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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-N-(2-(2-(((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)amino)methyl)pyrrolidin-1-yl)ethyl)methanesulfonamide 1445705-49-6 C16H25ClN8O2S
(R)-N-(2-(2-(((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)amino)methyl)pyrrolidin-1-yl)ethyl)methanesulfonamide
—— (E)-6-(3-oxo-3-(4-(phenoxymethyl)-5,6-dihydropyridin-1(2H)-yl)prop-1-en-1-yl)-3,4-dihydro-1,8-naphthyridin-2(1H)-one 1441350-58-8 C23H23N3O3
(E)-6-(3-oxo-3-(4-(phenoxymethyl)-5,6-dihydropyridin-1(2H)-yl)prop-1-en-1-yl)-3,4-dihydro-1,8-naphthyridin-2(1H)-one
—— (R)-N<sup>2</sup>-(1-(1H-pyrrolo[2,3-c]pyridin-5-yl)ethyl)-N<sup>4</sup>-(5-cyclopropyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine 1445855-50-4 C19H20N8
(R)-N<sup>2</sup>-(1-(1H-pyrrolo[2,3-c]pyridin-5-yl)ethyl)-N<sup>4</sup>-(5-cyclopropyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
—— 1-(cyclohexylmethyl)-5-(3,5-ditert-butylphenyl)-2-methyl-N-(2-propan-2-yloxyethyl)pyrrole-3-carboxamide 1442423-61-1 C32H50N2O2
1-(cyclohexylmethyl)-5-(3,5-ditert-butylphenyl)-2-methyl-N-(2-propan-2-yloxyethyl)pyrrole-3-carboxamide
—— 2-pyridin-4-yl-N-[5-[4-[6-[[2-[3-(trifluoromethoxy)phenyl]acetyl]amino]pyridazin-3-yl]butyl]-1,3,4-thiadiazol-2-yl]acetamide 1439399-60-6 C26H24F3N7O3S
2-pyridin-4-yl-N-[5-[4-[6-[[2-[3-(trifluoromethoxy)phenyl]acetyl]amino]pyridazin-3-yl]butyl]-1,3,4-thiadiazol-2-yl]acetamide
—— (E)-(1-(penta-2,4-dienyl)cyclohexyl)methanol 1380544-63-7 C12H20O
(E)-(1-(penta-2,4-dienyl)cyclohexyl)methanol
—— diethyl (4-oxo-4H-chromen-3-yl)methylphosphonate 1384987-08-9 C14H17O5P
diethyl (4-oxo-4H-chromen-3-yl)methylphosphonate
—— 2-Amino-4-(4-aminophenyl)-5,6,7,8-tetrahydronaphthalene-1,3-dicarbonitrile 1399697-87-0 C18H16N4
2-Amino-4-(4-aminophenyl)-5,6,7,8-tetrahydronaphthalene-1,3-dicarbonitrile
—— 6-[4-[13-(2,5-Ditert-butylphenyl)-5,7,12,14-tetraoxo-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaen-6-yl]-2,5-dimethylphenyl]-13-[4-(2,3,5,6-tetramethyl-4-perylen-3-ylphenyl)phenyl]-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaene-5,7,12,14-tetrone 1391420-77-1 C86H64N4O8
6-[4-[13-(2,5-Ditert-butylphenyl)-5,7,12,14-tetraoxo-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaen-6-yl]-2,5-dimethylphenyl]-13-[4-(2,3,5,6-tetramethyl-4-perylen-3-ylphenyl)phenyl]-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaene-5,7,12,14-tetrone
—— (R)-9-(3-(2-Fluorophenyl)benzyl)-2-(pyrrolidin-3-ylmethylamino)-7H-purin-8(9H)-one 1152086-26-4 C23H23FN6O
(R)-9-(3-(2-Fluorophenyl)benzyl)-2-(pyrrolidin-3-ylmethylamino)-7H-purin-8(9H)-one
—— N-[5-(2,2-dimethylpropylamino)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 1142937-55-0 C15H21N5O
N-[5-(2,2-dimethylpropylamino)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide
—— N3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1-(isoquinolin-1-yl)-1H-1,2,4-triazole-3,5-diamine 1038404-32-8 C19H16N6O2
N3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1-(isoquinolin-1-yl)-1H-1,2,4-triazole-3,5-diamine
—— 1-{6-[3-(trifluoromethyl)phenyl]-2-pyridinyl}-5-(trifluoromethyl)-1H-pyrazole-4-carboxylic acid 1158984-23-6 C17H9F6N3O2
1-{6-[3-(trifluoromethyl)phenyl]-2-pyridinyl}-5-(trifluoromethyl)-1H-pyrazole-4-carboxylic acid
—— 2-((adamantan-1-ylamino)methyl)quinolin-8-ol 1443122-40-4 C20H24N2O
2-((adamantan-1-ylamino)methyl)quinolin-8-ol
—— 5-[3-tert-butyl-4-(dimethylcarbamoyl)phenyl]-1-(cyclohexylmethyl)-2-methyl-N-(oxan-4-yl)pyrrole-3-carboxamide 1442424-75-0 C31H45N3O3
5-[3-tert-butyl-4-(dimethylcarbamoyl)phenyl]-1-(cyclohexylmethyl)-2-methyl-N-(oxan-4-yl)pyrrole-3-carboxamide
—— ethyl 5,5-dimethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydroisoxazolo[4,5-h]quinazoline-3-carboxylate 1356410-80-4 C25H30N6O3
ethyl 5,5-dimethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydroisoxazolo[4,5-h]quinazoline-3-carboxylate
—— 1-(1-(5-ethylpyrimidin-2-yl)piperidin-4-yl)-3-(4-(2-methyl-2H-tetrazol-5-yl)phenoxy)pyrrolidin-2-one 1351166-79-4 C23H28N8O2
1-(1-(5-ethylpyrimidin-2-yl)piperidin-4-yl)-3-(4-(2-methyl-2H-tetrazol-5-yl)phenoxy)pyrrolidin-2-one
—— 2-[3-(4-Fluoro-3-methylphenyl)-5-phenylpyrazol-1-yl]-1-(2-methyl-4,5,7,8-tetrahydro-[1,3]oxazolo[4,5-d]azepin-6-yl)ethanone 1440953-08-1 C26H25FN4O2
2-[3-(4-Fluoro-3-methylphenyl)-5-phenylpyrazol-1-yl]-1-(2-methyl-4,5,7,8-tetrahydro-[1,3]oxazolo[4,5-d]azepin-6-yl)ethanone
—— 2-[5-Ethyl-3-(4-fluoro-3-methylphenyl)pyrazol-1-yl]-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]ethanone 1440953-63-8 C22H26FN5O2
2-[5-Ethyl-3-(4-fluoro-3-methylphenyl)pyrazol-1-yl]-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]ethanone
—— N-(4-benzoyl-3,4-dihydro-2H-benzo[b][1,4]thiazin-6-yl)-4-(dimethylamino)butanamide 1438406-12-2 C21H25N3O2S
N-(4-benzoyl-3,4-dihydro-2H-benzo[b][1,4]thiazin-6-yl)-4-(dimethylamino)butanamide
—— 5-(4-pyridyl)-4-[4-(2-pyrrolidin-1-ylethoxymethyl)-1-piperidyl]thieno[2,3-d]pyrimidine 1437773-50-6 C23H29N5OS
5-(4-pyridyl)-4-[4-(2-pyrrolidin-1-ylethoxymethyl)-1-piperidyl]thieno[2,3-d]pyrimidine
—— US9598416, Example 51 1443617-10-4 C22H25N5OS
US9598416, Example 51
—— N-(2-methoxyethyl)-4-methyl-2-({1-[(3-phenylisoxazol-5-yl)-carbonyl]piperidin-4-yl}methyl)-2H-indazol-5-carboxamide 1442116-16-6 C28H31N5O4
N-(2-methoxyethyl)-4-methyl-2-({1-[(3-phenylisoxazol-5-yl)-carbonyl]piperidin-4-yl}methyl)-2H-indazol-5-carboxamide
—— 2-[3-(4-fluoro-3-methylphenyl)-5-phenylpyrazol-1-yl]-1-[4-(3-methoxyphenyl)-3,6-dihydro-2H-pyridin-1-yl]ethanone 1440953-39-8 C30H28FN3O2
2-[3-(4-fluoro-3-methylphenyl)-5-phenylpyrazol-1-yl]-1-[4-(3-methoxyphenyl)-3,6-dihydro-2H-pyridin-1-yl]ethanone
—— 4-(4-cyclopropyl-3-methyl-2-oxobenzimidazol-1-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-2-carboxamide 1150102-05-8 C24H25N7O2S
4-(4-cyclopropyl-3-methyl-2-oxobenzimidazol-1-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-2-carboxamide
—— 1-(3-methoxy-phenyl)carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan] 1028048-23-8 C21H24N2O3
1-(3-methoxy-phenyl)carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan]
—— 2-[(5-Chloropyridine-2-carbonyl)-propan-2-ylamino]-4-fluoro-5-[3-(trifluoromethyl)pyridin-2-yl]oxybenzoic acid 1113049-03-8 C22H16ClF4N3O4
2-[(5-Chloropyridine-2-carbonyl)-propan-2-ylamino]-4-fluoro-5-[3-(trifluoromethyl)pyridin-2-yl]oxybenzoic acid
—— (2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[2-(4-heptoxyphenyl)-1,3-oxazol-4-yl]phenyl]propanoic acid 1443789-00-1 C36H42N2O5
(2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[2-(4-heptoxyphenyl)-1,3-oxazol-4-yl]phenyl]propanoic acid
—— 1-(cyclohexylmethyl)-5-(3,5-ditert-butylphenyl)-2-methyl-N-(thietan-3-yl)pyrrole-3-carboxamide 1442423-12-2 C30H44N2OS
1-(cyclohexylmethyl)-5-(3,5-ditert-butylphenyl)-2-methyl-N-(thietan-3-yl)pyrrole-3-carboxamide
—— (R)-1-(4-methoxybenzyl)-2-(2-pyridin-4-yl-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4-yloxy)ethylamine 1438883-00-1 C25H26N4O2S
(R)-1-(4-methoxybenzyl)-2-(2-pyridin-4-yl-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4-yloxy)ethylamine
—— 4-[5-(1-methyl-5-{[4-(trifluoromethyl)phenoxy]methyl}-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyrimidine-2-amine 1359028-17-3 C18H14F3N7O2
4-[5-(1-methyl-5-{[4-(trifluoromethyl)phenoxy]methyl}-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyrimidine-2-amine
—— (6-benzo(b)thiophen-2-ylthieno[3,2-d]pyrimidin-4-yl)-(2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethyl)amine 1099820-54-8 C26H21FN4S2
(6-benzo(b)thiophen-2-ylthieno[3,2-d]pyrimidin-4-yl)-(2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethyl)amine
—— (3S,5R,10S,13S,16S,17S)-17-(2,2-Diiodo-acetyl)-3-hydroxy-10,13-dimethyl-hexadecahydro-cyclopropa[16,17]cyclopenta[a]phenanthren-11-one 100323-03-3 C22H30I2O3
(3S,5R,10S,13S,16S,17S)-17-(2,2-Diiodo-acetyl)-3-hydroxy-10,13-dimethyl-hexadecahydro-cyclopropa[16,17]cyclopenta[a]phenanthren-11-one
—— —— 1034281-39-4 C16H8F9N5O2
—— —— 1034286-22-0 C17H16BrN5
—— Z-Glu(NH2)-Arg(NO2)-Leu-Leu-Glu(NH2)-Gly-Leu-Val-NH2 14611-20-2 C49H81N15O14
Z-Glu(NH2)-Arg(NO2)-Leu-Leu-Glu(NH2)-Gly-Leu-Val-NH2
—— 3-Ethoxycholest-3-en 16159-06-1 C29H50O
3-Ethoxycholest-3-en
—— 1,6-Bis-<N'-(3,4-dichlor-benzyl)-guanidino>-hexan 105792-53-8 C22H28Cl4N6
1,6-Bis-<N'-(3,4-dichlor-benzyl)-guanidino>-hexan
—— (E)-3-Allyloxyamino-1-(3,4,5-trimethoxy-phenyl)-propenone 10120-67-9 C15H19NO5
(E)-3-Allyloxyamino-1-(3,4,5-trimethoxy-phenyl)-propenone
—— 2.4-Dichlor-5-sulfamoylbenzoyl-aethoxyamid 13013-76-8 C9H10Cl2N2O4S
2.4-Dichlor-5-sulfamoylbenzoyl-aethoxyamid
—— methyl 2,2-dimethyl-8-((4'-methylbiphenyl-2-yl)oxy)octanoate 1003959-89-4 C24H32O3
methyl 2,2-dimethyl-8-((4'-methylbiphenyl-2-yl)oxy)octanoate
—— N-[3-(dimethylamino)propyl]-N-methyl-6-(5-methyl-2-phenyl-4,5,6,7-tetrahydro-1H-indol-1-yl)pyridine-3-carboxamide 1065529-76-1 C27H34N4O
N-[3-(dimethylamino)propyl]-N-methyl-6-(5-methyl-2-phenyl-4,5,6,7-tetrahydro-1H-indol-1-yl)pyridine-3-carboxamide
—— 7-fluoro-6-(6-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-3-ylmethyl)-quinoline 1086330-17-7 C14H10FN5S
7-fluoro-6-(6-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-3-ylmethyl)-quinoline
—— N-(4-(5-ethyl-2-(trifluoromethyl)oxazol-4-yl)phenyl)-2,6-difluorobenzamide 1582285-95-7 C19H13F5N2O2
N-(4-(5-ethyl-2-(trifluoromethyl)oxazol-4-yl)phenyl)-2,6-difluorobenzamide
—— Boc-[(S)-β-Caa(diFP)-(R)-β-Caa(diFP)]2-OMe 1093295-16-9 C70H80F8N4O19
Boc-[(S)-β-Caa(diFP)-(R)-β-Caa(diFP)]2-OMe
—— (R)-2-hexanol p-toluenesulfonate 1393538-39-0 C13H20O3S
(R)-2-hexanol p-toluenesulfonate
—— 2-(naphthalen-2-yl)-1-(2,2,6,6-tetramethylpiperidin-1-yl)ethanone 1360789-09-8 C21H27NO
2-(naphthalen-2-yl)-1-(2,2,6,6-tetramethylpiperidin-1-yl)ethanone
—— 3α-acetoxy-17,21-dibromo-5β-pregnane-11,20-dione 114397-95-4 C23H32Br2O4
3α-acetoxy-17,21-dibromo-5β-pregnane-11,20-dione
—— ethyl 2-diazo-2-(1-hydroxy-4-methylcyclohexyl)acetate 1290044-63-1 C11H18N2O3
ethyl 2-diazo-2-(1-hydroxy-4-methylcyclohexyl)acetate
—— 3,3,4-triphenyl-1-(p-tolyl)azetidin-2-one 116028-05-8 C28H23NO
3,3,4-triphenyl-1-(p-tolyl)azetidin-2-one