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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[4-(4-Methyl-piperazin-1-yl)-piperidin-1-yl]-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417181-45-3 C29H35N5O
7-[4-(4-Methyl-piperazin-1-yl)-piperidin-1-yl]-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— 4-Difluoromethoxy-7-pyridin-4-yl-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417184-27-0 C25H19F2N3O2
4-Difluoromethoxy-7-pyridin-4-yl-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— 5-[3-(6-acetamido-1,3-benzoxazol-2-yl)phenyl]-2-(4-fluorophenyl)-N-methyl-6-[methyl(methylsulfonyl)amino]-1-benzofuran-3-carboxamide 1333242-85-5 C33H27FN4O6S
5-[3-(6-acetamido-1,3-benzoxazol-2-yl)phenyl]-2-(4-fluorophenyl)-N-methyl-6-[methyl(methylsulfonyl)amino]-1-benzofuran-3-carboxamide
—— (3aR,5S,6R,7R,7aR)-2-(ethylamino)-7-fluoro-5-((R)-1,1,1-trifluoro-2-hydroxypropan-2-yl)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-6-ol 1416709-19-7 C11H16F4N2O3S
(3aR,5S,6R,7R,7aR)-2-(ethylamino)-7-fluoro-5-((R)-1,1,1-trifluoro-2-hydroxypropan-2-yl)-5,6,7,7a-tetrahydro-3aH-pyrano[3,2-d]thiazol-6-ol
—— 1-{[1-(2-chlorophenyl)-4-methyl[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl}-N,Ndimethylpiperidin-4-amine 1417410-69-5 C24H27ClN6
1-{[1-(2-chlorophenyl)-4-methyl[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl}-N,Ndimethylpiperidin-4-amine
—— 7-(3,4-Difluoro-phenyl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417180-78-9 C25H18F2N2O
7-(3,4-Difluoro-phenyl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— 4-Ethoxy-7-pyridin-4-yl-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417183-08-4 C26H23N3O2
4-Ethoxy-7-pyridin-4-yl-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— 6-(5-methyl-1H-pyrazol-4-yl)-2-[(4-phenylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3H)-one 1330781-18-4 C21H22N6OS
6-(5-methyl-1H-pyrazol-4-yl)-2-[(4-phenylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3H)-one
—— 7-(1H-Indazol-6-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417181-42-0 C26H20N4O
7-(1H-Indazol-6-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— 7-(2-Methyl-morpholin-4-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one trifluoroacetate 1417183-80-2 C2HF3O2*C24H25N3O2
7-(2-Methyl-morpholin-4-yl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one trifluoroacetate
—— (3Z)-6-methoxy-3-[(2-methyl-1H-imidazol-5-yl)methylene]indolin-2-one 1416817-94-1 C14H13N3O2
(3Z)-6-methoxy-3-[(2-methyl-1H-imidazol-5-yl)methylene]indolin-2-one
—— 1-(2-chlorophenyl)-N,N,4-trimethyl[1,2,4]triazolo[4,3-a]quinoxalin-8-amine 1417409-86-9 C18H16ClN5
1-(2-chlorophenyl)-N,N,4-trimethyl[1,2,4]triazolo[4,3-a]quinoxalin-8-amine
—— 7-(4-Methoxy-phenyl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one 1417180-68-7 C26H22N2O2
7-(4-Methoxy-phenyl)-2-(2-quinolin-2-yl-ethyl)-2,3-dihydro-isoindol-1-one
—— N-[1-[3-(5-fluoro-1H-indol-3-yl)propyl]pyrrolidin-3-yl]-1-methyl-indole-5-sulphonamide 1417311-39-7 C24H27FN4O2S
N-[1-[3-(5-fluoro-1H-indol-3-yl)propyl]pyrrolidin-3-yl]-1-methyl-indole-5-sulphonamide
—— 6-chloro-N-[[1-[2-(1-naphthyloxy)ethyl]pyrrolidin-3-yl]methyl]benzothiophene-2-sulphonamide 1417310-43-0 C25H25ClN2O3S2
6-chloro-N-[[1-[2-(1-naphthyloxy)ethyl]pyrrolidin-3-yl]methyl]benzothiophene-2-sulphonamide
—— 4-fluoro-N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]methyl]benzenesulphonamide 1417310-26-9 C21H23F2N3O3S
4-fluoro-N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]methyl]benzenesulphonamide
—— (S)-ethyl 2-(3-(4-(5-methyl-1,3,4-oxadiazol-2-yl)phenoxy)-5-((1-methyl-2-oxopyrrolidin-3-yl)oxy)benzamido)thiazole-4-carboxylate 1263402-78-3 C27H25N5O7S
(S)-ethyl 2-(3-(4-(5-methyl-1,3,4-oxadiazol-2-yl)phenoxy)-5-((1-methyl-2-oxopyrrolidin-3-yl)oxy)benzamido)thiazole-4-carboxylate
—— 4-[4-Cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2-oxazol-3-yl]-6-(2,5-dimethylanilino)-6-oxohexanoic acid 1404378-00-2 C28H38N2O4
4-[4-Cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2-oxazol-3-yl]-6-(2,5-dimethylanilino)-6-oxohexanoic acid
—— (3-fluoro-4-morpholin-4-yl-phenyl)-(8-methoxy-2H-pyrazolo[3,4-c]quinolin-4-yl)-amine 1403886-72-5 C21H20FN5O2
(3-fluoro-4-morpholin-4-yl-phenyl)-(8-methoxy-2H-pyrazolo[3,4-c]quinolin-4-yl)-amine
—— (phenylmethyl) cis,cis-9-[(3(R)-carboxy-1-oxobutyl)ethylamino]-1,2,3,3a,9,9a-hexahydro-4H-cyclopenta[b]quinoline-4-carboxylate 1416606-47-7 C27H32N2O5
(phenylmethyl) cis,cis-9-[(3(R)-carboxy-1-oxobutyl)ethylamino]-1,2,3,3a,9,9a-hexahydro-4H-cyclopenta[b]quinoline-4-carboxylate
—— (E)-4-(6-(2-(2,4-difluorophenyl)-1,1-difluoro-2-hydroxy-3-(1H-tetrazol-1-yl)propyl)pyridin-3-yl)but-3-en-2-ol 1416732-80-3 C19H17F4N5O2
(E)-4-(6-(2-(2,4-difluorophenyl)-1,1-difluoro-2-hydroxy-3-(1H-tetrazol-1-yl)propyl)pyridin-3-yl)but-3-en-2-ol
—— (8R,11S,14R,17S)-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-14-[[3-(trifluoromethyl)phenyl]methyl]-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211436-73-5 C45H42F3N5O7S
(8R,11S,14R,17S)-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-14-[[3-(trifluoromethyl)phenyl]methyl]-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— (S)-N-((8-chloro-quinolin-3-yl)(3-(trifluoromethyl)pyridin-2-yl)-methyl)quinoline-7-carboxamide 1416794-52-9 C26H16ClF3N4O
(S)-N-((8-chloro-quinolin-3-yl)(3-(trifluoromethyl)pyridin-2-yl)-methyl)quinoline-7-carboxamide
—— 4-fluoro-N-[1-[2-(1H-indol-4-yloxy)ethyl]azetidin-3-yl]benzenesulphonamide 1417308-16-7 C19H20FN3O3S
4-fluoro-N-[1-[2-(1H-indol-4-yloxy)ethyl]azetidin-3-yl]benzenesulphonamide
—— 1-(((5S,7S)-2-oxo-3-(3-(trifluoromethyl)benzyl)-1-oxa-3-azaspiro[4.5]decan-7-yl)methyl)-1H-benzo[d]imidazole-6-carbonitrile 1416323-76-6 C25H23F3N4O2
1-(((5S,7S)-2-oxo-3-(3-(trifluoromethyl)benzyl)-1-oxa-3-azaspiro[4.5]decan-7-yl)methyl)-1H-benzo[d]imidazole-6-carbonitrile
—— cyclopentyl (2S)-{[2-(1-{[2,4-dihydroxy-5-(propan-2-yl)phenyl]carbonyl}piperidin-4-yl)ethyl]amino}(phenyl)ethanoate 1351814-49-7 C30H40N2O5
cyclopentyl (2S)-{[2-(1-{[2,4-dihydroxy-5-(propan-2-yl)phenyl]carbonyl}piperidin-4-yl)ethyl]amino}(phenyl)ethanoate
—— 2,2,2-trifluoro-1-(1-methyl-1H-imidazol-2-yl)ethyl {2-[1-(6-chloroquinolin-2-yl)piperidin-4-yl]ethyl}carbamate 1227245-37-5 C23H25ClF3N5O2
2,2,2-trifluoro-1-(1-methyl-1H-imidazol-2-yl)ethyl {2-[1-(6-chloroquinolin-2-yl)piperidin-4-yl]ethyl}carbamate
—— (3S)-3-(4-fluorophenyl)-10-[[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]methylidene]-3,4,5,7,8,9-hexahydropyrido[2,1-c][1,2,4]oxadiazepine 1227081-91-5 C26H27FN4O2
(3S)-3-(4-fluorophenyl)-10-[[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]methylidene]-3,4,5,7,8,9-hexahydropyrido[2,1-c][1,2,4]oxadiazepine
—— (S)-N-((3-fluoro-pyridin-2-yl)(4-(trifluoromethyl)phenyl)methyl)-6-methylnicotinamide 1416794-99-4 C20H15F4N3O
(S)-N-((3-fluoro-pyridin-2-yl)(4-(trifluoromethyl)phenyl)methyl)-6-methylnicotinamide
—— 4-[3-(Fluoromethyl)pyrrolidin-1-yl]-6-[2-(2-quinolyl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one 1417186-25-4 C23H23FN4O
4-[3-(Fluoromethyl)pyrrolidin-1-yl]-6-[2-(2-quinolyl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (4R,5R,8S,11R,14S,17R)-14-benzyl-4,5-dihydroxy-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211439-54-1 C44H43N5O9S
(4R,5R,8S,11R,14S,17R)-14-benzyl-4,5-dihydroxy-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— 4-[[[2-[2-Methoxy-4-[4-[4-(oxan-4-yl)piperazin-1-yl]piperidin-1-yl]anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-1,3-dihydroindol-2-one 1383681-37-5 C35H43F3N8O3
4-[[[2-[2-Methoxy-4-[4-[4-(oxan-4-yl)piperazin-1-yl]piperidin-1-yl]anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-1,3-dihydroindol-2-one
—— 3-fluoro-N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]azetidin-3-yl]methyl]benzenesulphonamide 1417309-18-2 C20H21F2N3O3S
3-fluoro-N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]azetidin-3-yl]methyl]benzenesulphonamide
—— (4R,9R,12R,15S,18R,21S)-18-benzyl-3,10,13,16,19-pentaoxo-15-[(4-phenylphenyl)methyl]-12-(thiophen-2-ylmethyl)-2,11,14,17,20-pentazatricyclo[21.2.2.04,9]heptacosa-1(26),23(27),24-triene-21-carboxylic acid 1211435-73-2 C48H49N5O7S
(4R,9R,12R,15S,18R,21S)-18-benzyl-3,10,13,16,19-pentaoxo-15-[(4-phenylphenyl)methyl]-12-(thiophen-2-ylmethyl)-2,11,14,17,20-pentazatricyclo[21.2.2.04,9]heptacosa-1(26),23(27),24-triene-21-carboxylic acid
—— 5-(2,4-Dimethylanilino)-3-[4-ethyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2-oxazol-3-yl]-5-oxopentanoic acid 1404377-73-6 C26H36N2O4
5-(2,4-Dimethylanilino)-3-[4-ethyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2-oxazol-3-yl]-5-oxopentanoic acid
—— 1-(((5S,7S)-3-(2,2-dimethylbutyl)-2-oxo-1-oxa-3-azaspiro[4.5]decan-7-yl)methyl)-1H-benzo[d]imidazole-6-carbonitrile 1416507-07-7 C23H30N4O2
1-(((5S,7S)-3-(2,2-dimethylbutyl)-2-oxo-1-oxa-3-azaspiro[4.5]decan-7-yl)methyl)-1H-benzo[d]imidazole-6-carbonitrile
—— (8R,11S,14R,17S)-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-14-(thiophen-3-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211436-70-2 C42H41N5O7S2
(8R,11S,14R,17S)-3,6,9,12,15-pentaoxo-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-14-(thiophen-3-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— 1-{1-[2-(2,3-dihydro-1,4-benzodioxan-5-yloxy)ethyl]piperidin-4-yl}methaneamine 1417311-89-7 C16H24N2O3
1-{1-[2-(2,3-dihydro-1,4-benzodioxan-5-yloxy)ethyl]piperidin-4-yl}methaneamine
—— N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]azetidin-3-yl]methyl]-1-methyl-indole-4-sulphonamide 1417309-26-2 C23H25FN4O3S
N-[[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]azetidin-3-yl]methyl]-1-methyl-indole-4-sulphonamide
—— N-[1-[2-(1H-indol-4-yloxy)ethyl]-4-piperidine]-4-(trifluoromethyl)benzene-1-sulphonamide 1417308-29-2 C22H24F3N3O3S
N-[1-[2-(1H-indol-4-yloxy)ethyl]-4-piperidine]-4-(trifluoromethyl)benzene-1-sulphonamide
—— N-[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]-6-methoxynaphthalene-2-sulphonamide 1417310-01-0 C25H26FN3O4S
N-[1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]pyrrolidin-3-yl]-6-methoxynaphthalene-2-sulphonamide
—— 4-bromo-5-methyl-[3,4']bipyridinyl 1417190-16-9 C11H9BrN2
4-bromo-5-methyl-[3,4']bipyridinyl
—— (3,5-Difluoro-2-iodophenyl)-di(propan-2-yl)-pyridin-2-ylsilane 1312936-53-0 C17H20F2INSi
(3,5-Difluoro-2-iodophenyl)-di(propan-2-yl)-pyridin-2-ylsilane
—— ethyl 2-diazo-2-(4-tert-butyl-1-hydroxycyclohexyl)acetate 1290044-64-2 C14H24N2O3
ethyl 2-diazo-2-(4-tert-butyl-1-hydroxycyclohexyl)acetate
—— 1-(4-methanesulfonylphenyl)-3,6-dimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid ethyl ester 1417332-93-4 C18H19N3O4S
1-(4-methanesulfonylphenyl)-3,6-dimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid ethyl ester
—— (S)-N-((3-fluoro-pyridin-2-yl)(4-(trifluoromethyl)phenyl)methyl)-2-oxo-2,3-dihydrobenzo[d]oxazole-5-carboxamide 1416795-23-7 C21H13F4N3O3
(S)-N-((3-fluoro-pyridin-2-yl)(4-(trifluoromethyl)phenyl)methyl)-2-oxo-2,3-dihydrobenzo[d]oxazole-5-carboxamide
—— 1-(4-{3-[(4,4-difluoro-1,4'-bipiperidin-1'-yl)carbonyl]-2-methyl-1H-indol-1-yl}phenyl)-3-(pyridin-3-ylmethyl)urea 1416890-71-5 C33H36F2N6O2
1-(4-{3-[(4,4-difluoro-1,4'-bipiperidin-1'-yl)carbonyl]-2-methyl-1H-indol-1-yl}phenyl)-3-(pyridin-3-ylmethyl)urea
—— 4-(4-methoxyphenyl)-1-[(E)-2-(3-methoxyphenyl)ethenyl]triazole 1293362-76-1 C18H17N3O2
4-(4-methoxyphenyl)-1-[(E)-2-(3-methoxyphenyl)ethenyl]triazole
—— 5-bromo-3-hydroxy-3-(2-hydroxyethyl)indolin-2-one 1214919-15-9 C10H10BrNO3
5-bromo-3-hydroxy-3-(2-hydroxyethyl)indolin-2-one
—— diethyl 3-methyl-4-phenyl-4,5-dihydroisoxazole-5,5-dicarboxylate 2-oxide 1354650-84-2 C16H19NO6
diethyl 3-methyl-4-phenyl-4,5-dihydroisoxazole-5,5-dicarboxylate 2-oxide