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中文名称 英文名称 CAS号 化学式 结构式图片
—— (chloro-5-nitrophenyl)furo[3,2-c]pyridine 1609356-09-3 C13H7ClN2O3
(chloro-5-nitrophenyl)furo[3,2-c]pyridine
—— 1-(7-Fluoro-1-benzothiophen-3-yl)prop-2-en-1-one 1569083-98-2 C11H7FOS
1-(7-Fluoro-1-benzothiophen-3-yl)prop-2-en-1-one
—— 8-methyl-3-(2-oxo-2H-chromen-3-yl)-4H-furo[3,2-c]chromen-4-one 1237713-05-1 C21H12O5
8-methyl-3-(2-oxo-2H-chromen-3-yl)-4H-furo[3,2-c]chromen-4-one
—— 11-methyl-6-(pyridin-3'-yl)pyrido[2,3-b][1,4]benzodiazepine 1012065-96-1 C18H14N4
11-methyl-6-(pyridin-3'-yl)pyrido[2,3-b][1,4]benzodiazepine
—— 2-Butenamide, N-[(1R)-2-[[5-[2-[(4-cyanophenyl)amino]-4-(propylamino)-5-pyrimidinyl]-4-pentyn-1-yl]amino]-1-methyl-2-oxoethyl]-4-(dimethylamino)-N-methyl-, (2E)- 1472797-95-7 C29H38N8O2
2-Butenamide, N-[(1R)-2-[[5-[2-[(4-cyanophenyl)amino]-4-(propylamino)-5-pyrimidinyl]-4-pentyn-1-yl]amino]-1-methyl-2-oxoethyl]-4-(dimethylamino)-N-methyl-, (2E)-
—— (methoxy-4 phenylazo)-6 phenylimino-2 benzoxazin-1,3 one-4 134260-03-0 C21H16N4O3
(methoxy-4 phenylazo)-6 phenylimino-2 benzoxazin-1,3 one-4
—— 4-[3-(2-Benzoyloxy-ethyl)-imidazo[1,2-a]pyrazin-8-yl]-piperazine-1-carboxylic acid tert-butyl ester 143591-78-0 C24H29N5O4
4-[3-(2-Benzoyloxy-ethyl)-imidazo[1,2-a]pyrazin-8-yl]-piperazine-1-carboxylic acid tert-butyl ester
—— 4-{[4-(4,6-dimethylpyrimidin-5-yl)-1H-indol-7-yl]oxy}furo[3,2-c]pyridine 1609577-47-0 C21H16N4O2
4-{[4-(4,6-dimethylpyrimidin-5-yl)-1H-indol-7-yl]oxy}furo[3,2-c]pyridine
—— ethyl 4-chloro-1-(2-{[(5-chloro-[1,3]thiazolo[5,4-b]pyridin-2-yl)carbamoyl]amino}phenyl)-7-hydroxy-3-methyl-2,3-dihydro-1H-indole-3-carboxylate 1555694-41-1 C25H21Cl2N5O4S
ethyl 4-chloro-1-(2-{[(5-chloro-[1,3]thiazolo[5,4-b]pyridin-2-yl)carbamoyl]amino}phenyl)-7-hydroxy-3-methyl-2,3-dihydro-1H-indole-3-carboxylate
—— 2-(1-(6-(difluoromethoxy)naphthalen-2-yl)-2-methylpropyl)-2H-tetrazole 1313885-93-6 C16H16F2N4O
2-(1-(6-(difluoromethoxy)naphthalen-2-yl)-2-methylpropyl)-2H-tetrazole
—— Methyl 3-butyl-2-[2-(4-methylpiperazin-1-yl)-1,3-thiazol-5-yl]imidazole-4-carboxylate 1542223-10-8 C17H25N5O2S
Methyl 3-butyl-2-[2-(4-methylpiperazin-1-yl)-1,3-thiazol-5-yl]imidazole-4-carboxylate
—— tert-butyl (2S)-2-[6-[4-[6-[2-[(2S)-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]phenyl]-1H-benzimidazol-2-yl]pyrrolidine-1-carboxylate 1560646-21-0 C45H52N6O4
tert-butyl (2S)-2-[6-[4-[6-[2-[(2S)-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]phenyl]-1H-benzimidazol-2-yl]pyrrolidine-1-carboxylate
—— 5,6-dihydroxy-8,8-dimethyl-2-phenyl-9,10-dihydropyrano[2,3-f]chromen-4(8H)-one 1310461-31-4 C20H18O5
5,6-dihydroxy-8,8-dimethyl-2-phenyl-9,10-dihydropyrano[2,3-f]chromen-4(8H)-one
—— [2-[[Anthracen-9-ylmethyl-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]amino]methyl]phenyl]boronic acid 1417895-72-7 C29H33BN2O4
[2-[[Anthracen-9-ylmethyl-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]amino]methyl]phenyl]boronic acid
—— methyl N-[(2S)-1-[(2S,4S)-2-[5-[6-[4-[2-[(2S,4S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-4-methylpyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]-3-tricyclo[6.2.2.02,7]dodeca-2,4,6-trienyl]-1H-imidazol-2-yl]-4-methylpyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1560640-11-0 C48H62N8O6
methyl N-[(2S)-1-[(2S,4S)-2-[5-[6-[4-[2-[(2S,4S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-4-methylpyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]-3-tricyclo[6.2.2.02,7]dodeca-2,4,6-trienyl]-1H-imidazol-2-yl]-4-methylpyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 11-methyl-6-(4'-fluorophenyl)pyrido[2,3-b][1,4]benzodiazepine 1012065-95-0 C19H14FN3
11-methyl-6-(4'-fluorophenyl)pyrido[2,3-b][1,4]benzodiazepine
—— (S)-(+)-dimethyl (3-methyl-2-oxo-6-phenylhex-5-yn-1-yl)phosphonate 1544279-90-4 C15H19O4P
(S)-(+)-dimethyl (3-methyl-2-oxo-6-phenylhex-5-yn-1-yl)phosphonate
—— 2-(5-((4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl)-amino)-1-methyl-1H-pyrazol-3-yl)-2-methylpropanenitrile 1481690-43-0 C15H18F3N7
2-(5-((4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl)-amino)-1-methyl-1H-pyrazol-3-yl)-2-methylpropanenitrile
—— methyl N-[(2S)-1-[(2S)-2-[5-[4-[6-[3-[[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]phenyl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1560639-35-1 C49H59N7O7
methyl N-[(2S)-1-[(2S)-2-[5-[4-[6-[3-[[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]phenyl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[5-[5-[6-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-3H-benzimidazol-5-yl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]thiophen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1560649-59-3 C47H56N8O6S
methyl N-[(2S)-1-[(2S)-2-[5-[5-[6-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-3H-benzimidazol-5-yl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]thiophen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 2,3-Dibromo-1-(tert-butyl-dimethyl-silanyl)-propan-1-one 1027575-51-4 C9H18Br2OSi
2,3-Dibromo-1-(tert-butyl-dimethyl-silanyl)-propan-1-one
—— 1-(5-Chlorothiophen-2-yl)-2-(2,4-difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)propan-2-ol 1416805-27-0 C14H9ClF4N4OS
1-(5-Chlorothiophen-2-yl)-2-(2,4-difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)propan-2-ol
—— tert-butyl (5-{[(2-chloropyridin-3-yl)sulfonyl]amino}-2-methoxypyridin-3-yl)methylcarbamate 1534390-33-4 C17H21ClN4O5S
tert-butyl (5-{[(2-chloropyridin-3-yl)sulfonyl]amino}-2-methoxypyridin-3-yl)methylcarbamate
—— 2-Chloro-4-(β-hydroxyethylamino)pyrrolo<3,2-d>pyrimidine 114684-99-0 C8H9ClN4O
2-Chloro-4-(β-hydroxyethylamino)pyrrolo<3,2-d>pyrimidine
—— 4-[(7-bromo-1,3-benzodioxol-4-yl)oxy]furo[3,2-c]pyridine 1609581-68-1 C14H8BrNO4
4-[(7-bromo-1,3-benzodioxol-4-yl)oxy]furo[3,2-c]pyridine
—— 4-(5-bromo-2-pyridin-4-ylpyrido[3,4-d]pyrimidin-4-yl)piperazine-1-carboxylic acid tert-butyl ester 1589084-51-4 C21H23BrN6O2
4-(5-bromo-2-pyridin-4-ylpyrido[3,4-d]pyrimidin-4-yl)piperazine-1-carboxylic acid tert-butyl ester
—— methyl N-[(2S)-1-[(2S)-2-[5-[4-[6-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-3H-benzimidazol-5-yl]-4,5-diazatricyclo[6.2.2.02,7]dodeca-2(7),3,5-trien-3-yl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1560649-14-0 C48H58N10O6
methyl N-[(2S)-1-[(2S)-2-[5-[4-[6-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-3H-benzimidazol-5-yl]-4,5-diazatricyclo[6.2.2.02,7]dodeca-2(7),3,5-trien-3-yl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 3-(2-(2-(cyclooctylidene)hydrazynyl)thiazol-4-yl)-2H-chromen-2-one 1262238-77-6 C20H21N3O2S
3-(2-(2-(cyclooctylidene)hydrazynyl)thiazol-4-yl)-2H-chromen-2-one
—— (2S,3R)-N-((3-(dimethylamino)-1-pyrrolidinyl)methyl)-N'-((3S)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-1,4-benzodiazepin-3-yl)-2,3-bis(3,3,3-trifluoropropyl)succinamide 1581704-52-0 C33H40F6N6O3
(2S,3R)-N-((3-(dimethylamino)-1-pyrrolidinyl)methyl)-N'-((3S)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-1,4-benzodiazepin-3-yl)-2,3-bis(3,3,3-trifluoropropyl)succinamide
—— (2-bromophenyl)((2R,3S)-3-phenyloxiran-2-yl)methanone 1314140-40-3 C15H11BrO2
(2-bromophenyl)((2R,3S)-3-phenyloxiran-2-yl)methanone
—— 4-(5-isopropenyl-2-pyridin-4-ylpyrido[3,4-d]pyrimidin-4-yl)piperazine-1-carboxylic acid tert-butyl ester 1589084-55-8 C24H28N6O2
4-(5-isopropenyl-2-pyridin-4-ylpyrido[3,4-d]pyrimidin-4-yl)piperazine-1-carboxylic acid tert-butyl ester
—— 1-<2-(trimethylsilyl)ethoxy>methyl-1H-tetrazole 146535-87-7 C7H16N4OSi
1-<2-(trimethylsilyl)ethoxy>methyl-1H-tetrazole
—— 4,4,5,5-Tetramethyl-2-[6-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)naphthalen-1-yl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]-1,3,2-dioxaborolane 1560648-08-9 C33H40B2O4
4,4,5,5-Tetramethyl-2-[6-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)naphthalen-1-yl]-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl]-1,3,2-dioxaborolane
—— (E)-3-Methyl-4-{(2S,3S,4R,5S)-5-[(2S,3S)-3-((1R,2S)-1-methyl-2-trimethylsilanyloxy-propyl)-oxiranylmethyl]-3,4-bis-trimethylsilanyloxy-tetrahydro-pyran-2-yl}-but-2-enoic acid N'-(4-nitro-phenyl)-hydrazide 1055041-26-3 C32H57N3O8Si3
(E)-3-Methyl-4-{(2S,3S,4R,5S)-5-[(2S,3S)-3-((1R,2S)-1-methyl-2-trimethylsilanyloxy-propyl)-oxiranylmethyl]-3,4-bis-trimethylsilanyloxy-tetrahydro-pyran-2-yl}-but-2-enoic acid N'-(4-nitro-phenyl)-hydrazide
—— methyl 2-((1H-tetrazol-1-yl)methyl)-4-(2-chloro-4-fluorophenyl)-5-cyano-6-methyl-1,4-dihydropyridine-3-carboxylate 1240289-94-4 C17H14ClFN6O2
methyl 2-((1H-tetrazol-1-yl)methyl)-4-(2-chloro-4-fluorophenyl)-5-cyano-6-methyl-1,4-dihydropyridine-3-carboxylate
—— Methyl 3-butyl-2-[5-(4-methylpiperazin-1-yl)-1,3,4-thiadiazol-2-yl]imidazole-4-carboxylate 1542223-17-5 C16H24N6O2S
Methyl 3-butyl-2-[5-(4-methylpiperazin-1-yl)-1,3,4-thiadiazol-2-yl]imidazole-4-carboxylate
—— 2-Chloro-4-piperidin-1-yl-5H-pyrrolo[3,2-d]pyrimidine 114684-95-6 C11H13ClN4
2-Chloro-4-piperidin-1-yl-5H-pyrrolo[3,2-d]pyrimidine
—— N-(2-hydrazinyl-2-oxoethyl)-2-hydroxy-3,4-dimethoxybenzamide 1569083-95-9 C11H15N3O5
N-(2-hydrazinyl-2-oxoethyl)-2-hydroxy-3,4-dimethoxybenzamide
—— 6-(3-methyl-butyl)-2-thioxo-2,3-dihydro-1H-pyrimidin-4-one 138836-05-2 C9H14N2OS
6-(3-methyl-butyl)-2-thioxo-2,3-dihydro-1H-pyrimidin-4-one
—— US10335409, Example 79 1535215-66-7 C36H48Cl2N4O6
US10335409, Example 79
—— 3-(4-bromorophenylaminoacetyl)coumarin 164590-65-2 C17H12BrNO3
3-(4-bromorophenylaminoacetyl)coumarin
—— N<sup>2</sup>,N<sup>4</sup>-Bis-(4-methoxy-phenyl)-5H-pyrrolo[3,2-d]pyrimidine-2,4-diamine 114685-02-8 C20H19N5O2
N<sup>2</sup>,N<sup>4</sup>-Bis-(4-methoxy-phenyl)-5H-pyrrolo[3,2-d]pyrimidine-2,4-diamine
—— 4-(imidazo[1,2-a]pyridin-5-yl)-3-methylaniline 1609581-23-8 C14H13N3
4-(imidazo[1,2-a]pyridin-5-yl)-3-methylaniline
—— 2-(3-nitrophenyl)-1-phenylquinolin-4(1H)-one 1380424-20-3 C21H14N2O3
2-(3-nitrophenyl)-1-phenylquinolin-4(1H)-one
—— 5-[[5-[(1,3-Dimethyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]thieno[3,2-b]thiophen-2-yl]methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione 1566578-97-9 C20H16N4O4S4
5-[[5-[(1,3-Dimethyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]thieno[3,2-b]thiophen-2-yl]methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 4-(3,5-dimethylphenylsulfanyl)-3-iodo-6-methyl-5-(tetrazol-2-ylmethyl)pyridin-2(1H)-one 1185190-17-3 C16H16IN5OS
4-(3,5-dimethylphenylsulfanyl)-3-iodo-6-methyl-5-(tetrazol-2-ylmethyl)pyridin-2(1H)-one
—— 6-(trifluoromethyl)biphenyl-3-ol 1214364-82-5 C13H9F3O
6-(trifluoromethyl)biphenyl-3-ol
—— tert-butyl (2S)-1-oxo-1-((3S)-(8-fluoro-4-oxo-2',3',4,5,5',6'-hexahydro-3H-spiro[benzo[b][1,4]oxazepine-2,4'-pyran]-3-ylamino))propan-2-yl carbamate 1562191-95-0 C22H30FN3O6
tert-butyl (2S)-1-oxo-1-((3S)-(8-fluoro-4-oxo-2',3',4,5,5',6'-hexahydro-3H-spiro[benzo[b][1,4]oxazepine-2,4'-pyran]-3-ylamino))propan-2-yl carbamate
—— 1-[4-(furo[3,2-c]pyridin-4-yloxy)phenyl]-2-methyl-1H-imidazo[4,5-c]pyridine 1609577-60-7 C20H14N4O2
1-[4-(furo[3,2-c]pyridin-4-yloxy)phenyl]-2-methyl-1H-imidazo[4,5-c]pyridine
—— [(4S,7R)-10-[tert-butyl(diphenyl)silyl]oxy-7-chloro-4-hydroxy-5-methylidenedecyl] benzoate 1192815-37-4 C34H43ClO4Si
[(4S,7R)-10-[tert-butyl(diphenyl)silyl]oxy-7-chloro-4-hydroxy-5-methylidenedecyl] benzoate