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—— (2S)-3-[4-[5-(4-acetylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-[(4-tert-butylbenzoyl)amino]propanoic acid 1443788-68-8 C30H29N3O5
(2S)-3-[4-[5-(4-acetylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-[(4-tert-butylbenzoyl)amino]propanoic acid
—— tert-butyl N-[8-tert-butyl-2-(1,4-dioxa-8-thiaspiro[4.5]decan-6-ylmethylcarbamoyl)-4-methylquinolin-6-yl]-N-(2,2,2-trifluoroethyl)carbamate 1453860-37-1 C30H40F3N3O5S
tert-butyl N-[8-tert-butyl-2-(1,4-dioxa-8-thiaspiro[4.5]decan-6-ylmethylcarbamoyl)-4-methylquinolin-6-yl]-N-(2,2,2-trifluoroethyl)carbamate
—— 2-[2-Cyclohexyl-4-(4-fluoro-3-methylphenyl)imidazol-1-yl]-1-[4-(4-methoxypyridin-2-yl)piperazin-1-yl]ethanone 1443145-10-5 C28H34FN5O2
2-[2-Cyclohexyl-4-(4-fluoro-3-methylphenyl)imidazol-1-yl]-1-[4-(4-methoxypyridin-2-yl)piperazin-1-yl]ethanone
—— 1-(1-methyl-2-oxo-1,2-dihydroquinolin-5-yl)-3-[(4S)-7-(trifluoromethoxy)-3,4-dihydro-2H-chromen-4-yl]urea 1444789-80-3 C21H18F3N3O4
1-(1-methyl-2-oxo-1,2-dihydroquinolin-5-yl)-3-[(4S)-7-(trifluoromethoxy)-3,4-dihydro-2H-chromen-4-yl]urea
—— 3-{[4-(cyclohexyl{2-ethyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}methoxy)benzoyl]amino}propanoic acid 1150211-42-9 C30H32F3NO5
3-{[4-(cyclohexyl{2-ethyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}methoxy)benzoyl]amino}propanoic acid
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(2,2-difluoroethylcarbamoyl)-6-methylphenyl]-5-[[5-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide 1229658-31-4 C25H16ClF9N10O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(2,2-difluoroethylcarbamoyl)-6-methylphenyl]-5-[[5-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide
—— 3-[({3-(4-chlorophenyl)-5-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]-4,5-dihydro-1H-1,2,4-triazol-1-yl}acetyl)amino]-3-(2,3-dichlorophenyl)propyl carbamate 1245620-71-6 C23H21Cl3F3N5O5
3-[({3-(4-chlorophenyl)-5-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]-4,5-dihydro-1H-1,2,4-triazol-1-yl}acetyl)amino]-3-(2,3-dichlorophenyl)propyl carbamate
—— 1-[4-(aminosulfonyl)phenyl]-5-cyclopentyl-1H-1,2,4-triazole-3-carboxylic acid 1006905-20-9 C14H16N4O4S
1-[4-(aminosulfonyl)phenyl]-5-cyclopentyl-1H-1,2,4-triazole-3-carboxylic acid
—— 3-[{[4-({cyclohexyl[2-ethyl-5-(2-methylpropyl)thiophen-3-yl]methyl}amino)phenyl]carbonyl}(methyl)amino]propanoic acid 1150213-66-3 C28H40N2O3S
3-[{[4-({cyclohexyl[2-ethyl-5-(2-methylpropyl)thiophen-3-yl]methyl}amino)phenyl]carbonyl}(methyl)amino]propanoic acid
—— (1R,3aS,3bS,10aR,10bS,11S,12aS)-1-{[(dimethylcarbamoyl)sulfanyl]carbonyl}-7-{3-[(1,1-dioxidotetrahydrothiophen-3-yl)carbamoyl]phenyl}-11-hydroxy-10a,12a-dimethyl-1,2,3,3a,3b,4,5,7,10,10a,10b,11,12,12a-tetradecahydrocyclopenta[5,6]naphtho[1,2-f]indazol-1-yl propanoate 1246779-25-8 C38H48N4O8S2
(1R,3aS,3bS,10aR,10bS,11S,12aS)-1-{[(dimethylcarbamoyl)sulfanyl]carbonyl}-7-{3-[(1,1-dioxidotetrahydrothiophen-3-yl)carbamoyl]phenyl}-11-hydroxy-10a,12a-dimethyl-1,2,3,3a,3b,4,5,7,10,10a,10b,11,12,12a-tetradecahydrocyclopenta[5,6]naphtho[1,2-f]indazol-1-yl propanoate
—— N-[(1S)-1-[4-[1-(4-bromopyridin-2-yl)azetidin-3-yl]oxyphenyl]ethyl]acetamide 1443669-25-7 C18H20BrN3O2
N-[(1S)-1-[4-[1-(4-bromopyridin-2-yl)azetidin-3-yl]oxyphenyl]ethyl]acetamide
—— 5-Amino-N1,N1-dimethylisophthalamide 1251529-89-1 C10H13N3O2
5-Amino-N1,N1-dimethylisophthalamide
—— 2-(2-chlorophenyl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide 1229657-64-0 C23H17ClF3N9O2
2-(2-chlorophenyl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide
—— 5-(cyclopropylsulfonyl)-8-fluoro-7-(2-fluoro-4-iodophenyl)-3-methyl-5H-imidazo[4,5-b]isoxazolo[3,4-e]pyridin-6(7H)-one 1040247-05-9 C17H11F2IN4O4S
5-(cyclopropylsulfonyl)-8-fluoro-7-(2-fluoro-4-iodophenyl)-3-methyl-5H-imidazo[4,5-b]isoxazolo[3,4-e]pyridin-6(7H)-one
—— 3-amino-benzoic acid-[2-(1(3)<i>H</i>-imidazol-4-yl)-ethylamide] 108996-93-6 C12H14N4O
3-amino-benzoic acid-[2-(1(3)<i>H</i>-imidazol-4-yl)-ethylamide]
—— 2-[5-cyclopropyl-1-(2-fluorobenzyl)-4-methyl-1H-pyrazol-3-yl]-5-methoxypyrimidin-4-amine 1445831-30-0 C19H20FN5O
2-[5-cyclopropyl-1-(2-fluorobenzyl)-4-methyl-1H-pyrazol-3-yl]-5-methoxypyrimidin-4-amine
—— 8-(5-carboxymethyl-2-methoxyphenyl)-5-fluoro-3,4-dihydro-1H-isoquinoline-2-carboxylic acid 2-methylthiazol-4-ylmethyl ester 1445885-85-7 C24H23FN2O5S
8-(5-carboxymethyl-2-methoxyphenyl)-5-fluoro-3,4-dihydro-1H-isoquinoline-2-carboxylic acid 2-methylthiazol-4-ylmethyl ester
—— N-((5'-methyl-[2,2'-bithiophen]-5-yl)methyl)adamantan-1-amine 1443122-84-6 C20H25NS2
N-((5'-methyl-[2,2'-bithiophen]-5-yl)methyl)adamantan-1-amine
—— 1-[(4R)-6,8-difluoro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)urea 1444795-72-5 C21H19F4N3O3
1-[(4R)-6,8-difluoro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)urea
—— (S)-N-(4-((3-chloro-4-(4-isopropylpiperazin-1-yl)phenyl)amino)-7-methoxyquinazolin-6-yl)-1-((S)-3,3-dimethyl-2-((S)-2-(methylamino)propanamido)butanoyl)pyrrolidine-2-carboxamide hydrochloride 1363153-35-8 C37H52ClN9O4*ClH
(S)-N-(4-((3-chloro-4-(4-isopropylpiperazin-1-yl)phenyl)amino)-7-methoxyquinazolin-6-yl)-1-((S)-3,3-dimethyl-2-((S)-2-(methylamino)propanamido)butanoyl)pyrrolidine-2-carboxamide hydrochloride
—— [4-[1-(3-Chlorophenyl)-1,2,4-triazole-3-carbonyl]-3-methylpiperazin-1-yl]-[3-(methoxymethyl)-1-benzofuran-2-yl]methanone 1443758-49-3 C25H24ClN5O4
[4-[1-(3-Chlorophenyl)-1,2,4-triazole-3-carbonyl]-3-methylpiperazin-1-yl]-[3-(methoxymethyl)-1-benzofuran-2-yl]methanone
—— (R)-2-[N-(carbamoylmethyl)sulfamoyl]-6-(2-chlorophenyl)-7-(4-chlorophenyl)-3-[N-(1,1-dioxotetrahydrothien-3-yl)carbamoyl]pyrazolo[1,5-a]pyrimidine 1001425-04-2 C25H22Cl2N6O6S2
(R)-2-[N-(carbamoylmethyl)sulfamoyl]-6-(2-chlorophenyl)-7-(4-chlorophenyl)-3-[N-(1,1-dioxotetrahydrothien-3-yl)carbamoyl]pyrazolo[1,5-a]pyrimidine
—— 1-(2-Amino-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-6-yl)-2-[3-(4-fluoro-3-methylphenyl)-5-propan-2-yl-1,2,4-triazol-1-yl]ethanone 1443255-83-1 C21H25FN6OS
1-(2-Amino-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-6-yl)-2-[3-(4-fluoro-3-methylphenyl)-5-propan-2-yl-1,2,4-triazol-1-yl]ethanone
—— (2S,5R)-5-(2-chlorophenyl)-1-(2-fluoro-3'-(methylsulfonamido)-[1,1'-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid 1312802-90-6 C25H22ClFN2O5S
(2S,5R)-5-(2-chlorophenyl)-1-(2-fluoro-3'-(methylsulfonamido)-[1,1'-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid
—— 4-chloro-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-3-[4-(1-propyl-piperidin-4-ylcarbamoyl)-phenyl]-pyrrolo[2,3-b]pyridine-1-carboxylic acid ethylamide 1312580-84-9 C36H44ClN7O2
4-chloro-2-[4-(4-methyl-piperazin-1-yl)-phenyl]-3-[4-(1-propyl-piperidin-4-ylcarbamoyl)-phenyl]-pyrrolo[2,3-b]pyridine-1-carboxylic acid ethylamide
—— 2-(4-chloro-3-fluorophenyl)-N-[4-(4-chlorophenyl)-1-oxophthalazin-2(1H)-yl]acetamide 1309193-61-0 C22H14Cl2FN3O2
2-(4-chloro-3-fluorophenyl)-N-[4-(4-chlorophenyl)-1-oxophthalazin-2(1H)-yl]acetamide
—— 4-bromo-N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(cyclopropylmethyl)-1H-benzotriazol-5-amine 1247947-79-0 C20H18BrClN6
4-bromo-N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(cyclopropylmethyl)-1H-benzotriazol-5-amine
—— tert-butyl 4-(5-fluoro-3-(6-methylimidazo[1,2-a]pyridin-2-yl)-2-oxo-2H-chromen-7-yl)piperazine-1-carboxylate 1446332-81-5 C26H27FN4O4
tert-butyl 4-(5-fluoro-3-(6-methylimidazo[1,2-a]pyridin-2-yl)-2-oxo-2H-chromen-7-yl)piperazine-1-carboxylate
—— 7-(1,4-diazepan-1-yl)-3-(imidazo[2,1-b][1,3]thiazol-6-yl)-2H-chromen-2-one 1446329-41-4 C19H18N4O2S
7-(1,4-diazepan-1-yl)-3-(imidazo[2,1-b][1,3]thiazol-6-yl)-2H-chromen-2-one
—— [4-Amino-6-(ethoxymethyl)-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-(1,1-dioxo-1,3-thiazolidin-3-yl)methanone 1443531-47-2 C23H25N5O5S2
[4-Amino-6-(ethoxymethyl)-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,1-f][1,2,4]triazin-7-yl]-(1,1-dioxo-1,3-thiazolidin-3-yl)methanone
—— 2-[7-(4-methylpiperazin-1-yl)-2-oxo-2H-chromen-3-yl]imidazo[1,2-a]pyridine-6-carbonitrile 1446329-43-6 C22H19N5O2
2-[7-(4-methylpiperazin-1-yl)-2-oxo-2H-chromen-3-yl]imidazo[1,2-a]pyridine-6-carbonitrile
—— 6-(2-Chloro-4-pyridin-3-ylphenyl)-8-ethyl-2-[3-fluoro-4-(4-propan-2-ylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one 1428758-55-7 C33H33ClFN7O
6-(2-Chloro-4-pyridin-3-ylphenyl)-8-ethyl-2-[3-fluoro-4-(4-propan-2-ylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— (3R,3aR,6S,6aR)-6-[5-[5-[5-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-3-yl]pyridin-2-yl]pyridin-2-yl]oxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol 1445206-82-5 C25H20F3N5O4
(3R,3aR,6S,6aR)-6-[5-[5-[5-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-3-yl]pyridin-2-yl]pyridin-2-yl]oxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol
—— {(S)-3-[4-(6-methoxy-5-methylpyridin-3-yl)quinolin-6-yloxy]pyrrolidin-1-yl} (tetrahydropyran-4-yl)methanone 1445650-98-5 C26H29N3O4
{(S)-3-[4-(6-methoxy-5-methylpyridin-3-yl)quinolin-6-yloxy]pyrrolidin-1-yl} (tetrahydropyran-4-yl)methanone
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3,6-dihydro-2H-pyran-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate 1428666-82-3 C26H33N3O4
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3,6-dihydro-2H-pyran-4-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— 1-[(4R)-7-bromo-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)urea 1444799-25-0 C22H24BrN3O3
1-[(4R)-7-bromo-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)urea
—— [4-[5-fluoro-2-((1R,2R)-2-phenylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-3-(2,2,2-trifluoroethoxy)phenyl]acetic acid 1445887-90-0 C29H25F4NO4
[4-[5-fluoro-2-((1R,2R)-2-phenylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-3-(2,2,2-trifluoroethoxy)phenyl]acetic acid
—— 2-(6-chloro-3-pyridyl)-2-imidazoline 154753-13-6 C8H8ClN3
2-(6-chloro-3-pyridyl)-2-imidazoline
—— (R)-4-amino-2-ethyl-isoxazolidin-3-one trifluoroacetate 1309958-90-4 C2HF3O2*C5H10N2O2
(R)-4-amino-2-ethyl-isoxazolidin-3-one trifluoroacetate
—— rac-1,3-dimethyl-1H-pyrazole-4-carboxylic acid [3-(2-methyl-5-m-tolyl-thiazole-4-carbonyl)-thiazolidin-2-ylmethyl]-amide 1204584-88-2 C22H25N5O2S2
rac-1,3-dimethyl-1H-pyrazole-4-carboxylic acid [3-(2-methyl-5-m-tolyl-thiazole-4-carbonyl)-thiazolidin-2-ylmethyl]-amide
—— 1-[(2R,4R)-2-(1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]-3-pyridin-4-ylurea hydrochloride 1095173-37-7 C19H22N6O*ClH
1-[(2R,4R)-2-(1H-benzimidazol-2-yl)-1-methylpiperidin-4-yl]-3-pyridin-4-ylurea hydrochloride
—— N-[(1S)-1-[4-[1-(3-methylquinoxalin-2-yl)azetidin-3-yl]oxyphenyl]ethyl]acetamide 1443669-46-2 C22H24N4O2
N-[(1S)-1-[4-[1-(3-methylquinoxalin-2-yl)azetidin-3-yl]oxyphenyl]ethyl]acetamide
—— 4-Thiazolidinecarboxylic acid, 3-[3-(2-chlorophenyl)-1-oxopropyl]-, (4R)- 1284804-95-0 C13H14ClNO3S
4-Thiazolidinecarboxylic acid, 3-[3-(2-chlorophenyl)-1-oxopropyl]-, (4R)-
—— 3-(8-bromoimidazo[1,2-a]pyridin-2-yl)-7-(4-methylpiperazin-1-yl)-2H-chromen-2-one 1446329-82-3 C21H19BrN4O2
3-(8-bromoimidazo[1,2-a]pyridin-2-yl)-7-(4-methylpiperazin-1-yl)-2H-chromen-2-one
—— 1-[(4R)-6-fluoro-2,2-dipropyl-3,4-dihydro-2H-chromen-4-yl]-3-[3-(2-hydroxyethyl)-2-oxo-1,2,3,4-tetrahydroquinazolin-7-yl]urea 1444799-85-2 C26H33FN4O4
1-[(4R)-6-fluoro-2,2-dipropyl-3,4-dihydro-2H-chromen-4-yl]-3-[3-(2-hydroxyethyl)-2-oxo-1,2,3,4-tetrahydroquinazolin-7-yl]urea
—— (3R,3aR,6S,6aR)-6-[5-[5-[5-(4-chlorophenyl)-1H-1,2,4-triazol-3-yl]pyridin-2-yl]pyridin-2-yl]oxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol 1445206-80-3 C24H20ClN5O4
(3R,3aR,6S,6aR)-6-[5-[5-[5-(4-chlorophenyl)-1H-1,2,4-triazol-3-yl]pyridin-2-yl]pyridin-2-yl]oxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol
—— 2-(3-chlorophenoxy)-N-{4-ethoxy-2-[(2-methylpropyl)amino]phenyl}acetamide 1446338-36-8 C20H25ClN2O3
2-(3-chlorophenoxy)-N-{4-ethoxy-2-[(2-methylpropyl)amino]phenyl}acetamide
—— 6-methyl-4-[5-(methylsulfonyl)-2-(tetrahydrofuran-3-ylamino)phenyl]-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one 1446233-81-3 C19H21N3O4S
6-methyl-4-[5-(methylsulfonyl)-2-(tetrahydrofuran-3-ylamino)phenyl]-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one
—— 1-[(2R,4R)-2-(difluoromethyl)-2-methyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)urea 1444799-09-0 C22H23F2N3O3
1-[(2R,4R)-2-(difluoromethyl)-2-methyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)urea
—— (S)-2,5-dichloro-N-(piperidin-3-ylmethyl)pyrimidin-4-amine 1445705-80-5 C10H14Cl2N4
(S)-2,5-dichloro-N-(piperidin-3-ylmethyl)pyrimidin-4-amine