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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-benzyl-2-(4-[5-bromo-2-(2-chloro-6-fluoro-phenyl)-1H-imidazol-4-yl]-phenyl)-6-methyl-1H-benzoimidazole 1038843-07-0 C30H21BrClFN4
1-benzyl-2-(4-[5-bromo-2-(2-chloro-6-fluoro-phenyl)-1H-imidazol-4-yl]-phenyl)-6-methyl-1H-benzoimidazole
—— 8-[4-[5-Chloro-2-[[2-methyl-4-(piperidine-1-carbonyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid 1423067-76-8 C31H34ClN3O4S
8-[4-[5-Chloro-2-[[2-methyl-4-(piperidine-1-carbonyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 3-methyl-N-[(6-methyl-2-oxo-4-propyl-1H-pyridin-3-yl)methyl]-1-propan-2-yl-6-(1H-pyrazol-4-yl)indazole-4-carboxamide 1346704-42-4 C25H30N6O2
3-methyl-N-[(6-methyl-2-oxo-4-propyl-1H-pyridin-3-yl)methyl]-1-propan-2-yl-6-(1H-pyrazol-4-yl)indazole-4-carboxamide
—— 1-(2-Thiazolyl)-3-methyl-2-oxo-tetrahydroimidazol 14746-92-0 C7H9N3OS
1-(2-Thiazolyl)-3-methyl-2-oxo-tetrahydroimidazol
—— N-(1-(3-((propylamino)methyl)benzyl)-1H-pyrazol-4-yl)-1H-indazole-3-carboxamide 1422980-57-1 C22H24N6O
N-(1-(3-((propylamino)methyl)benzyl)-1H-pyrazol-4-yl)-1H-indazole-3-carboxamide
—— 7,7-diethyl-5,5-dimethyl-N-[1-(1-methylpyrazole-4-carbonyl)pyrrolidin-3-yl]-8-oxo-6,9-dihydrocarbazole-3-carboxamide 1424994-04-6 C28H35N5O3
7,7-diethyl-5,5-dimethyl-N-[1-(1-methylpyrazole-4-carbonyl)pyrrolidin-3-yl]-8-oxo-6,9-dihydrocarbazole-3-carboxamide
—— 1-cyclobutyl-4-(4-{[(5-methyl-1,2-oxazol-3-yl)oxy]methyl}benzylidene)piperidine 1425971-08-9 C21H26N2O2
1-cyclobutyl-4-(4-{[(5-methyl-1,2-oxazol-3-yl)oxy]methyl}benzylidene)piperidine
—— methyl 1-benzo[f][1,3]benzodioxol-6-yl-6-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylate 1071422-38-2 C25H22N2O4
methyl 1-benzo[f][1,3]benzodioxol-6-yl-6-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylate
—— (R)-1-(3-((5-methyl-2-(4-trifluoromethylphenyl)oxazol-4-yl)methoxy)benzyl)piperidine-2-carboxylic acid methyl ester 1065334-39-5 C26H27F3N2O4
(R)-1-(3-((5-methyl-2-(4-trifluoromethylphenyl)oxazol-4-yl)methoxy)benzyl)piperidine-2-carboxylic acid methyl ester
—— 11-ethyl-2-methyl-10,11-dihydrodibenzo[b,f]thiepine 5,5-dioxide 1027351-61-6 C17H18O2S
11-ethyl-2-methyl-10,11-dihydrodibenzo[b,f]thiepine 5,5-dioxide
—— S-(2-acetylphenyl) thiophene-2-carbothioate 1314533-43-1 C13H10O2S2
S-(2-acetylphenyl) thiophene-2-carbothioate
—— (4R)-4-(cyclopropylmethoxymethyl)-5-quinolin-8-ylsulfonyl-1,3,4,6-tetrahydro-2,5-benzoxazocine 1333115-08-4 C24H26N2O4S
(4R)-4-(cyclopropylmethoxymethyl)-5-quinolin-8-ylsulfonyl-1,3,4,6-tetrahydro-2,5-benzoxazocine
—— 1-[4-[4-[5-[[(1R)-1-(2-chlorophenyl)ethoxy]carbonylamino]-1,3-thiazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid 1423685-42-0 C28H23ClN2O4S
1-[4-[4-[5-[[(1R)-1-(2-chlorophenyl)ethoxy]carbonylamino]-1,3-thiazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
—— 5-(2-trifluoromethoxy-phenyl)-2H-pyrazol-3-ylamine 1040724-28-4 C10H8F3N3O
5-(2-trifluoromethoxy-phenyl)-2H-pyrazol-3-ylamine
—— 2-(1-(5-methylpyrazin-2-yl)piperidin-4-yloxy)-6-(1,2,3,6-tetrahydropyridin-4-yl)benzo[d]thiazole 1346627-28-8 C22H25N5OS
2-(1-(5-methylpyrazin-2-yl)piperidin-4-yloxy)-6-(1,2,3,6-tetrahydropyridin-4-yl)benzo[d]thiazole
—— 5-fluoro-3-phenyl-5-[4-(trifluoromethyl)phenyl]-7H-thieno[2,3-b]pyridine-4,6-dione 1313503-93-3 C20H11F4NO2S
5-fluoro-3-phenyl-5-[4-(trifluoromethyl)phenyl]-7H-thieno[2,3-b]pyridine-4,6-dione
—— N-(3-chloro-4-fluorophenyl)-7-(2-fluorophenyl)-2-pyridin-3-ylquinazolin-4-amine 1313896-14-8 C25H15ClF2N4
N-(3-chloro-4-fluorophenyl)-7-(2-fluorophenyl)-2-pyridin-3-ylquinazolin-4-amine
—— 1-[4-{4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}-4-hydroxyhexahydrocyclopenta[c]pyrrol-2(1H)-yl]ethanone 1425971-51-2 C25H34N2O2
1-[4-{4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}-4-hydroxyhexahydrocyclopenta[c]pyrrol-2(1H)-yl]ethanone
—— cyclopentyl(4-((1-ethylpiperidin-4-ylidene)methyl)phenyl)methanol 1425971-39-6 C20H29NO
cyclopentyl(4-((1-ethylpiperidin-4-ylidene)methyl)phenyl)methanol
—— 1-{1-(benzylsulfonyl)piperidin-4-yl}-3,4-dihydro-1H-pyrrolo[3’,2’:5,6]pyrido[4,3-d]pyrimidin-2(7H)-one 1423054-32-3 C21H23N5O3S
1-{1-(benzylsulfonyl)piperidin-4-yl}-3,4-dihydro-1H-pyrrolo[3’,2’:5,6]pyrido[4,3-d]pyrimidin-2(7H)-one
—— N-[2-{[(4-cyanophenyl)carbamoyl]amino}-1-(3-hydroxypropyl)-1H-benzimidazol-5-yl]-N,3-dimethylbutanamide 1424297-11-9 C24H28N6O3
N-[2-{[(4-cyanophenyl)carbamoyl]amino}-1-(3-hydroxypropyl)-1H-benzimidazol-5-yl]-N,3-dimethylbutanamide
—— 4-[4-[2-[1-(5-Fluoropyrimidin-2-yl)piperidin-4-yl]oxy-1,3-benzothiazol-6-yl]piperazin-1-yl]sulfonyl-2-methylbutan-2-ol 1346625-88-4 C25H33FN6O4S2
4-[4-[2-[1-(5-Fluoropyrimidin-2-yl)piperidin-4-yl]oxy-1,3-benzothiazol-6-yl]piperazin-1-yl]sulfonyl-2-methylbutan-2-ol
—— 2-Amino-8-methylmercapto-purin 10179-92-7 C6H7N5S
2-Amino-8-methylmercapto-purin
—— 2-amino-4-methyl-7-(2-pyridin-4-yl-phenyl)-7,8-dihydro-6H-quinazolin-5-one oxime 1087140-50-8 C20H19N5O
2-amino-4-methyl-7-(2-pyridin-4-yl-phenyl)-7,8-dihydro-6H-quinazolin-5-one oxime
—— 3-(benzo[d][1,3]dioxol-5-ylmethyl)-5-((1-methyl-1H-benzo[d]imidazol-2-yl)methylene)-2-thioxothiazolidin-4-one 1019776-54-5 C20H15N3O3S2
3-(benzo[d][1,3]dioxol-5-ylmethyl)-5-((1-methyl-1H-benzo[d]imidazol-2-yl)methylene)-2-thioxothiazolidin-4-one
—— N-Tert-butyl-6-(4-fluorophenyl)-2-{4-[(3-methoxyphenyl)methyl]piperazin-1-YL}imidazo[2,1-B][1,3,4]thiadiazol-5-amine 1058676-69-9 C26H31FN6OS
N-Tert-butyl-6-(4-fluorophenyl)-2-{4-[(3-methoxyphenyl)methyl]piperazin-1-YL}imidazo[2,1-B][1,3,4]thiadiazol-5-amine
—— 3-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(thiazol-2-ylmethylene)-2-thioxothiazolidin-4-one 1019776-61-4 C15H10N2O3S3
3-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(thiazol-2-ylmethylene)-2-thioxothiazolidin-4-one
—— methyl 1-(2-tert-butoxy-2-oxoethyl)-2-(2-aminophenyl)-3-cyclohexyl-1H-indole-6-carboxylate 1160266-58-9 C28H34N2O4
methyl 1-(2-tert-butoxy-2-oxoethyl)-2-(2-aminophenyl)-3-cyclohexyl-1H-indole-6-carboxylate
—— 5-(2-(3,4-dimethoxyphenyl)propan-2-yl)-1-(4-fluorophenyl)-2-((2-(4-(2-methyl-1H-imidazol-1-yl)phenoxy)ethyl)sulfinyl)-1H-imidazole 1430211-38-3 C32H33FN4O4S
5-(2-(3,4-dimethoxyphenyl)propan-2-yl)-1-(4-fluorophenyl)-2-((2-(4-(2-methyl-1H-imidazol-1-yl)phenoxy)ethyl)sulfinyl)-1H-imidazole
—— 8-[4-[5-Cyano-2-[[2-methyl-4-(morpholin-4-ylmethyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid 1423067-46-2 C31H34N4O4S
8-[4-[5-Cyano-2-[[2-methyl-4-(morpholin-4-ylmethyl)phenyl]methoxy]phenyl]-1,3-thiazol-2-yl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— ethyl 1-(3-chloro-2,6-difluorophenyl)-1H-imidazole-4-carboxylate 1422386-59-1 C12H9ClF2N2O2
ethyl 1-(3-chloro-2,6-difluorophenyl)-1H-imidazole-4-carboxylate
—— 4-[4-(3-Chloro-4-fluoroanilino)-2-pyridin-3-ylquinazolin-6-yl]benzamide 1313895-74-7 C26H17ClFN5O
4-[4-(3-Chloro-4-fluoroanilino)-2-pyridin-3-ylquinazolin-6-yl]benzamide
—— N-[1-[[5-(methylcarbamoyl)-2-furyl]methyl]pyrazol-4-yl]-6-(3-pyridyl)-1H-indazole-3-carboxamide 1422979-93-8 C23H19N7O3
N-[1-[[5-(methylcarbamoyl)-2-furyl]methyl]pyrazol-4-yl]-6-(3-pyridyl)-1H-indazole-3-carboxamide
—— 4-Brom-3-methyl-1-phenyl-pyrazol-carbonsaeure-(5) 16146-35-3 C11H9BrN2O2
4-Brom-3-methyl-1-phenyl-pyrazol-carbonsaeure-(5)
—— methyl (3R,4R,5S,6R)-5,6-bis[[tert-butyl(dimethyl)silyl]oxy]-3-hydroxy-4-methyl-2-methylideneheptanoate 1196871-18-7 C22H46O5Si2
methyl (3R,4R,5S,6R)-5,6-bis[[tert-butyl(dimethyl)silyl]oxy]-3-hydroxy-4-methyl-2-methylideneheptanoate
—— 2,3,4-tri-O-acetyl-5-bromo-5-deoxy-N-hexyl-D-ribonamide 1190205-39-0 C17H28BrNO7
2,3,4-tri-O-acetyl-5-bromo-5-deoxy-N-hexyl-D-ribonamide
—— (5-Undecyl-[1,3,4]oxadiazol-2-yl)-acetonitrile 120634-27-7 C15H25N3O
(5-Undecyl-[1,3,4]oxadiazol-2-yl)-acetonitrile
—— (Z)-1-(tert-butylthio)-2-(4-isobutylphenyl)diazene 140244-84-4 C14H22N2S
(Z)-1-(tert-butylthio)-2-(4-isobutylphenyl)diazene
—— (6aS,12bR)-10,10-dimethyl-7,12b-dihydro-[1,3]dioxolo[4',5':5,6]indeno[2,1-c]chromene-3,4,6a(6H)-triol 1261995-43-0 C19H18O6
(6aS,12bR)-10,10-dimethyl-7,12b-dihydro-[1,3]dioxolo[4',5':5,6]indeno[2,1-c]chromene-3,4,6a(6H)-triol
—— [RhH(CO)2(1-(2,8-dimethylphenoxaphosphino)-1'-bis(diphenylphosphino)ferrocene)] 1215039-34-1 C38H31FeO3P2Rh
[RhH(CO)2(1-(2,8-dimethylphenoxaphosphino)-1'-bis(diphenylphosphino)ferrocene)]
—— (S)-[(4R,5S)-5-((2R,4S)-1-Benzyl-4-hydroxy-piperidin-2-yl)-2,2-dimethyl-[1,3]dioxolan-4-yl]-benzyloxy-acetaldehyde 163456-92-6 C26H33NO5
(S)-[(4R,5S)-5-((2R,4S)-1-Benzyl-4-hydroxy-piperidin-2-yl)-2,2-dimethyl-[1,3]dioxolan-4-yl]-benzyloxy-acetaldehyde
—— methyl 4-[[5-methoxy-2-[(trimethylsilyl)ethynyl]phenyl]-ethynyl]benzoate 1378284-26-4 C22H22O3Si
methyl 4-[[5-methoxy-2-[(trimethylsilyl)ethynyl]phenyl]-ethynyl]benzoate
—— 2-ethyl-6-[2-(4-morpholino)ethoxy]-4-[-(2'-(2-triphenylmethyl-2H-tetrazol-5-yl)biphenyl-4-yl)methoxy]-1,5-naphthyridine 143071-87-8 C49H45N7O3
2-ethyl-6-[2-(4-morpholino)ethoxy]-4-[-(2'-(2-triphenylmethyl-2H-tetrazol-5-yl)biphenyl-4-yl)methoxy]-1,5-naphthyridine
—— 1-(2-chloro-4-trifluoromethylphenyl)-4-trifluoromethylsulfinylimidazole 132897-07-5 C11H5ClF6N2OS
1-(2-chloro-4-trifluoromethylphenyl)-4-trifluoromethylsulfinylimidazole
—— 3-[2-[4-(6-fluoro-1-methyl-1H-indazol-3-yl)-1-piperidinyl]-ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one 129014-66-0 C24H26FN5O
3-[2-[4-(6-fluoro-1-methyl-1H-indazol-3-yl)-1-piperidinyl]-ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
—— (E)-N-(6,6-dimethyl-2-hepten-4-ynyl)-N-ethyl-3-[3-(1-pyrrolyl)benzylthio]benzylamine 155294-27-2 C29H34N2S
(E)-N-(6,6-dimethyl-2-hepten-4-ynyl)-N-ethyl-3-[3-(1-pyrrolyl)benzylthio]benzylamine
—— 2-[2,3-dichloro-4-[(8R)-2-[6-methoxy-5-(4-methylimidazol-1-yl)pyridin-2-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]phenyl]-2-methylpropanenitrile 1242311-59-6 C26H25Cl2N7O
2-[2,3-dichloro-4-[(8R)-2-[6-methoxy-5-(4-methylimidazol-1-yl)pyridin-2-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-8-yl]phenyl]-2-methylpropanenitrile
—— (3S,4R,5R)-5-(aminomethyl)-2-[[3-[3-(dimethylamino)-5-[[(2R)-1-ethylpyrrolidin-2-yl]methylcarbamoyl]phenyl]-2-methoxyphenyl]methyl]-4-[(1S)-1-hydroxyethyl]-N-[(1S,2S,3S,5R)-2,6,6-trimethyl-3-bicyclo[3.1.1]heptanyl]-1,2-oxazolidine-3-carboxamide 1009092-21-0 C41H62N6O5
(3S,4R,5R)-5-(aminomethyl)-2-[[3-[3-(dimethylamino)-5-[[(2R)-1-ethylpyrrolidin-2-yl]methylcarbamoyl]phenyl]-2-methoxyphenyl]methyl]-4-[(1S)-1-hydroxyethyl]-N-[(1S,2S,3S,5R)-2,6,6-trimethyl-3-bicyclo[3.1.1]heptanyl]-1,2-oxazolidine-3-carboxamide
—— 5-[3-[1-(4-bromophenyl)cyclobutyl]-1,2,4-oxadiazol-5-yl]-N-(2-methoxyethyl)pyridine-2-carboxamide 1361190-09-1 C21H21BrN4O3
5-[3-[1-(4-bromophenyl)cyclobutyl]-1,2,4-oxadiazol-5-yl]-N-(2-methoxyethyl)pyridine-2-carboxamide
—— US10202379, Reference Example 498 1370242-30-0 C24H25N3O3
US10202379, Reference Example 498