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哌啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-ethylpiperidine-1-carboxylic acid —— C19H21FN6O3
(3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-ethylpiperidine-1-carboxylic acid
—— (1-aminocyclopropyl)methyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H24FN7O3
(1-aminocyclopropyl)methyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— 6-(Methoxymethyl)-5-[2-[(4-piperidin-4-ylbenzoyl)amino]pyridin-4-yl]oxyindole-1-carboxamide —— C28H29N5O4
6-(Methoxymethyl)-5-[2-[(4-piperidin-4-ylbenzoyl)amino]pyridin-4-yl]oxyindole-1-carboxamide
—— 2,2,2-trifluoroethyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C19H18F4N6O3
2,2,2-trifluoroethyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2-methylpropyl)piperidine-1-carboxylic acid —— C21H25FN6O3
(3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2-methylpropyl)piperidine-1-carboxylic acid
—— (1-aminocyclopropyl)methyl (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H24FN7O3
(1-aminocyclopropyl)methyl (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— oxetan-3-yl (3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C20H21FN6O4
oxetan-3-yl (3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— 5-[2-[[4-(1-Ethylpiperidin-4-yl)benzoyl]amino]pyridin-4-yl]oxy-6-(3-fluoropropoxy)-2-methylindole-1-carboxamide —— C32H36FN5O4
5-[2-[[4-(1-Ethylpiperidin-4-yl)benzoyl]amino]pyridin-4-yl]oxy-6-(3-fluoropropoxy)-2-methylindole-1-carboxamide
—— (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-[[1-(cyanomethyl)cyclopropyl]methyl]piperidine-1-carboxylic acid —— C23H24FN7O3
(3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-[[1-(cyanomethyl)cyclopropyl]methyl]piperidine-1-carboxylic acid
—— [1-(cyanomethyl)cyclopropyl]methyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C23H24FN7O3
[1-(cyanomethyl)cyclopropyl]methyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(2-morpholin-4-ylethyl)piperidine-1-carboxylic acid —— C23H28FN7O4
(3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(2-morpholin-4-ylethyl)piperidine-1-carboxylic acid
—— 1,1,1-trifluoropropan-2-yl (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate —— C20H20F4N6O3
1,1,1-trifluoropropan-2-yl (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate
—— 6-(Difluoromethoxy)-5-[2-[[4-[(4-hydroxypiperidin-1-yl)methyl]benzoyl]amino]pyridin-4-yl]oxy-2-methylindole-1-carboxamide —— C29H29F2N5O5
6-(Difluoromethoxy)-5-[2-[[4-[(4-hydroxypiperidin-1-yl)methyl]benzoyl]amino]pyridin-4-yl]oxy-2-methylindole-1-carboxamide
—— oxan-4-yl (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C22H25FN6O4
oxan-4-yl (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— cyclopentyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C22H25FN6O3
cyclopentyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— 2,2-dimethylpropyl (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate —— C22H27FN6O3
2,2-dimethylpropyl (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate
—— (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxylic acid —— C23H26FN7O4
(3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxylic acid
—— (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2,2-difluoroethyl)piperidine-1-carboxylic acid —— C19H19F3N6O3
(3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2,2-difluoroethyl)piperidine-1-carboxylic acid
—— but-3-ynyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H21FN6O3
but-3-ynyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— cyclopropylmethyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H23FN6O3
cyclopropylmethyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(1-cyclopropylethyl)piperidine-1-carboxylic acid —— C22H25FN6O3
(3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(1-cyclopropylethyl)piperidine-1-carboxylic acid
—— 2-methylpropyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H25FN6O3
2-methylpropyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3-methyloxetan-3-yl)methyl (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C22H25FN6O4
(3-methyloxetan-3-yl)methyl (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (1-methylpiperidin-4-yl)methyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C24H30FN7O3
(1-methylpiperidin-4-yl)methyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(cyclopropylmethyl)piperidine-1-carboxylic acid —— C21H23FN6O3
(3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(cyclopropylmethyl)piperidine-1-carboxylic acid
—— (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-ethylpiperidine-1-carboxylic acid —— C19H21FN6O3
(3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-ethylpiperidine-1-carboxylic acid
—— (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid —— C22H27FN6O3
(3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid
—— cyclopropylmethyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H23FN6O3
cyclopropylmethyl (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid —— C22H27FN6O3
(3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid
—— (1-methylpiperidin-4-yl) (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C23H28FN7O3
(1-methylpiperidin-4-yl) (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— tert-butyl (3R,4S)-3-(3-anilino-4-carbamoylpyrazol-1-yl)-4-cyanopiperidine-1-carboxylate —— C21H26N6O3
tert-butyl (3R,4S)-3-(3-anilino-4-carbamoylpyrazol-1-yl)-4-cyanopiperidine-1-carboxylate
—— 1,1,1-Trifluoropropan-2-yl 3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate —— C20H20F4N6O3
1,1,1-Trifluoropropan-2-yl 3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate
—— ethyl (3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C19H21FN6O3
ethyl (3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— 2-methylpropyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H25FN6O3
2-methylpropyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(1-cyclopropylethyl)piperidine-1-carboxylic acid —— C22H25FN6O3
(3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(1-cyclopropylethyl)piperidine-1-carboxylic acid
—— tert-butyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C21H25FN6O3
tert-butyl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2-methoxyethyl)piperidine-1-carboxylic acid —— C20H23FN6O4
(3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2-methoxyethyl)piperidine-1-carboxylic acid
—— oxan-4-yl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate —— C22H25FN6O4
oxan-4-yl (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyanopiperidine-1-carboxylate
—— (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-2,3-dicyano-2-(2-methylpropyl)piperidine-1-carboxylic acid —— C22H24FN7O3
(3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-2,3-dicyano-2-(2-methylpropyl)piperidine-1-carboxylic acid
—— (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(1-methylpiperidin-4-yl)piperidine-1-carboxylic acid —— C23H28FN7O3
(3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(1-methylpiperidin-4-yl)piperidine-1-carboxylic acid
—— 4-[4-Carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-3-(dimethylamino)-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid —— C24H32FN7O3
4-[4-Carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-3-(dimethylamino)-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid
—— (3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-[(1-methylcyclopropyl)methyl]piperidine-1-carboxylic acid —— C22H25FN6O3
(3S,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-[(1-methylcyclopropyl)methyl]piperidine-1-carboxylic acid
—— (2-cyano-2-methylpropyl) (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate —— C22H24FN7O3
(2-cyano-2-methylpropyl) (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyanopiperidine-1-carboxylate
—— (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(2,2,2-trifluoroethyl)piperidine-1-carboxylic acid —— C19H18F4N6O3
(3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(2,2,2-trifluoroethyl)piperidine-1-carboxylic acid
—— (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(oxan-4-yl)piperidine-1-carboxylic acid —— C22H25FN6O4
(3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-(oxan-4-yl)piperidine-1-carboxylic acid
—— (3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-ethoxy-2-(2-oxoethyl)piperidine-1-carboxylic acid —— C21H23FN6O5
(3R,4S)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-ethoxy-2-(2-oxoethyl)piperidine-1-carboxylic acid
—— (3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-[2-(dimethylamino)ethyl]piperidine-1-carboxylic acid —— C21H26FN7O3
(3S,4R)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-[2-(dimethylamino)ethyl]piperidine-1-carboxylic acid
—— (3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-[[1-(cyanomethyl)cyclopropyl]methyl]piperidine-1-carboxylic acid —— C23H24FN7O3
(3R,4S)-3-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-4-cyano-2-[[1-(cyanomethyl)cyclopropyl]methyl]piperidine-1-carboxylic acid
—— (3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid —— C22H27FN6O3
(3S,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2,2-dimethylpropyl)piperidine-1-carboxylic acid
—— (3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2-methylpropyl)piperidine-1-carboxylic acid —— C21H25FN6O3
(3R,4R)-4-[4-carbamoyl-3-(4-fluoroanilino)pyrazol-1-yl]-3-cyano-2-(2-methylpropyl)piperidine-1-carboxylic acid