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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-4-[4-Cyano-2-(ethylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164203-82-0 C22H17F3N4O3S
(4S)-4-[4-Cyano-2-(ethylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— 3-(4-Hydroxy-2,2,6,6-tetramethylpiperidin-1-yl)oxybutan-2-one 1001081-05-5 C13H25NO3
3-(4-Hydroxy-2,2,6,6-tetramethylpiperidin-1-yl)oxybutan-2-one
—— (4S)-4-(4-cyano-2-methylsulfonylphenyl)-3-(1-ethyl-3-methylpyrazol-4-yl)sulfonyl-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carbonitrile 1164203-03-5 C27H23F3N6O5S2
(4S)-4-(4-cyano-2-methylsulfonylphenyl)-3-(1-ethyl-3-methylpyrazol-4-yl)sulfonyl-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carbonitrile
—— (2-Aminopyridin-3-yl)-cyclopentylmethanone 1344224-96-9 C11H14N2O
(2-Aminopyridin-3-yl)-cyclopentylmethanone
—— (1-Amino-5-furan-2-yl-8,8-dimethyl-8,9-dihydro-6H-3,7-dioxa-4-aza-cyclopenta[a]naphthalen-2-yl)-(4-chloro-phenyl)-methanone 172985-29-4 C23H19ClN2O4
(1-Amino-5-furan-2-yl-8,8-dimethyl-8,9-dihydro-6H-3,7-dioxa-4-aza-cyclopenta[a]naphthalen-2-yl)-(4-chloro-phenyl)-methanone
—— 1-(4-methylbenzyl)-1H-1,2,4-triazole 143131-65-1 C10H11N3
1-(4-methylbenzyl)-1H-1,2,4-triazole
—— (rac)-4-{4-Cyano-2-[(1-methylethyl)sulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid 1164204-79-8 C23H20F3N3O5S
(rac)-4-{4-Cyano-2-[(1-methylethyl)sulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid
—— (7-methoxy-2-oxo-2<i>H</i>-chromen-4-yl)-acetic acid hydrazide 143951-95-5 C12H12N2O4
(7-methoxy-2-oxo-2<i>H</i>-chromen-4-yl)-acetic acid hydrazide
—— 3-amino-6-(1-phenylcyclopropyl)pyridine-2(1H)-thione 1202075-99-7 C14H14N2S
3-amino-6-(1-phenylcyclopropyl)pyridine-2(1H)-thione
—— Hydroxy-di-p-tolyl-acetic acid [1-(4-methoxy-phenyl)-meth-(E)-ylidene]-hydrazide 128462-80-6 C24H24N2O3
Hydroxy-di-p-tolyl-acetic acid [1-(4-methoxy-phenyl)-meth-(E)-ylidene]-hydrazide
—— 2-(N-tert-butylamino)-3'-iodo-4'-azidopropiophenone 1354635-87-2 C13H17IN4O
2-(N-tert-butylamino)-3'-iodo-4'-azidopropiophenone
—— 2-(3,4-Dihydro-3,3-dimethyl-1(2H)-isoquinolinylidene)-N-2-thienylacetamide 170658-17-0 C17H18N2OS
2-(3,4-Dihydro-3,3-dimethyl-1(2H)-isoquinolinylidene)-N-2-thienylacetamide
—— (rac)-4-{4-Cyano-2-[phenylsulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164204-09-4 C26H17F3N4O3S
(rac)-4-{4-Cyano-2-[phenylsulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— 3-(9,10-dihydro-9-oxoacridine-2-yl)propionic acid 126862-61-1 C16H13NO3
3-(9,10-dihydro-9-oxoacridine-2-yl)propionic acid
—— 7-Chloro-4-(3,4,5-trimethyl-pyrazol-1-yl)-quinoline 124833-70-1 C15H14ClN3
7-Chloro-4-(3,4,5-trimethyl-pyrazol-1-yl)-quinoline
—— 4-hydroxy-2-({2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}sulfanyl)-6-phenylpyrimidine-5-carbonitrile 1448163-14-1 C21H19N7O2S
4-hydroxy-2-({2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}sulfanyl)-6-phenylpyrimidine-5-carbonitrile
—— 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-5-hydroxybenzoic acid 1032614-17-7 C15H9FN2O4
3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-5-hydroxybenzoic acid
—— 12-(2-Fluor-phenyl)-benz<a>anthracen 1789-53-3 C24H15F
12-(2-Fluor-phenyl)-benz<a>anthracen
—— (2-Fluoro-phenyl)-(2,3,4,5-tetrahydro-benzo[b]oxepin-7-yl)-methanone 147394-49-8 C17H15FO2
(2-Fluoro-phenyl)-(2,3,4,5-tetrahydro-benzo[b]oxepin-7-yl)-methanone
—— (6S)-5-Cyano-6-[4-cyano-2-(methylsulfonyl)phenyl]-N-(2-hydroxy-1,1-dimethylethyl)-4-methyl-2-oxo-3-[3-(trifluoromethyl)phenyl]-3,6-dihydropyrimidine-1(2H)-carboxamide 1161921-62-5 C26H24F3N5O5S
(6S)-5-Cyano-6-[4-cyano-2-(methylsulfonyl)phenyl]-N-(2-hydroxy-1,1-dimethylethyl)-4-methyl-2-oxo-3-[3-(trifluoromethyl)phenyl]-3,6-dihydropyrimidine-1(2H)-carboxamide
—— ethyl 3-nitroimidazo[1,2-a]pyridine-5-carboxylate 177485-57-3 C10H9N3O4
ethyl 3-nitroimidazo[1,2-a]pyridine-5-carboxylate
—— (rac)-4-[4-Cyano-2-(ethylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide 1164203-78-4 C22H19F3N4O4S
(rac)-4-[4-Cyano-2-(ethylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
—— Butanediamide, N'-(4-(aminosulfonyl)phenyl)-N,N-bis(2-hydroxyethyl)- 171088-67-8 C14H21N3O6S
Butanediamide, N'-(4-(aminosulfonyl)phenyl)-N,N-bis(2-hydroxyethyl)-
—— 3(S)-9-{6-[Ethyl-(4-methoxy-benzyl)-amino]-pyridin-2-yl}-3-(2-methyl-pyrimidin-5-yl)-nonanoic acid ethyl ester 1429492-21-6 C31H42N4O3
3(S)-9-{6-[Ethyl-(4-methoxy-benzyl)-amino]-pyridin-2-yl}-3-(2-methyl-pyrimidin-5-yl)-nonanoic acid ethyl ester
—— (rac)-4-[4-Cyano-2-((2-hydroxyethyl)sulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid 1164204-65-2 C22H18F3N3O6S
(rac)-4-[4-Cyano-2-((2-hydroxyethyl)sulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid
—— (2R,3R)-3-[3-(2,5-Dimethyl-pyrrol-1-yl)-2,5-dimethoxy-phenyl]-3-methoxy-2-methyl-propionic acid methyl ester 115820-54-7 C20H27NO5
(2R,3R)-3-[3-(2,5-Dimethyl-pyrrol-1-yl)-2,5-dimethoxy-phenyl]-3-methoxy-2-methyl-propionic acid methyl ester
—— (4S)-4-(4-cyano-2-methylsulfonylphenyl)-6-methyl-2-oxo-3-(thiomorpholine-4-carbonyl)-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carbonitrile 1164202-30-5 C26H22F3N5O4S2
(4S)-4-(4-cyano-2-methylsulfonylphenyl)-6-methyl-2-oxo-3-(thiomorpholine-4-carbonyl)-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carbonitrile
—— methyl 1H-pyrazolo[3,4-b]pyridine-4-carboxylate 1638769-07-9 C8H7N3O2
methyl 1H-pyrazolo[3,4-b]pyridine-4-carboxylate
—— (rac)-4-[4-Cyano-2-(ethylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid 1164204-57-2 C22H18F3N3O5S
(rac)-4-[4-Cyano-2-(ethylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid
—— (rac)-4-{4-Cyano-2-[phenylsulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid 1164204-86-7 C26H18F3N3O5S
(rac)-4-{4-Cyano-2-[phenylsulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid
—— (rac)-4-{2-[(2-{[tert-Butyl(dimethyl)silyl]oxy}ethyl)sulfonyl]-4-cyanophenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164204-70-9 C28H31F3N4O4SSi
(rac)-4-{2-[(2-{[tert-Butyl(dimethyl)silyl]oxy}ethyl)sulfonyl]-4-cyanophenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— 2-[(6S)-5-cyano-6-[4-cyano-2-(methylsulfonyl)phenyl]-4-methyl-2-oxo-3-[3-(trifluoromethyl)phenyl]-3,6-dihydropyrimidin-1(2H)-yl]acetamide 1161921-71-6 C23H18F3N5O4S
2-[(6S)-5-cyano-6-[4-cyano-2-(methylsulfonyl)phenyl]-4-methyl-2-oxo-3-[3-(trifluoromethyl)phenyl]-3,6-dihydropyrimidin-1(2H)-yl]acetamide
—— 3(S)-9-[6-(4-Methoxy-benzylamino)-pyridin-2-yl]-3-(2-methyl-pyrimidin-5-yl)-nonanoic acid ethyl ester 1429483-05-5 C29H38N4O3
3(S)-9-[6-(4-Methoxy-benzylamino)-pyridin-2-yl]-3-(2-methyl-pyrimidin-5-yl)-nonanoic acid ethyl ester
—— 2-Hydroxyethyl (4S)-4-[4-cyano-2-(methylsulfonyl)phenyl]-3,6-dimethyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylate 1164204-19-6 C24H22F3N3O6S
2-Hydroxyethyl (4S)-4-[4-cyano-2-(methylsulfonyl)phenyl]-3,6-dimethyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxylate
—— (2-(4-(difluoromethoxy)-3-isopropoxyphenyl)oxazol-4-yl)methanol 1574285-36-1 C14H15F2NO4
(2-(4-(difluoromethoxy)-3-isopropoxyphenyl)oxazol-4-yl)methanol
—— (4S)-4-[4-Cyano-2-(methylsulfonyl)phenyl]-6-methyl-2-oxo-1,3-bis[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164203-63-7 C28H18F6N4O3S
(4S)-4-[4-Cyano-2-(methylsulfonyl)phenyl]-6-methyl-2-oxo-1,3-bis[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— (rac)-4-{4-Cyano-2-[(1-methylethyl)sulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164204-00-5 C23H19F3N4O3S
(rac)-4-{4-Cyano-2-[(1-methylethyl)sulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— N-(2-(1-[2-(4-chloro-phenoxy)-phenylamino]-butyl)-phenyl)-acetamide 1158909-96-6 C24H25ClN2O2
N-(2-(1-[2-(4-chloro-phenoxy)-phenylamino]-butyl)-phenyl)-acetamide
—— N-(2-aminoethyl)-2,3,4,5,6-pentamethylbenzenesulfonamide 1155143-72-8 C13H22N2O2S
N-(2-aminoethyl)-2,3,4,5,6-pentamethylbenzenesulfonamide
—— (4S)-4-[4-cyano-2-(ethylsulfonyl)phenyl]-3,6-dimethyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164203-84-2 C23H19F3N4O3S
(4S)-4-[4-cyano-2-(ethylsulfonyl)phenyl]-3,6-dimethyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— (2R,3R)-3-(2,5-Dimethoxy-3-nitro-phenyl)-3-hydroxy-2-methyl-propionic acid methyl ester 128836-47-5 C13H17NO7
(2R,3R)-3-(2,5-Dimethoxy-3-nitro-phenyl)-3-hydroxy-2-methyl-propionic acid methyl ester
—— (4S)-3-[(3R)-3-Aminopiperidin-1-yl]carbonyl-4-[4-cyano-2-(methylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1164202-26-9 C27H25F3N6O4S
(4S)-3-[(3R)-3-Aminopiperidin-1-yl]carbonyl-4-[4-cyano-2-(methylsulfonyl)phenyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile
—— (2R,3R)-3-(2,5-Dimethoxy-3-nitro-phenyl)-3-methoxy-2-methyl-propionic acid methyl ester 122911-29-9 C14H19NO7
(2R,3R)-3-(2,5-Dimethoxy-3-nitro-phenyl)-3-methoxy-2-methyl-propionic acid methyl ester
—— 3-(4-bromophenyl)-5-hydroxy-7-methoxyquinolin-4(1H)-one 1528669-19-3 C16H12BrNO3
3-(4-bromophenyl)-5-hydroxy-7-methoxyquinolin-4(1H)-one
—— (rac)-4-{4-Cyano-2-[(1-methylethyl)sulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide 1164203-98-8 C23H21F3N4O4S
(rac)-4-{4-Cyano-2-[(1-methylethyl)sulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
—— (rac)-4-{4-Cyano-2-[phenylsulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide 1164204-05-0 C26H19F3N4O4S
(rac)-4-{4-Cyano-2-[phenylsulfonyl]phenyl}-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
—— tert-butyl (R,E)-2,2-dimethyl-4-[2,3-bis-trimethylsilanyl-prop-1-enyl]-oxazolidine-3-carbamate 1140504-33-1 C19H39NO3Si2
tert-butyl (R,E)-2,2-dimethyl-4-[2,3-bis-trimethylsilanyl-prop-1-enyl]-oxazolidine-3-carbamate
—— methyl 2-{[4-(2-fuorophenyl)-4-oxobut-2-yn-1-yl](methyl)amino}-2-(trifluoromethyl)pent-4-enoate 1456821-88-7 C18H17F4NO3
methyl 2-{[4-(2-fuorophenyl)-4-oxobut-2-yn-1-yl](methyl)amino}-2-(trifluoromethyl)pent-4-enoate
—— N-[2-(([2-(4-chloro-phenoxy)-phenyl]-methyl-amino)-methyl)-phenyl]-N-methylacetamide 1158909-97-7 C23H23ClN2O2
N-[2-(([2-(4-chloro-phenoxy)-phenyl]-methyl-amino)-methyl)-phenyl]-N-methylacetamide
—— (4S)-4-[4-cyano-2-(methylsulfonyl)phenyl]-6-methyl-3-(methylsulfonyl)-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile 1161921-76-1 C22H17F3N4O5S2
(4S)-4-[4-cyano-2-(methylsulfonyl)phenyl]-6-methyl-3-(methylsulfonyl)-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile