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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[N-(4-amidinobenzoyl)-L-4-nitrophenylalanyl]-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridin-2-acetic acid.trifluoroacetate 220386-57-2 C2HF3O2*C25H25N7O6
5-[N-(4-amidinobenzoyl)-L-4-nitrophenylalanyl]-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridin-2-acetic acid.trifluoroacetate
—— NNC 26-1187 267225-30-9 C39H47N5O3
NNC 26-1187
—— 6-methoxy-3-methoxycarbonyl-2-morpholino-7-(4-pyridylmethyloxy)-4-(3,4,5-trimethoxyphenyl)-1(2H)isoquinolinone 212500-17-9 C31H33N3O9
6-methoxy-3-methoxycarbonyl-2-morpholino-7-(4-pyridylmethyloxy)-4-(3,4,5-trimethoxyphenyl)-1(2H)isoquinolinone
—— [2S,4S] 4-[(3,5-bis-trifluoromethyl-benzyl)-formyl-amino]-2-cyclopropyl-6-trifluoromethyl-3,4-dihydro-2H-quinoline-1-carboxylic acid isopropyl ester 261947-35-7 C27H25F9N2O3
[2S,4S] 4-[(3,5-bis-trifluoromethyl-benzyl)-formyl-amino]-2-cyclopropyl-6-trifluoromethyl-3,4-dihydro-2H-quinoline-1-carboxylic acid isopropyl ester
—— N-Methyl-N-[1-[5-(3,4-difluorophenylmethoxy)pentyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine Hydrogen Fumarate 286440-41-3 C4H4O4*C26H33F2N3OS
N-Methyl-N-[1-[5-(3,4-difluorophenylmethoxy)pentyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine Hydrogen Fumarate
—— N-Methyl-N-[1-[4-[2-(3,4-difluorophenyl)ethoxy]butyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine Hydrogen Fumarate 286440-47-9 C4H4O4*C26H33F2N3OS
N-Methyl-N-[1-[4-[2-(3,4-difluorophenyl)ethoxy]butyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine Hydrogen Fumarate
—— N-(2,6-dichlorobenzoyl)-4-[2,6-dimethoxy-4-(morpholinomethyl)phenyl]-L-phenylalanine 232272-67-2 C29H30Cl2N2O6
N-(2,6-dichlorobenzoyl)-4-[2,6-dimethoxy-4-(morpholinomethyl)phenyl]-L-phenylalanine
—— N-Methyl-N-[1-[4-(3,4-difluorophenylmethoxy)butyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine Hydrogen Fumarate 286440-43-5 C4H4O4*C25H31F2N3OS
N-Methyl-N-[1-[4-(3,4-difluorophenylmethoxy)butyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine Hydrogen Fumarate
—— 4-({5-(benzylamino)-3-chloro-2-[(2-naphthylsulfanyl)methyl]-1H-indol-1-yl}methyl)benzoic acid 241492-89-7 C34H27ClN2O2S
4-({5-(benzylamino)-3-chloro-2-[(2-naphthylsulfanyl)methyl]-1H-indol-1-yl}methyl)benzoic acid
—— 2-[5-amino-6-oxo-2-(4-fluorophenyl)-1,6-dihydro-1-pyrimidinyl]-N-[1-[[5-(α,α-dimethyl-3,4-methylenedioxybenzyl)-1,3,4-oxadiazole-2-yl]carbonyl]-2-methylpropyl]acetamide 251958-28-8 C29H29FN6O6
2-[5-amino-6-oxo-2-(4-fluorophenyl)-1,6-dihydro-1-pyrimidinyl]-N-[1-[[5-(α,α-dimethyl-3,4-methylenedioxybenzyl)-1,3,4-oxadiazole-2-yl]carbonyl]-2-methylpropyl]acetamide
—— N-[3-[2-[Bis(1-methylethyl)amino]ethoxy]-4-methoxyphenyl]-3',5'-bis(methoxycarbonyl)-1,1'-biphenyl-4-carboxamide 282727-17-7 C32H38N2O7
N-[3-[2-[Bis(1-methylethyl)amino]ethoxy]-4-methoxyphenyl]-3',5'-bis(methoxycarbonyl)-1,1'-biphenyl-4-carboxamide
—— Leu Asn Tyr Arg 243121-61-1 C25H40N8O7
Leu Asn Tyr Arg
—— 2-[2-(4-{4-[(R)-1-[(2S,5R)-4-benzyl-2,5-dimethylhexahydropyrazin-1-yl]1(3-hydroxyphenyl)methyl]phenyl}-2H-1,2,3-triazol-2-yl)ethoxy]acetic acid 254113-46-7 C32H37N5O4
2-[2-(4-{4-[(R)-1-[(2S,5R)-4-benzyl-2,5-dimethylhexahydropyrazin-1-yl]1(3-hydroxyphenyl)methyl]phenyl}-2H-1,2,3-triazol-2-yl)ethoxy]acetic acid
—— propyl (1R,2E,4S,5R,9R,11S,12S)-1-methoxy-8,12-dimethyl-11-[(E)-3-(1-methylimidazol-4-yl)prop-2-enoyl]oxy-5-propan-2-yl-15-oxatricyclo[10.2.1.04,9]pentadeca-2,7,13-triene-2-carboxylate 216317-77-0 C31H42N2O6
propyl (1R,2E,4S,5R,9R,11S,12S)-1-methoxy-8,12-dimethyl-11-[(E)-3-(1-methylimidazol-4-yl)prop-2-enoyl]oxy-5-propan-2-yl-15-oxatricyclo[10.2.1.04,9]pentadeca-2,7,13-triene-2-carboxylate
—— N-[3-[2-[bis(1-methylethyl)amino]ethoxy]-4-methoxyphenyl]-3'-isopropoxycarbonyl-1,1'-biphenyl-4-carboxamide 282727-16-6 C32H40N2O5
N-[3-[2-[bis(1-methylethyl)amino]ethoxy]-4-methoxyphenyl]-3'-isopropoxycarbonyl-1,1'-biphenyl-4-carboxamide
—— (2R,3R,4S,5S)-2-{6-(3,3-Dimethyl-butylamino)-2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-purin-9-yl}-5-(3-ethyl-[1,2,4]oxadiazol-5-yl)-tetrahydro-furan-3,4-diol 235415-69-7 C25H36N10O4
(2R,3R,4S,5S)-2-{6-(3,3-Dimethyl-butylamino)-2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-purin-9-yl}-5-(3-ethyl-[1,2,4]oxadiazol-5-yl)-tetrahydro-furan-3,4-diol
—— 2-{3-[(Benzylsulfonyl)amino]-6-Methyl-2-Oxopyridin-1(2h)-Yl}-N-({1-[2-(Tert-Butylamino)-2-Oxoethyl]-4-Methyl-1h-Imidazol-5-Yl}methyl)acetamide 214152-91-7 C26H34N6O5S
2-{3-[(Benzylsulfonyl)amino]-6-Methyl-2-Oxopyridin-1(2h)-Yl}-N-({1-[2-(Tert-Butylamino)-2-Oxoethyl]-4-Methyl-1h-Imidazol-5-Yl}methyl)acetamide
—— 2-(4,6-Dimethyl-2-pyrimidinyloxy)-3-(2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethoxy)-3,3-diphenylpropionic acid 224455-10-1 C32H31N3O5
2-(4,6-Dimethyl-2-pyrimidinyloxy)-3-(2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethoxy)-3,3-diphenylpropionic acid
—— 3-(2-chloro-4-(2-phenylethyl)benzyl)-2-methyl-5-((4-methylbenzene)sulfonylcarbamoyl)indole 245367-87-7 C32H29ClN2O3S
3-(2-chloro-4-(2-phenylethyl)benzyl)-2-methyl-5-((4-methylbenzene)sulfonylcarbamoyl)indole
—— (S)-7-[[N-4-piperidinylpropyl-N-(1H-benzimidazol-2-ylmethyl)]-aminocarbonyl]-2,3,4,5-tetrahydro-4-methyl-3-oxo-1H-1,4-benzodiazepine-2-acetic acid 220437-17-2 C29H36N6O4
(S)-7-[[N-4-piperidinylpropyl-N-(1H-benzimidazol-2-ylmethyl)]-aminocarbonyl]-2,3,4,5-tetrahydro-4-methyl-3-oxo-1H-1,4-benzodiazepine-2-acetic acid
—— 1-(2-Amino-benzothiazol-6-yl)-3-phenylsulphonylamino-2-(4-benzyl-piperidin-1-yl)-propan-1-one 226996-47-0 C28H30N4O3S2
1-(2-Amino-benzothiazol-6-yl)-3-phenylsulphonylamino-2-(4-benzyl-piperidin-1-yl)-propan-1-one
—— N-[(2-hydroxy-2-phenyl)ethyl]-3-{[(1S,2R)-2-(4,5-diphenyloxazol-2-yl)-1-cyclopentyl]methyl}benzamide 262595-40-4 C36H34N2O3
N-[(2-hydroxy-2-phenyl)ethyl]-3-{[(1S,2R)-2-(4,5-diphenyloxazol-2-yl)-1-cyclopentyl]methyl}benzamide
—— 5-(2-(5-Chloro-2-methoxybenzamido)ethyl)-N-(isopropylaminocarbonyl)-2-phenylbenzenesulfonamide 254973-83-6 C26H28ClN3O5S
5-(2-(5-Chloro-2-methoxybenzamido)ethyl)-N-(isopropylaminocarbonyl)-2-phenylbenzenesulfonamide
—— (2S)-2-{[(Z)-1-ethyl-3-oxo-3-phenyl-1-propenyl]amino}-3-(4-{2-[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy}phenyl)propanoic acid 258345-48-1 C32H31FN2O5
(2S)-2-{[(Z)-1-ethyl-3-oxo-3-phenyl-1-propenyl]amino}-3-(4-{2-[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy}phenyl)propanoic acid
—— 4-[({4-[-(3-fluorophenyl)-6-(trifluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]phenyl}sulfonyl)amino]-4-oxobutanoic acid 267235-74-5 C24H17F4N3O5S
4-[({4-[-(3-fluorophenyl)-6-(trifluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]phenyl}sulfonyl)amino]-4-oxobutanoic acid
—— 2-{4-[(2,6-Dichlorobenzoyl)amino]benzyl}3-(2,6-dimethoxyanilino)-3-oxopropanoic acid 263356-12-3 C25H22Cl2N2O6
2-{4-[(2,6-Dichlorobenzoyl)amino]benzyl}3-(2,6-dimethoxyanilino)-3-oxopropanoic acid
—— 1-Cyclopentyl-7-{4-[4-(3-morpholin-4-ylpropyl)piperidin-1-yl]phenylamino}pyrimido[4,5-d]pyrimidin-2(1H)-one 251369-85-4 C29H39N7O2
1-Cyclopentyl-7-{4-[4-(3-morpholin-4-ylpropyl)piperidin-1-yl]phenylamino}pyrimido[4,5-d]pyrimidin-2(1H)-one
—— 3-{4-[3-(8,9-Dihydro-3,5-dithia-4-aza-cyclopenta[f]azulen-4-yl)-propoxy]-phenyl}-2-benzyloxy-propionic acid 265318-18-1 C29H29NO4S2
3-{4-[3-(8,9-Dihydro-3,5-dithia-4-aza-cyclopenta[f]azulen-4-yl)-propoxy]-phenyl}-2-benzyloxy-propionic acid
—— 6-(3-dimethylaminopropylamino)-N-[2-methyl-5-(2-morpholinopyrid-4-ylcarbonylamino)phenyl]pyridine-3-carboxamide 258503-26-3 C28H35N7O3
6-(3-dimethylaminopropylamino)-N-[2-methyl-5-(2-morpholinopyrid-4-ylcarbonylamino)phenyl]pyridine-3-carboxamide
—— 1-[2-Methylcarbamoyl-5-tert-butyl-3-thienyl]-3-[4-(2-morpholin-4-yl-ethoxy)naphthalen-1-yl]-urea 294639-46-6 C27H34N4O4S
1-[2-Methylcarbamoyl-5-tert-butyl-3-thienyl]-3-[4-(2-morpholin-4-yl-ethoxy)naphthalen-1-yl]-urea
—— (2R,S)-3-[3'-(3-iso-propyl-ureido)-biphenyl-3-yl]-2-(4-ethyl-benzenesulfonylamino)-propanoic acid 276258-13-0 C27H31N3O5S
(2R,S)-3-[3'-(3-iso-propyl-ureido)-biphenyl-3-yl]-2-(4-ethyl-benzenesulfonylamino)-propanoic acid
—— rac-3-[3-[(2-guanidino-4-methyl-thiazol-5-yl-carbonyl)-amino]benzenesulphonylamino]-3-phenyl-propionic acid 232593-59-8 C21H22N6O5S2
rac-3-[3-[(2-guanidino-4-methyl-thiazol-5-yl-carbonyl)-amino]benzenesulphonylamino]-3-phenyl-propionic acid
—— (S)-N-[4-[[2-(acetylamino)-6-amino-1-oxohexyl]amino]-2-phenylbenzoyl]-L-α-asparagine 250789-43-6 C25H31N5O6
(S)-N-[4-[[2-(acetylamino)-6-amino-1-oxohexyl]amino]-2-phenylbenzoyl]-L-α-asparagine
—— 2-[N-(2-Chloropyrid-3-oyl)-amino]-3-[N'-(2,6-dichlorobenzoyl)-6-amino-pyrid-3-yl]propionic acid 251458-87-4 C21H15Cl3N4O4
2-[N-(2-Chloropyrid-3-oyl)-amino]-3-[N'-(2,6-dichlorobenzoyl)-6-amino-pyrid-3-yl]propionic acid
—— [7-Ethyl-3-methyl-8-oxamoyl-6-(2-phenylethynylbenzyl)pyrrolo [1,2-a]pyrazin-1-yl]oxyacetic acid 245757-25-9 C29H25N3O5
[7-Ethyl-3-methyl-8-oxamoyl-6-(2-phenylethynylbenzyl)pyrrolo [1,2-a]pyrazin-1-yl]oxyacetic acid
—— 5-[2-hydroxy-4-(2-difluoromethoxy-5-fluorophenyl)-4-methyl-2-trifluoromethyl-valeroylamino]-phthalide 271587-31-6 C22H19F6NO5
5-[2-hydroxy-4-(2-difluoromethoxy-5-fluorophenyl)-4-methyl-2-trifluoromethyl-valeroylamino]-phthalide
—— [7-Ethyl-3-methyl-8-oxamoyl-6-(2-phenyloxybenzyl) pyrrolo [1,2-a]pyrazin-1-yl]oxyacetic acid 245757-27-1 C27H25N3O6
[7-Ethyl-3-methyl-8-oxamoyl-6-(2-phenyloxybenzyl) pyrrolo [1,2-a]pyrazin-1-yl]oxyacetic acid
—— 3,4,7,8-tetrahydro-2,2,8,8-tetramethyl-4-morpholino-6-(3-trifluoromethylphenyl)-2H,6H-benzo[1,2-b:5,4-b']dipyran 292081-92-6 C27H32F3NO3
3,4,7,8-tetrahydro-2,2,8,8-tetramethyl-4-morpholino-6-(3-trifluoromethylphenyl)-2H,6H-benzo[1,2-b:5,4-b']dipyran
—— N-tetradecyl-N,N-dimethyl-N-[(3-trimethoxysilyl) propyl]ammonium bromide 271799-62-3 Br*C22H50NO3Si
N-tetradecyl-N,N-dimethyl-N-[(3-trimethoxysilyl) propyl]ammonium bromide
—— N-(4-amino-2-methyl-6-quinolyl)-2-[(4-methoxymethoxyphenoxy)methyl]benzamide hydrochloride 244218-64-2 C26H25N3O4*ClH
N-(4-amino-2-methyl-6-quinolyl)-2-[(4-methoxymethoxyphenoxy)methyl]benzamide hydrochloride
—— 1-[[(5S,8S)-5-(3,4-dichlorophenyl)-8-(methylamino)-5,6,7,8-tetrahydronaphthalen-2-yl]sulfonyl]piperidin-4-ol 291305-15-2 C22H26Cl2N2O3S
1-[[(5S,8S)-5-(3,4-dichlorophenyl)-8-(methylamino)-5,6,7,8-tetrahydronaphthalen-2-yl]sulfonyl]piperidin-4-ol
—— 4-[3-Chloro-4-(3,3,3-trifluoro-2-hydroxy-2-methylpropanamido)benzenesulfonyl]-n,n-dimethylbenzamide 252017-04-2 C19H18ClF3N2O5S
4-[3-Chloro-4-(3,3,3-trifluoro-2-hydroxy-2-methylpropanamido)benzenesulfonyl]-n,n-dimethylbenzamide
—— Boronic acid, [1,3-phenylenebis(sulfonylimino-3,1-phenylene)]bis- 277295-54-2 C18H18B2N2O8S2
Boronic acid, [1,3-phenylenebis(sulfonylimino-3,1-phenylene)]bis-
—— cyclohexanecarboxylic acid-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-naphthalen-2-ylmethyl-amide 277300-34-2 C31H39N3O2
cyclohexanecarboxylic acid-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-naphthalen-2-ylmethyl-amide
—— (S)-2-{4-[(1H-Imidazol-2-ylmethyl)-amino]-2-naphthalen-1-yl-benzoylamino}-4-methyl-pentanoic acid methyl ester 225938-64-7 C28H30N4O3
(S)-2-{4-[(1H-Imidazol-2-ylmethyl)-amino]-2-naphthalen-1-yl-benzoylamino}-4-methyl-pentanoic acid methyl ester
—— 3-[4-[2-(1-Piperidinyl)ethoxy]phenoxy]-2-cyclohexylbenzo[b]thiophene Hydrochloride 205814-27-3 C27H33NO2S*ClH
3-[4-[2-(1-Piperidinyl)ethoxy]phenoxy]-2-cyclohexylbenzo[b]thiophene Hydrochloride
—— (S)-4-[[4-[(3,5-dimethylphenyl)methoxy]phenyl]sulfonyl]-N-hydroxy-2,2-dimethyl-3-thiomorpholinecarboxamide 250581-19-2 C22H28N2O5S2
(S)-4-[[4-[(3,5-dimethylphenyl)methoxy]phenyl]sulfonyl]-N-hydroxy-2,2-dimethyl-3-thiomorpholinecarboxamide
—— (3R,6S)-4-[4-(2,5-dimethyl-benzyloxy)-benzenesulfonyl]-2,2,6-trimethyl-morpholine-3-carboxylic acid hydroxyamide 259132-71-3 C23H30N2O6S
(3R,6S)-4-[4-(2,5-dimethyl-benzyloxy)-benzenesulfonyl]-2,2,6-trimethyl-morpholine-3-carboxylic acid hydroxyamide
—— N-(2, 4-difluorophenyl)carbonyl-2-(3, 4-methylenedioxyphenyl)-3, 3-diphenylpropylamine 229973-29-9 C29H23F2NO3
N-(2, 4-difluorophenyl)carbonyl-2-(3, 4-methylenedioxyphenyl)-3, 3-diphenylpropylamine
—— 1-Methyl-7-{4-[4-(3-morpholin-4-ylpropyl)piperidin-1-yl]phenylamino}pyrimido[4,5-d]pyrimidin-2(1H)-one 251369-84-3 C25H33N7O2
1-Methyl-7-{4-[4-(3-morpholin-4-ylpropyl)piperidin-1-yl]phenylamino}pyrimido[4,5-d]pyrimidin-2(1H)-one