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中文名称 英文名称 CAS号 化学式 结构式图片
—— [3,5,3",5"-Tetrachloro-5'-(8-phenyl-octylcarbamoyl)-[1,1';3',1"]terphenyl-2'-yloxy]acetic acid 251476-58-1 C35H33Cl4NO4
[3,5,3",5"-Tetrachloro-5'-(8-phenyl-octylcarbamoyl)-[1,1';3',1"]terphenyl-2'-yloxy]acetic acid
—— N-(2-fluorobenzyl)-1-(4-aminomethylphenyl)-5-[4-(3-thienyl)benzyl]-2,4-dioxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepine-3-acetamide hydrochloride 264915-52-8 C36H31FN4O3S*ClH
N-(2-fluorobenzyl)-1-(4-aminomethylphenyl)-5-[4-(3-thienyl)benzyl]-2,4-dioxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepine-3-acetamide hydrochloride
—— (2R,3R)-3-[4-(4-cyanophenyl)thiazol-2-yl]-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)-2-[[p-[(3RS-hydroxy)-1-pyrrolidinylmethyl]benzoyloxy]methoxy]butane 251295-40-6 C35H32F2N6O4S
(2R,3R)-3-[4-(4-cyanophenyl)thiazol-2-yl]-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)-2-[[p-[(3RS-hydroxy)-1-pyrrolidinylmethyl]benzoyloxy]methoxy]butane
—— (2R)-N-(1-benzylpiperidin-4-yl)-3-cyclohexylmethylthio-((4R)-3-(3,3-dimethyl-1,2-dioxobutyl)thiazolidin-4-ylcarbonylamino)propanamide · hydrochloride 255735-60-5 C32H48N4O4S2*ClH
(2R)-N-(1-benzylpiperidin-4-yl)-3-cyclohexylmethylthio-((4R)-3-(3,3-dimethyl-1,2-dioxobutyl)thiazolidin-4-ylcarbonylamino)propanamide · hydrochloride
—— (2S)-3-[4-({[4-(Aminocarbonyl)-1-piperidinyl]carbonyl}oxy)phenyl]-2-({(2S)-2-[(dibenzo[b,d]furan-4-ylcarbonyl)amino]-4-methylpentanoyl}amino) propanoic acid 278598-54-2 C35H38N4O8
(2S)-3-[4-({[4-(Aminocarbonyl)-1-piperidinyl]carbonyl}oxy)phenyl]-2-({(2S)-2-[(dibenzo[b,d]furan-4-ylcarbonyl)amino]-4-methylpentanoyl}amino) propanoic acid
—— 3-[7-[(benzimidazol-2-ylamino)methyl]-1-methyl-6,8-difluoroquinoline-4-one-3-ylcarbonylamino]-2-((2,4,6-trimethylphenyl)sulfonylamino)propionic acid 208580-66-9 C31H30F2N6O6S
3-[7-[(benzimidazol-2-ylamino)methyl]-1-methyl-6,8-difluoroquinoline-4-one-3-ylcarbonylamino]-2-((2,4,6-trimethylphenyl)sulfonylamino)propionic acid
—— (1S,3R,7S,8S,8aR)-1,2,3,7,8,8a-Hexahydro-3,7-dimethyl-8-(2-((4R,6R)-tetrahydro-4-(2-((2-hydroxyethyl)amino)-2-oxoethyl)-3-((4-hydroxy-3-methoxyphenyl)methyl)-2-oxo-2H-1,3-oxazin-6-yl)ethyl)-1-naphthalenyl (2S)-2-methylbutanoate 288323-74-0 C35H50N2O8
(1S,3R,7S,8S,8aR)-1,2,3,7,8,8a-Hexahydro-3,7-dimethyl-8-(2-((4R,6R)-tetrahydro-4-(2-((2-hydroxyethyl)amino)-2-oxoethyl)-3-((4-hydroxy-3-methoxyphenyl)methyl)-2-oxo-2H-1,3-oxazin-6-yl)ethyl)-1-naphthalenyl (2S)-2-methylbutanoate
—— 3-[7-[(pyridin-2-ylamino)methyl]-1-methyl-6,8-difluoroquinoline-4-one-3-ylcarbonylamino]-2-((2,4,6-trimethylphenyl)sulfonylamino)propionic acid 208580-70-5 C29H29F2N5O6S
3-[7-[(pyridin-2-ylamino)methyl]-1-methyl-6,8-difluoroquinoline-4-one-3-ylcarbonylamino]-2-((2,4,6-trimethylphenyl)sulfonylamino)propionic acid
—— (2R,S)-3-[3'-(3-(pyridin-2-yl-methyl)ureido)-biphenyl-4-yl]-2-[2,4,6-trimethylbenzenesulfonylamino]-propanoic acid 276257-78-4 C31H32N4O5S
(2R,S)-3-[3'-(3-(pyridin-2-yl-methyl)ureido)-biphenyl-4-yl]-2-[2,4,6-trimethylbenzenesulfonylamino]-propanoic acid
—— N-[2-(Benzo[1,3]dioxol-5-yl)-3-hydroxy-4-oxo-4H-chromen-6-yl]-4-(4-morpholinyl)-3-nitrobenzenesulfonamide 260064-14-0 C26H21N3O10S
N-[2-(Benzo[1,3]dioxol-5-yl)-3-hydroxy-4-oxo-4H-chromen-6-yl]-4-(4-morpholinyl)-3-nitrobenzenesulfonamide
—— n-(4-(2-benzoyl-4-hydroxy-5-isopropyl-phenoxy)-3,5-dibromo-phenyl)oxamic acid methyl ester 258819-87-3 C25H21Br2NO6
n-(4-(2-benzoyl-4-hydroxy-5-isopropyl-phenoxy)-3,5-dibromo-phenyl)oxamic acid methyl ester
—— 4-{3-benzoyl-5-(benzyloxy)-2-[(2-naphthyloxy)methyl]-1H-indol-1-yl}butanoic acid 241493-18-5 C37H31NO5
4-{3-benzoyl-5-(benzyloxy)-2-[(2-naphthyloxy)methyl]-1H-indol-1-yl}butanoic acid
—— (2S)-2-({(Z)-1-ethyl-3-oxo-3-[4-(trifluoromethyl)phenyl]-1-propenyl}amino)-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl}propanoic acid 258345-58-3 C33H31F3N2O5
(2S)-2-({(Z)-1-ethyl-3-oxo-3-[4-(trifluoromethyl)phenyl]-1-propenyl}amino)-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl}propanoic acid
—— 6-(2-chlorophenyl)-7,8,9,10-tetrahydro-1-methyl-9-[2-(2-trifluoromethylphenyl)-1-thioxoethyl]-4H-pyrido[4',3';4,5]thieno[3,2-f][1,2,4]triazolo[3,2-a][1,4]diazepine 252754-63-5 C27H21ClF3N5S2
6-(2-chlorophenyl)-7,8,9,10-tetrahydro-1-methyl-9-[2-(2-trifluoromethylphenyl)-1-thioxoethyl]-4H-pyrido[4',3';4,5]thieno[3,2-f][1,2,4]triazolo[3,2-a][1,4]diazepine
—— (2S)-N2-{(3S)-1-[6-Methoxy-2-phenylquinolin-4-ylcarbonyl]pyrrolidin-3-yl}-1-(1,3-benzoxazol-2-yl)-2-piperidinecarboxamide 256526-37-1 C34H33N5O4
(2S)-N2-{(3S)-1-[6-Methoxy-2-phenylquinolin-4-ylcarbonyl]pyrrolidin-3-yl}-1-(1,3-benzoxazol-2-yl)-2-piperidinecarboxamide
—— ethyl 7-[3-[[(4-bromophenyl)carbamoylamino]methyl]pyrrol-1-yl]-6-chloro-3-oxo-4H-quinoxaline-2-carboxylate 288840-83-5 C23H19BrClN5O4
ethyl 7-[3-[[(4-bromophenyl)carbamoylamino]methyl]pyrrol-1-yl]-6-chloro-3-oxo-4H-quinoxaline-2-carboxylate
—— (2S)-N-[4-[(Aminoiminomethyl)amino]-1-(2-benzothiazolylcarbonyl)butyl]-1-[(4-methylphenyl)sulfonyl]-2-pyrrolidinecarboxamide 287182-58-5 C25H30N6O4S2
(2S)-N-[4-[(Aminoiminomethyl)amino]-1-(2-benzothiazolylcarbonyl)butyl]-1-[(4-methylphenyl)sulfonyl]-2-pyrrolidinecarboxamide
—— 4-{4-[3-(N,N-Dimethyl)amino-2-hydroxy-propoxy]anilino}-6-(N-(4,4,4-trifluorobutyl)-2,5-dichloroanilino)pyrimidine 260054-11-3 C25H28Cl2F3N5O2
4-{4-[3-(N,N-Dimethyl)amino-2-hydroxy-propoxy]anilino}-6-(N-(4,4,4-trifluorobutyl)-2,5-dichloroanilino)pyrimidine
—— (4-(2-benzoyl-4-hydroxy-5-isopropyl-phenoxy)-3,5-dibromo-phenyl)-acetic acid 258819-47-5 C24H20Br2O5
(4-(2-benzoyl-4-hydroxy-5-isopropyl-phenoxy)-3,5-dibromo-phenyl)-acetic acid
—— 2-amino-N-{2-[3-benzyl-3-(N',N'-dimethylhydrazinocarbonyl)piperidin-1-yl]-1-((2-naphthyl)methyl)-2-oxo-ethyl}-2-methyl-propionamide 249921-13-9 C32H41N5O3
2-amino-N-{2-[3-benzyl-3-(N',N'-dimethylhydrazinocarbonyl)piperidin-1-yl]-1-((2-naphthyl)methyl)-2-oxo-ethyl}-2-methyl-propionamide
—— 2-[(4'-Methoxy-[1,1'-biphenyl]-4-yl)-sulfonyl]-amino-3-[2-(2-oxo-azepan-1-ylmethyl)-[1,3]dioxan-2-yl]-propionic acid 291541-41-8 C27H34N2O8S
2-[(4'-Methoxy-[1,1'-biphenyl]-4-yl)-sulfonyl]-amino-3-[2-(2-oxo-azepan-1-ylmethyl)-[1,3]dioxan-2-yl]-propionic acid
—— N-[(S)-1-(N-cyclopentylamino)-1,2-dioxo-3-heptyl]-1-[N-(quinoline-8-sulfonyl)amino]cyclohexanecarboxamide 274684-82-1 C28H38N4O5S
N-[(S)-1-(N-cyclopentylamino)-1,2-dioxo-3-heptyl]-1-[N-(quinoline-8-sulfonyl)amino]cyclohexanecarboxamide
—— 5-Chloro-2-(4-chlorophenylsulfonylamino)-N-(4-(4-chlorophenoxy)phenyl)benzamide 254432-22-9 C25H17Cl3N2O4S
5-Chloro-2-(4-chlorophenylsulfonylamino)-N-(4-(4-chlorophenoxy)phenyl)benzamide
—— (2S,3S,5S)-5-[N-[2-(2,6-dimethylphenoxy)acetyl]amino]-2-[N-(3-hydroxy-2-methylbenzoyl)amino]-3-hydroxy-7-methyl-1-phenyloctane 282539-75-7 C33H42N2O5
(2S,3S,5S)-5-[N-[2-(2,6-dimethylphenoxy)acetyl]amino]-2-[N-(3-hydroxy-2-methylbenzoyl)amino]-3-hydroxy-7-methyl-1-phenyloctane
—— 4-(4-(4-Fluorophenylcarbonyl)-1-piperazinyl)-3-trifluoromethyl-benzoylguanidine methanesulphonate 261505-83-3 CH4O3S*C20H19F4N5O2
4-(4-(4-Fluorophenylcarbonyl)-1-piperazinyl)-3-trifluoromethyl-benzoylguanidine methanesulphonate
—— ethyl 6-chloro-3-oxo-7-[3-[[[4-(trifluoromethyl)phenyl]carbamoylamino]methyl]pyrrol-1-yl]-4H-quinoxaline-2-carboxylate 288840-86-8 C24H19ClF3N5O4
ethyl 6-chloro-3-oxo-7-[3-[[[4-(trifluoromethyl)phenyl]carbamoylamino]methyl]pyrrol-1-yl]-4H-quinoxaline-2-carboxylate
—— 3-(N,N-Dimethylamino)methyl-1-[3-(4-methoxyphenyl)propanoyl]-1,2,3,4-tetrahydroquinoline p-toluenesulfonate 246864-43-7 C7H8O3S*C22H28N2O2
3-(N,N-Dimethylamino)methyl-1-[3-(4-methoxyphenyl)propanoyl]-1,2,3,4-tetrahydroquinoline p-toluenesulfonate
—— rel-2-[4-[(4R,5R)-3,3-Dibutyl-7-(dimethylamino)-2,3,4,5-tetrahydro-4-hydroxy-1,1-dioxido-1-benzothiepin-5-yl]phenoxy]acetic acid 289039-86-7 C28H39NO6S
rel-2-[4-[(4R,5R)-3,3-Dibutyl-7-(dimethylamino)-2,3,4,5-tetrahydro-4-hydroxy-1,1-dioxido-1-benzothiepin-5-yl]phenoxy]acetic acid
—— 2-[5-amino-6-oxo-2-(4-fluorophenyl)-1,6-dihydro-1-pyrimidinyl]-N-[(1R)-1-[[5-(3-methylbenzyl)-1,3,4-oxadiazole-2-yl]carbonyl]-2-methylpropyl]acetamide 251988-66-6 C27H27FN6O4
2-[5-amino-6-oxo-2-(4-fluorophenyl)-1,6-dihydro-1-pyrimidinyl]-N-[(1R)-1-[[5-(3-methylbenzyl)-1,3,4-oxadiazole-2-yl]carbonyl]-2-methylpropyl]acetamide
—— (3-{4-[4-(4-Benzyl-phenylamino)-quinazolin-6-yl]-benzyl}-3-aza-bicyclo[3.1.0]hex-6-yl)-methanol 289036-77-7 C34H32N4O
(3-{4-[4-(4-Benzyl-phenylamino)-quinazolin-6-yl]-benzyl}-3-aza-bicyclo[3.1.0]hex-6-yl)-methanol
—— (2R,3R,4S,5S)-2-{6-(1-Ethyl-propylamino)-2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-purin-9-yl}-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-tetrahydro-furan-3,4-diol 235415-07-3 C23H32N10O4
(2R,3R,4S,5S)-2-{6-(1-Ethyl-propylamino)-2-[2-(1-methyl-1H-imidazol-4-yl)-ethylamino]-purin-9-yl}-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-tetrahydro-furan-3,4-diol
—— 2-(4,6-Dimethyl-2-pyrimidinyloxy)-3-(N-methyl-N-phenylcarbamoylmethoxy)-3,3-diphenylpropionic acid 224455-02-1 C30H29N3O5
2-(4,6-Dimethyl-2-pyrimidinyloxy)-3-(N-methyl-N-phenylcarbamoylmethoxy)-3,3-diphenylpropionic acid
—— 1-[2-Oxo-3-(4-phenyl-butyl)-3,10-diaza-bicyclo[4.3.1]dec-4-en-10-yl]-2-(3,4,5-trimethoxy-phenyl)-ethane-1,2-dione 255910-73-7 C29H34N2O6
1-[2-Oxo-3-(4-phenyl-butyl)-3,10-diaza-bicyclo[4.3.1]dec-4-en-10-yl]-2-(3,4,5-trimethoxy-phenyl)-ethane-1,2-dione
—— (+/-)-N-hydroxy-Nα-methyl-Nα-(4-phenoxybenzenesulfonyl)-2-(2-phthalimidoethyl)glycinamide 246262-73-7 C25H23N3O7S
(+/-)-N-hydroxy-Nα-methyl-Nα-(4-phenoxybenzenesulfonyl)-2-(2-phthalimidoethyl)glycinamide
—— N-[2-methyl-5-(3-trifluoromethylbenzamido)phenyl]-3-(4-methylpiperazin-1-yl)methylbenzamide 221875-34-9 C28H29F3N4O2
N-[2-methyl-5-(3-trifluoromethylbenzamido)phenyl]-3-(4-methylpiperazin-1-yl)methylbenzamide
—— N-(5-Chloropyridin-2-yl)-2-[(piperidin-4-ylmethoxycarbonyl)amino]benzamide Trifluoroacetic Acid Salt 280769-36-0 C2HF3O2*C19H21ClN4O3
N-(5-Chloropyridin-2-yl)-2-[(piperidin-4-ylmethoxycarbonyl)amino]benzamide Trifluoroacetic Acid Salt
—— (N-4-Carboxybenzoyl)-(N'-3,5-dichloroisonicotinoyl)-L-4-aminophenylalanine 240482-17-1 C23H17Cl2N3O6
(N-4-Carboxybenzoyl)-(N'-3,5-dichloroisonicotinoyl)-L-4-aminophenylalanine
—— 1-(1,1-diphenyl)methyl-2-ethyl-4-(2,4,5-trichlorophenyl)-1H-benzimidazole 254876-47-6 C28H21Cl3N2
1-(1,1-diphenyl)methyl-2-ethyl-4-(2,4,5-trichlorophenyl)-1H-benzimidazole
—— N-[2-methyl-5-(3-morpholinobenzamido)phenyl]-4-diethylaminomethylbenzamide 250680-84-3 C30H36N4O3
N-[2-methyl-5-(3-morpholinobenzamido)phenyl]-4-diethylaminomethylbenzamide
—— 9-bromo-2-(3-hydroxypropyloxy)-5-(3-pyridylmethyl)-4H-pyrido[3,2,1-jk]carbazole-4-one hydrochloride 216856-45-0 C24H19BrN2O3*ClH
9-bromo-2-(3-hydroxypropyloxy)-5-(3-pyridylmethyl)-4H-pyrido[3,2,1-jk]carbazole-4-one hydrochloride
—— N-[4-(5-cyano-3-pyridin-3-yl-pyrazol-1-yl)phenyl]-4-(3-[1,3]dioxolan-2-yl-propoxy)benzamide 251655-57-9 C28H25N5O4
N-[4-(5-cyano-3-pyridin-3-yl-pyrazol-1-yl)phenyl]-4-(3-[1,3]dioxolan-2-yl-propoxy)benzamide
—— 1-(4-chlorobenzyl)-4-[[(N-(2-amino-5-trifluoromethylbenzoyl)glycyl)amino]methyl]piperidine 226242-85-9 C23H26ClF3N4O2
1-(4-chlorobenzyl)-4-[[(N-(2-amino-5-trifluoromethylbenzoyl)glycyl)amino]methyl]piperidine
—— 4-[(6-benzenesulphonylamino-1-n-propyl-1H-benzimidazol-2-yl)-methyl]-benzamidine-hydrochloride 236414-36-1 C24H25N5O2S*ClH
4-[(6-benzenesulphonylamino-1-n-propyl-1H-benzimidazol-2-yl)-methyl]-benzamidine-hydrochloride
—— 3,4,7,8-tetrahydro-4-(4-methylpiperazin-1-yl)-2,2,8,8-tetramethyl-6-(3-trifluoromethylphenyl)-2H,6H-benzo[1,2-b:5,4-b']dipyran 292081-95-9 C28H35F3N2O2
3,4,7,8-tetrahydro-4-(4-methylpiperazin-1-yl)-2,2,8,8-tetramethyl-6-(3-trifluoromethylphenyl)-2H,6H-benzo[1,2-b:5,4-b']dipyran
—— (2S)-N2-[(3S)-1-benzylpyrrolidin-3-yl]-1-(6-bromo-1,3-benzoxazol-2-yl)-2-piperidinecarboxamide 256526-28-0 C24H27BrN4O2
(2S)-N2-[(3S)-1-benzylpyrrolidin-3-yl]-1-(6-bromo-1,3-benzoxazol-2-yl)-2-piperidinecarboxamide
—— 4'-[2-(Diethylamino)ethoxy]-2-(isopropanesulfonamido)benzanilide Hydrochloride 253338-84-0 C22H31N3O4S*ClH
4'-[2-(Diethylamino)ethoxy]-2-(isopropanesulfonamido)benzanilide Hydrochloride
—— 2-[4-(Ethanesulfonyl-(1-propyl)amino)-2,2-dimethylchroman-6-yloxy]-N-(3-ethoxypropyl)acetamide 221552-57-4 C23H38N2O6S
2-[4-(Ethanesulfonyl-(1-propyl)amino)-2,2-dimethylchroman-6-yloxy]-N-(3-ethoxypropyl)acetamide
—— 1-(2-Hydroxyethyl)-3-[1-(3-hydroxymethylbenzyl)piperidin-4-yl]-4-phenyl-3,4-dihydro-2(1H)-quinazolinone 265328-88-9 C29H33N3O3
1-(2-Hydroxyethyl)-3-[1-(3-hydroxymethylbenzyl)piperidin-4-yl]-4-phenyl-3,4-dihydro-2(1H)-quinazolinone
—— 3,4,7,8-Tetrahydro-N,N-dimethyl-2,2,8,8-tetramethyl-6-(3-trifluoromethylphenyl)-2H,6H-benzo[1,2-b:5,4-b']dipyran-4-amine hydrochloride 292082-07-6 C25H30F3NO2*ClH
3,4,7,8-Tetrahydro-N,N-dimethyl-2,2,8,8-tetramethyl-6-(3-trifluoromethylphenyl)-2H,6H-benzo[1,2-b:5,4-b']dipyran-4-amine hydrochloride
—— (2-bromophenyl)[2-chloro-4-(E-((2-(hydroxymethyl)piperidin-1-yl)carbonyl)ethenyl)phenyl]sulfide 280748-83-6 C21H21BrClNO2S
(2-bromophenyl)[2-chloro-4-(E-((2-(hydroxymethyl)piperidin-1-yl)carbonyl)ethenyl)phenyl]sulfide