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有机酸及其衍生物

中文名称 英文名称 CAS号 化学式 结构式图片
—— (5,5-Dichloro-4-methoxy-1,4,6,7-tetrahydroindol-2-yl)-(4-methylpiperazin-1-yl)methanone 1263084-75-8 C15H21Cl2N3O2
(5,5-Dichloro-4-methoxy-1,4,6,7-tetrahydroindol-2-yl)-(4-methylpiperazin-1-yl)methanone
—— N2-[4-({5,5-dimethyl-7-[(1S)-1-methylpropyl]-6-oxo-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzyl]-N1,N1-dimethylglycinamide 1201361-49-0 C23H32N6O2
N2-[4-({5,5-dimethyl-7-[(1S)-1-methylpropyl]-6-oxo-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzyl]-N1,N1-dimethylglycinamide
—— 3-t-Butoxycarbonylamino-3-methyl-N-[2,3,4,5-tetrahydro-2-oxo-1-[[2'-(thiazol-2-yl)[1,1'-biphenyl]-4-yl]methyl]-1H-1-benzazepin-3(R)-yl]-butanamide 162356-52-7 C36H40N4O4S
3-t-Butoxycarbonylamino-3-methyl-N-[2,3,4,5-tetrahydro-2-oxo-1-[[2'-(thiazol-2-yl)[1,1'-biphenyl]-4-yl]methyl]-1H-1-benzazepin-3(R)-yl]-butanamide
—— 3-[2(S),3-Dihydroxypropyl]amino-3-methyl-N-[1-[[2'-(ethylamino)sulfonyl[1,1'-biphenyl]-4-yl]methyl]-7-trifluoromethyl-2,3,4,5-tetrahydro-2-oxo-1H-1-benzazepin-3(R)-yl]butanamide 169188-56-1 C34H41F3N4O6S
3-[2(S),3-Dihydroxypropyl]amino-3-methyl-N-[1-[[2'-(ethylamino)sulfonyl[1,1'-biphenyl]-4-yl]methyl]-7-trifluoromethyl-2,3,4,5-tetrahydro-2-oxo-1H-1-benzazepin-3(R)-yl]butanamide
—— 2-{2-diethylamino-5-[(2-fluorobenzenesulfonyl)methylamino]-pyrimidin-4-ylamino}-3-(4-dimethylcarbamoyloxyphenyl)propionic acid 1055312-73-6 C27H33FN6O6S
2-{2-diethylamino-5-[(2-fluorobenzenesulfonyl)methylamino]-pyrimidin-4-ylamino}-3-(4-dimethylcarbamoyloxyphenyl)propionic acid
—— N-hydroxy-N-[(2R)-5-methyl-2-({N'-[7-(methyloxy)-1,2,4-benzotriazin-3-yl]-hydrazino}-carbonyl)-hexyl]-formamide 634608-43-8 C17H24N6O4
N-hydroxy-N-[(2R)-5-methyl-2-({N'-[7-(methyloxy)-1,2,4-benzotriazin-3-yl]-hydrazino}-carbonyl)-hexyl]-formamide
—— N-{(1S,2S,4R)-2-azido-1-benzyl-4-[(1S)-1-benzylcarbamoyl-2-methylpropylcarbamoyl]-pentyl}-N',N'-dipropyl-isophthalamide 637024-80-7 C39H51N7O4
N-{(1S,2S,4R)-2-azido-1-benzyl-4-[(1S)-1-benzylcarbamoyl-2-methylpropylcarbamoyl]-pentyl}-N',N'-dipropyl-isophthalamide
—— H-D-Ala-Phe-Ψ(CH2S)-Gly-NH2 118780-14-6 C14H21N3O2S
H-D-Ala-Phe-Ψ(CH2S)-Gly-NH2
—— (+/-)-2t-Brom-cyclopropan-r-carbonsaeure-dimethylamid 17824-40-7 C6H10BrNO
(+/-)-2t-Brom-cyclopropan-r-carbonsaeure-dimethylamid
—— 1338812-11-5 C54H44O15
—— (R)-4-amino-1-(4-methylpiperazin-1-yl)-5-phenylpentan-1-one 1616684-83-3 C16H25N3O
(R)-4-amino-1-(4-methylpiperazin-1-yl)-5-phenylpentan-1-one
—— (R)-2-acetylamino-4-methyl-oct-7-enoic acid methyl ester 1146119-54-1 C12H21NO3
(R)-2-acetylamino-4-methyl-oct-7-enoic acid methyl ester
—— (S)-N-(4-methyl-1-(1-methyl-2-phenethylhydrazineyl)-1-oxopentan-2-yl)-2,3-dihydrobenzo[b][1,4]dioxine-6-carboxamide 1391932-14-1 C24H31N3O4
(S)-N-(4-methyl-1-(1-methyl-2-phenethylhydrazineyl)-1-oxopentan-2-yl)-2,3-dihydrobenzo[b][1,4]dioxine-6-carboxamide
—— (S)-2-((S)-1-((9S,15S)-9,15-dibenzyl-2,2-dimethyl-4,7,10,13-tetraoxo-3-oxa-5,8,11,14-tetraazahexadecan-16-oyl)pyrrolidine-2-carboxamido)-3-phenylpropyl acetate 1374975-58-2 C43H54N6O9
(S)-2-((S)-1-((9S,15S)-9,15-dibenzyl-2,2-dimethyl-4,7,10,13-tetraoxo-3-oxa-5,8,11,14-tetraazahexadecan-16-oyl)pyrrolidine-2-carboxamido)-3-phenylpropyl acetate
—— butyl 2-(4-(4-(cyclobutylamino)-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino)-N-methylphenylsulfonamido)acetate 1192708-53-4 C23H30N6O4S
butyl 2-(4-(4-(cyclobutylamino)-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino)-N-methylphenylsulfonamido)acetate
—— N-(2,6-Dimethyl-phenyl)-2-(2-hydroxy-1,1-bis-hydroxymethyl-ethylamino)-acetamide 845-36-3 C14H22N2O4
N-(2,6-Dimethyl-phenyl)-2-(2-hydroxy-1,1-bis-hydroxymethyl-ethylamino)-acetamide
—— 1608113-29-6 C50H56N6O12
—— 108998-95-4 C45H68N13O10S3*Cl
—— N-[[6-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-azaspiro[2.5]octan2-yl]methyl]furo[2,3-c]pyridine-2-carboxamide 1453268-62-6 C22H26N4O4
N-[[6-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-azaspiro[2.5]octan2-yl]methyl]furo[2,3-c]pyridine-2-carboxamide
—— (+/-)-(2R,3R,5R,1'S)-1-benzyl-2-(1-acetamido-3-methyl)butyl-3-bromoacetyl-pyrrolidine-5-carboxylic acid t-butyl ester 854986-64-4 C25H37BrN2O4
(+/-)-(2R,3R,5R,1'S)-1-benzyl-2-(1-acetamido-3-methyl)butyl-3-bromoacetyl-pyrrolidine-5-carboxylic acid t-butyl ester
—— N-[4-amino-5-(5-iodo-2-isopropyl-4-methoxy-phenoxy)-pyrimidin-2-yl]-2-tert-butylamino-acetamide 1050370-94-9 C20H28IN5O3
N-[4-amino-5-(5-iodo-2-isopropyl-4-methoxy-phenoxy)-pyrimidin-2-yl]-2-tert-butylamino-acetamide
—— 4-[3-(2-cyano-pyrrol-1-yl)-1-(4-methyl-piperidine-1-carbonyl)-propylsulfamoyl]-5-fluoro-indole-1-carboxylic acid tert-butyl ester 1191032-51-5 C28H34FN5O5S
4-[3-(2-cyano-pyrrol-1-yl)-1-(4-methyl-piperidine-1-carbonyl)-propylsulfamoyl]-5-fluoro-indole-1-carboxylic acid tert-butyl ester
—— N-(3-bromo-4-fluorobenzyl)-N-(2-methoxyethyl)-1-methyl-1H-imidazole-4-carboxamide 1262237-79-5 C15H17BrFN3O2
N-(3-bromo-4-fluorobenzyl)-N-(2-methoxyethyl)-1-methyl-1H-imidazole-4-carboxamide
—— 1-(4-fluorobenzyl)-3-furan-2-yl-4-methyl-1H-pyrrole-2-carboxylic acid (2-morpholin-4-ylethyl)-amide 959846-99-2 C23H26FN3O3
1-(4-fluorobenzyl)-3-furan-2-yl-4-methyl-1H-pyrrole-2-carboxylic acid (2-morpholin-4-ylethyl)-amide
—— [Mn(isopropyl methyl ketone semicarbazone)2]SO4 864915-86-6 C12H26MnN6O2*O4S
[Mn(isopropyl methyl ketone semicarbazone)2]SO4
—— diethyl 2-(4,10-diethoxy-3,11-dioxa-6,8-dithiatridecan-7-ylidene)malonate 1290127-88-6 C20H36O8S2
diethyl 2-(4,10-diethoxy-3,11-dioxa-6,8-dithiatridecan-7-ylidene)malonate
—— t-butyl 1,3-dioxo-1H-pyrazolo<1,2-a>pyrazolidine-5-carboxylate 111709-26-3 C11H16N2O4
t-butyl 1,3-dioxo-1H-pyrazolo<1,2-a>pyrazolidine-5-carboxylate
—— LIAPEA 207345-04-8 C28H48N6O9
LIAPEA
—— ethyl 2-hydroxy-2-(methyl-d3)propanoate-3,3,3-d3 1034976-71-0 C6H12O3
ethyl 2-hydroxy-2-(methyl-d3)propanoate-3,3,3-d3
—— 2-methyl-4-morpholino-5-isopropyl-3(2H)-pyridazinone 78920-19-1 C12H21N3O2
2-methyl-4-morpholino-5-isopropyl-3(2H)-pyridazinone
—— (RS)-N-(4-carbamimidoyl-2-methylcarbamoylmethoxy-benzyl)-2-(2,6-difluoro-4-methoxy-phenyl)-2-methoxy-acetamide hydrochloride 701266-17-3 C21H24F2N4O5*ClH
(RS)-N-(4-carbamimidoyl-2-methylcarbamoylmethoxy-benzyl)-2-(2,6-difluoro-4-methoxy-phenyl)-2-methoxy-acetamide hydrochloride
—— 2-diazo-3-(1-diethylcarbamoylcyclopropyl)-3-oxopropionic acid ethyl ester 190900-58-4 C13H19N3O4
2-diazo-3-(1-diethylcarbamoylcyclopropyl)-3-oxopropionic acid ethyl ester
—— DL-2-(p-Benzyloxyphenyl)glycinoctylesterhydrochlorid 126746-16-5 C23H31NO3*ClH
DL-2-(p-Benzyloxyphenyl)glycinoctylesterhydrochlorid
—— (S)-1,1,1-trifluoro-2-methyl-3-oxopropan-2-yl acetate 1425924-49-7 C6H7F3O3
(S)-1,1,1-trifluoro-2-methyl-3-oxopropan-2-yl acetate
—— [(E)-3-dicyclohexylboranylprop-2-enyl] acetate 209607-10-3 C17H29BO2
[(E)-3-dicyclohexylboranylprop-2-enyl] acetate
—— Acetic acid (3aR,5R,6R,6aS)-5-acetoxymethyl-2-oxo-hexahydro-furo[2,3-d]oxazol-6-yl ester 81026-83-7 C10H13NO7
Acetic acid (3aR,5R,6R,6aS)-5-acetoxymethyl-2-oxo-hexahydro-furo[2,3-d]oxazol-6-yl ester
—— 4-{[4-methyl-3-(4-pyridin-2-yl-pyrimidin-2-ylamino)-phenyl-carbamoyl]-methyl}-piperazine-1-carboxylic acid ethyl ester 881676-23-9 C25H29N7O3
4-{[4-methyl-3-(4-pyridin-2-yl-pyrimidin-2-ylamino)-phenyl-carbamoyl]-methyl}-piperazine-1-carboxylic acid ethyl ester
—— 2-(3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamido)-N1-(5-hydroxy-8-(3-hydroxy-1-(isobutylamino)-1-oxopropan-2-ylamino)-2,7-dimethyl-8-oxooctan-4-yl)succinamide 881009-64-9 C29H51N7O7
2-(3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamido)-N1-(5-hydroxy-8-(3-hydroxy-1-(isobutylamino)-1-oxopropan-2-ylamino)-2,7-dimethyl-8-oxooctan-4-yl)succinamide
—— N-tetrachlorophthaloyl-L-glutamic acid 5-methyl ester 915156-59-1 C14H9Cl4NO6
N-tetrachlorophthaloyl-L-glutamic acid 5-methyl ester
—— 2-{4-[(2R)-hydroxy-3-(2-methylbenzothiazol-5-yloxy)propyl]piperazinyl}-N-(3-quinolyl)acetamide 1082299-27-1 C26H29N5O3S
2-{4-[(2R)-hydroxy-3-(2-methylbenzothiazol-5-yloxy)propyl]piperazinyl}-N-(3-quinolyl)acetamide
—— (S)-N-((S)-9-bromo-5-((2-methylnaphthalen-1-yl)methyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-2-(methylamino)propanamide hydrochloride 1562201-42-6 C25H26BrN3O3*ClH
(S)-N-((S)-9-bromo-5-((2-methylnaphthalen-1-yl)methyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-2-(methylamino)propanamide hydrochloride
—— (2S)-1-benzoyl-2-tert-butyl-3-methyl-5-methylideneimidazolidin-4-one 822521-14-2 C16H20N2O2
(2S)-1-benzoyl-2-tert-butyl-3-methyl-5-methylideneimidazolidin-4-one
—— ethyl {2-acetyl-1-[(6-amino-9-{2-[2-{[3-(2-{2-[(6-amino-9-{2-[2-{[3-(2-{2-[(6-amino-9-{2-[2-{[3-(2-{2-[(6-amino-9-{2-[2-{[3-(2-amino-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]-2-(2-ethoxy-2-oxoethyl)hydrazinyl}-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]-2-(2-ethoxy-2-oxoethyl)hydrazinyl}-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]-2-(2-ethoxy-2-oxoethyl)hydrazinyl}-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]hydrazinyl}acetate 1328885-86-4 C94H121N45O33
ethyl {2-acetyl-1-[(6-amino-9-{2-[2-{[3-(2-{2-[(6-amino-9-{2-[2-{[3-(2-{2-[(6-amino-9-{2-[2-{[3-(2-{2-[(6-amino-9-{2-[2-{[3-(2-amino-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]-2-(2-ethoxy-2-oxoethyl)hydrazinyl}-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]-2-(2-ethoxy-2-oxoethyl)hydrazinyl}-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]-2-(2-ethoxy-2-oxoethyl)hydrazinyl}-2-oxoethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl]methyl}-2-(2-ethoxy-2-oxoethyl)hydrazinyl]-2-oxoethyl}-9H-purin-8-yl)methyl]hydrazinyl}acetate
—— (2S,3S,4S,5S)-2-((S)-1-((S)-1-(tert-butoxycarbonyl)pyrrolidine-2-carboxamido)-2-(ethanoyl-oxy)ethyl)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-3,4-diyl diethanoate 1104734-01-1 C26H36N4O12
(2S,3S,4S,5S)-2-((S)-1-((S)-1-(tert-butoxycarbonyl)pyrrolidine-2-carboxamido)-2-(ethanoyl-oxy)ethyl)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-3,4-diyl diethanoate
—— (2S)-N-[(2S)-1-(2,4-dimethoxyanilino)-4-methylsulfonylbutan-2-yl]-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-(4-methylsulfonylphenyl)ethyl]amino]pentanamide 1190741-93-5 C28H40F3N3O7S2
(2S)-N-[(2S)-1-(2,4-dimethoxyanilino)-4-methylsulfonylbutan-2-yl]-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-(4-methylsulfonylphenyl)ethyl]amino]pentanamide
—— ethyl (E)-2-((3aR,7aR)-3a-hydroxy-7a-methylhexahydro-1H-inden-4(2H)-ylidene)acetate 1372790-24-3 C14H22O3
ethyl (E)-2-((3aR,7aR)-3a-hydroxy-7a-methylhexahydro-1H-inden-4(2H)-ylidene)acetate
—— N-(3-benzyl-4-(3-chlorophenylamino)-2-oxochroman-3-yl)benzamide 1322617-44-6 C29H23ClN2O3
N-(3-benzyl-4-(3-chlorophenylamino)-2-oxochroman-3-yl)benzamide
—— [(7-hydroxy[1,2,4]triazolo[1,5-a]pyridine-8-carbonyl)amino]acetic acid hydrochloride 1262131-72-5 C9H8N4O4*ClH
[(7-hydroxy[1,2,4]triazolo[1,5-a]pyridine-8-carbonyl)amino]acetic acid hydrochloride
—— 4-[2-(2-oxo-2λ<sup>5</sup>-[1,3,2]dioxaphospholan-2-yloxy)-ethyl]-morpholine 39683-73-3 C8H16NO5P
4-[2-(2-oxo-2λ<sup>5</sup>-[1,3,2]dioxaphospholan-2-yloxy)-ethyl]-morpholine
—— N-<(cis-4-Isopropylcyclohexyl)carbonyl>-D-phenylalanine methyl ester 958230-60-9 C20H29NO3
N-<(cis-4-Isopropylcyclohexyl)carbonyl>-D-phenylalanine methyl ester