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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[4-(5-isopropyl-pyridine-2-sulfonylamino)-6-methoxy-5-(2-methoxy-phenoxy)-pyrimidin-2-yl]-pyridine-2-carboxylic acid 285135-05-9 C26H25N5O7S
4-[4-(5-isopropyl-pyridine-2-sulfonylamino)-6-methoxy-5-(2-methoxy-phenoxy)-pyrimidin-2-yl]-pyridine-2-carboxylic acid
—— N-Methyl-N-[1-[3-(4-fluorobenzyloxy)propyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine hydrogen fumarate 286440-28-6 C4H4O4*C24H30FN3OS
N-Methyl-N-[1-[3-(4-fluorobenzyloxy)propyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine hydrogen fumarate
—— (2S)-2-{[(Z)-1-butyl-3-oxo-3-phenyl-1-propenyl]amino}-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl}propanoic acid 258345-63-0 C34H36N2O5
(2S)-2-{[(Z)-1-butyl-3-oxo-3-phenyl-1-propenyl]amino}-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl}propanoic acid
—— ethyl 7-[3-[[(2-bromophenyl)carbamoylamino]methyl]pyrrol-1-yl]-6-chloro-3-oxo-4H-quinoxaline-2-carboxylate 288840-85-7 C23H19BrClN5O4
ethyl 7-[3-[[(2-bromophenyl)carbamoylamino]methyl]pyrrol-1-yl]-6-chloro-3-oxo-4H-quinoxaline-2-carboxylate
—— TAK-622 216260-16-1 C27H21F6N3O2
TAK-622
—— N-Methyl-N-[1-[2-[2-(4-fluorophenyl)ethoxy]ethyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine 286440-38-8 C24H30FN3OS
N-Methyl-N-[1-[2-[2-(4-fluorophenyl)ethoxy]ethyl]-4-piperidyl]-4H-3,1-benzothiazin-2-amine
—— N-[[(3E)-3-cyanomethylene-2,6,6-trimethyl-1-cyclohexen-1-yl]carbonyl]-4-[(2,6-dichlorobenzoyl)amino]-L-phenylalanine 279240-14-1 C28H27Cl2N3O4
N-[[(3E)-3-cyanomethylene-2,6,6-trimethyl-1-cyclohexen-1-yl]carbonyl]-4-[(2,6-dichlorobenzoyl)amino]-L-phenylalanine
—— 3-{3-[4-(2-t-Butyl-6-trifluoromethylpyrimidin-4-yl-)piperazin-1-yl]propylmercapto}-4-methyl-5-phenyl-1,2,4-(4H)-triazole 219600-01-8 C25H32F3N7S
3-{3-[4-(2-t-Butyl-6-trifluoromethylpyrimidin-4-yl-)piperazin-1-yl]propylmercapto}-4-methyl-5-phenyl-1,2,4-(4H)-triazole
—— (2S,3S,4R,5R)-2-(3-Ethyl-[1,2,4]oxadiazol-5-yl)-5-{6-(1-ethyl-propylamino)-2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-purin-9-yl}-tetrahydro-furan-3,4-diol 235415-05-1 C24H34N10O4
(2S,3S,4R,5R)-2-(3-Ethyl-[1,2,4]oxadiazol-5-yl)-5-{6-(1-ethyl-propylamino)-2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-purin-9-yl}-tetrahydro-furan-3,4-diol
—— N-[2-(Benzo[1,3]dioxol-5-yl)-3-hydroxy-4-oxo-4H-chromen-6-yl]-4-bromobenzenesulfonamide 260063-95-4 C22H14BrNO7S
N-[2-(Benzo[1,3]dioxol-5-yl)-3-hydroxy-4-oxo-4H-chromen-6-yl]-4-bromobenzenesulfonamide
—— N-[(1-carboxymethyl)cyclopentaneacetyl]-O-[(2,6-dichlorophenyl)methyl]-L-tyrosine 279240-04-9 C25H27Cl2NO6
N-[(1-carboxymethyl)cyclopentaneacetyl]-O-[(2,6-dichlorophenyl)methyl]-L-tyrosine
—— 4-bromo-N-[2-(3,4-dihydroxyphenyl)-3-hydroxy-4-oxo-4H-chromen-6-yl]benzenesulfonamide 260063-42-1 C21H14BrNO7S
4-bromo-N-[2-(3,4-dihydroxyphenyl)-3-hydroxy-4-oxo-4H-chromen-6-yl]benzenesulfonamide
—— N-[3-(4-diethylaminomethylbenzamido)-4-methylphenyl]-2-morpholinopyridine-4-carboxamide 263268-75-3 C29H35N5O3
N-[3-(4-diethylaminomethylbenzamido)-4-methylphenyl]-2-morpholinopyridine-4-carboxamide
—— N-(4, 5-dichlorophenyl)carbonyl-2-(3, 4-methylenedioxyphenyl)-3, 3-diphenylpropylamine 229973-34-6 C29H23Cl2NO3
N-(4, 5-dichlorophenyl)carbonyl-2-(3, 4-methylenedioxyphenyl)-3, 3-diphenylpropylamine
—— (6,7-Dichloro-3-pyridin-2-yl-quinoxalin-2-yl)-(1-phenyl-4-piperidin-1-yl-butyl)-amine 239095-27-3 C28H29Cl2N5
(6,7-Dichloro-3-pyridin-2-yl-quinoxalin-2-yl)-(1-phenyl-4-piperidin-1-yl-butyl)-amine
—— 3-{4-[1-(8,9-Dihydro-3,5-dithia-4-aza-cyclopenta[f]azulen-4-yl)-methoxy]-phenyl}-2-benzyloxy-propionic acid 265318-15-8 C27H25NO4S2
3-{4-[1-(8,9-Dihydro-3,5-dithia-4-aza-cyclopenta[f]azulen-4-yl)-methoxy]-phenyl}-2-benzyloxy-propionic acid
—— 2-(2-butoxyphenyl)-7-((2-(4-cyanophenylmethyl)-imidazol-5-yl)-1-oxo-ethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine 280775-13-5 C29H30N6O2
2-(2-butoxyphenyl)-7-((2-(4-cyanophenylmethyl)-imidazol-5-yl)-1-oxo-ethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine
—— (2-bromophenyl)[2-chloro-4-(E-((2-tetrahydroisoquinolinyl)carbonyl)ethenyl)phenyl]sulfide 280748-92-7 C24H19BrClNOS
(2-bromophenyl)[2-chloro-4-(E-((2-tetrahydroisoquinolinyl)carbonyl)ethenyl)phenyl]sulfide
—— 4-{4-[1-(3-Chlorobenzylamino)-2,2-dicyanovinyl]-1-piperazinyl}-6,7-dimethoxyquinazoline 245449-73-4 C25H24ClN7O2
4-{4-[1-(3-Chlorobenzylamino)-2,2-dicyanovinyl]-1-piperazinyl}-6,7-dimethoxyquinazoline
—— 3(S)-(Pyrimidin-5-yl)-9-(5,6,7,8-tetrahydro[1,8]naphthyridin-2-yl)-nonanoic acid 227753-43-7 C21H28N4O2
3(S)-(Pyrimidin-5-yl)-9-(5,6,7,8-tetrahydro[1,8]naphthyridin-2-yl)-nonanoic acid
—— 2-trifluoroacetamido-3-(4-trifluoromethoxyphenyl)-6-benzoyl-imidazo[1,2-a]pyridine 251367-63-2 C23H13F6N3O3
2-trifluoroacetamido-3-(4-trifluoromethoxyphenyl)-6-benzoyl-imidazo[1,2-a]pyridine
—— (R,S)-[1-(4'-Chlorobiphenyl-4-sulfonylamino)-2-(1H-indol-3-yl)-ethyl]phosphonic Acid 254886-90-3 C22H20ClN2O5PS
(R,S)-[1-(4'-Chlorobiphenyl-4-sulfonylamino)-2-(1H-indol-3-yl)-ethyl]phosphonic Acid
—— 1-Cyclopropyl-7-fluoro-8-[4-(4-fluoroanilino)piperidino]-4-oxo-1,4-dihydrobenzo[b][1,8]-naphthyridine-3-carboxylic Acid 278796-06-8 C27H24F2N4O3
1-Cyclopropyl-7-fluoro-8-[4-(4-fluoroanilino)piperidino]-4-oxo-1,4-dihydrobenzo[b][1,8]-naphthyridine-3-carboxylic Acid
—— 1-[4-[2-(1-piperidinyl)acetylamido]phenoxy]-2-(4-methoxyphenyl)-6-hydroxynaphthalene 205752-26-7 C30H30N2O4
1-[4-[2-(1-piperidinyl)acetylamido]phenoxy]-2-(4-methoxyphenyl)-6-hydroxynaphthalene
—— N-[5-{[amino(2-thienyl)methylidene]amino}-2-(1H-pyrrol-1-yl)benzyl]-5-(1,2-dithiolan-3-yl)pentanamide 299189-09-6 C24H28N4OS3
N-[5-{[amino(2-thienyl)methylidene]amino}-2-(1H-pyrrol-1-yl)benzyl]-5-(1,2-dithiolan-3-yl)pentanamide
—— 1-(4-Cyanobenzyl)-5-[1-(2-hydroxy-2-(adamant-1-yl)ethyl)-2-oxo-piperazin-4-yl-methyl]imidazole 291751-11-6 C28H35N5O2
1-(4-Cyanobenzyl)-5-[1-(2-hydroxy-2-(adamant-1-yl)ethyl)-2-oxo-piperazin-4-yl-methyl]imidazole
—— 2-methoxy-N-(2-methyl-1H-benzimidazol-4-yl)-4-(2,3,4,5-tetrahydro-5-oxo-1H-1-benzazepin-1-yl)carbonylbenzamide 233262-78-7 C27H24N4O4
2-methoxy-N-(2-methyl-1H-benzimidazol-4-yl)-4-(2,3,4,5-tetrahydro-5-oxo-1H-1-benzazepin-1-yl)carbonylbenzamide
—— 1-(1-Benzyl-1H-indol-4-yl)-4-(2-(6-chloro-1H-indol-3-yl)ethyl)piperazine 252978-07-7 C29H29ClN4
1-(1-Benzyl-1H-indol-4-yl)-4-(2-(6-chloro-1H-indol-3-yl)ethyl)piperazine
—— 2-[(4'-Methoxy[1,1'-biphenyl]-4-yl)sulfonyl]amino-4-hydroxy-5-(phenylamino)-pentanoic acid 291540-88-0 C24H26N2O6S
2-[(4'-Methoxy[1,1'-biphenyl]-4-yl)sulfonyl]amino-4-hydroxy-5-(phenylamino)-pentanoic acid
—— (cis)-4-[2-([(2S)-1-(1,3-benzoxazol-2-yl)-2-piperidinyl]carbonylamino)ethyl]-N1-isopropyl-3,5-dimethyl-1-piperazinecarboxamide 256518-28-2 C25H38N6O3
(cis)-4-[2-([(2S)-1-(1,3-benzoxazol-2-yl)-2-piperidinyl]carbonylamino)ethyl]-N1-isopropyl-3,5-dimethyl-1-piperazinecarboxamide
—— 5-(4-chlorophenylcarbonyl)amino-3-phenylsulfonyl-2,3-dihydro-1,1-dioxidebenzo[b]thiophene 246171-52-8 C21H16ClNO5S2
5-(4-chlorophenylcarbonyl)amino-3-phenylsulfonyl-2,3-dihydro-1,1-dioxidebenzo[b]thiophene
—— N-hydroxy-1-{4-[4-(3-methoxyphenyl)-3-methylphenyl]piperidin-1-ylsulphonyl}cyclobutanecarboxamide 227304-53-2 C24H30N2O5S
N-hydroxy-1-{4-[4-(3-methoxyphenyl)-3-methylphenyl]piperidin-1-ylsulphonyl}cyclobutanecarboxamide
—— (5S,8S)-5-(3,4-dichlorophenyl)-N-(1,3-dihydroxypropan-2-yl)-8-(methylamino)-5,6,7,8-tetrahydronaphthalene-2-sulfonamide 291305-17-4 C20H24Cl2N2O4S
(5S,8S)-5-(3,4-dichlorophenyl)-N-(1,3-dihydroxypropan-2-yl)-8-(methylamino)-5,6,7,8-tetrahydronaphthalene-2-sulfonamide
—— 2(R)-1-[4-(biphenyl-4-yl)oxybenzenesulfonyl]-N-hydroxy-piperidine-2-carboxamide 215921-24-7 C24H24N2O5S
2(R)-1-[4-(biphenyl-4-yl)oxybenzenesulfonyl]-N-hydroxy-piperidine-2-carboxamide
—— 5-(4-Fluorophenyl)-2-[2-(4-methylsulfonylphenyl)ethylthio]-4-(4-pyridyl)imidazole 262589-67-3 C23H20FN3O2S2
5-(4-Fluorophenyl)-2-[2-(4-methylsulfonylphenyl)ethylthio]-4-(4-pyridyl)imidazole
—— 2-(S)-t-butoxycarbonylamino-3-[4'-(1''-trimethylsilylethyloxycarbonyl-1''-methyl)ethyl]benzenepropanoic acid 228410-26-2 C23H37NO6Si
2-(S)-t-butoxycarbonylamino-3-[4'-(1''-trimethylsilylethyloxycarbonyl-1''-methyl)ethyl]benzenepropanoic acid
—— 5-Propyl-5-phenyl-2-(6-chloro-3-methoxy-2-phenylquinolin-4-yl)-imidazoline 298689-10-8 C28H26ClN3O
5-Propyl-5-phenyl-2-(6-chloro-3-methoxy-2-phenylquinolin-4-yl)-imidazoline
—— N-(2,4,4-Trimethyl-1,2,3,4-tetrahydroisoquinolin-5-yl)-5-bromo-4-ethoxy-2-methoxybenzamide 259146-01-5 C22H27BrN2O3
N-(2,4,4-Trimethyl-1,2,3,4-tetrahydroisoquinolin-5-yl)-5-bromo-4-ethoxy-2-methoxybenzamide
—— N-(4-chlorobenzyl)-8-(2-hydroxyethoxy)-6-(3-hydroxypropyl)-1-methyl-4-oxo-1,4-dihydro-3-quinolinecarboxamide 281650-69-9 C23H25ClN2O5
N-(4-chlorobenzyl)-8-(2-hydroxyethoxy)-6-(3-hydroxypropyl)-1-methyl-4-oxo-1,4-dihydro-3-quinolinecarboxamide
—— 1-N-(n-Butylsulfonyl)-4-phenyl-4-(3-(2-methoxyphenyl)-3-oxo-2-azaprop-1-yl)piperidine 266341-43-9 C24H32N2O4S
1-N-(n-Butylsulfonyl)-4-phenyl-4-(3-(2-methoxyphenyl)-3-oxo-2-azaprop-1-yl)piperidine
—— (2R,5R)-1-[4-(2,5-DIFLUORO-BENZYLOXY)-BENZENESULFONYL]-5-HYDROXY-PIPERIDINE-2-CARBOXYLIC ACID HYDROXYAMIDE 258860-90-1 C19H20F2N2O6S
(2R,5R)-1-[4-(2,5-DIFLUORO-BENZYLOXY)-BENZENESULFONYL]-5-HYDROXY-PIPERIDINE-2-CARBOXYLIC ACID HYDROXYAMIDE
—— (2S)-N2-{(3S)-1-[3-(Aminocarbonyl)phenylmethyl]pyrrolidin-3-yl}-1-(1,3-benzoxazol-2-yl)-2-piperidinecarboxamide 256526-57-5 C25H29N5O3
(2S)-N2-{(3S)-1-[3-(Aminocarbonyl)phenylmethyl]pyrrolidin-3-yl}-1-(1,3-benzoxazol-2-yl)-2-piperidinecarboxamide
—— N-(2,4,4-Trimethyl-1,2,3,4-tetrahydroisoquinolin-5-yl)-4-ethoxy-2-methoxy-5-trifluoromethylbenzamide 259146-05-9 C23H27F3N2O3
N-(2,4,4-Trimethyl-1,2,3,4-tetrahydroisoquinolin-5-yl)-4-ethoxy-2-methoxy-5-trifluoromethylbenzamide
—— N-(4-{1-[2-(2-oxo-2,3-dihydrobenzooxazol-6-sulfinyl) ethyl]piperidin-4-ylmethyl}phenyl) acetamide 253450-24-7 C23H27N3O4S
N-(4-{1-[2-(2-oxo-2,3-dihydrobenzooxazol-6-sulfinyl) ethyl]piperidin-4-ylmethyl}phenyl) acetamide
—— 4'-[2-(Diethylamino)ethoxy]-2,6-diethoxybenzanilide Hydrochloride 253338-80-6 C23H32N2O4*ClH
4'-[2-(Diethylamino)ethoxy]-2,6-diethoxybenzanilide Hydrochloride
—— 3,7-bis(2-fluorophenyl)-2-(4-methylthiazol-2-ylmethoxy)pyrazolo[1,5-d][1,2,4]triazine 265643-40-1 C22H15F2N5OS
3,7-bis(2-fluorophenyl)-2-(4-methylthiazol-2-ylmethoxy)pyrazolo[1,5-d][1,2,4]triazine
—— N-hydroxy-2(R)-[(1H-indol-5-ylmethyl)-(4-methoxybenzenesulfonyl)amino]-3-methylbutyramide 279254-35-2 C21H25N3O5S
N-hydroxy-2(R)-[(1H-indol-5-ylmethyl)-(4-methoxybenzenesulfonyl)amino]-3-methylbutyramide
—— 4-(3-Difluoromethoxy-4-methoxyphenyl)-2-(2-phenyl-2-oxoethyl)-2H-phthalazin-1-one 234780-16-6 C24H18F2N2O4
4-(3-Difluoromethoxy-4-methoxyphenyl)-2-(2-phenyl-2-oxoethyl)-2H-phthalazin-1-one
—— 5-Isobutyl-5-phenyl-2-(3-methoxy-2-phenylquinolin-4-yl)-imidazoline 298688-97-8 C29H29N3O
5-Isobutyl-5-phenyl-2-(3-methoxy-2-phenylquinolin-4-yl)-imidazoline
—— 1-(3,5-dichloropyridin-4-ylmethyl)-6-methoxy-5-(tetrahydropyran-2-yl-methoxy)-phthalazine 228869-18-9 C21H21Cl2N3O3
1-(3,5-dichloropyridin-4-ylmethyl)-6-methoxy-5-(tetrahydropyran-2-yl-methoxy)-phthalazine