-2-[(1-methylpyrrolidin-1-ium-1-yl)methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[2-[3-(1-azoniabicyclo[2.2.2]octan-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C33H35F3N6O5
Methyl 5-[2-[3-(1-azoniabicyclo[2.2.2]octan-1-yl)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— Methyl 5-[4-cyano-2-[3-(4-methylmorpholin-4-ium-4-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C31H33F3N6O6
Methyl 5-[4-cyano-2-[3-(4-methylmorpholin-4-ium-4-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl (5R)-5-[4-cyano-2-[[1-(2-formyloxyethyl)pyrrolidin-1-ium-1-yl]methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C30H30F3N6O5+
methyl (5R)-5-[4-cyano-2-[[1-(2-formyloxyethyl)pyrrolidin-1-ium-1-yl]methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-(5-hydroxypentyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C27H26F3N5O4
Methyl 5-[4-cyano-2-(5-hydroxypentyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-[[3-(hydroxymethyl)pyridin-1-ium-1-yl]methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate —— C30H25F3N6O6
Methyl 5-[4-cyano-2-[[3-(hydroxymethyl)pyridin-1-ium-1-yl]methyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;formate
—— methyl (5R)-5-[2-[3-(1-adamantylamino)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C35H37F3N6O3
methyl (5R)-5-[2-[3-(1-adamantylamino)propyl]-4-cyanophenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate
—— Methyl 5-[4-cyano-2-(2-pyridin-1-ium-1-ylethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;bromide —— C29H24BrF3N6O3
Methyl 5-[4-cyano-2-(2-pyridin-1-ium-1-ylethyl)phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate;bromide
—— Methyl 5-[4-cyano-2-[3-(3-methylpyridin-1-ium-1-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate —— C31H28F3N6O3+
Methyl 5-[4-cyano-2-[3-(3-methylpyridin-1-ium-1-yl)propyl]phenyl]-7-methyl-3-oxo-8-[3-(trifluoromethyl)phenyl]-2,5-dihydro-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylate