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中文名称 英文名称 CAS号 化学式 结构式图片
—— [4-(2,6-dimethylpyridin-3-yl)piperazin-1-yl][4-(1,1-dioxo-1λ<sup>6</sup>-isothiazolidin-2-yl)-2-methanesulfonylphenyl]methanone 1346115-45-4 C22H28N4O5S2
[4-(2,6-dimethylpyridin-3-yl)piperazin-1-yl][4-(1,1-dioxo-1λ<sup>6</sup>-isothiazolidin-2-yl)-2-methanesulfonylphenyl]methanone
—— (R)-1-(6-(5-(pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridine-3-yl)pyridin-2-yl)piperidin-3-amine 1422438-61-6 C21H21N7
(R)-1-(6-(5-(pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridine-3-yl)pyridin-2-yl)piperidin-3-amine
—— 1-((3,5-dimethylisoxazol-4-yl)(5-(2-(((2,4-dimethylphenyl)(phenyl)methyl)amino)-2-oxoethyl)benzofuran-2-yl)methyl)azetidine-3-carboxylic acid 1422167-24-5 C35H35N3O5
1-((3,5-dimethylisoxazol-4-yl)(5-(2-(((2,4-dimethylphenyl)(phenyl)methyl)amino)-2-oxoethyl)benzofuran-2-yl)methyl)azetidine-3-carboxylic acid
—— 4-amino-6-[[(1S)-1-[8-(1-methyl-6-oxopyridin-3-yl)-1-oxo-2-phenylisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile 1425044-35-4 C28H23N7O2
4-amino-6-[[(1S)-1-[8-(1-methyl-6-oxopyridin-3-yl)-1-oxo-2-phenylisoquinolin-3-yl]ethyl]amino]pyrimidine-5-carbonitrile
—— 6-(4-((2-(azepan-1-yl)-5-oxo-5,6-dihydropyrimido[4,5-d]pyridazin-4-yl)amino)-2-fluorophenyl)-6-azaspiro[2.5]octane-1-carboxylic acid 1425381-03-8 C26H30FN7O3
6-(4-((2-(azepan-1-yl)-5-oxo-5,6-dihydropyrimido[4,5-d]pyridazin-4-yl)amino)-2-fluorophenyl)-6-azaspiro[2.5]octane-1-carboxylic acid
—— 1-{4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}-4-methylcyclohexane-1,4-diol 1425971-63-6 C23H33NO2
1-{4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}-4-methylcyclohexane-1,4-diol
—— 2-(2,6-difluorophenyl)-N-(5-((4-hydroxy-4-methylpentyl)oxy)isothiazol-4-yl)-5-(methylamino)thiazole-4-carboxamide 1422395-24-1 C20H22F2N4O3S2
2-(2,6-difluorophenyl)-N-(5-((4-hydroxy-4-methylpentyl)oxy)isothiazol-4-yl)-5-(methylamino)thiazole-4-carboxamide
—— 2-{[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-7-fluoro-6-methylquinolin-4-yl]amino}ethanol 1422498-32-5 C21H22FN3O3S
2-{[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-7-fluoro-6-methylquinolin-4-yl]amino}ethanol
—— (S)-2-(1-benzyl-2-piperidinyl)pyridine 1061659-71-9 C17H20N2
(S)-2-(1-benzyl-2-piperidinyl)pyridine
—— N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-6-piperazin-1-yl-pyridine-3-carboxamide 1027354-13-7 C30H32N6O2
N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-6-piperazin-1-yl-pyridine-3-carboxamide
—— (2-(2-amino-3-morpholinoquinolin-6-yl)-3-methylphenyl)(3,3-difluoroazetidin-1-yl)methanone 1319195-25-9 C24H24F2N4O2
(2-(2-amino-3-morpholinoquinolin-6-yl)-3-methylphenyl)(3,3-difluoroazetidin-1-yl)methanone
—— 5-methoxy-3-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-1H-quinazoline-2,4-dione 1422209-28-6 C23H22N4O6S
5-methoxy-3-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-1H-quinazoline-2,4-dione
—— 6-(3-cyano-1-methyl-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid 1426524-50-6 C18H15N3O3
6-(3-cyano-1-methyl-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid
—— 6-[3-chloro-4-(methylsulfinyl)phenyl]pyrimidine-4-carboxylic acid 1426320-13-9 C12H9ClN2O3S
6-[3-chloro-4-(methylsulfinyl)phenyl]pyrimidine-4-carboxylic acid
—— 1-[4-[3-Methyl-2-[[2-methyl-4-(morpholin-4-ylmethyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylic acid 1423066-81-2 C29H35N3O4S
1-[4-[3-Methyl-2-[[2-methyl-4-(morpholin-4-ylmethyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]piperidine-4-carboxylic acid
—— 5-ethyl-6-[4-(3-fluoropyrrolidin-1-yl)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxylic acid 1426662-70-5 C18H19FN2O3
5-ethyl-6-[4-(3-fluoropyrrolidin-1-yl)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxylic acid
—— 6-(2-((benzyl(methyl)amino)methyl)-1-methyl-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid 1426524-93-7 C26H27N3O3
6-(2-((benzyl(methyl)amino)methyl)-1-methyl-1H-indol-5-yl)-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid
—— (S)-2-(methoxycarbonyl)amino-N-(1-(6-(4-(2-((S)-1-((S)-2-((methoxycarbonyl)amino)-3-methylbutanoyl)pyrrolidin-2-yl)-1H-naphtho[1,2-d]imidazol-7-yl)phenyl)-1H-benzo[d]imidazol-2-yl)cyclobutyl)-3-methylbutanamide 1426330-59-7 C46H52N8O6
(S)-2-(methoxycarbonyl)amino-N-(1-(6-(4-(2-((S)-1-((S)-2-((methoxycarbonyl)amino)-3-methylbutanoyl)pyrrolidin-2-yl)-1H-naphtho[1,2-d]imidazol-7-yl)phenyl)-1H-benzo[d]imidazol-2-yl)cyclobutyl)-3-methylbutanamide
—— 6-{4-[3-(aminomethyl)pyrrolidin-1-yl]phenyl}-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid trifluoroacetate 1426664-11-0 C2HF3O2*C19H23N3O3
6-{4-[3-(aminomethyl)pyrrolidin-1-yl]phenyl}-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid trifluoroacetate
—— 6-[5-(dimethylamino)thiophen-2-yl]-5-ethyl-4-hydroxy-2-oxo-1,2-dihydropyridine-3-carboxylic acid 1426668-74-7 C14H16N2O4S
6-[5-(dimethylamino)thiophen-2-yl]-5-ethyl-4-hydroxy-2-oxo-1,2-dihydropyridine-3-carboxylic acid
—— 6-[4-(7-amino-5-azaspiro[2.4]hept-5-yl)phenyl]-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid trifluoroacetate 1426665-44-2 C2HF3O2*C20H23N3O3
6-[4-(7-amino-5-azaspiro[2.4]hept-5-yl)phenyl]-5-ethyl-2-oxo-1,2-dihydropyridine-3-carboxylic acid trifluoroacetate
—— (4aR,8aS)-8a-(2,6-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-amine 1425947-69-8 C13H14F2N2OS
(4aR,8aS)-8a-(2,6-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-amine
—— 2-(3-phenyl-2-[(5-pyridino[3,4-b]pyridin-3-yl(1,3,4-thiadiazol-2-yl))amino]propyl)benzo[c]azolidine-1,3-dione 1015070-02-6 C27H20N6O2S
2-(3-phenyl-2-[(5-pyridino[3,4-b]pyridin-3-yl(1,3,4-thiadiazol-2-yl))amino]propyl)benzo[c]azolidine-1,3-dione
—— 3-((3-hydroxyazetidin-1-ylsulfonyl)methyl)phenylamine 1219824-82-4 C10H14N2O3S
3-((3-hydroxyazetidin-1-ylsulfonyl)methyl)phenylamine
—— (1R,6S)-3-[4-[2-[[4-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]-2-methylphenyl]methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]-3-azabicyclo[4.1.0]heptane-6-carboxylic acid 1423068-82-9 C30H35N3O5S2
(1R,6S)-3-[4-[2-[[4-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]-2-methylphenyl]methoxy]-5-methylphenyl]-1,3-thiazol-2-yl]-3-azabicyclo[4.1.0]heptane-6-carboxylic acid
—— 6,8-dichloro-1-(methyl(2-oxo-2-((pyridin-3-ylmethyl)amino)ethyl)amino)isoquinoline-3-carboxylic acid 1426383-34-7 C19H16Cl2N4O3
6,8-dichloro-1-(methyl(2-oxo-2-((pyridin-3-ylmethyl)amino)ethyl)amino)isoquinoline-3-carboxylic acid
—— 3-[(1S)-1-[(2-amino-5-pyridin-4-ylpyrimidin-4-yl)amino]ethyl]-8-(2-methoxypyridin-4-yl)-2-phenylisoquinolin-1-one 1425042-91-6 C32H27N7O2
3-[(1S)-1-[(2-amino-5-pyridin-4-ylpyrimidin-4-yl)amino]ethyl]-8-(2-methoxypyridin-4-yl)-2-phenylisoquinolin-1-one
—— 2-(azepan-1-yl)-4-((4-(((2S,5S)-5-(hydroxymethyl)-1,4-dioxan-2-yl)methoxy)phenyl)amino)pyrimido[4,5-d]pyridazin-5(6H)-one 1425380-80-8 C24H30N6O5
2-(azepan-1-yl)-4-((4-(((2S,5S)-5-(hydroxymethyl)-1,4-dioxan-2-yl)methoxy)phenyl)amino)pyrimido[4,5-d]pyridazin-5(6H)-one
—— 5-[(4-fluoroanilino)methylene]-1-(2-furylmethyl)-3-isopropyl-2,4,6(1H,3H,5H)-pyrimidinetrione 1164454-84-5 C19H18FN3O4
5-[(4-fluoroanilino)methylene]-1-(2-furylmethyl)-3-isopropyl-2,4,6(1H,3H,5H)-pyrimidinetrione
—— 2-amino-7-benzo[1,3]dioxol-4-yl-7,8-dihydro-6H-quinazolin-5-one oxime 1087139-19-2 C15H14N4O3
2-amino-7-benzo[1,3]dioxol-4-yl-7,8-dihydro-6H-quinazolin-5-one oxime
—— 2-(ethylideneamino)oxy-5-fluoro-N-[(2-fluorophenyl)methyl]pyrimidin-4-amine 1312324-14-3 C13H12F2N4O
2-(ethylideneamino)oxy-5-fluoro-N-[(2-fluorophenyl)methyl]pyrimidin-4-amine
—— 5-Fluoro-2-[(4-methylphenyl)methylideneamino]oxypyrimidin-4-amine 1312323-96-8 C12H11FN4O
5-Fluoro-2-[(4-methylphenyl)methylideneamino]oxypyrimidin-4-amine
—— 1-(3,5-Bis-trifluoromethyl-phenyl)-3-(4-chloro-2-trifluoromethyl-phenyl)-urea 1682-89-9 C16H8ClF9N2O
1-(3,5-Bis-trifluoromethyl-phenyl)-3-(4-chloro-2-trifluoromethyl-phenyl)-urea
—— (E)-N-cyclopropylpent-3-enamide 1443734-95-9 C8H13NO
(E)-N-cyclopropylpent-3-enamide
—— 4,4-diethoxy-2-methyl-pyrrolidine 1431885-70-9 C9H19NO2
4,4-diethoxy-2-methyl-pyrrolidine
—— 3-nitro-benzenesulfonic acid-(3-nitro-benzylidenehydrazide) 120167-59-1 C13H10N4O6S
3-nitro-benzenesulfonic acid-(3-nitro-benzylidenehydrazide)
—— 2-(4-benzoylpiperazin-1-yl)-N'-(5-fluoro-2-hydroxy-3-propylbenzylidene)acetohydrazide 1554476-31-1 C23H27FN4O3
2-(4-benzoylpiperazin-1-yl)-N'-(5-fluoro-2-hydroxy-3-propylbenzylidene)acetohydrazide
—— 6-tert-butyl 3-ethyl 5,5-dimethyl-2-(methylsulfinyl)-7-oxo-4,7-dihydrothieno[2,3-c]pyridine-3,6(5H)-dicarboxylate 1008526-81-5 C18H25NO6S2
6-tert-butyl 3-ethyl 5,5-dimethyl-2-(methylsulfinyl)-7-oxo-4,7-dihydrothieno[2,3-c]pyridine-3,6(5H)-dicarboxylate
—— (2-Bromo-phenylmethanesulfonyl)-acetic acid methyl ester 122504-97-6 C10H11BrO4S
(2-Bromo-phenylmethanesulfonyl)-acetic acid methyl ester
—— (5,5-diphenyl-pent-4-enyl)-(4-trifluoromethylbenzyl)amine hydrochloride 1379523-69-9 C24H24FN
(5,5-diphenyl-pent-4-enyl)-(4-trifluoromethylbenzyl)amine hydrochloride
—— 2-(4-<i>tert</i>-butyl-phenyl)-5-<i>p</i>-tolyl-[1,3,4]thiadiazole 17453-11-1 C19H20N2S
2-(4-<i>tert</i>-butyl-phenyl)-5-<i>p</i>-tolyl-[1,3,4]thiadiazole
—— 3-chloro-2-(3-chlorophenyl)tetrahydrofuran 1426692-56-9 C10H10Cl2O
3-chloro-2-(3-chlorophenyl)tetrahydrofuran
—— —— 1384353-08-5 C22H30BrNO2
—— [Pd(η3-2-MeC3H4)(1,10-phenanthroline)]BPh4 1196131-99-3 C16H15N2Pd*C24H20B
[Pd(η3-2-MeC3H4)(1,10-phenanthroline)]BPh4
—— 9,12,17-trioxo-5,6,7,9,12,14,15,16-octahydro-6,15-methanobenzo<a>naphtho<2,3-f>cyclodecene 134591-78-9 C23H18O3
9,12,17-trioxo-5,6,7,9,12,14,15,16-octahydro-6,15-methanobenzo<a>naphtho<2,3-f>cyclodecene
—— spiro[1,3-diazabicyclo[1.2.2]heptane-2,3'-(1,2-diferrocenylcyclopropene)] 1449573-17-4 C27H26Fe2N2
spiro[1,3-diazabicyclo[1.2.2]heptane-2,3'-(1,2-diferrocenylcyclopropene)]
—— N4-cyclohexyl-5,6-dimethyl-N2-[(1R)-1-phenylethyl]pyrimidine-2,4-diamine 1450808-99-7 C20H28N4
N4-cyclohexyl-5,6-dimethyl-N2-[(1R)-1-phenylethyl]pyrimidine-2,4-diamine
—— p-trifluoromethylphenyl 2E,6E,10E-geranylgeranyl carbamate 1453112-85-0 C28H38F3NO2
p-trifluoromethylphenyl 2E,6E,10E-geranylgeranyl carbamate
—— N4-cyclohexyl-5,6-dimethyl-N2-[(5-methylpyridin-2-yl)methyl]pyrimidine-2,4-diamine 1450809-79-6 C19H27N5
N4-cyclohexyl-5,6-dimethyl-N2-[(5-methylpyridin-2-yl)methyl]pyrimidine-2,4-diamine
—— {1-[(S)-4-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridin-3-yl)-benzyl]-piperidin-4-yl}-(3-hydroxy-azetidin-1-yl)-methanone 1454648-62-4 C23H27N3O4
{1-[(S)-4-(2,3-dihydro-[1,4]dioxino[2,3-b]pyridin-3-yl)-benzyl]-piperidin-4-yl}-(3-hydroxy-azetidin-1-yl)-methanone