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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl 5-iodo-7-(3-nitrophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylcarbamate 1422828-23-6 C17H16IN5O4
tert-butyl 5-iodo-7-(3-nitrophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylcarbamate
—— (2S,5R)-methyl 5-(2,4-dichlorophenyl)pyrrolidine-2-carboxylate 1312804-35-5 C12H13Cl2NO2
(2S,5R)-methyl 5-(2,4-dichlorophenyl)pyrrolidine-2-carboxylate
—— 4-tert-butyl-N-{3-[6-(4-dimethylamino-cyclohex-1-enyl)-7H-pyrrolo[2,3-d]pyrimidine-4-yl]-2-methyl-phenyl}-benzamide 1418128-30-9 C32H37N5O
4-tert-butyl-N-{3-[6-(4-dimethylamino-cyclohex-1-enyl)-7H-pyrrolo[2,3-d]pyrimidine-4-yl]-2-methyl-phenyl}-benzamide
—— 2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-6-phenyl-8-(pyridin-3-yl)pyrimido[4,5-d]pyridazin-5(6H)-one 1419770-46-9 C28H26N8O
2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-6-phenyl-8-(pyridin-3-yl)pyrimido[4,5-d]pyridazin-5(6H)-one
—— {3-[2-{[(cyclopropylcarbonyl)(ethyl)amino]methyl}-4-(trifluoromethyl)phenyl]-4,5-difluoro-1H-indol-1-yl}acetic acid 1420070-17-2 C24H21F5N2O3
{3-[2-{[(cyclopropylcarbonyl)(ethyl)amino]methyl}-4-(trifluoromethyl)phenyl]-4,5-difluoro-1H-indol-1-yl}acetic acid
—— 6-(2-chloro-6-methylphenyl)-8-methyl-2-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)pyrimido[4,5-d]pyridazin-5(6H)-one 1419789-39-1 C23H21ClN6O
6-(2-chloro-6-methylphenyl)-8-methyl-2-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)pyrimido[4,5-d]pyridazin-5(6H)-one
—— methyl-1H-[1,2,3]triazole-4-carboxylic acid (7-chloro-4-oxo-1-phenyl-1,4-dihydro-quinolin-3-ylmethyl)amide 1418024-05-1 C20H16ClN5O2
methyl-1H-[1,2,3]triazole-4-carboxylic acid (7-chloro-4-oxo-1-phenyl-1,4-dihydro-quinolin-3-ylmethyl)amide
—— 1-{[(5S,7S)-3-({4-[3-methyl-4-(methyloxy)phenyl]-1,3-thiazol-2-yl}methyl)-2-oxo-1-oxa-3-azaspiro[4.5]dec-7-yl]methyl}-1H-benzimidazole-6-carbonitrile 1419609-18-9 C29H29N5O3S
1-{[(5S,7S)-3-({4-[3-methyl-4-(methyloxy)phenyl]-1,3-thiazol-2-yl}methyl)-2-oxo-1-oxa-3-azaspiro[4.5]dec-7-yl]methyl}-1H-benzimidazole-6-carbonitrile
—— 6-(2,6-dichlorophenyl)-8-methyl-2-{[2-(methylsulfonyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]amino}pyrimido[4,5-d]pyridazin-5(6H)-one 1419788-44-5 C23H20Cl2N6O3S
6-(2,6-dichlorophenyl)-8-methyl-2-{[2-(methylsulfonyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]amino}pyrimido[4,5-d]pyridazin-5(6H)-one
—— (3-hydroxy-1-piperidyl)-[2-(4-isopropylsulfonylphenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]methanone 1416773-56-2 C21H24N4O4S
(3-hydroxy-1-piperidyl)-[2-(4-isopropylsulfonylphenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]methanone
—— [4-[2-(dimethylamino)ethyl]piperazin-1-yl]-[5-[(4-pyridin-2-ylpyrimidin-2-yl)amino]-1H-indol-2-yl]methanone 1391600-71-7 C26H30N8O
[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-[5-[(4-pyridin-2-ylpyrimidin-2-yl)amino]-1H-indol-2-yl]methanone
—— N-benzyl-4-(3-chloro-4-methoxybenzyloxy)-2-(6-azaspiro[2.5]octan-6-yl)pyrimidine-5-carboxamide 1418759-20-2 C27H29ClN4O3
N-benzyl-4-(3-chloro-4-methoxybenzyloxy)-2-(6-azaspiro[2.5]octan-6-yl)pyrimidine-5-carboxamide
—— 6-(2,6-dichlorophenyl)-2-(2',3'-dihydro-1'H-spiro[cyclopropane-1,4'-isoquinolin]-7'-ylamino)-8-(1-methyl-1H-imidazol-4-yl)pyrimido[4,5-d]pyridazin-5(6H)-one 1419781-24-0 C27H22Cl2N8O
6-(2,6-dichlorophenyl)-2-(2',3'-dihydro-1'H-spiro[cyclopropane-1,4'-isoquinolin]-7'-ylamino)-8-(1-methyl-1H-imidazol-4-yl)pyrimido[4,5-d]pyridazin-5(6H)-one
—— (R)-N-(1-(dimethylamino)-3-methylbutan-2-yl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide 1418292-66-6 C17H21F3N4O2
(R)-N-(1-(dimethylamino)-3-methylbutan-2-yl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide
—— 2-[4-(4-fluoro-2-methoxyphenyl)piperazin-1-ylmethyl]pyrrolo[1,2-a]quinazolin-5(4H)-one 1417562-76-5 C23H23FN4O2
2-[4-(4-fluoro-2-methoxyphenyl)piperazin-1-ylmethyl]pyrrolo[1,2-a]quinazolin-5(4H)-one
—— N-{2-[1-(4,4-Difluoro-tetrahydro-pyran-3-yl)-1,6-dihydro-1,3,5,6-tetraaza-as-indacen-2-yl]-ethyl}-methanesulfonamide 1418199-55-9 C16H19F2N5O3S
N-{2-[1-(4,4-Difluoro-tetrahydro-pyran-3-yl)-1,6-dihydro-1,3,5,6-tetraaza-as-indacen-2-yl]-ethyl}-methanesulfonamide
—— 6-(2,6-dichlorophenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-8-[3-(piperidin-1-ylmethyl)phenyl]pyrimido[4,5-d]pyridazin-5(6H)-one 1419773-31-1 C35H36Cl2N8O
6-(2,6-dichlorophenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-8-[3-(piperidin-1-ylmethyl)phenyl]pyrimido[4,5-d]pyridazin-5(6H)-one
—— (2R,3R,4R,5R)-2-(4-aminopyrrolo[2,3-d]pyrimidin-7-yl)-5-[(1R)-1-hydroxypropyl]-3-methyloxolane-3,4-diol 1417563-25-7 C14H20N4O4
(2R,3R,4R,5R)-2-(4-aminopyrrolo[2,3-d]pyrimidin-7-yl)-5-[(1R)-1-hydroxypropyl]-3-methyloxolane-3,4-diol
—— N-[4-(4-methylpiperazin-1-yl)phenyl]-9-phenyl-6-propyl-6H-pyrimido[5,4-c][2,1]benzothiazin-2-amine 5,5-dioxide 1418315-79-3 C30H32N6O2S
N-[4-(4-methylpiperazin-1-yl)phenyl]-9-phenyl-6-propyl-6H-pyrimido[5,4-c][2,1]benzothiazin-2-amine 5,5-dioxide
—— N-(2-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)propyl)-3-methyloxetane-3-carboxamide 1419214-99-5 C27H26F3N7O3
N-(2-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)propyl)-3-methyloxetane-3-carboxamide
—— 2-{[4-(4-isopropylpiperazin-1-yl)-3-methylphenyl]amino}-6-(2-methylphenyl)-8-(2-thienyl)pyrimido[4,5-d]pyridazin-5(6H)-one 1419771-71-3 C31H33N7OS
2-{[4-(4-isopropylpiperazin-1-yl)-3-methylphenyl]amino}-6-(2-methylphenyl)-8-(2-thienyl)pyrimido[4,5-d]pyridazin-5(6H)-one
—— 6-(2,6-dichlorophenyl)-2-[(1,1-dimethyl-1,2,3,4-tetrahydroisoquinolin-6-yl)amino]-8-methylpyrimido[4,5-d]pyridazin-5(6H)-one 1419788-52-5 C24H22Cl2N6O
6-(2,6-dichlorophenyl)-2-[(1,1-dimethyl-1,2,3,4-tetrahydroisoquinolin-6-yl)amino]-8-methylpyrimido[4,5-d]pyridazin-5(6H)-one
—— 6-(3-chloropyridin-2-yl)-8-(1-methyl-1H-imidazol-4-yl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimido[4,5-d]pyridazin-5(6H)-one 1419781-36-4 C26H25ClN10O
6-(3-chloropyridin-2-yl)-8-(1-methyl-1H-imidazol-4-yl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimido[4,5-d]pyridazin-5(6H)-one
—— N-(4-carbamoylphenyl)-2-(4-isopropylsulfonylphenyl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 1416773-81-3 C23H21N5O4S
N-(4-carbamoylphenyl)-2-(4-isopropylsulfonylphenyl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide
—— N-[4-(4-methylpiperazin-1-yl)phenyl]-6-propyl-8-(1H-pyrazol-4-yl)-6H-pyrimido[5,4-c][2,1]benzothiazin-2-amine 5,5-dioxide 1418315-52-2 C27H30N8O2S
N-[4-(4-methylpiperazin-1-yl)phenyl]-6-propyl-8-(1H-pyrazol-4-yl)-6H-pyrimido[5,4-c][2,1]benzothiazin-2-amine 5,5-dioxide
—— [3-(3,4-dimethoxyphenyl)-4,5-dihydropyrazol-1-yl]-(3-trifluoromethoxyphenyl)methanone 1417707-28-8 C19H17F3N2O4
[3-(3,4-dimethoxyphenyl)-4,5-dihydropyrazol-1-yl]-(3-trifluoromethoxyphenyl)methanone
—— 6-(2-chlorophenyl)-2-({3-methyl-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-8-phenylpyrimido[4,5-d]pyridazin-5(6H)-one 1419775-69-1 C32H32ClN7O
6-(2-chlorophenyl)-2-({3-methyl-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-8-phenylpyrimido[4,5-d]pyridazin-5(6H)-one
—— 3-tert-butyl-1-(1-methyl-1H-indol-5-yl)imidazo[1,5-a]pyrazin-8-amine 1320266-66-7 C19H21N5
3-tert-butyl-1-(1-methyl-1H-indol-5-yl)imidazo[1,5-a]pyrazin-8-amine
—— N-(2-(4-(isopropylsulfonyl)phenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl)-2-methoxybenzamide 1416739-81-5 C23H22N4O4S
N-(2-(4-(isopropylsulfonyl)phenyl)-5H-pyrrolo[2,3-b]pyrazin-7-yl)-2-methoxybenzamide
—— (R)-4-(4-amino-1-(1-isobutyrylpiperidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide 1419217-09-6 C27H27F3N8O2
(R)-4-(4-amino-1-(1-isobutyrylpiperidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-4-(8-amino-3-(1-(4-(dimethylamino)butanoyl)pyrrolidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide 1419214-88-2 C28H32N8O2
(R)-4-(8-amino-3-(1-(4-(dimethylamino)butanoyl)pyrrolidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide
—— 2-(4-isopropylsulfonylphenyl)-N-(4-pyridylmethyl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide 1416773-94-8 C22H21N5O3S
2-(4-isopropylsulfonylphenyl)-N-(4-pyridylmethyl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxamide
—— 8-chloro-3-[(1S)-1-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)amino]ethyl]-2-phenylisoquinolin-1-one 1420829-95-3 C25H21ClN4OS
8-chloro-3-[(1S)-1-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)amino]ethyl]-2-phenylisoquinolin-1-one
—— (5R)-5-{4-[4-(1H-pyrazol-3-yl)phenoxy]phenoxy}piperidin-2-one 1419210-66-4 C20H19N3O3
(5R)-5-{4-[4-(1H-pyrazol-3-yl)phenoxy]phenoxy}piperidin-2-one
—— (13S)-3-fluoro-8-methoxy-13-methyl-11-propan-2-yl-1,4,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2(7),3,8-triene-6,10-dione 1338075-11-8 C14H17FN4O3
(13S)-3-fluoro-8-methoxy-13-methyl-11-propan-2-yl-1,4,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2(7),3,8-triene-6,10-dione
—— N-(5-hydroxyadamantane-2-yl)-2-methyl-2-(2-methyl-5-nitrophenylsulfonamido)propanamide 1422025-18-0 C21H29N3O6S
N-(5-hydroxyadamantane-2-yl)-2-methyl-2-(2-methyl-5-nitrophenylsulfonamido)propanamide
—— 5'-(2-chloro-oxazol-5-yl)-[1,3']bipyridinyl-2-one 1420998-68-0 C13H8ClN3O2
5'-(2-chloro-oxazol-5-yl)-[1,3']bipyridinyl-2-one
—— N-(2,3-Dihydro-furo[2,3-b]pyridin-3-yl)-2-(2,4,6-trifluoro-phenyl)-acetamide 1421618-97-4 C15H11F3N2O2
N-(2,3-Dihydro-furo[2,3-b]pyridin-3-yl)-2-(2,4,6-trifluoro-phenyl)-acetamide
—— 5-{4-[4-(tetrahydrofuran-3-ylmethoxy)phenoxy]phenyl}-1H-pyrazole 1419211-42-9 C20H20N2O3
5-{4-[4-(tetrahydrofuran-3-ylmethoxy)phenoxy]phenyl}-1H-pyrazole
—— 6-(2-chloro-6-fluorophenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-8-(pyridin-4-yl)pyrimido[4,5-d]pyridazin-5(6H)-one 1419779-39-7 C28H24ClFN8O
6-(2-chloro-6-fluorophenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-8-(pyridin-4-yl)pyrimido[4,5-d]pyridazin-5(6H)-one
—— 6-(5-isopropyl-2-methylphenyl)-2-(5-methyl-1H-indazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine 1421251-42-4 C26H28N4
6-(5-isopropyl-2-methylphenyl)-2-(5-methyl-1H-indazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine
—— 2-(2-bromo-5-methylbenzyl)-1-cyclopropylbutane-1,3-dione 1420532-68-8 C15H17BrO2
2-(2-bromo-5-methylbenzyl)-1-cyclopropylbutane-1,3-dione
—— N4-(5-fluoro-1H-indazol-3-yl)-N2-[2-methyl-3-(methylsulfonyl)phenyl]-2,4-pyrimidinediamine 1335499-88-1 C19H17FN6O2S
N4-(5-fluoro-1H-indazol-3-yl)-N2-[2-methyl-3-(methylsulfonyl)phenyl]-2,4-pyrimidinediamine
—— tert-butyl 4-(2-(1H-indol-3-yl)-2-oxoacetyl)-3-(1H-indol-3-yl)piperazine-1-carboxylate 1420071-96-0 C27H28N4O4
tert-butyl 4-(2-(1H-indol-3-yl)-2-oxoacetyl)-3-(1H-indol-3-yl)piperazine-1-carboxylate
—— 4-cyclopropyl-N-(5-fluoro-2-methyl-3-{6-[1-(pyrrolidine-1-carbonyl)-1,2,3,6-tetrahydro-pyridine-4-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-yl}-phenyl)-benzamide 1418127-92-0 C33H33FN6O2
4-cyclopropyl-N-(5-fluoro-2-methyl-3-{6-[1-(pyrrolidine-1-carbonyl)-1,2,3,6-tetrahydro-pyridine-4-yl]-7H-pyrrolo[2,3-d]pyrimidine-4-yl}-phenyl)-benzamide
—— 7-((3-fluoro-4-((5-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-1-methyl-2,3-dihydroimidazo[1,2-c]pyrimidin-5(1H)-one 1421433-53-5 C20H16F4N4O3
7-((3-fluoro-4-((5-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-1-methyl-2,3-dihydroimidazo[1,2-c]pyrimidin-5(1H)-one
—— 3-[(1S)-1-[(2-aminopyrido[3,2-d]pyrimidin-4-yl)amino]ethyl]-8-(1-methylpyrazol-4-yl)-2-phenylisoquinolin-1-one 1420618-87-6 C28H24N8O
3-[(1S)-1-[(2-aminopyrido[3,2-d]pyrimidin-4-yl)amino]ethyl]-8-(1-methylpyrazol-4-yl)-2-phenylisoquinolin-1-one
—— 5-Methyl-furan-2-carboxylic acid [5-cyclopropylcarbamoyl-2-(4-o-tolyl-piperazin-1-yl)-phenyl]amide 1419867-83-6 C27H30N4O3
5-Methyl-furan-2-carboxylic acid [5-cyclopropylcarbamoyl-2-(4-o-tolyl-piperazin-1-yl)-phenyl]amide
—— (S)-4-(8-amino-3-(pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-propylpyridin-2-yl)benzamide 1420478-93-8 C25H27N7O
(S)-4-(8-amino-3-(pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-propylpyridin-2-yl)benzamide
—— N-[5-[2-[2-(2-acetamidoethoxy)ethoxy]ethylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]-2-cyclopropyl-1,3-oxazole-4-carboxamide 1419869-76-3 C33H42N6O6
N-[5-[2-[2-(2-acetamidoethoxy)ethoxy]ethylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]-2-cyclopropyl-1,3-oxazole-4-carboxamide