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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (3S,4R)-1-[1-(2-chloro-6-cyclopropylbenzoyl)-4-fluoroindazol-3-yl]-3-hydroxy-4-methylpiperidine-4-carboxylate 1561773-30-5 C26H27ClFN3O4
ethyl (3S,4R)-1-[1-(2-chloro-6-cyclopropylbenzoyl)-4-fluoroindazol-3-yl]-3-hydroxy-4-methylpiperidine-4-carboxylate
—— 5,6-dihydroxy-8,9,9-trimethyl-2-phenyl-8,9-dihydro-4H-furo[2,3-h]chromen-4-one 1310461-30-3 C20H18O5
5,6-dihydroxy-8,9,9-trimethyl-2-phenyl-8,9-dihydro-4H-furo[2,3-h]chromen-4-one
—— 4-tetrazol-2-ylmethyl-benzaldehyde 1260599-31-2 C9H8N4O
4-tetrazol-2-ylmethyl-benzaldehyde
—— 3,8-bis[(2R)-1-(1H-tetrazol-1-yl)propan-2-yl]-3,8-dihydrobenzo[1,2-d:4,5-d']bis[1,2,3]triazine-4,9-dione 1134102-01-4 C16H16N14O2
3,8-bis[(2R)-1-(1H-tetrazol-1-yl)propan-2-yl]-3,8-dihydrobenzo[1,2-d:4,5-d']bis[1,2,3]triazine-4,9-dione
—— BMS-824 1265278-71-4 C31H27FN4O4S
BMS-824
—— [(2R,3S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-4-phenylmethoxybutan-2-yl] (2S)-2-hydroxy-3-methylbutanoate 1416772-64-9 C21H31NO7
[(2R,3S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-4-phenylmethoxybutan-2-yl] (2S)-2-hydroxy-3-methylbutanoate
—— 2-Amino-4-methoxy-6-methyl-5,8-dihydro-6H-pyrido[2,3-d]pyrimidin-7-one 117530-55-9 C9H12N4O2
2-Amino-4-methoxy-6-methyl-5,8-dihydro-6H-pyrido[2,3-d]pyrimidin-7-one
—— N,N-dimethyl-2H-tetrazole-2-carboxamide 1188418-96-3 C4H7N5O
N,N-dimethyl-2H-tetrazole-2-carboxamide
—— 8-cyclopropyl-3-[(2R)-1-(2H-tetrazol-2-yl)propan-2-yl]-7,8-dihydro-3H-[1,3]oxazino[6,5-g][1,2,3]benzotriazine-4,9-dione 1039453-38-7 C16H16N8O3
8-cyclopropyl-3-[(2R)-1-(2H-tetrazol-2-yl)propan-2-yl]-7,8-dihydro-3H-[1,3]oxazino[6,5-g][1,2,3]benzotriazine-4,9-dione
—— 3-Phenyl-5-pyridin-2-ylaniline 1546890-21-4 C17H14N2
3-Phenyl-5-pyridin-2-ylaniline
—— N-n-butyl-4,5-dinitro-2-methoxyaniline 111611-41-7 C11H15N3O5
N-n-butyl-4,5-dinitro-2-methoxyaniline
—— (R)-N-(1-Hydrazinocarbonylethyl)-3,4-dimethoxybenzamide 1569084-06-5 C12H17N3O4
(R)-N-(1-Hydrazinocarbonylethyl)-3,4-dimethoxybenzamide
—— 2-Amino-4-hydrazino-6-methyl-5,8-dihydro-6H-pyrido[2,3-d]pyrimidin-7-one 117530-57-1 C8H12N6O
2-Amino-4-hydrazino-6-methyl-5,8-dihydro-6H-pyrido[2,3-d]pyrimidin-7-one
—— 4-ethenyl-6-fluoro-N-methyl-2-(2-methylpyrimidin-5-yl)oxy-5-prop-2-enyl-9H-pyrimido[4,5-b]indol-8-amine 1581683-99-9 C21H19FN6O
4-ethenyl-6-fluoro-N-methyl-2-(2-methylpyrimidin-5-yl)oxy-5-prop-2-enyl-9H-pyrimido[4,5-b]indol-8-amine
—— 2,4-bi(tetrazolo)-6-chloro-1,3,5-triazine 1026023-89-1 C5H2ClN11
2,4-bi(tetrazolo)-6-chloro-1,3,5-triazine
—— (4-Butoxy-2-fluorophenyl)boronic acid 1107603-52-0 C10H14BFO3
(4-Butoxy-2-fluorophenyl)boronic acid
—— 4-cyclohexylmethyloxy-2-benzyl-benzoic acid 1099484-37-3 C21H24O3
4-cyclohexylmethyloxy-2-benzyl-benzoic acid
—— 4,5-di(hexadecyloxy)-1,2-dinitrobenzene 1315454-15-9 C38H68N2O6
4,5-di(hexadecyloxy)-1,2-dinitrobenzene
—— 3-[(2R)-1-(1H-tetrazol-1-yl)propan-2-yl]-8-[(2R)-1-(2H-tetrazol-2-yl)propan-2-yl]-3,8-dihydrobenzo[1,2-d:4,5-d']bis[1,2,3]triazine-4,9-dione 1134102-00-3 C16H16N14O2
3-[(2R)-1-(1H-tetrazol-1-yl)propan-2-yl]-8-[(2R)-1-(2H-tetrazol-2-yl)propan-2-yl]-3,8-dihydrobenzo[1,2-d:4,5-d']bis[1,2,3]triazine-4,9-dione
—— 9H-fluoren-9-ylmethyl (2S)-2-[1-[5-chloro-2-[[(2-methylpropan-2-yl)oxycarbonylamino]methyl]phenyl]ethylcarbamoyl]pyrrolidine-1-carboxylate 1567185-53-8 C34H38ClN3O5
9H-fluoren-9-ylmethyl (2S)-2-[1-[5-chloro-2-[[(2-methylpropan-2-yl)oxycarbonylamino]methyl]phenyl]ethylcarbamoyl]pyrrolidine-1-carboxylate
—— (2S,3R)-3-((5-(3-chlorophenyl)-9-ethyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)carbamoyl)-6,6,6-trifluoro-2-(3,3,3-trifluoropropyl)hexanoic acid 1584647-29-9 C27H26ClF6N3O4
(2S,3R)-3-((5-(3-chlorophenyl)-9-ethyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)carbamoyl)-6,6,6-trifluoro-2-(3,3,3-trifluoropropyl)hexanoic acid
—— methyl 4-(2-{1-benzhydryl-5-chloro-2-[2-({[2-(2H-tetrazol-2-yl)ethyl]sulfonyl}amino)ethyl]-1H-indol-3-yl}ethoxy)benzoate 1125597-94-5 C36H35ClN6O5S
methyl 4-(2-{1-benzhydryl-5-chloro-2-[2-({[2-(2H-tetrazol-2-yl)ethyl]sulfonyl}amino)ethyl]-1H-indol-3-yl}ethoxy)benzoate
—— 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-((4-fluorophenyl)ethynyl)pyrazin-2-yl)-3-(2H-tetrazol-2-yl)propan-2-ol 1416805-76-9 C22H13F5N6O
2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-((4-fluorophenyl)ethynyl)pyrazin-2-yl)-3-(2H-tetrazol-2-yl)propan-2-ol
—— 3-(5-bromopyridin-2-yl)-2-(2,4-difluorophenyl)-3-fluoro-1-(1H-tetrazol-1-yl)butan-2-ol 1416733-51-1 C16H13BrF3N5O
3-(5-bromopyridin-2-yl)-2-(2,4-difluorophenyl)-3-fluoro-1-(1H-tetrazol-1-yl)butan-2-ol
—— 1-(3,4-dichlorophenyl)-3-(dimethylamino)propan-1-ol 1225932-01-3 C11H15Cl2NO
1-(3,4-dichlorophenyl)-3-(dimethylamino)propan-1-ol
—— Amino-N-[5-[4-aminotetrahydropyran-2-yl]-1-methyl-pyrazol-4-yl]-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1586039-96-4 C19H20F2N6O2S
Amino-N-[5-[4-aminotetrahydropyran-2-yl]-1-methyl-pyrazol-4-yl]-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— PZ1051-1 1272246-56-6 C13H16BrN3
PZ1051-1
—— (E)-3-(2-(2-(3,4,5-trimethoxybenzylidene)hydrazinyl)thiazol-4-yl)-2H-chromen-2-one 1408316-05-1 C22H19N3O5S
(E)-3-(2-(2-(3,4,5-trimethoxybenzylidene)hydrazinyl)thiazol-4-yl)-2H-chromen-2-one
—— 2-(2,4-Difluorophenyl)-1,1-difluoro-1-(5-((4-fluorophenyl)ethynyl)pyrazin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol 1416805-75-8 C22H13F5N6O
2-(2,4-Difluorophenyl)-1,1-difluoro-1-(5-((4-fluorophenyl)ethynyl)pyrazin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol
—— US10335409, Example 55 1535213-53-6 C36H49F3N4O7
US10335409, Example 55
—— 4-Cyclopropyl-N1-methyl-1,2-benzenediamine 1267635-63-1 C10H14N2
4-Cyclopropyl-N1-methyl-1,2-benzenediamine
—— tert-butyl (2S)-1-oxo-1-((3S)-(9-fluoro-4-oxo-2',3',4,5,5',6'-hexahydro-3H-spiro[benzo[b][1,4]oxazepine-2,4'-pyran]-3-ylamino))propan-2-yl carbamate 1562191-76-7 C22H30FN3O6
tert-butyl (2S)-1-oxo-1-((3S)-(9-fluoro-4-oxo-2',3',4,5,5',6'-hexahydro-3H-spiro[benzo[b][1,4]oxazepine-2,4'-pyran]-3-ylamino))propan-2-yl carbamate
—— 1-(1,1-dimethylethyl) 3-ethyl 4-(7-chloro-4-quinolinyl)-5,6-dihydro-1,3(2H)-pyridinedicarboxylate 1197213-86-7 C22H25ClN2O4
1-(1,1-dimethylethyl) 3-ethyl 4-(7-chloro-4-quinolinyl)-5,6-dihydro-1,3(2H)-pyridinedicarboxylate
—— tert-butyl (2S)-2-[1-[5-chloro-2-(tetrazol-1-yl)phenyl]ethylcarbamoyl]pyrrolidine-1-carboxylate 1567184-83-1 C19H25ClN6O3
tert-butyl (2S)-2-[1-[5-chloro-2-(tetrazol-1-yl)phenyl]ethylcarbamoyl]pyrrolidine-1-carboxylate
—— 7-chloro-4-(trifluoromethyl)quinoline 1300746-83-1 C10H5ClF3N
7-chloro-4-(trifluoromethyl)quinoline
—— 2-(2,4-Difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)-1-(6-vinylquinoxalin-2-yl)propan-2-ol 1416805-84-9 C20H14F4N6O
2-(2,4-Difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)-1-(6-vinylquinoxalin-2-yl)propan-2-ol
—— (3S,4S)-4-hydroxy-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-4-[4-((S)-2-methyl-3-tetrazol-1-yl-propoxymethyl)-phenyl]-piperidine-1-carboxylic acid tert-butyl ester 1147886-69-8 C35H50N6O7
(3S,4S)-4-hydroxy-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-4-[4-((S)-2-methyl-3-tetrazol-1-yl-propoxymethyl)-phenyl]-piperidine-1-carboxylic acid tert-butyl ester
—— (2S,3R)-1-(methylamino)hex-5-ene-2,3-diol 1256091-46-9 C7H15NO2
(2S,3R)-1-(methylamino)hex-5-ene-2,3-diol
—— dimethyl 1-(naphthalen-1-yl)vinyl phosphate 1374846-74-8 C14H15O4P
dimethyl 1-(naphthalen-1-yl)vinyl phosphate
—— tert-butyl N-[3-fluoro-4-[5-methyl-2-(trifluoromethyl)-1,3-oxazol-4-yl]phenyl]carbamate 1582286-29-0 C16H16F4N2O3
tert-butyl N-[3-fluoro-4-[5-methyl-2-(trifluoromethyl)-1,3-oxazol-4-yl]phenyl]carbamate
—— 7-chloro-N-[3-(4,5-dihydrooxazol-2-yl)phenyl]quinolin-4-amine 1322669-55-5 C18H14ClN3O
7-chloro-N-[3-(4,5-dihydrooxazol-2-yl)phenyl]quinolin-4-amine
—— (3S,4S)-4-hydroxy-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-4-{4-[(R)-2-methyl-3-(toluene-4-sulfonyloxy)-propoxymethyl]-phenyl}-piperidine-1-carboxylic acid tert-butyl ester 1147886-55-2 C41H56N2O10S
(3S,4S)-4-hydroxy-3-[4-(3-methoxy-propyl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethoxy]-4-{4-[(R)-2-methyl-3-(toluene-4-sulfonyloxy)-propoxymethyl]-phenyl}-piperidine-1-carboxylic acid tert-butyl ester
—— tert-butyl (2S,3S,4R)-4-(3-ethenyl-7-methoxyquinoxalin-2-yl)oxy-3-methyl-1-[(2S)-2-(1-methylcyclopentyl)-2-[[(1R,2R)-2-pent-4-enylcyclopropyl]oxycarbonylamino]acetyl]pyrrolidine-2-carboxylate 1535212-86-2 C38H52N4O7
tert-butyl (2S,3S,4R)-4-(3-ethenyl-7-methoxyquinoxalin-2-yl)oxy-3-methyl-1-[(2S)-2-(1-methylcyclopentyl)-2-[[(1R,2R)-2-pent-4-enylcyclopropyl]oxycarbonylamino]acetyl]pyrrolidine-2-carboxylate
—— methyl 4-(2-{1-benzhydryl-5-chloro-2-[2-({[2-(1H-tetrazol-1-yl)ethyl]sulfonyl}amino)ethyl]-1H-indol-3-yl}ethoxy)benzoate 1125597-96-7 C36H35ClN6O5S
methyl 4-(2-{1-benzhydryl-5-chloro-2-[2-({[2-(1H-tetrazol-1-yl)ethyl]sulfonyl}amino)ethyl]-1H-indol-3-yl}ethoxy)benzoate
—— 1-(3'-hydroxyphenyl)-2-(4'-methylbenzoyl)-6,7-dioxolo-1,2,3,4-tetrahydroisoquinoline 1188392-67-7 C24H21NO4
1-(3'-hydroxyphenyl)-2-(4'-methylbenzoyl)-6,7-dioxolo-1,2,3,4-tetrahydroisoquinoline
—— 2-(2,4-Difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)-1-(6-(4-(trifluoromethyl)phenyl)pyridazin-3-yl)propan-2-ol 1416805-81-6 C21H13F7N6O
2-(2,4-Difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)-1-(6-(4-(trifluoromethyl)phenyl)pyridazin-3-yl)propan-2-ol
—— N-[3-(3-azabicyclo[3.1.0]hexan-3-yl)-5-bromopyridin-2-yl]-2-chloro-6-fluoro-N-methylbenzamide 1532518-44-7 C18H16BrClFN3O
N-[3-(3-azabicyclo[3.1.0]hexan-3-yl)-5-bromopyridin-2-yl]-2-chloro-6-fluoro-N-methylbenzamide
—— (R)-3-chloro-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridine-7-carbonitrile 1214265-76-5 C16H17ClN6
(R)-3-chloro-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridine-7-carbonitrile
—— (2S,3R)-3-[(2R)-2-[(2R,3S,4S)-4-amino-3-hydroxy-2-methyl-5-pyridin-3-ylpentanoyl]oxy-3-methylbutanoyl]oxy-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoic acid 1416772-45-6 C25H39N3O9
(2S,3R)-3-[(2R)-2-[(2R,3S,4S)-4-amino-3-hydroxy-2-methyl-5-pyridin-3-ylpentanoyl]oxy-3-methylbutanoyl]oxy-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoic acid
—— (E)‑3‑(2‑(2‑(4‑(dimethylamino)benzylidene)hydrazinyl)thiazol‑4‑yl)‑2H‑chromen‑2‑one 1408316-04-0 C21H18N4O2S
(E)‑3‑(2‑(2‑(4‑(dimethylamino)benzylidene)hydrazinyl)thiazol‑4‑yl)‑2H‑chromen‑2‑one