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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(3-chloro-4-fluorophenyl)-7-(2-methoxyphenyl)-2-pyridin-3-ylquinazolin-4-amine 1313896-05-7 C26H18ClFN4O
N-(3-chloro-4-fluorophenyl)-7-(2-methoxyphenyl)-2-pyridin-3-ylquinazolin-4-amine
—— 2-amino-4-[[(1S)-1-[8-(4-fluorophenyl)-1-oxo-2-phenylisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile 1425042-06-3 C28H21FN6O
2-amino-4-[[(1S)-1-[8-(4-fluorophenyl)-1-oxo-2-phenylisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile
—— (2-(2-amino-3-morpholinoquinolin-6-yl)-3-(trifluoromethyl)phenyl)(pyrrolidin-1-yl)methanone 1319195-84-0 C25H25F3N4O2
(2-(2-amino-3-morpholinoquinolin-6-yl)-3-(trifluoromethyl)phenyl)(pyrrolidin-1-yl)methanone
—— 7,7-dimethyl-8-oxo-N-[1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidin-3-yl]spiro[6,9-dihydrocarbazole-5,1'-cyclobutane]-3-carboxamide 1424994-27-3 C25H28N6O3
7,7-dimethyl-8-oxo-N-[1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidin-3-yl]spiro[6,9-dihydrocarbazole-5,1'-cyclobutane]-3-carboxamide
—— ethyl 5-chloro-1-[2'-hydroxy-3'-(methyloxy)-4-biphenylyl]-3-({[(2-methylphenyl)amino]carbonyl}amino)-1H-pyrrole-2-carboxylate 1346607-67-7 C28H26ClN3O5
ethyl 5-chloro-1-[2'-hydroxy-3'-(methyloxy)-4-biphenylyl]-3-({[(2-methylphenyl)amino]carbonyl}amino)-1H-pyrrole-2-carboxylate
—— 6-(Bromomethyl)-2,4-diamino-5-propylpyrido [2,3-d]pyrimidine 153802-80-3 C11H14BrN5
6-(Bromomethyl)-2,4-diamino-5-propylpyrido [2,3-d]pyrimidine
—— Sodium [3-[3-(4,5-diphenyloxazol-2-yl)cyclohexylmethyl]phenoxy]acetate 171046-11-0 C30H28NO4*Na
Sodium [3-[3-(4,5-diphenyloxazol-2-yl)cyclohexylmethyl]phenoxy]acetate
—— 3-[(1S)-1-[[2-amino-5-(morpholine-4-carbonyl)pyrimidin-4-yl]amino]ethyl]-8-chloro-2-phenylisoquinolin-1-one 1425044-73-0 C26H25ClN6O3
3-[(1S)-1-[[2-amino-5-(morpholine-4-carbonyl)pyrimidin-4-yl]amino]ethyl]-8-chloro-2-phenylisoquinolin-1-one
—— 1-{4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}-3-(methoxymethyl)cyclobutanol 1425971-73-8 C22H31NO2
1-{4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}-3-(methoxymethyl)cyclobutanol
—— N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)-2,3-dihydro-1,4-benzodioxine-6-sulfonamide 1425927-59-8 C17H17N3O5S
N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
—— (2-methoxy-5-(2-((methylsulfonyl)methyl)-4-morpholinopyrido[2,3-d]pyrimidin-7-yl)phenyl)methanol 1421658-57-2 C21H24N4O5S
(2-methoxy-5-(2-((methylsulfonyl)methyl)-4-morpholinopyrido[2,3-d]pyrimidin-7-yl)phenyl)methanol
—— (S)-N-cyclopropyl-2-(5-fluoro-2-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-ylamino)-3,3-dimethylbutane-1-sulfonamide 1422050-91-6 C20H24F2N6O2S
(S)-N-cyclopropyl-2-(5-fluoro-2-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-ylamino)-3,3-dimethylbutane-1-sulfonamide
—— isopropyl 4-{5-[3-methyl-4-(methylcarbamoyl)phenyl]benzo[d]oxazol-2-yl}piperidine-1-carboxylate 1415991-78-4 C25H29N3O4
isopropyl 4-{5-[3-methyl-4-(methylcarbamoyl)phenyl]benzo[d]oxazol-2-yl}piperidine-1-carboxylate
—— 3-(3-fluoro-4-bromophenyl)-5-fluoro-2-mercaptoquinazolin-4(3H)-one 1423009-63-5 C14H7BrF2N2OS
3-(3-fluoro-4-bromophenyl)-5-fluoro-2-mercaptoquinazolin-4(3H)-one
—— methyl ((S)-1-(((1S,2S)-2-(5-(7-(2-((S)-1-((S)-2-(methoxycarbonyl)amino-3-methylbutanoyl)pyrrolidin-2-yl)-1H-imidazol-5-yl)-9,9-dimethyl-9H-fluoren-2-yl)-1H-imidazol-2-yl)cyclopentyl)amino)-3-methyl-1-oxobutan-2-yl)carbamate 1422429-20-6 C44H56N8O6
methyl ((S)-1-(((1S,2S)-2-(5-(7-(2-((S)-1-((S)-2-(methoxycarbonyl)amino-3-methylbutanoyl)pyrrolidin-2-yl)-1H-imidazol-5-yl)-9,9-dimethyl-9H-fluoren-2-yl)-1H-imidazol-2-yl)cyclopentyl)amino)-3-methyl-1-oxobutan-2-yl)carbamate
—— N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-fluoroquinolin-4-yl]ethane-1,2-diamine 1422498-12-1 C20H21FN4O2S
N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-fluoroquinolin-4-yl]ethane-1,2-diamine
—— N-({2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}methyl)-2-(tetrahydro-2H-pyran-4-yl)acetamide 1421848-62-5 C24H29FN4O2S
N-({2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}methyl)-2-(tetrahydro-2H-pyran-4-yl)acetamide
—— 1-[4-[4-[4-[[(1R)-1-(2-chlorophenyl)ethoxy]carbonylamino]-3-methyl-1,2-thiazol-5-yl]-3-methylphenyl]phenyl]cyclopropane-1-carboxylic acid 1423685-58-8 C30H27ClN2O4S
1-[4-[4-[4-[[(1R)-1-(2-chlorophenyl)ethoxy]carbonylamino]-3-methyl-1,2-thiazol-5-yl]-3-methylphenyl]phenyl]cyclopropane-1-carboxylic acid
—— 4-{[3-(cyclohexylmethylsulfamoyl)benzenesulfonylamino]methyl}-piperidine-1-carboxylic acid tert-butyl ester 1332527-67-9 C24H39N3O6S2
4-{[3-(cyclohexylmethylsulfamoyl)benzenesulfonylamino]methyl}-piperidine-1-carboxylic acid tert-butyl ester
—— N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-methylquinolin-4-yl]ethane-1,2-diamine 1422498-24-5 C21H24N4O2S
N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-methylquinolin-4-yl]ethane-1,2-diamine
—— N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-ethylquinolin-4-yl]ethane-1,2-diamine 1422498-14-3 C22H26N4O2S
N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-ethylquinolin-4-yl]ethane-1,2-diamine
—— 4-(2-methyl-5-oxopyrrolidin-1-yl)benzoic acid 1346123-50-9 C12H13NO3
4-(2-methyl-5-oxopyrrolidin-1-yl)benzoic acid
—— 1-[4-(4-chlorophenyl)butyl]-3-[7-(1H-pyrazol-4-yl)-1,5-naphthyridin-2-yl]urea 1422125-06-1 C22H21ClN6O
1-[4-(4-chlorophenyl)butyl]-3-[7-(1H-pyrazol-4-yl)-1,5-naphthyridin-2-yl]urea
—— 1-[4-[5-Methyl-2-[[2-methyl-4-(piperidine-1-carbonyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]-2-(trifluoromethyl)piperidine-4-carboxylic acid 1423068-00-1 C31H34F3N3O4S
1-[4-[5-Methyl-2-[[2-methyl-4-(piperidine-1-carbonyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]-2-(trifluoromethyl)piperidine-4-carboxylic acid
—— 2-(4-methoxyphenyl)-5-(piperidine-1-yl)oxazolo[5,4-b]pyridine 1422199-06-1 C18H19N3O2
2-(4-methoxyphenyl)-5-(piperidine-1-yl)oxazolo[5,4-b]pyridine
—— (R)-4-(4-methyl-2-oxooxazolidin-3-ylmethyl)benzoic acid 1346123-61-2 C12H13NO4
(R)-4-(4-methyl-2-oxooxazolidin-3-ylmethyl)benzoic acid
—— 2-[3-(4-fluorophenyl)-5 (1-phenylpiperidin-4-yl)-1H-pyrazol-1-yl]pyridine 1349862-83-4 C25H23FN4
2-[3-(4-fluorophenyl)-5 (1-phenylpiperidin-4-yl)-1H-pyrazol-1-yl]pyridine
—— 3-chloro-N-[5'-methanesulfonyl-4-((1S,4S)-2-2-oxa-5-aza-bicyclo[2..2.1]hept-5-yl-2-oxo-ethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-3'-yl]-benzamide 1314529-81-1 C25H29ClN4O5S
3-chloro-N-[5'-methanesulfonyl-4-((1S,4S)-2-2-oxa-5-aza-bicyclo[2..2.1]hept-5-yl-2-oxo-ethyl)-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-3'-yl]-benzamide
—— N-benzyl-2-(4-chlorophenyl)-N-methyloxazolo[5,4-b]pyridine-5-amine 1422199-25-4 C20H16ClN3O
N-benzyl-2-(4-chlorophenyl)-N-methyloxazolo[5,4-b]pyridine-5-amine
—— tert-butyl ((1S,2R)-2-(5-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-1H-imidazol-2-yl)cyclopentyl)carbamate 1422428-20-3 C25H36BN3O4
tert-butyl ((1S,2R)-2-(5-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-1H-imidazol-2-yl)cyclopentyl)carbamate
—— 2'-(3,5-dimethylisoxazol-4-yl)-3'-(hydroxymethyl)-5'-(trifluoromethyl)-[1,1'-biphenyl]-4-ol 1422021-52-0 C19H16F3NO3
2'-(3,5-dimethylisoxazol-4-yl)-3'-(hydroxymethyl)-5'-(trifluoromethyl)-[1,1'-biphenyl]-4-ol
—— 3-{[4-{[(1S)-1-(5-fluoropyridin-2-yl)ethyl]amino}-6-(4-hydroxypiperidin-1-yl) pyrimidin-2-yl]amino}pyridin-2(1H)-one 1421757-94-9 C21H24FN7O2
3-{[4-{[(1S)-1-(5-fluoropyridin-2-yl)ethyl]amino}-6-(4-hydroxypiperidin-1-yl) pyrimidin-2-yl]amino}pyridin-2(1H)-one
—— N-(5-(piperazin-1-yl)isothiazol-4-yl)-2-(piperidin-1-yl)thiazole-4-carboxamide 1422394-64-6 C16H22N6OS2
N-(5-(piperazin-1-yl)isothiazol-4-yl)-2-(piperidin-1-yl)thiazole-4-carboxamide
—— 5-(1H-imidazol-1-yl)-3-phenyl-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[3,4-c]pyridine 1422442-96-3 C20H19N5O
5-(1H-imidazol-1-yl)-3-phenyl-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[3,4-c]pyridine
—— 4-[6-methyl-4-(4-methylpiperazin-1-yl)quinolin-2-yl]-2,3,4,5-tetrahydro-1,4-benzothiazepine 1,1-dioxide 1422497-83-3 C24H28N4O2S
4-[6-methyl-4-(4-methylpiperazin-1-yl)quinolin-2-yl]-2,3,4,5-tetrahydro-1,4-benzothiazepine 1,1-dioxide
—— N-{1-[3-(1-ethyl-5-{[5-fluoropyrimidin-2-yl]oxy}-1H-pyrazol-3-yl)phenyl]cyclopropyl}-2,2,2-trifluoroethanesulfonamide 1289202-19-2 C20H19F4N5O3S
N-{1-[3-(1-ethyl-5-{[5-fluoropyrimidin-2-yl]oxy}-1H-pyrazol-3-yl)phenyl]cyclopropyl}-2,2,2-trifluoroethanesulfonamide
—— 4-[(1-cyclobutylpiperidin-4-ylidene)methyl]-N-methyl-N-(tetrahydro-2H-pyran-4-yl)benzenesulfonamide 1425972-81-1 C22H32N2O3S
4-[(1-cyclobutylpiperidin-4-ylidene)methyl]-N-methyl-N-(tetrahydro-2H-pyran-4-yl)benzenesulfonamide
—— 6-bromo-N-(2-fluoro-5-(2-(4-methylpiperazin-1-yl)benzylcarbamoyl)phenyl)pyrazolo[1,5-a]pyridine-3-carboxamide 1426531-79-4 C27H26BrFN6O2
6-bromo-N-(2-fluoro-5-(2-(4-methylpiperazin-1-yl)benzylcarbamoyl)phenyl)pyrazolo[1,5-a]pyridine-3-carboxamide
—— cyclobutyl 1-[[2,3-dimethoxy-6-(1-oxoindan-4-yl)phenoxy]methyl]cyclopropanecarboxylate 1345881-59-5 C26H28O6
cyclobutyl 1-[[2,3-dimethoxy-6-(1-oxoindan-4-yl)phenoxy]methyl]cyclopropanecarboxylate
—— 8-bromo-5-oxo-2,3,4,5-tetrahydrobenzo[b]oxepin-4-yl 1-((tert-butoxycarbonyl)amino)cyclobutanecarboxylate 1426331-53-4 C20H24BrNO6
8-bromo-5-oxo-2,3,4,5-tetrahydrobenzo[b]oxepin-4-yl 1-((tert-butoxycarbonyl)amino)cyclobutanecarboxylate
—— 5-amino-2-(2,6-difluorophenyl)-N-(5-((2,2-dimethyl-1,3-dioxolan-4-yl)methoxy)isothiazol-4-yl)thiazole-4-carboxamide 1422395-17-2 C19H18F2N4O4S2
5-amino-2-(2,6-difluorophenyl)-N-(5-((2,2-dimethyl-1,3-dioxolan-4-yl)methoxy)isothiazol-4-yl)thiazole-4-carboxamide
—— 6-(4-(benzyloxy)-1-methyl-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid 1426527-40-3 C24H22N2O4
6-(4-(benzyloxy)-1-methyl-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid
—— isobutyl 1-[[2,3-dimethoxy-6-(1-oxoindan-4-yl)phenoxy]methyl]cyclopropanecarboxylate 1345881-60-8 C26H30O6
isobutyl 1-[[2,3-dimethoxy-6-(1-oxoindan-4-yl)phenoxy]methyl]cyclopropanecarboxylate
—— 1-(5-oxo-4-((4-(piperazin-1-ylmethyl)phenyl)amino)-5,6-dihydropyrimido[4,5-d]pyridazin-2-yl)piperidine-4-carboxylic acid hydrochloride 1425380-21-7 C23H28N8O3*ClH
1-(5-oxo-4-((4-(piperazin-1-ylmethyl)phenyl)amino)-5,6-dihydropyrimido[4,5-d]pyridazin-2-yl)piperidine-4-carboxylic acid hydrochloride
—— (3aR,6aS)-5-(2-methoxyphenyl)-2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrole 1422449-82-8 C13H18N2O
(3aR,6aS)-5-(2-methoxyphenyl)-2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrole
—— N-{[3-(aminomethyl)oxetan-3-yl]methyl}-6-methyl-2-(1-oxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)quinolin-4-amine 1422498-96-1 C24H28N4O2S
N-{[3-(aminomethyl)oxetan-3-yl]methyl}-6-methyl-2-(1-oxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)quinolin-4-amine
—— 2-amino-4-[[(1S)-1-[8-(2-methylpyrimidin-5-yl)-2-(1,2-oxazol-3-yl)-1-oxoisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile 1425043-65-7 C24H19N9O2
2-amino-4-[[(1S)-1-[8-(2-methylpyrimidin-5-yl)-2-(1,2-oxazol-3-yl)-1-oxoisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile
—— Ethyl 1-[4-[2-[(4-bromo-2-cyanophenyl)methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylate 1423071-47-9 C26H26BrN3O3S
Ethyl 1-[4-[2-[(4-bromo-2-cyanophenyl)methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— methyl (S)-4-(1-methanesulfonylaminoethyl)benzoate 1346123-69-0 C11H15NO4S
methyl (S)-4-(1-methanesulfonylaminoethyl)benzoate
—— 6-{4-[3-(dimethylamino)pyrrolidin-1-yl]-2-fluorophenyl}-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid 1426665-85-1 C20H24FN3O3
6-{4-[3-(dimethylamino)pyrrolidin-1-yl]-2-fluorophenyl}-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid