中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
3-[[(2Z,4E)-3-amino-5-(ethylaminooxy)-2-methyl-1-(methylideneamino)hexa-2,4-dienylidene]amino]-N,N-dimethylpiperidine-1-carboxamide |
—— |
C18H32N6O2 |
|
—— |
methyl (2S,4S)-4-[[6-(3,5-dimethyl-1,2-oxazol-4-yl)-2,5-dimethylpyrimidin-4-yl]amino]-2-methylpiperidine-1-carboxylate |
—— |
C19H27N5O3 |
|
—— |
Tert-butyl 6-imino-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C11H18N2O2 |
|
—— |
N-[(E)-3-piperidin-4-ylprop-2-enylidene]methanimidamide |
—— |
C9H15N3 |
|
—— |
[4-[(1-Benzylpiperidin-4-yl)amino]-2-(2,2,2-trifluoroethyl)thieno[2,3-b]pyridin-5-yl]methanol |
—— |
C22H24F3N3OS |
|
—— |
N-[(3S,4S)-1-benzyl-3-phenylmethoxypiperidin-4-yl]-2-(2,2,2-trifluoroethyl)thieno[2,3-b]pyridin-4-amine |
—— |
C28H28F3N3OS |
|
—— |
N-[1-[(2-methylphenyl)methyl]piperidin-4-yl]-6-propylthieno[2,3-d]pyrimidin-4-amine |
—— |
C22H28N4S |
|
—— |
N-[1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl]-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-amine |
—— |
C22H25F3N4S |
|
—— |
3-Chloro-4-[[4-[[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino]piperidin-1-yl]methyl]benzenesulfonamide |
—— |
C20H21ClF3N5O2S2 |
|
—— |
(3R,4R)-1-benzyl-3-N-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-4-N-[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]piperidine-3,4-diamine |
—— |
C26H33F3N6S |
|
—— |
(3S,4S)-3-N,1-dibenzyl-4-N-[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]piperidine-3,4-diamine |
—— |
C27H28F3N5S |
|
—— |
N-((1-benzylpiperidin-4-yl)methyl)-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-amine |
—— |
C21H23F3N4S |
|
—— |
N-[[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]methyl]-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-amine |
—— |
C22H25F3N4OS |
|
—— |
N-[[1-[(2-chlorophenyl)methyl]piperidin-4-yl]methyl]-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-amine |
—— |
C21H22ClF3N4S |
|
—— |
(3S,4S)-1-benzyl-4-N-[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]piperidine-3,4-diamine |
—— |
C20H22F3N5S |
|
—— |
7-(1-Benzylpiperidin-4-yl)-3-(2,2,2-trifluoroethyl)-2-thia-6,7,9,11-tetrazatricyclo[6.3.1.04,12]dodeca-1(11),3,8(12),9-tetraene |
—— |
C21H22F3N5S |
|
—— |
[4-[[4-[[[6-(2,2,2-Trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino]methyl]piperidin-1-yl]methyl]phenyl]methanol |
—— |
C22H25F3N4OS |
|
—— |
N-[1-[[4-(aminomethyl)phenyl]methyl]piperidin-4-yl]-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-amine |
—— |
C21H24F3N5S |
|
—— |
[2-(2,4-Dimethylpyrazol-3-yl)phenyl]-[6-(5-methylpyridin-2-yl)oxy-2-azabicyclo[2.2.1]heptan-2-yl]methanone |
—— |
C24H26N4O2 |
|
—— |
US9611277, Example 32 |
—— |
C23H23N3O3 |
|
—— |
[6-(5-Methylpyridin-2-yl)oxy-2-azabicyclo[2.2.1]heptan-2-yl]-[2-(1,2,4-triazol-4-yl)phenyl]methanone |
—— |
C21H21N5O2 |
|
—— |
(2-Methoxy-6-pyrimidin-2-ylphenyl)-[6-(5-methylpyridin-2-yl)oxy-2-azabicyclo[2.2.1]heptan-2-yl]methanone |
—— |
C24H24N4O3 |
|
—— |
(4R)-3-[2-[[(1S)-1-[4-[(4,4-difluoropiperidin-1-yl)methyl]-3-fluorophenyl]ethyl]amino]pyrimidin-4-yl]-4-[(1R)-1-hydroxyethyl]-1,3-oxazolidin-2-one |
—— |
C23H28F3N5O3 |
|
—— |
(3-Fluoro-2-pyrimidin-2-ylphenyl)-[6-(5-methylpyrimidin-2-yl)oxy-2-azabicyclo[2.2.2]octan-2-yl]methanone |
—— |
C23H22FN5O2 |
|
—— |
US9611277, Example 221 |
—— |
C20H21N7O |
|
—— |
(3-Fluoro-2-pyrimidin-2-ylphenyl)-[6-[(5-methylpyrimidin-2-yl)amino]-2-azabicyclo[2.2.2]octan-2-yl]methanone |
—— |
C23H23FN6O |
|
—— |
(S)-1-(4-((4,4-difluoropiperidin-1-yl)methyl)-3-fluorophenyl)ethanamine |
—— |
C14H19F3N2 |
|
—— |
1-(4-Tert-butyl-3-fluoro-5-methylphenyl)-4-fluoro-4-methylpiperidine |
—— |
C17H25F2N |
|
—— |
(2-Fluoro-6-pyrimidin-2-ylphenyl)-[6-(5-methylpyridin-2-yl)oxy-2-azabicyclo[2.2.1]heptan-2-yl]methanone |
—— |
C23H21FN4O2 |
|
—— |
(7-Ethoxyquinolin-8-yl)-[6-(5-methylpyridin-2-yl)oxy-2-azabicyclo[2.2.1]heptan-2-yl]methanone |
—— |
C24H25N3O3 |
|
—— |
1-(4-Tert-butylphenyl)-3-fluoro-3-methylpiperidine |
—— |
C16H24FN |
|
—— |
1-(4-Tert-butyl-3-methylphenyl)-4-(1,1-difluoroethyl)piperidine |
—— |
C18H27F2N |
|
—— |
methyl-N-[(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-piperidin-2-ylpyrrolidin-3-yl]boronamidic acid |
—— |
C14H26BN5O3S |
|
—— |
[1-[[4-[5-(3-Fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]-4-(morpholine-4-carbonyl)piperidin-4-yl] hydrogen carbonate |
—— |
C32H31FN4O6 |
|
—— |
methyl-N-[(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-(1-methylpiperidin-2-yl)pyrrolidin-3-yl]boronamidic acid |
—— |
C15H28BN5O3S |
|
—— |
[4-Carboxyoxy-1-[[4-[5-(4-ethoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] hydrogen carbonate |
—— |
C24H25N3O8 |
|
—— |
[4-Carboxyoxy-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] 2-phenylethyl carbonate |
—— |
C36H32FN3O7 |
|
—— |
[4-Carboxyoxy-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] pentyl carbonate |
—— |
C33H34FN3O7 |
|
—— |
1-[[4-[5-(2,2-dimethyl-3H-1-benzofuran-5-yl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]-2-methylpiperidine-4,4-dicarboxylic acid |
—— |
C27H29N3O6 |
|
—— |
[4-[(1-Ethylpyrrolidin-2-yl)methylcarbamoyl]-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] hydrogen carbonate |
—— |
C35H38FN5O5 |
|
—— |
1-(4-Tert-butyl-3-methylphenyl)-4-(trifluoromethyl)piperidine |
—— |
C17H24F3N |
|
—— |
[4-(Ethylcarbamoyl)-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] hydrogen carbonate |
—— |
C30H29FN4O5 |
|
—— |
2,2-Dimethyl-1-[[4-[5-[4-(2-methylpropyl)phenyl]-1,2,4-oxadiazol-3-yl]phenyl]methyl]-3-propan-2-yloxycarbonyloxypiperidine-4,4-dicarboxylic acid;2-(1,3-dioxole-4-carbonyl)-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]-5-methyl-4-phenylmethoxycarbonylpiperidine-4-carboxylic acid |
—— |
C72H73FN6O16 |
|
—— |
2,2-Dimethyl-1-[[4-[5-[4-(2-methylpropyl)phenyl]-1,2,4-oxadiazol-3-yl]phenyl]methyl]-3-propan-2-yloxycarbonyloxypiperidine-4,4-dicarboxylic acid |
—— |
C32H39N3O8 |
|
—— |
[4-Carboxyoxy-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] 2-oxopropyl carbonate |
—— |
C31H28FN3O8 |
|
—— |
[4-Carboxyoxy-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] [2-(4-methoxyphenyl)-2-oxoethyl] carbonate |
—— |
C37H32FN3O9 |
|
—— |
[1-[[4-[5-(3-Fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]-4-(pyrrolidine-1-carbonyl)piperidin-4-yl] hydrogen carbonate |
—— |
C32H31FN4O5 |
|
—— |
2-(1,3-Dioxole-4-carbonyl)-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]-5-methyl-4-phenylmethoxycarbonylpiperidine-4-carboxylic acid |
—— |
C40H34FN3O8 |
|
—— |
[4-(Cyclobutylcarbamoyl)-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] hydrogen carbonate |
—— |
C32H31FN4O5 |
|
—— |
[4-(Dimethylcarbamoyl)-1-[[4-[5-(3-fluoro-4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]piperidin-4-yl] ethyl carbonate |
—— |
C32H33FN4O5 |
|