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—— ethyl (5S)-1-acetyl-7-(3-chlorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C17H16ClN3O5
ethyl (5S)-1-acetyl-7-(3-chlorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide —— C19H21N5O3
(E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide
—— (E)-N-[(2S)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-3-pyridin-3-ylprop-2-enamide —— C21H23N3O2
(E)-N-[(2S)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-3-pyridin-3-ylprop-2-enamide
—— (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide —— C18H19N5O3
(E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide
—— (E)-N-[(1S)-2-phenoxy-1-phenylethyl]-3-pyrazin-2-ylprop-2-enamide —— C21H19N3O2
(E)-N-[(1S)-2-phenoxy-1-phenylethyl]-3-pyrazin-2-ylprop-2-enamide
—— (E)-N-[(2R)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-3-pyridin-3-ylprop-2-enamide —— C21H23N3O2
(E)-N-[(2R)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-3-pyridin-3-ylprop-2-enamide
—— (E)-N-(4-benzylpiperazin-4-ium-1-yl)-1-(4-chlorophenyl)ethanimine —— C19H23ClN3+
(E)-N-(4-benzylpiperazin-4-ium-1-yl)-1-(4-chlorophenyl)ethanimine
—— (E)-2-benzamido-3-(3,4-diethoxyphenyl)prop-2-enoate —— C20H20NO5-
(E)-2-benzamido-3-(3,4-diethoxyphenyl)prop-2-enoate
—— ethyl N-[(3R)-1-(4-cyano-2-fluorophenyl)piperidin-3-yl]carbamate —— C15H18FN3O2
ethyl N-[(3R)-1-(4-cyano-2-fluorophenyl)piperidin-3-yl]carbamate
—— (E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2R)-2-methylmorpholin-4-yl]ethyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C26H29ClFN3O3
(E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2R)-2-methylmorpholin-4-yl]ethyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide —— C21H23N5O3
(E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide
—— (E)-1-(3-bromophenyl)-N-[4-[(4-chlorophenyl)methyl]piperazin-4-ium-1-yl]ethanimine —— C19H22BrClN3+
(E)-1-(3-bromophenyl)-N-[4-[(4-chlorophenyl)methyl]piperazin-4-ium-1-yl]ethanimine
—— (E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C26H29ClFN3O3
(E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-1-(4-bromophenyl)-N-[4-(4-chlorophenyl)piperazin-1-yl]ethanimine —— C18H19BrClN3
(E)-1-(4-bromophenyl)-N-[4-(4-chlorophenyl)piperazin-1-yl]ethanimine
—— ethyl (5S)-1-acetyl-6,8-dioxo-7-(2,4,6-trimethylphenyl)-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C20H23N3O5
ethyl (5S)-1-acetyl-6,8-dioxo-7-(2,4,6-trimethylphenyl)-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— (E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide —— C19H21N5O3
(E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide
—— (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-ethylprop-2-enamide —— C20H23N5O3
(E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-ethylprop-2-enamide
—— ethyl 5-[[2-[(2R)-butan-2-yl]pyrazol-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C17H24N4O3
ethyl 5-[[2-[(2R)-butan-2-yl]pyrazol-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-2-(1H-benzimidazol-2-yl)-3-[2-(4-methylpiperazin-4-ium-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enenitrile —— C23H22N7O+
(E)-2-(1H-benzimidazol-2-yl)-3-[2-(4-methylpiperazin-4-ium-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enenitrile
—— (E)-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-2-(morpholine-4-carbonyl)prop-2-enenitrile —— C22H25N5O4
(E)-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-2-(morpholine-4-carbonyl)prop-2-enenitrile
—— (E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-ethylprop-2-enamide —— C20H23N5O3
(E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-ethylprop-2-enamide
—— ethyl (4R,5R)-4-(4-methoxyphenyl)-5-(4-methylbenzoyl)-4,5-dihydro-1H-pyrazole-3-carboxylate —— C21H22N2O4
ethyl (4R,5R)-4-(4-methoxyphenyl)-5-(4-methylbenzoyl)-4,5-dihydro-1H-pyrazole-3-carboxylate
—— (E)-2-cyano-3-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide —— C21H23N5O3
(E)-2-cyano-3-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide
—— ethyl (5R)-1-acetyl-7-(4-fluorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C17H16FN3O5
ethyl (5R)-1-acetyl-7-(4-fluorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— ethyl (5S)-1-acetyl-7-(4-fluorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C17H16FN3O5
ethyl (5S)-1-acetyl-7-(4-fluorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— ethyl (5R)-1-acetyl-6,8-dioxo-7-(2,4,6-trimethylphenyl)-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C20H23N3O5
ethyl (5R)-1-acetyl-6,8-dioxo-7-(2,4,6-trimethylphenyl)-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— ethyl 5-[[2-[(2S)-butan-2-yl]pyrazol-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C17H24N4O3
ethyl 5-[[2-[(2S)-butan-2-yl]pyrazol-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide —— C21H23N5O3
(E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide
—— ethyl 3-[[2-[(2S)-butan-2-yl]pyrazol-3-yl]carbamoyl]-5-nitrobenzoate —— C17H20N4O5
ethyl 3-[[2-[(2S)-butan-2-yl]pyrazol-3-yl]carbamoyl]-5-nitrobenzoate
—— ethyl (4R,5S)-4-(4-methoxyphenyl)-5-(4-methylbenzoyl)-4,5-dihydro-1H-pyrazole-3-carboxylate —— C21H22N2O4
ethyl (4R,5S)-4-(4-methoxyphenyl)-5-(4-methylbenzoyl)-4,5-dihydro-1H-pyrazole-3-carboxylate
—— (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-methylprop-2-enamide —— C20H23N5O3
(E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-methylprop-2-enamide
—— ethyl 3-[[2-[(2R)-butan-2-yl]pyrazol-3-yl]carbamoyl]-5-nitrobenzoate —— C17H20N4O5
ethyl 3-[[2-[(2R)-butan-2-yl]pyrazol-3-yl]carbamoyl]-5-nitrobenzoate
—— ethyl (5R)-1-acetyl-7-(3,5-dimethylphenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C19H21N3O5
ethyl (5R)-1-acetyl-7-(3,5-dimethylphenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— ethyl (5R)-1-acetyl-7-(3-chloro-4-methylphenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C18H18ClN3O5
ethyl (5R)-1-acetyl-7-(3-chloro-4-methylphenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— (E)-2-cyano-3-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-methylprop-2-enamide —— C19H21N5O3
(E)-2-cyano-3-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-methylprop-2-enamide
—— (E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-methylprop-2-enamide —— C19H21N5O3
(E)-2-cyano-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-methylprop-2-enamide
—— ethyl 4-[(3S)-3-(1-adamantylamino)-2,5-dioxopyrrolidin-1-yl]benzoate —— C23H28N2O4
ethyl 4-[(3S)-3-(1-adamantylamino)-2,5-dioxopyrrolidin-1-yl]benzoate
—— (E)-2-cyano-3-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-(2-methoxyethyl)prop-2-enamide —— C21H25N5O4
(E)-2-cyano-3-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-(2-methoxyethyl)prop-2-enamide
—— ethyl (3aS,6aS)-5-(2-methoxyphenyl)-1-(3-methylphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C22H21N3O5
ethyl (3aS,6aS)-5-(2-methoxyphenyl)-1-(3-methylphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— ethyl (3aR,6aS)-5-(2-methoxyphenyl)-1-(3-methylphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C22H21N3O5
ethyl (3aR,6aS)-5-(2-methoxyphenyl)-1-(3-methylphenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— ethyl (5R)-1-acetyl-7-(3,5-dichlorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C17H15Cl2N3O5
ethyl (5R)-1-acetyl-7-(3,5-dichlorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— (E)-4-[2,5-diethoxy-4-[(4-methylbenzoyl)amino]anilino]-4-oxobut-2-enoate —— C22H23N2O6-
(E)-4-[2,5-diethoxy-4-[(4-methylbenzoyl)amino]anilino]-4-oxobut-2-enoate
—— ethyl 4-[(3R)-3-(1-adamantylamino)-2,5-dioxopyrrolidin-1-yl]benzoate —— C23H28N2O4
ethyl 4-[(3R)-3-(1-adamantylamino)-2,5-dioxopyrrolidin-1-yl]benzoate
—— (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-(2-methoxyethyl)prop-2-enamide —— C22H27N5O4
(E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-(2-methoxyethyl)prop-2-enamide
—— (E)-N-benzyl-3-((4-butylphenyl)amino)-2-cyanoacrylamide —— C21H23N3O
(E)-N-benzyl-3-((4-butylphenyl)amino)-2-cyanoacrylamide
—— (E)-N-(3-chlorophenyl)-2-cyano-3-(2,4-dimethoxyanilino)prop-2-enamide —— C18H16ClN3O3
(E)-N-(3-chlorophenyl)-2-cyano-3-(2,4-dimethoxyanilino)prop-2-enamide
—— ethyl 4-[[(E)-3-(3-chloroanilino)-2-cyano-3-oxoprop-1-enyl]amino]benzoate —— C19H16ClN3O3
ethyl 4-[[(E)-3-(3-chloroanilino)-2-cyano-3-oxoprop-1-enyl]amino]benzoate
—— ethyl (5S)-1-acetyl-7-(4-chlorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate —— C17H16ClN3O5
ethyl (5S)-1-acetyl-7-(4-chlorophenyl)-6,8-dioxo-1,2,7-triazaspiro[4.4]non-2-ene-3-carboxylate
—— (E)-2-cyano-3-(3,5-dimethoxyanilino)-N-(2-methoxyethyl)prop-2-enamide —— C15H19N3O4
(E)-2-cyano-3-(3,5-dimethoxyanilino)-N-(2-methoxyethyl)prop-2-enamide
—— ethyl (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enoate —— C20H22N4O4
ethyl (E)-2-cyano-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enoate