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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-(3-chlorophenyl)piperidin-1-yl)-N-(6-(4-(2-fluorophenylcarbamoyl)piperazin-1-yl)pyridin-3-yl)-4-(trifluoromethyl)oxazole-5-carboxamide 1228003-16-4 C32H30ClF4N7O3
2-(4-(3-chlorophenyl)piperidin-1-yl)-N-(6-(4-(2-fluorophenylcarbamoyl)piperazin-1-yl)pyridin-3-yl)-4-(trifluoromethyl)oxazole-5-carboxamide
—— 4-(2-methylphenyl)-1-(3-(1-naphthyloxy)propyl)-3-((3-(trifluoromethoxy)phenyl)amino)-1H-indole-2-carboxylic acid 1072900-67-4 C36H29F3N2O4
4-(2-methylphenyl)-1-(3-(1-naphthyloxy)propyl)-3-((3-(trifluoromethoxy)phenyl)amino)-1H-indole-2-carboxylic acid
—— (E)-4-(1-(acetoxyimino)ethyl)benzonitrile 1426021-82-0 C11H10N2O2
(E)-4-(1-(acetoxyimino)ethyl)benzonitrile
—— 5-chloro-N-(2-hydroxyphenyl)pentanamide 1610700-32-7 C11H14ClNO2
5-chloro-N-(2-hydroxyphenyl)pentanamide
—— ethyl 2-isopropyl-3-oxopentanoate 118793-28-5 C10H18O3
ethyl 2-isopropyl-3-oxopentanoate
—— 6-(3-(2-bromophenyl)triaz-2-en-1-yl)quinoline 1256156-67-8 C15H11BrN4
6-(3-(2-bromophenyl)triaz-2-en-1-yl)quinoline
—— 22β-(4-iodobenzyloxy)-3β,24-isopropylidenedioxyolean-12-ene 1311130-41-2 C40H59IO3
22β-(4-iodobenzyloxy)-3β,24-isopropylidenedioxyolean-12-ene
—— 4-(2-bromo-1,1-dimethoxyethyl)benzonitrile 164594-65-4 C11H12BrNO2
4-(2-bromo-1,1-dimethoxyethyl)benzonitrile
—— 4,5,6,7-Tetrachloro-2,2-diethyl-2λ<sup>4</sup>-benzo[1,3,2]dioxatellurole 145593-02-8 C10H10Cl4O2Te
4,5,6,7-Tetrachloro-2,2-diethyl-2λ<sup>4</sup>-benzo[1,3,2]dioxatellurole
—— 4-[Benzyl(propan-2-yl)amino]-1-naphthalen-2-ylbutan-1-ol 1146191-29-8 C24H29NO
4-[Benzyl(propan-2-yl)amino]-1-naphthalen-2-ylbutan-1-ol
—— 4,5,6,7-tetrahydro-benzo[b]thiophene-2-carboxylic acid {3-[5-(6-cyclopropylamino-pyridazin-3-ylamino)-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl]-2-methyl-phenyl}-amide 1013116-57-8 C29H30N6O2S
4,5,6,7-tetrahydro-benzo[b]thiophene-2-carboxylic acid {3-[5-(6-cyclopropylamino-pyridazin-3-ylamino)-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl]-2-methyl-phenyl}-amide
—— N-[1-(4-chlorobenzyl)-2-hydroxyethyl]-4-ethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide 1104273-12-2 C19H19ClN4O2S
N-[1-(4-chlorobenzyl)-2-hydroxyethyl]-4-ethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— 4-(5-tert-butyl-1H-pyrazol-4-yl)-N-(2,3-dihydro-1H-inden-1-yl)pyridin-2-amine 1160104-13-1 C21H24N4
4-(5-tert-butyl-1H-pyrazol-4-yl)-N-(2,3-dihydro-1H-inden-1-yl)pyridin-2-amine
—— 5-[(4-acetyl-2-methylphenoxy)methyl]-3-phenyl-1,3-oxazolidin-2-one 1174338-11-4 C19H19NO4
5-[(4-acetyl-2-methylphenoxy)methyl]-3-phenyl-1,3-oxazolidin-2-one
—— 5-(3-butyl-5-methyl-isoxazol-4-ylmethoxy)-2H-pyrazole-3-carboxylic acid (2-hydroxy-1-hydroxymethyl-ethyl)-amide 1254964-64-1 C16H24N4O5
5-(3-butyl-5-methyl-isoxazol-4-ylmethoxy)-2H-pyrazole-3-carboxylic acid (2-hydroxy-1-hydroxymethyl-ethyl)-amide
—— 4-[2-Ethyl-4-(2-fluoro-4-methylphenyl)phenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one 1160560-11-1 C24H27FO3
4-[2-Ethyl-4-(2-fluoro-4-methylphenyl)phenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one
—— 3-[3-(3-chloro-4-isopropoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-1-thiophen-2-yl-propan-1-one 1035213-51-4 C18H17ClN2O3S
3-[3-(3-chloro-4-isopropoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-1-thiophen-2-yl-propan-1-one
—— (2S)-2-({[(3S)-3-(pent-4-en-1-yloxy)pyrrolidin-1-yl]carbonyl}amino)non-8-enoic acid 1025369-10-1 C19H32N2O4
(2S)-2-({[(3S)-3-(pent-4-en-1-yloxy)pyrrolidin-1-yl]carbonyl}amino)non-8-enoic acid
—— N,N-diethyl-6,9,12-trioxa-3,15,21-triazabicyclo[15.3.1]henicosa-1(20),17(21),18-trien-19-amine 135456-41-6 C19H34N4O3
N,N-diethyl-6,9,12-trioxa-3,15,21-triazabicyclo[15.3.1]henicosa-1(20),17(21),18-trien-19-amine
—— 2-phenylselanylpyridine-3-carbaldehyde 1350431-58-1 C12H9NOSe
2-phenylselanylpyridine-3-carbaldehyde
—— (E)-2-(bis(ethylthio)methylene)-5-(4-methoxyphenyl)-3-oxo-N-phenylpent-4-enamide 1262340-25-9 C23H25NO3S2
(E)-2-(bis(ethylthio)methylene)-5-(4-methoxyphenyl)-3-oxo-N-phenylpent-4-enamide
—— (3Z,5E)-6-[tert-butyl(dimethyl)silyl]-2,2-dimethyl-N-trimethylsilylhexa-3,5-dien-3-amine 181211-08-5 C17H37NSi2
(3Z,5E)-6-[tert-butyl(dimethyl)silyl]-2,2-dimethyl-N-trimethylsilylhexa-3,5-dien-3-amine
—— 4-(2-hydroxyphenyl)-8-methyl-7-nitroquinoline-3-carboxylic acid 1394232-20-2 C17H12N2O5
4-(2-hydroxyphenyl)-8-methyl-7-nitroquinoline-3-carboxylic acid
—— (1R)-1-(4-fluoronaphthalen-1-yl)ethanamine hydrochloride 1211473-33-4 C12H12FN*ClH
(1R)-1-(4-fluoronaphthalen-1-yl)ethanamine hydrochloride
—— 4-[2-Ethyl-4-(4-fluorophenyl)phenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one 1160559-69-2 C23H25FO3
4-[2-Ethyl-4-(4-fluorophenyl)phenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one
—— [4-[4-(3,4-Dichlorophenyl)-2-ethylphenyl]-2,2,6,6-tetramethyl-5-oxopyran-3-yl] acetate 1160560-89-3 C25H26Cl2O4
[4-[4-(3,4-Dichlorophenyl)-2-ethylphenyl]-2,2,6,6-tetramethyl-5-oxopyran-3-yl] acetate
—— ethyl 3-[3-(2-tert-butyl-4-fluorophenoxy)pyrrolidin-1-yl]-3-oxopropanoate 1146959-44-5 C19H26FNO4
ethyl 3-[3-(2-tert-butyl-4-fluorophenoxy)pyrrolidin-1-yl]-3-oxopropanoate
—— 3-(2,4-Dihydroxy-3-methylbenzoyl)-1-methyl-2-piperidone 152428-32-5 C14H17NO4
3-(2,4-Dihydroxy-3-methylbenzoyl)-1-methyl-2-piperidone
—— 5-[2-(4-fluorophenyl)-2H-pyrazol-3-yl]-3-thiophen-2-yl-benzo[c]isoxazole 1539280-88-0 C20H12FN3OS
5-[2-(4-fluorophenyl)-2H-pyrazol-3-yl]-3-thiophen-2-yl-benzo[c]isoxazole
—— (R)-2-(1-((6-((4,4-difluorocyclohexyl)oxy)-5-(trifluoromethyl)naphthalen-2-yl)methyl)piperidin-3-yl)acetic acid 1548145-20-5 C25H28F5NO3
(R)-2-(1-((6-((4,4-difluorocyclohexyl)oxy)-5-(trifluoromethyl)naphthalen-2-yl)methyl)piperidin-3-yl)acetic acid
—— US10138229, Example 20 1558036-47-7 C25H24Cl2N4O4
US10138229, Example 20
—— (S)-isopropyl 2-(((6-methylpyridin-2-yl)methyl)carbamoyl)pyrrolidine-1-carboxylate 1422467-54-6 C16H23N3O3
(S)-isopropyl 2-(((6-methylpyridin-2-yl)methyl)carbamoyl)pyrrolidine-1-carboxylate
—— methyl 3-(2-phenylcyclopent-1-enyl)propanoate 1380523-83-0 C15H18O2
methyl 3-(2-phenylcyclopent-1-enyl)propanoate
—— 5-(3-(6-chloro-1H-benzoimidazol-2-yl)phenyl)-5-methylmorpholin-3-one 1392106-05-6 C18H16ClN3O2
5-(3-(6-chloro-1H-benzoimidazol-2-yl)phenyl)-5-methylmorpholin-3-one
—— 17α-mercapto-androst-5-en-3β-ol 109836-12-6 C19H30OS
17α-mercapto-androst-5-en-3β-ol
—— 2,4-Dimethyl-6-p-tolyl-4,7,8,9-tetrahydro-cyclopenta[4,5]pyrido[2,3-d]pyrimidine-1,3-dione 113290-26-9 C19H19N3O2
2,4-Dimethyl-6-p-tolyl-4,7,8,9-tetrahydro-cyclopenta[4,5]pyrido[2,3-d]pyrimidine-1,3-dione
—— 3-(1-methyl-5-(4-methyl-cyclohexyl)-1,2,3,6-tetrahydro-pyridin-4-yl)-5-(4-thiazol-4-ylethynyl-phenyl)-thiophene-2-carboxylic acid 1383526-58-6 C29H30N2O2S2
3-(1-methyl-5-(4-methyl-cyclohexyl)-1,2,3,6-tetrahydro-pyridin-4-yl)-5-(4-thiazol-4-ylethynyl-phenyl)-thiophene-2-carboxylic acid
—— 6-ethyl-6-nitro-1-(2-nitro-butyl)-hexahydro-[1,4]diazepine 105974-27-4 C11H22N4O4
6-ethyl-6-nitro-1-(2-nitro-butyl)-hexahydro-[1,4]diazepine
—— 4-<1-Methyl-hepten-(1)-yl>-phenol 17404-16-9 C14H20O
4-<1-Methyl-hepten-(1)-yl>-phenol
—— (+/-)-N-[5-(4-bromo-phenyl)-1-(2,4-dichloro-phenyl)-4,5-dihydro-1H-pyrazol-3-ylmethyl]-3-cyclohexyl-acrylamide 1029695-06-4 C25H26BrCl2N3O
(+/-)-N-[5-(4-bromo-phenyl)-1-(2,4-dichloro-phenyl)-4,5-dihydro-1H-pyrazol-3-ylmethyl]-3-cyclohexyl-acrylamide
—— N-phenyl-6-(2-phenylethenyl)-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide 1214926-93-8 C22H19N3O2
N-phenyl-6-(2-phenylethenyl)-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide
—— 3-chloro-5-(6-chloro-3-((5-(2,4-dimethyloxazol-5-yl)-1,3,4-oxadiazol-2-yl)methyl)-2-fluorophenoxy)benzonitrile 1094343-17-5 C21H13Cl2FN4O3
3-chloro-5-(6-chloro-3-((5-(2,4-dimethyloxazol-5-yl)-1,3,4-oxadiazol-2-yl)methyl)-2-fluorophenoxy)benzonitrile
—— (3'Z,5'Z)-celaxanthin 1173048-20-8 C40H54O
(3'Z,5'Z)-celaxanthin
—— US10138229, Example 70 1558037-01-6 C24H23ClN4O3
US10138229, Example 70
—— (S)-methyl 1-((R)-1-(naphthalen-2-yl)-2-nitroethyl)-2-oxocyclopentanecarboxylate 1167427-81-7 C19H19NO5
(S)-methyl 1-((R)-1-(naphthalen-2-yl)-2-nitroethyl)-2-oxocyclopentanecarboxylate
—— —— 143267-60-1 C18H27NO6
—— 1,3-bis[[4-(phenoxymethyl)-1H-1,2,3-triazol-1-yl]methyl]benzene 1451257-00-3 C26H24N6O2
1,3-bis[[4-(phenoxymethyl)-1H-1,2,3-triazol-1-yl]methyl]benzene
—— 10-chloro-2-fluoro-5,12-dihydroindolo[3,2-b][1,5]benzodiazepine 1346156-86-2 C15H9ClFN3
10-chloro-2-fluoro-5,12-dihydroindolo[3,2-b][1,5]benzodiazepine
—— 2-methoxydibenzofuran-3-sulfonic acid 190522-68-0 C13H10O5S
2-methoxydibenzofuran-3-sulfonic acid
—— methyl 3(5)-<(2-benzyloxy)ethoxymethyl>-4-(benzyloxymethyl)pyrazole-5(3)-carboxylate 149125-66-6 C23H26N2O5
methyl 3(5)-<(2-benzyloxy)ethoxymethyl>-4-(benzyloxymethyl)pyrazole-5(3)-carboxylate