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中文名称 英文名称 CAS号 化学式 结构式图片
—— —— 125107-73-5 C11H14ClNO2
—— 2,2-Dimethoxy-3,3,3-trifluorpropansaeuremethylester 14918-87-7 C6H9F3O4
2,2-Dimethoxy-3,3,3-trifluorpropansaeuremethylester
—— 4'-hydroxy-5'-(4-methoxy-phenyl)-1-methyl-2',4'-dihydro-1<i>H</i>-spiro[indole-3,3'-pyrazol]-2-one 15970-16-8 C18H17N3O3
4'-hydroxy-5'-(4-methoxy-phenyl)-1-methyl-2',4'-dihydro-1<i>H</i>-spiro[indole-3,3'-pyrazol]-2-one
—— 4-[(2E,4E)-5-Dimethylamino-4-(4-octyl-phenyl)-penta-2,4-dienoyl]-benzonitrile 101667-69-0 C28H34N2O
4-[(2E,4E)-5-Dimethylamino-4-(4-octyl-phenyl)-penta-2,4-dienoyl]-benzonitrile
—— 2-iodophenyl 4-methoxyphenylsulfonate 136859-43-3 C13H11IO4S
2-iodophenyl 4-methoxyphenylsulfonate
—— dimethylamino-[dimethyl-[(C-methyl-N-propan-2-ylcarbonimidoyl)-propan-2-ylamino]silyl]azanide;1,2,3,4,5-pentamethylcyclopenta-1,3-diene;titanium(4+);dichloride 1361315-73-2 C22H44Cl2N4SiTi
dimethylamino-[dimethyl-[(C-methyl-N-propan-2-ylcarbonimidoyl)-propan-2-ylamino]silyl]azanide;1,2,3,4,5-pentamethylcyclopenta-1,3-diene;titanium(4+);dichloride
—— 4-[5-(1-{[(3S,4R)-1-tertbutyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl]carbonyl}-piperidin-4-yl)-3-methyl-1H-pyrazol-1-yl]-3-chloro-benzonitrile 1352245-61-4 C31H34ClF2N5O
4-[5-(1-{[(3S,4R)-1-tertbutyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl]carbonyl}-piperidin-4-yl)-3-methyl-1H-pyrazol-1-yl]-3-chloro-benzonitrile
—— 6-biphenyl-3-ylpyridin-3-ylamine 1357165-91-3 C17H14N2
6-biphenyl-3-ylpyridin-3-ylamine
—— (±)-2-{3-[5-fluoro-2-((1R,2R)-2-phenylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-4-methoxyphenyl}propionic acid 1445885-55-1 C29H28FNO4
(±)-2-{3-[5-fluoro-2-((1R,2R)-2-phenylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-4-methoxyphenyl}propionic acid
—— (R)-2-(5-(tert-butyl)thiophene-2-carboxamido)-3-(4-(5-(4-(heptyloxy)phenyl)pyrimidin-2-yl)phenyl)propanoic acid 1443789-99-8 C35H41N3O4S
(R)-2-(5-(tert-butyl)thiophene-2-carboxamido)-3-(4-(5-(4-(heptyloxy)phenyl)pyrimidin-2-yl)phenyl)propanoic acid
—— methyl 3-(3-methoxy-4-propoxyphenyl)-3-(4,6-dioxo-4H-thiophene[3,4-c]pyrrole-5(6H)-yl)propionate 1026995-80-1 C20H21NO6S
methyl 3-(3-methoxy-4-propoxyphenyl)-3-(4,6-dioxo-4H-thiophene[3,4-c]pyrrole-5(6H)-yl)propionate
—— N-[(1R,2R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]-6-[4-(2-methoxyethoxy)phenyl]-6-oxohexanamide 1092470-17-1 C30H40N2O7
N-[(1R,2R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]-6-[4-(2-methoxyethoxy)phenyl]-6-oxohexanamide
—— methyl N-benzyl-N-[(1-{[(tert-butoxycarbonyl)amino]methyl}cyclopropyl)carbonyl]-L-alaninate 1149352-56-6 C21H30N2O5
methyl N-benzyl-N-[(1-{[(tert-butoxycarbonyl)amino]methyl}cyclopropyl)carbonyl]-L-alaninate
—— N-[[(5S)-3-[3,5-difluoro-4-[2-(5-nitrofuran-2-carbonyl)-1,2,5-oxadiazepan-5-yl]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]acetamide 1138150-23-8 C21H21F2N5O8
N-[[(5S)-3-[3,5-difluoro-4-[2-(5-nitrofuran-2-carbonyl)-1,2,5-oxadiazepan-5-yl]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]acetamide
—— 6-benzyl-N-(cycloheptylmethyl)-2,6,7,8-tetrahydro-1,2,3,5,6-pentaazaacenaphthylen-4-amine 1246670-14-3 C22H28N6
6-benzyl-N-(cycloheptylmethyl)-2,6,7,8-tetrahydro-1,2,3,5,6-pentaazaacenaphthylen-4-amine
—— 2-chloro-4-{[(2,4-difluorophenyl)methyl][(3S)-1-(1-methylpropyl)-5-oxo-3-pyrrolidinyl]amino}benzonitrile 1006035-23-9 C22H22ClF2N3O
2-chloro-4-{[(2,4-difluorophenyl)methyl][(3S)-1-(1-methylpropyl)-5-oxo-3-pyrrolidinyl]amino}benzonitrile
—— (6-Methoxy-3-methyl-4-phenylmethoxyquinolin-2-yl)methyl acetate 1135033-21-4 C21H21NO4
(6-Methoxy-3-methyl-4-phenylmethoxyquinolin-2-yl)methyl acetate
—— 1-(5-Methoxy-1,3-dihydroisoindol-2-yl)-2-[3-(4-methoxyphenyl)-5-propan-2-ylpyrazol-1-yl]ethanone 1440952-33-9 C24H27N3O3
1-(5-Methoxy-1,3-dihydroisoindol-2-yl)-2-[3-(4-methoxyphenyl)-5-propan-2-ylpyrazol-1-yl]ethanone
—— 1-(4-(8-(1-methyl-1H-pyrazol-4-yl)-2-phenyl-9H-purin-9-yl)phenyl)cyclobutanamine 1439392-57-0 C25H23N7
1-(4-(8-(1-methyl-1H-pyrazol-4-yl)-2-phenyl-9H-purin-9-yl)phenyl)cyclobutanamine
—— N-[[1-[5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl]-4-piperidyl]methyl]cyclopropanamine 1437771-23-7 C21H23FN4S
N-[[1-[5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl]-4-piperidyl]methyl]cyclopropanamine
—— tert-butyl [(1R)-2-({4-[2-({4-[(3-fluoroazetidin-1-yl)carbonyl]-2-(2,2,2-trifluoroethoxy)phenyl}amino)[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl}amino)-1-(4-fluorophenyl)-2-oxoethyl]carbamate 1443764-29-1 C37H34F5N7O5
tert-butyl [(1R)-2-({4-[2-({4-[(3-fluoroazetidin-1-yl)carbonyl]-2-(2,2,2-trifluoroethoxy)phenyl}amino)[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl}amino)-1-(4-fluorophenyl)-2-oxoethyl]carbamate
—— methyl 3-(3-isopropoxy-4-methoxyphenyl)-3-(4,6-dioxo-4H-thiophene[3,4-c]pyrrole-5(6H)-yl)propionate 1026995-76-5 C20H21NO6S
methyl 3-(3-isopropoxy-4-methoxyphenyl)-3-(4,6-dioxo-4H-thiophene[3,4-c]pyrrole-5(6H)-yl)propionate
—— 2-[3-(4-Fluoro-3-methylphenyl)-5-propylpyrazol-1-yl]-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperazin-1-yl]ethanone 1440954-30-2 C22H27FN6O2
2-[3-(4-Fluoro-3-methylphenyl)-5-propylpyrazol-1-yl]-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperazin-1-yl]ethanone
—— US9598416, Example 76 1443617-35-3 C22H25N5O2S
US9598416, Example 76
—— (1R,6S)-tert-butyl 3-(6-nitropyridin-3-yl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate 1331847-75-6 C17H22N4O5
(1R,6S)-tert-butyl 3-(6-nitropyridin-3-yl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
—— 4-[5-[5-chloro-1-(4-methoxy-benzyl)-2-oxo-1,2-dihydro-pyridin-3-yl]-2-(2,4-dimethoxy-pyrimidin-5-yl)-3-isopropyl-6-oxo-2,4,5,6-tetrahydro-pyrrolo[3,4-c]pyrazol-4-yl]-benzonitrile 1441764-24-4 C34H30ClN7O5
4-[5-[5-chloro-1-(4-methoxy-benzyl)-2-oxo-1,2-dihydro-pyridin-3-yl]-2-(2,4-dimethoxy-pyrimidin-5-yl)-3-isopropyl-6-oxo-2,4,5,6-tetrahydro-pyrrolo[3,4-c]pyrazol-4-yl]-benzonitrile
—— N<sup>2</sup>-(5-fluoropyridin-3-yl)-N<sup>4</sup>-isopropyl-6-phenyl-1,3,5-triazine-2,4-diamine 1446501-16-1 C17H17FN6
N<sup>2</sup>-(5-fluoropyridin-3-yl)-N<sup>4</sup>-isopropyl-6-phenyl-1,3,5-triazine-2,4-diamine
—— (1,1-dioxo-tetrahydro-1lambda*6*-thiophen-3-yl)-{(S)-3-[4-(5-fluoro-6-methoxy-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-methanone 1446000-16-3 C23H26FN3O6S
(1,1-dioxo-tetrahydro-1lambda*6*-thiophen-3-yl)-{(S)-3-[4-(5-fluoro-6-methoxy-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-methanone
—— SR-3306 1128096-91-2 C28H26N8O
SR-3306
—— N-{4-[(cyclopentylmethyl)carbamoyl]phenyl}-5-fluoro-1,3-dihydro-2H-isoindole-2-carboxamide 1375542-67-8 C22H24FN3O2
N-{4-[(cyclopentylmethyl)carbamoyl]phenyl}-5-fluoro-1,3-dihydro-2H-isoindole-2-carboxamide
—— 5-amino-1-(2-deoxy-3,5-di-O-tert-butyldimethylsilyl-β-D-ribofuranosyl)imidazole-4-carboxamide 170871-02-0 C21H42N4O4Si2
5-amino-1-(2-deoxy-3,5-di-O-tert-butyldimethylsilyl-β-D-ribofuranosyl)imidazole-4-carboxamide
—— ethyl 2-(dibenzylamino)-4-[(2-methoxy-2-oxoethyl)amino]-4-oxobutanoate 1018684-17-7 C23H28N2O5
ethyl 2-(dibenzylamino)-4-[(2-methoxy-2-oxoethyl)amino]-4-oxobutanoate
—— (1R,2R,4S)-1-tert-butyl 2-methyl 4-hydroxycyclopentane-1,2-dicarboxylate 1067648-60-5 C12H20O5
(1R,2R,4S)-1-tert-butyl 2-methyl 4-hydroxycyclopentane-1,2-dicarboxylate
—— (<S>-1,2-dimethylpropyl)(3-methylbutyl)(3-(trimethylsiloxy)propoxy)borane 109529-40-0 C16H37BO2Si
(<S>-1,2-dimethylpropyl)(3-methylbutyl)(3-(trimethylsiloxy)propoxy)borane
—— (R)-2-((2R,3R)-7-(3-(benzyloxy)phenyl)-3-((4-methoxybenzyl)oxy)heptan-2-yl)oxirane 1380328-05-1 C30H36O4
(R)-2-((2R,3R)-7-(3-(benzyloxy)phenyl)-3-((4-methoxybenzyl)oxy)heptan-2-yl)oxirane
—— allyl 6-O-benzyloxycarbonyl-2-<(2S,3R)-3-(benzyloxycarbonyloxy-2-fluorotetradecanoyl)amino>-2-deoxy-3-O-<(3R)-3-tetradecanoyloxytetradecanoyl>-α-D-glucopyranoside 4-(diphenyl phosphate) 132791-90-3 C79H115FNO17P
allyl 6-O-benzyloxycarbonyl-2-<(2S,3R)-3-(benzyloxycarbonyloxy-2-fluorotetradecanoyl)amino>-2-deoxy-3-O-<(3R)-3-tetradecanoyloxytetradecanoyl>-α-D-glucopyranoside 4-(diphenyl phosphate)
—— (2S,3S,4S,4aS,9R,9aR)-3,4,9-tris(benzyloxy)-2-((R)-1-(benzyloxy)propan-2-yl)octahydro-6H-pyrano[3,2-b]oxepin-6-one 1227264-81-4 C40H44O7
(2S,3S,4S,4aS,9R,9aR)-3,4,9-tris(benzyloxy)-2-((R)-1-(benzyloxy)propan-2-yl)octahydro-6H-pyrano[3,2-b]oxepin-6-one
—— Acetic acid (2R,3R,4S,5S,6R)-4,5-diacetoxy-6-acetoxymethyl-2-[6-(4-amino-phenyl)-3-cyano-4-furan-2-yl-2-oxo-2H-pyridin-1-yl]-tetrahydro-pyran-3-yl ester 171071-18-4 C30H29N3O11
Acetic acid (2R,3R,4S,5S,6R)-4,5-diacetoxy-6-acetoxymethyl-2-[6-(4-amino-phenyl)-3-cyano-4-furan-2-yl-2-oxo-2H-pyridin-1-yl]-tetrahydro-pyran-3-yl ester
—— —— 158020-21-4 C15H8Co2O6
—— 3-(8-methylimidazo[1,2-a]pyridin-2-yl)-7-(4-methylpiperazin-1-yl)-2H-chromen-2-one 1446328-16-0 C22H22N4O2
3-(8-methylimidazo[1,2-a]pyridin-2-yl)-7-(4-methylpiperazin-1-yl)-2H-chromen-2-one
—— 1-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-7-yl)-3-[(4R)-8-(trifluoromethyl)-3,4-dihydro-2H-chromen-4-yl]urea 1444795-02-1 C20H19F3N4O3
1-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-7-yl)-3-[(4R)-8-(trifluoromethyl)-3,4-dihydro-2H-chromen-4-yl]urea
—— 2(R)-(2-amino-6-ethoxy-9(H)-purinyl)-4(R)-(4(S)-(3,5-dichlorophenyl)-2-oxo-1,3,2-dioxaphosphorinan-2(R)-yloxymethyl)-1(R)-methyl-7-oxo-3,6,8-trioxa-cis-bicyclo[3.3.0]octane 1447584-26-0 C23H24Cl2N5O9P
2(R)-(2-amino-6-ethoxy-9(H)-purinyl)-4(R)-(4(S)-(3,5-dichlorophenyl)-2-oxo-1,3,2-dioxaphosphorinan-2(R)-yloxymethyl)-1(R)-methyl-7-oxo-3,6,8-trioxa-cis-bicyclo[3.3.0]octane
—— N<sup>2</sup>-(4,4-difluorocyclohexyl)-6-phenyl-N<sup>4</sup>-(pyridin-4-yl)-1,3,5-triazine-2,4-diamine 1446503-39-4 C20H20F2N6
N<sup>2</sup>-(4,4-difluorocyclohexyl)-6-phenyl-N<sup>4</sup>-(pyridin-4-yl)-1,3,5-triazine-2,4-diamine
—— 3-((R)-2-(((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)amino)methyl)pyrrolidin-1-yl) tetrahydrothiophene 1,1-dioxide 1445705-38-3 C17H24ClN7O2S
3-((R)-2-(((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)amino)methyl)pyrrolidin-1-yl) tetrahydrothiophene 1,1-dioxide
—— ethyl N-[5-chloro-2-(1-methylpyrazole-4-carbonyl)furo[3,2-b]pyridin-3-yl]-N-[(2S,4S,6R)-2-ethyl-6-methyloxan-4-yl]carbamate 1445970-90-0 C23H27ClN4O5
ethyl N-[5-chloro-2-(1-methylpyrazole-4-carbonyl)furo[3,2-b]pyridin-3-yl]-N-[(2S,4S,6R)-2-ethyl-6-methyloxan-4-yl]carbamate
—— MeOCO-Gly-DL-N(Ph(4-F))Phg(2-Me)-NHcHex 1355327-37-5 C25H30FN3O4
MeOCO-Gly-DL-N(Ph(4-F))Phg(2-Me)-NHcHex
—— (R)-tert-butyl 4-((2-chloro-5-(5-(3-hydroxypyrrolidine-1-carbonyl)-1,3,4-thiadiazol-2-yl)pyridin-4-yl)amino)benzoate 1447226-57-4 C23H24ClN5O4S
(R)-tert-butyl 4-((2-chloro-5-(5-(3-hydroxypyrrolidine-1-carbonyl)-1,3,4-thiadiazol-2-yl)pyridin-4-yl)amino)benzoate
—— N-(2-nitrophenyl)sulfanylfluoren-9-imine 1423604-19-6 C19H12N2O2S
N-(2-nitrophenyl)sulfanylfluoren-9-imine
—— N-{4-[(3-ethoxypropyl)carbamoyl]phenyl}-1,3-dihydro-2H-isoindole-2-carboxamide 1375544-42-5 C21H25N3O3
N-{4-[(3-ethoxypropyl)carbamoyl]phenyl}-1,3-dihydro-2H-isoindole-2-carboxamide
—— 1-trifluoromethyl-cyclopentanecarboxylic acid {1-[4-(4-fluoro-phenyl)-5-morpholin-4-yl-thiazol-2-ylcarbamoyl]-1-methyl-ethyl}-amide 1205601-67-7 C24H28F4N4O3S
1-trifluoromethyl-cyclopentanecarboxylic acid {1-[4-(4-fluoro-phenyl)-5-morpholin-4-yl-thiazol-2-ylcarbamoyl]-1-methyl-ethyl}-amide