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—— (6aR)-5-(3-phenylpropanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C22H22N2O3
(6aR)-5-(3-phenylpropanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(3-fluorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17FN2O3
(6aS)-5-(3-fluorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— 6-[(4-benzylpiperazin-1-yl)methyl]-2-[4-[(2R)-2-ethylhexanoyl]piperazin-1-yl]-1H-pyrimidin-4-one —— C28H42N6O2
6-[(4-benzylpiperazin-1-yl)methyl]-2-[4-[(2R)-2-ethylhexanoyl]piperazin-1-yl]-1H-pyrimidin-4-one
—— (6aR)-5-(3-methylbutanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C18H22N2O3
(6aR)-5-(3-methylbutanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-[2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C17H17N5O3S
(6aS)-5-[2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(4-fluorobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C19H15FN2O3
(6aS)-5-(4-fluorobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aR)-5-[2-(1-phenyltetrazol-5-yl)sulfanylacetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C21H18N6O3S
(6aR)-5-[2-(1-phenyltetrazol-5-yl)sulfanylacetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aR)-5-[(E)-but-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C17H18N2O3
(6aR)-5-[(E)-but-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-(3-fluorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17FN2O3
(6aR)-5-(3-fluorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(2-chlorobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C19H15ClN2O3
(6aS)-5-(2-chlorobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(4-methoxybenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C21H20N2O4
(6aS)-5-(4-methoxybenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-[(E)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C22H18N2O5
(6aR)-5-[(E)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(3-fluorobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C19H15FN2O3
(6aS)-5-(3-fluorobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(2-bromobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17BrN2O3
(6aS)-5-(2-bromobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(3-phenylpropanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C22H22N2O3
(6aS)-5-(3-phenylpropanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(2-chlorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17ClN2O3
(6aS)-5-(2-chlorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(furan-2-carbonyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C18H16N2O4
(6aS)-5-(furan-2-carbonyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-[2-(1-methylimidazol-2-yl)sulfanylacetyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C19H20N4O3S
(6aS)-5-[2-(1-methylimidazol-2-yl)sulfanylacetyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(3,4-dimethoxybenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C22H22N2O5
(6aS)-5-(3,4-dimethoxybenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(3-methylbutanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C18H22N2O3
(6aS)-5-(3-methylbutanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-(3,5-dimethoxybenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C22H22N2O5
(6aR)-5-(3,5-dimethoxybenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-(4-bromobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C19H15BrN2O3
(6aR)-5-(4-bromobenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aR)-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C23H22N2O4
(6aR)-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-[2-(4-methylpiperazin-1-yl)acetyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H26N4O3
(6aS)-5-[2-(4-methylpiperazin-1-yl)acetyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-[(2R)-2-ethylhexanoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C21H28N2O3
(6aS)-5-[(2R)-2-ethylhexanoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-[2-(2,5-dioxopyrrolidin-1-yl)acetyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C19H19N3O5
(6aR)-5-[2-(2,5-dioxopyrrolidin-1-yl)acetyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-[(E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C24H24N2O5
(6aR)-5-[(E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-[(E)-but-2-enoyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C16H16N2O3
(6aS)-5-[(E)-but-2-enoyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— 6-[(2S)-pentan-2-yl]-1-phenyl-4-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]pyrazolo[3,4-d]pyrimidine —— C27H33N7
6-[(2S)-pentan-2-yl]-1-phenyl-4-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]pyrazolo[3,4-d]pyrimidine
—— (6aS)-5-[(2R)-2-ethylhexanoyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C20H26N2O3
(6aS)-5-[(2R)-2-ethylhexanoyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(2-pyrimidin-2-ylsulfanylacetyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C19H18N4O3S
(6aS)-5-(2-pyrimidin-2-ylsulfanylacetyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(2-pyrimidin-2-ylsulfanylacetyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C18H16N4O3S
(6aS)-5-(2-pyrimidin-2-ylsulfanylacetyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aR)-5-(4-chlorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17ClN2O3
(6aR)-5-(4-chlorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-[(E)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C23H20N2O5
(6aR)-5-[(E)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-[(E)-3-phenylprop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C22H20N2O3
(6aR)-5-[(E)-3-phenylprop-2-enoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— 6-(4-ethylphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-5-sulfanylidene-3H-pyrimido[4,5-d]pyrimidin-4-one —— C23H21N5OS
6-(4-ethylphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-5-sulfanylidene-3H-pyrimido[4,5-d]pyrimidin-4-one
—— (6aR)-5-(2-bromobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17BrN2O3
(6aR)-5-(2-bromobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(4-methoxybenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C20H18N2O4
(6aS)-5-(4-methoxybenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— 6-(4-ethylphenyl)-7-methyl-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-5-sulfanylidene-3H-pyrimido[4,5-d]pyrimidin-4-one —— C24H23N5OS
6-(4-ethylphenyl)-7-methyl-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-5-sulfanylidene-3H-pyrimido[4,5-d]pyrimidin-4-one
—— (6aR)-5-[2-(4-ethylpiperazin-1-yl)acetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C20H26N4O3
(6aR)-5-[2-(4-ethylpiperazin-1-yl)acetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(4-methylbenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C21H20N2O3
(6aS)-5-(4-methylbenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-(4-fluorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C20H17FN2O3
(6aR)-5-(4-fluorobenzoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aR)-5-(2-thiophen-2-ylacetyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C18H16N2O3S
(6aR)-5-(2-thiophen-2-ylacetyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-[(2R)-2-methylbutanoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C18H22N2O3
(6aS)-5-[(2R)-2-methylbutanoyl]-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(2-methylpropanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C17H20N2O3
(6aS)-5-(2-methylpropanoyl)-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-(2-methoxybenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C20H18N2O4
(6aS)-5-(2-methoxybenzoyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aR)-5-butanoyl-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione —— C17H20N2O3
(6aR)-5-butanoyl-7,8,9,10-tetrahydro-6aH-pyrido[2,1-c][1,4]benzodiazepine-6,12-dione
—— (6aS)-5-[2-(4-chlorophenyl)sulfanylacetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C20H17ClN2O3S
(6aS)-5-[2-(4-chlorophenyl)sulfanylacetyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— (6aS)-5-(thiophene-2-carbonyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C17H14N2O3S
(6aS)-5-(thiophene-2-carbonyl)-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— 6-(4-chlorophenyl)-7-methyl-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-5-sulfanylidene-3H-pyrimido[4,5-d]pyrimidin-4-one —— C22H18ClN5OS
6-(4-chlorophenyl)-7-methyl-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-5-sulfanylidene-3H-pyrimido[4,5-d]pyrimidin-4-one