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—— 4-[[[2-[4-[4-(cyclopropylmethyl)piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-3,3-dimethyl-1H-indol-2-one 1383680-50-9 C31H36F3N7O2
4-[[[2-[4-[4-(cyclopropylmethyl)piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-3,3-dimethyl-1H-indol-2-one
—— 2-(2'-cyclohexenyl)-2,2-diphenylethanol 1311320-04-3 C20H22O
2-(2'-cyclohexenyl)-2,2-diphenylethanol
—— N-[[1-[3-(6-fluoro 1,2-benzoxazol-3-yl)propyl]azetidin-3-yl]methyl]-1-methylindole-5-sulphonamide 1417309-24-0 C23H25FN4O3S
N-[[1-[3-(6-fluoro 1,2-benzoxazol-3-yl)propyl]azetidin-3-yl]methyl]-1-methylindole-5-sulphonamide
—— (S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(1-oxetan-3-yl-azetidin-3-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416909-06-2 C33H37ClN2O5
(S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(1-oxetan-3-yl-azetidin-3-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— N-[1-[2-(1H-indol-4-yloxy)ethyl]azetidin-3-yl]-3-methylbenzenesulphonamide 1417308-18-9 C20H23N3O3S
N-[1-[2-(1H-indol-4-yloxy)ethyl]azetidin-3-yl]-3-methylbenzenesulphonamide
—— ((3aR,5R,6R,7R,7aR)-6-(benzyloxy)-2-(dimethylamino)-7-fluoro-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)methanol 1416709-89-1 C16H21FN2O3S
((3aR,5R,6R,7R,7aR)-6-(benzyloxy)-2-(dimethylamino)-7-fluoro-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-5-yl)methanol
—— 7-(3-Methoxy-pyridin-4-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one trifluoroacetate 1417182-46-7 C2HF3O2*C25H21N3O2
7-(3-Methoxy-pyridin-4-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one trifluoroacetate
—— (2S,3S)-1',2-dimethyl-2-naphthalen-2-ylspiro[[1,3]oxazolo[2,3-b]quinazoline-3,3'-indole]-2',5-dione 1287715-62-1 C29H21N3O3
(2S,3S)-1',2-dimethyl-2-naphthalen-2-ylspiro[[1,3]oxazolo[2,3-b]quinazoline-3,3'-indole]-2',5-dione
—— N-[[1-[2-[(2,2-dimethyl-3H-benzofuran-7-yl)oxy]ethyl]pyrrolidin-3-yl]methyl]naphthalene-2-sulphonamide 1417308-86-1 C27H32N2O4S
N-[[1-[2-[(2,2-dimethyl-3H-benzofuran-7-yl)oxy]ethyl]pyrrolidin-3-yl]methyl]naphthalene-2-sulphonamide
—— 2-{2-[1-(3-Dimethylamino-propyl)-1H-benzoimidazol-2-yl]-ethyl}-7-pyridin-4-yl-2,3-dihydro-isoindol-1-one trifluoroacetate 1417184-59-8 C2HF3O2*C27H29N5O
2-{2-[1-(3-Dimethylamino-propyl)-1H-benzoimidazol-2-yl]-ethyl}-7-pyridin-4-yl-2,3-dihydro-isoindol-1-one trifluoroacetate
—— N-benzyl-3-nitro-4-(3,6,6-trimethyl-4-oxo-5,7-dihydroindazol-1-yl)benzamide 1329599-88-3 C24H24N4O4
N-benzyl-3-nitro-4-(3,6,6-trimethyl-4-oxo-5,7-dihydroindazol-1-yl)benzamide
—— (2S)-2-[[(2S,3S,5R)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)-3-[(2-methylpropan-2-yl)oxycarbonylamino]oxolane-2-carbonyl]amino]propanoic acid 1252667-88-1 C18H26N4O8
(2S)-2-[[(2S,3S,5R)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)-3-[(2-methylpropan-2-yl)oxycarbonylamino]oxolane-2-carbonyl]amino]propanoic acid
—— 6-[2-(1,5-Dimethyl-1H-benzoimidazol-2-yl)-ethyl]-4-morpholin-4-yl-6,7-dihydro-pyrrolo[3,4-b]pyridin-5-one 1417185-98-8 C22H25N5O2
6-[2-(1,5-Dimethyl-1H-benzoimidazol-2-yl)-ethyl]-4-morpholin-4-yl-6,7-dihydro-pyrrolo[3,4-b]pyridin-5-one
—— 7-(4-Pyrrolidin-1-yl-piperidin-1-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one trifluoroacetate 1417183-26-6 C2HF3O2*C28H32N4O
7-(4-Pyrrolidin-1-yl-piperidin-1-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one trifluoroacetate
—— N'-(3-fluoro-4-{[6-methoxy-7-({1-[(methylamino)-2-oxoethyl]piperidin-4-yl}oxy)quinolin-4-yl]oxy}phenyl)-N-(2-chloro-6-methylphenyl)cyclopropane-1,1-dicarboxamide 1416320-91-6 C36H37ClFN5O6
N'-(3-fluoro-4-{[6-methoxy-7-({1-[(methylamino)-2-oxoethyl]piperidin-4-yl}oxy)quinolin-4-yl]oxy}phenyl)-N-(2-chloro-6-methylphenyl)cyclopropane-1,1-dicarboxamide
—— 2-[[1-[4-Cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2-oxazol-3-yl]-3-(2,4-dimethylanilino)-3-oxopropyl]amino]acetic acid 1404377-37-2 C27H37N3O4
2-[[1-[4-Cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2-oxazol-3-yl]-3-(2,4-dimethylanilino)-3-oxopropyl]amino]acetic acid
—— ((1S)-1-phenylbutyl) cis,cis-[(3-carboxy-1-oxopropyl)cyclopropylamino]-1,2,3,3a,9,9a-hexahydro-4H-cyclopenta[b]quinoline-4-carboxylate 1416606-72-8 C30H36N2O5
((1S)-1-phenylbutyl) cis,cis-[(3-carboxy-1-oxopropyl)cyclopropylamino]-1,2,3,3a,9,9a-hexahydro-4H-cyclopenta[b]quinoline-4-carboxylate
—— N-[1-[2-(2,3-dihydro-1,4-benzodioxan-8-yloxy)ethyl]pyrrolidin-3-yl]naphthalene-1-sulphonamide 1417308-70-3 C24H26N2O5S
N-[1-[2-(2,3-dihydro-1,4-benzodioxan-8-yloxy)ethyl]pyrrolidin-3-yl]naphthalene-1-sulphonamide
—— 3-[3-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-1-yl)propyl]-5,5-diethyl-imidazolidine-2,4-dione 1417032-85-9 C27H33N5O2S
3-[3-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-1-yl)propyl]-5,5-diethyl-imidazolidine-2,4-dione
—— (4R,5R,8S,11S,14S,17S)-14-benzyl-4,5-dihydroxy-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211439-45-0 C44H43N5O9S
(4R,5R,8S,11S,14S,17S)-14-benzyl-4,5-dihydroxy-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— 2-methoxyethyl 2,3-di-O-benzyl-β-D-galactopyranoside 127874-04-8 C23H30O7
2-methoxyethyl 2,3-di-O-benzyl-β-D-galactopyranoside
—— 14-(3,3-dimethylbut-1-en-2-yl)-35-isopropyl-15,34,55,74-tetramethyl-54,75-bis(3-methylenepentyl)-1,3,5,7(1,3)-tetracyclopentanacyclooctaphane-11,14,34,51,54,71(75),73-heptaene 125453-70-5 C36H40N4O6
14-(3,3-dimethylbut-1-en-2-yl)-35-isopropyl-15,34,55,74-tetramethyl-54,75-bis(3-methylenepentyl)-1,3,5,7(1,3)-tetracyclopentanacyclooctaphane-11,14,34,51,54,71(75),73-heptaene
—— 3-[5-(hydroxymethyl)thiophen-2-yl]benzaldehyde 1242026-81-8 C12H10O2S
3-[5-(hydroxymethyl)thiophen-2-yl]benzaldehyde
—— (S)-2-((R)-1-(benzyloxy)-2,2-difluorobut-3-en-1-yl)oxirane 1369405-71-9 C13H14F2O2
(S)-2-((R)-1-(benzyloxy)-2,2-difluorobut-3-en-1-yl)oxirane
—— <1S-<1α(R<sup>*</sup>),3α,7β,8β(4S<sup>*</sup>,6R<sup>*</sup>),8aβ>>-8-<2-<2,2-dimethyl-6-(2-oxoethyl)-1,3-dioxan-4-yl>ethyl>-3,7-dimethyl-1,2,3,7,8,8a-hexahydro-1-naphthalenyl 2-methylbutanoate 116996-48-6 C27H42O5
<1S-<1α(R<sup>*</sup>),3α,7β,8β(4S<sup>*</sup>,6R<sup>*</sup>),8aβ>>-8-<2-<2,2-dimethyl-6-(2-oxoethyl)-1,3-dioxan-4-yl>ethyl>-3,7-dimethyl-1,2,3,7,8,8a-hexahydro-1-naphthalenyl 2-methylbutanoate
—— [Pd(2,6-dimethylphenylisocyanide)(triphenylphosphine)(allyl)]ClO4 1269182-47-9 C30H29NPPd*ClO4
[Pd(2,6-dimethylphenylisocyanide)(triphenylphosphine)(allyl)]ClO4
—— N2-{2-[1,3-dihydro-2H-isoindol-2-yl(methyl)amino]-2-oxoethyl}-N2-{4-[5-(ethoxycarbonyl)-1,3-thiazol-2-yl]-2-methylphenyl}-N1-{2-[(tert-butoxycarbonyl)(ethyl)amino]ethyl}glycinamide 1190897-01-8 C35H46N6O6S
N2-{2-[1,3-dihydro-2H-isoindol-2-yl(methyl)amino]-2-oxoethyl}-N2-{4-[5-(ethoxycarbonyl)-1,3-thiazol-2-yl]-2-methylphenyl}-N1-{2-[(tert-butoxycarbonyl)(ethyl)amino]ethyl}glycinamide
—— (R)-2-methyl-propane-2-sulfinic acid [(1S,3S)-3-cyanomethoxy-1-(2-fluoro-5-nitro-phenyl)-1-methyl-3-phenyl-propyl]amide 1346145-75-2 C22H26FN3O4S
(R)-2-methyl-propane-2-sulfinic acid [(1S,3S)-3-cyanomethoxy-1-(2-fluoro-5-nitro-phenyl)-1-methyl-3-phenyl-propyl]amide
—— N-[2-[2-(2,3-dihydrochromen-4-ylidene)hydrazinyl]-2-oxoethyl]-3,4-dimethoxybenzamide 1569078-30-3 C20H21N3O5
N-[2-[2-(2,3-dihydrochromen-4-ylidene)hydrazinyl]-2-oxoethyl]-3,4-dimethoxybenzamide
—— N-[N'-butan-2-yl-N-[5-(3,5-difluorophenyl)-1H-pyrazol-3-yl]carbamimidoyl]-4-(trifluoromethyl)benzamide 1381826-54-5 C22H20F5N5O
N-[N'-butan-2-yl-N-[5-(3,5-difluorophenyl)-1H-pyrazol-3-yl]carbamimidoyl]-4-(trifluoromethyl)benzamide
—— (trans)-{4-[hydroxy-(tetrahydro-pyran-4-yI)-methyl]-cyclohexyl}-carbamic acid tert-butyl ester 1416471-31-2 C17H31NO4
(trans)-{4-[hydroxy-(tetrahydro-pyran-4-yI)-methyl]-cyclohexyl}-carbamic acid tert-butyl ester
—— 4-[[[2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]spiro[1H-indole-3,1'-cyclopropane]-2-one 1383680-48-5 C28H30F3N7O2
4-[[[2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]spiro[1H-indole-3,1'-cyclopropane]-2-one
—— 2-(2-Benzothiazol-2-yl-ethyl)-7-pyridin-4-yl-2,3-dihydro-isoindol-1-one 1417183-71-1 C22H17N3OS
2-(2-Benzothiazol-2-yl-ethyl)-7-pyridin-4-yl-2,3-dihydro-isoindol-1-one
—— 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-(5-methoxythiophen-2-yl)pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol 1416734-09-2 C20H15F4N5O2S
2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-(5-methoxythiophen-2-yl)pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ol
—— 1-(2,2-dimethylpropyl)-5-[2-hydroxy-8-(isoxazol-3-ylcarbonyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-methyl-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1416312-14-5 C23H29N5O4
1-(2,2-dimethylpropyl)-5-[2-hydroxy-8-(isoxazol-3-ylcarbonyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-methyl-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— 5-ethyl-3,3-dimethyl-8-(1-(phenylsulfonyl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-07-4 C25H31NO4S
5-ethyl-3,3-dimethyl-8-(1-(phenylsulfonyl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 6-(5-methyl-1H-pyrazol-4-yl)-2-[(4R)-1,3-thiazolidin-4-yl]thieno[3,2-d]pyrimidin-4(3H)-one 1330782-16-5 C13H13N5OS2
6-(5-methyl-1H-pyrazol-4-yl)-2-[(4R)-1,3-thiazolidin-4-yl]thieno[3,2-d]pyrimidin-4(3H)-one
—— N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-4-piperidine]methyl]naphthalene-2-sulphonamide 1417308-08-7 C26H28FN3O3S
N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-4-piperidine]methyl]naphthalene-2-sulphonamide
—— 2-(2,4-difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)-1-(thiophen-2-yl)propan-2-ol 1416805-40-7 C14H10F4N4OS
2-(2,4-difluorophenyl)-1,1-difluoro-3-(1H-tetrazol-1-yl)-1-(thiophen-2-yl)propan-2-ol
—— (Z)-3-(2-bromooct-2-enoyl)oxazolidin-2-one 1276027-37-2 C11H16BrNO3
(Z)-3-(2-bromooct-2-enoyl)oxazolidin-2-one
—— N-tert-butyl-1-(2-ethynyl-5-methoxyphenyl)methanimine oxide 1333261-16-7 C14H17NO2
N-tert-butyl-1-(2-ethynyl-5-methoxyphenyl)methanimine oxide
—— 1-[(3aR,4R,6S,6aS)-6-[[3-[(3aR,4R,6S,6aS)-6-[[3-[(3aR,4R,6S,6aS)-6-[[3-[(3aR,4R,6R,6aR)-6-[[2,3-dimethylbutan-2-yl(dimethyl)silyl]oxymethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-6-amino-2-oxopyrimidin-4-yl]methylsulfanylmethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-6-amino-2-oxopyrimidin-4-yl]methylsulfanylmethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-6-amino-2-oxopyrimidin-4-yl]methylsulfanylmethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-4-amino-6-[[(4-methoxyphenyl)-diphenylmethoxy]methyl]pyrimidin-2-one 1309372-11-9 C80H104N12O19S3Si
1-[(3aR,4R,6S,6aS)-6-[[3-[(3aR,4R,6S,6aS)-6-[[3-[(3aR,4R,6S,6aS)-6-[[3-[(3aR,4R,6R,6aR)-6-[[2,3-dimethylbutan-2-yl(dimethyl)silyl]oxymethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-6-amino-2-oxopyrimidin-4-yl]methylsulfanylmethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-6-amino-2-oxopyrimidin-4-yl]methylsulfanylmethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-6-amino-2-oxopyrimidin-4-yl]methylsulfanylmethyl]-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-4-amino-6-[[(4-methoxyphenyl)-diphenylmethoxy]methyl]pyrimidin-2-one
—— N-[1-[(1S,2R,3S,4R,5R)-3-(2-cyanoethoxymethoxy)-4-hydroxy-5-(hydroxymethyl)-2-bicyclo[3.1.0]hexanyl]-2-oxopyrimidin-4-yl]benzamide 1309375-22-1 C22H24N4O6
N-[1-[(1S,2R,3S,4R,5R)-3-(2-cyanoethoxymethoxy)-4-hydroxy-5-(hydroxymethyl)-2-bicyclo[3.1.0]hexanyl]-2-oxopyrimidin-4-yl]benzamide
—— 4-[[[2-[4-[4-(2-Hydroxyethylamino)piperidin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-1,3-dihydroindol-2-one 1383681-28-4 C28H32F3N7O3
4-[[[2-[4-[4-(2-Hydroxyethylamino)piperidin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-1,3-dihydroindol-2-one
—— (8R,11S,14R,17S)-14-[3-[(2-methylpropan-2-yl)oxy]-3-oxopropyl]-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211436-60-0 C44H49N5O9S
(8R,11S,14R,17S)-14-[3-[(2-methylpropan-2-yl)oxy]-3-oxopropyl]-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— N-[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]-1-methylindole-5-sulphonamide 1417309-91-1 C23H25FN4O3S
N-[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]-1-methylindole-5-sulphonamide
—— N-[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]-4-(trifluoromethyl)benzenesulphonamide 1417307-86-8 C21H21F4N3O3S
N-[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]-4-(trifluoromethyl)benzenesulphonamide
—— (3aR,5S,6R,7R,7aR)-2-(dimethylamino)-7-fluoro-5-((R)-2,2,2-trifluoro-1-hydroxyethyl)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-6-ol 1416709-04-0 C10H14F4N2O3S
(3aR,5S,6R,7R,7aR)-2-(dimethylamino)-7-fluoro-5-((R)-2,2,2-trifluoro-1-hydroxyethyl)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-6-ol
—— 7-(2,4-Dimethoxy-phenyl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417180-82-5 C27H24N2O3
7-(2,4-Dimethoxy-phenyl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— (S)-(2-bromophenyl)(4-(trifluoro-methyl)-phenyl)-methanamine 1416847-70-5 C14H11BrF3N
(S)-(2-bromophenyl)(4-(trifluoro-methyl)-phenyl)-methanamine