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—— 2,6-difluoro-N-[3-[5-[2-(3-fluoro-4-morpholin-4-ylanilino)pyrimidin-4-yl]-2-piperidin-1-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide 1244645-06-4 C34H32F3N7O3S2
2,6-difluoro-N-[3-[5-[2-(3-fluoro-4-morpholin-4-ylanilino)pyrimidin-4-yl]-2-piperidin-1-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide
—— 2-(3,6-dichloro-2-fluoro-phenylamino)-N-(4,4-dimethyl-cyclohex-1-yl)-6-methoxy-1H-benzimidazole-5-carboxamide 1219123-95-1 C23H25Cl2FN4O2
2-(3,6-dichloro-2-fluoro-phenylamino)-N-(4,4-dimethyl-cyclohex-1-yl)-6-methoxy-1H-benzimidazole-5-carboxamide
—— 3-(2-Phenylethyl)-6-[3-(trifluoromethyl)anilino]-1-[[4-(trifluoromethyl)phenyl]methyl]-1,3,5-triazine-2,4-dione 1239686-30-6 C26H20F6N4O2
3-(2-Phenylethyl)-6-[3-(trifluoromethyl)anilino]-1-[[4-(trifluoromethyl)phenyl]methyl]-1,3,5-triazine-2,4-dione
—— 4-(cyclopropylmethoxy)-N-[(2S)-6-[[[1-(methoxymethyl)cyclopropyl]methylamino]methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-N-methylbenzamide 1240388-45-7 C29H38N2O3
4-(cyclopropylmethoxy)-N-[(2S)-6-[[[1-(methoxymethyl)cyclopropyl]methylamino]methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-N-methylbenzamide
—— Ac(1)-2Thi-Phe(Ph(4-OMe))(Ph(4-OMe))-Phe-Tyr(1)-OH 1211441-09-6 C43H42N4O8S
Ac(1)-2Thi-Phe(Ph(4-OMe))(Ph(4-OMe))-Phe-Tyr(1)-OH
—— 2-(1H-indol-3-yl)-N-(2-methoxymethyl-indan-2-yl)-acetamide 1015074-50-6 C21H22N2O2
2-(1H-indol-3-yl)-N-(2-methoxymethyl-indan-2-yl)-acetamide
—— 1-(6-chloroquinolin-2-yl)-1,1-difluoro-2-(4-fluorophenyl)-3-(1H-tetrazol-1-yl)propan-2-ol 1416805-58-7 C19H13ClF3N5O
1-(6-chloroquinolin-2-yl)-1,1-difluoro-2-(4-fluorophenyl)-3-(1H-tetrazol-1-yl)propan-2-ol
—— L-(2R,3R)-4-[(3-benzylcarbamoyl-2,3-dihydroxy-propionylamino)methyl]-cyclohexanecarboxylic acid 1040443-95-5 C19H26N2O6
L-(2R,3R)-4-[(3-benzylcarbamoyl-2,3-dihydroxy-propionylamino)methyl]-cyclohexanecarboxylic acid
—— —— 1192255-76-7 C21H24ClN7O2S
—— (S)-3-[(S)-1-(4-chloro-2,3-difluorophenoxy)-3-methylbutyl]pyrrolidine monotrifluoroacetate 1261128-21-5 C2HF3O2*C15H20ClF2NO
(S)-3-[(S)-1-(4-chloro-2,3-difluorophenoxy)-3-methylbutyl]pyrrolidine monotrifluoroacetate
—— 2-((1r,4r)-4-(4-(6-((2,6-dichlorobenzyl)carbamoyl)imidazo[2,1-b]thiazol-2-yl)phenyl)cyclohexyl)acetic acid 1449780-13-5 C27H25Cl2N3O3S
2-((1r,4r)-4-(4-(6-((2,6-dichlorobenzyl)carbamoyl)imidazo[2,1-b]thiazol-2-yl)phenyl)cyclohexyl)acetic acid
—— (S)-3-[(S)-cyclopropyl-(2,5-dichloro-3-fluorophenoxy)methyl]pyrrolidine monotrifluoroacetate 1261129-96-7 C2HF3O2*C14H16Cl2FNO
(S)-3-[(S)-cyclopropyl-(2,5-dichloro-3-fluorophenoxy)methyl]pyrrolidine monotrifluoroacetate
—— (S)-ethyl 2-(3-((S)-(4-(trifluoro-methyl)-phenyl)(3-(trifluoro-methyl)-pyridin-2-yl)-methyl)-ureido)-propanoate (2,2,2-trifluoro-acetate) 1416944-85-8 C2HF3O2*C20H19F6N3O3
(S)-ethyl 2-(3-((S)-(4-(trifluoro-methyl)-phenyl)(3-(trifluoro-methyl)-pyridin-2-yl)-methyl)-ureido)-propanoate (2,2,2-trifluoro-acetate)
—— 4-(5-Bromo-4-chloro-2-ethylthiophen-3-yl)-1,4-dihydroquinazoline;hydrochloride 1449703-56-3 C14H12BrClN2S*ClH
4-(5-Bromo-4-chloro-2-ethylthiophen-3-yl)-1,4-dihydroquinazoline;hydrochloride
—— (S)-3-[(R)-1-(2-chloro-3-fluorophenoxy)-2-isopropoxyethyl]pyrrolidine trifluoroacetate 1262114-07-7 C2HF3O2*C15H21ClFNO2
(S)-3-[(R)-1-(2-chloro-3-fluorophenoxy)-2-isopropoxyethyl]pyrrolidine trifluoroacetate
—— —— 1452185-03-3 C12H10Cl2O5
—— N,N'-Dibenzyl-N''-((E)-2-cyano-3-mercapto-3-methylsulfanyl-acryloyl)-guanidine 107426-14-2 C20H20N4OS2
N,N'-Dibenzyl-N''-((E)-2-cyano-3-mercapto-3-methylsulfanyl-acryloyl)-guanidine
—— 1-(2,2-dimethylpropyl)-3-methyl-5-{1-[(1-methyl-1H-pyrazol-3-yl)carbonyl]piperidin-3-yl}-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1416309-38-0 C22H30N6O2
1-(2,2-dimethylpropyl)-3-methyl-5-{1-[(1-methyl-1H-pyrazol-3-yl)carbonyl]piperidin-3-yl}-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— 6-(2-Chloro-4-methylanilino)-4-[5-cyclopropyl-1-[3-(2,2-dimethylpropyl)cyclobutyl]triazol-4-yl]-6-oxohexanoic acid 1404378-27-3 C27H37ClN4O3
6-(2-Chloro-4-methylanilino)-4-[5-cyclopropyl-1-[3-(2,2-dimethylpropyl)cyclobutyl]triazol-4-yl]-6-oxohexanoic acid
—— N-[4-({[2-chloro-5-(trifluoromethyl)benzyl]carbamoyl}amino)phenyl]biphenyl-2-sulfonamide 1333941-69-7 C27H21ClF3N3O3S
N-[4-({[2-chloro-5-(trifluoromethyl)benzyl]carbamoyl}amino)phenyl]biphenyl-2-sulfonamide
—— 5-bromo-N-(3,3-dimethylbutan-2-yl)-2-methoxypyridine-3-sulfonamide 1416336-28-1 C12H19BrN2O3S
5-bromo-N-(3,3-dimethylbutan-2-yl)-2-methoxypyridine-3-sulfonamide
—— 7-butoxymethyl-3-methyl-2H-furo[2,3-c]pyran-2-one 1238521-88-4 C13H16O4
7-butoxymethyl-3-methyl-2H-furo[2,3-c]pyran-2-one
—— 2-[(2,4-dichlorophenyl)oxy]-N-[(1R)-1-[(4-methylpiperazin-1-yl)carbonyl]-3-(phenyloxy)propyl]pyridine-3-carboxamide 1239354-42-7 C27H28Cl2N4O4
2-[(2,4-dichlorophenyl)oxy]-N-[(1R)-1-[(4-methylpiperazin-1-yl)carbonyl]-3-(phenyloxy)propyl]pyridine-3-carboxamide
—— (R)-(3-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)piperidin-1-yl)(3,3-difluoroazetidin-1-yl)methanone 1310724-99-2 C17H18F2N6O
(R)-(3-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)piperidin-1-yl)(3,3-difluoroazetidin-1-yl)methanone
—— 5-((1R,3R,4S)-3-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)-4-methylcyclopentylamino)pyrazine-2-carbonitrile 1310725-09-7 C19H18N8
5-((1R,3R,4S)-3-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)-4-methylcyclopentylamino)pyrazine-2-carbonitrile
—— 1-[4-[4-Chloro-3-(trifluoromethyl)phenyl]piperazin-1-yl]-3-[4-[4-nitro-3-(trifluoromethyl)anilino]piperidin-1-yl]propane-1,3-dione 1247030-98-3 C26H26ClF6N5O4
1-[4-[4-Chloro-3-(trifluoromethyl)phenyl]piperazin-1-yl]-3-[4-[4-nitro-3-(trifluoromethyl)anilino]piperidin-1-yl]propane-1,3-dione
—— N-{4-methoxy-3-[3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl}-3-(trifluoromethyl)benzamide 1202021-93-9 C24H17F3N6O2
N-{4-methoxy-3-[3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl}-3-(trifluoromethyl)benzamide
—— 1'-(cyclopropylmethyl)-5'-(2-fluorobenzoyl)spiro[1,3-dioxane-2,3'-indol]-2'(1'H)-one 1239671-99-8 C22H20FNO4
1'-(cyclopropylmethyl)-5'-(2-fluorobenzoyl)spiro[1,3-dioxane-2,3'-indol]-2'(1'H)-one
—— 2-propanyl ({(3R,5aR,6R,7R,8aS)-6-[(1E,3R)-4-(3-chloro-5-fluorophenoxy)-3-hydroxy-1-buten-1-yl]-7-hydroxyoctahydro-2H-cyclopenta[b]oxepin-3-yl}methoxy)acetate 1262873-98-2 C25H34ClFO7
2-propanyl ({(3R,5aR,6R,7R,8aS)-6-[(1E,3R)-4-(3-chloro-5-fluorophenoxy)-3-hydroxy-1-buten-1-yl]-7-hydroxyoctahydro-2H-cyclopenta[b]oxepin-3-yl}methoxy)acetate
—— 5-(2-(2-bromophenyl)hydrazono)-6-ethoxy-6-oxohexanoic acid 1585223-49-9 C14H17BrN2O4
5-(2-(2-bromophenyl)hydrazono)-6-ethoxy-6-oxohexanoic acid
—— ethyl 4-{{6-butyl-5-[(2'-cyano-[1,1'-biphenyl]-4-yl)methyl]-2-methylpyrimidin-4-yl}oxy}butanoate 1332766-56-9 C29H33N3O3
ethyl 4-{{6-butyl-5-[(2'-cyano-[1,1'-biphenyl]-4-yl)methyl]-2-methylpyrimidin-4-yl}oxy}butanoate
—— 4-(1-cyclohexyl-3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyric acid 1229515-45-0 C19H25NO3
4-(1-cyclohexyl-3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyric acid
—— tert-butyl 4-((5-formyl-2-(pyridin-2-yl)thiazol-4-yl)methyl)piperazine-1-carboxylate 1235474-16-4 C19H24N4O3S
tert-butyl 4-((5-formyl-2-(pyridin-2-yl)thiazol-4-yl)methyl)piperazine-1-carboxylate
—— N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-3-(2-oxoimidazolidin-1-yl)benzamide 1416310-89-8 C30H40N6O3
N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-3-(2-oxoimidazolidin-1-yl)benzamide
—— 5-Methoxy-1,2-dimethyl-3-(2-nitroethyl)indole 1292285-88-1 C13H16N2O3
5-Methoxy-1,2-dimethyl-3-(2-nitroethyl)indole
—— 2-(2-fluorobenzyl)-7-(m-tolylethynyl)-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one 1416220-77-3 C23H19FN2O
2-(2-fluorobenzyl)-7-(m-tolylethynyl)-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one
—— 1-(2,2-dimethylpropyl)-3-methyl-5-(2-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl}-2-azabicyclo[2.2.2]oct-5-en-5-yl)-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1416308-16-1 C24H27F3N6O2
1-(2,2-dimethylpropyl)-3-methyl-5-(2-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl}-2-azabicyclo[2.2.2]oct-5-en-5-yl)-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— N-((1,3-dimethyl-1H-pyrazol-4-yl)methyl)-1-(4-fluorophenyl)-N-methyl-2-((pyridine-4-ylmethyl)thio)-1H-imidazole-5-carboxamide 1416264-54-4 C23H23FN6OS
N-((1,3-dimethyl-1H-pyrazol-4-yl)methyl)-1-(4-fluorophenyl)-N-methyl-2-((pyridine-4-ylmethyl)thio)-1H-imidazole-5-carboxamide
—— —— 1416458-62-2 C15H8ClF5O2S
—— (E)-3-[(1α,3α,4α)-3,4-difluorocyclopentyl]-N-{5-[(2R)-1,2-dihydroxyethyl]pyrazin-2-yl}-2-(4-(methylsulfonyl)phenyl)acrylamide 1193393-87-1 C21H23F2N3O5S
(E)-3-[(1α,3α,4α)-3,4-difluorocyclopentyl]-N-{5-[(2R)-1,2-dihydroxyethyl]pyrazin-2-yl}-2-(4-(methylsulfonyl)phenyl)acrylamide
—— (S)-3-[(R)-1-(4-chloro-2-trifluoromethylphenoxy)butyl]pyrrolidine monotrifluoroacetate 1261124-65-5 C2HF3O2*C15H19ClF3NO
(S)-3-[(R)-1-(4-chloro-2-trifluoromethylphenoxy)butyl]pyrrolidine monotrifluoroacetate
—— 5,6-dimethoxy-2-((E)-6,10-dimethylundeca-1,5,9-trien-2-yl)-1H-indole 1459200-19-1 C23H31NO2
5,6-dimethoxy-2-((E)-6,10-dimethylundeca-1,5,9-trien-2-yl)-1H-indole
—— (1R)-N-((4-(m-tolyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-1-(naphthalen-1-yl)ethanamine 1401075-45-3 C28H28N2O
(1R)-N-((4-(m-tolyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-yl)methyl)-1-(naphthalen-1-yl)ethanamine
—— 4-ethoxy-2-(piperazin-1-yl)-7-(pyridin-4-yl)-5H-pyrimido[5,4-b]indol-9-ol 1043489-75-3 C21H22N6O2
4-ethoxy-2-(piperazin-1-yl)-7-(pyridin-4-yl)-5H-pyrimido[5,4-b]indol-9-ol
—— —— 1300610-33-6 C42H30Si
—— 3-(3-methoxy-4-hydroxystyryl)-1-(pyridin-2-yl)-1H-pyrazole-5-thiol 1270044-22-8 C17H15N3O2S
3-(3-methoxy-4-hydroxystyryl)-1-(pyridin-2-yl)-1H-pyrazole-5-thiol
—— ethyl 3-{2-[(1R)-1-({(2R)-3-[(2S)-2-(3-fluoro-4-methylbenzyl)pyrrolidin-1-y1]-2-hydroxypropyl}oxy)ethyl]-4-methylphenyl}propanoate 1232829-05-8 C29H40FNO4
ethyl 3-{2-[(1R)-1-({(2R)-3-[(2S)-2-(3-fluoro-4-methylbenzyl)pyrrolidin-1-y1]-2-hydroxypropyl}oxy)ethyl]-4-methylphenyl}propanoate
—— 4-amino-5-cyano-6-ethoxy-N-((1-(3-(pyridin-4-yl)benzyl)piperidin-4-yl)methyl)picolinamide 1235473-32-1 C27H30N6O2
4-amino-5-cyano-6-ethoxy-N-((1-(3-(pyridin-4-yl)benzyl)piperidin-4-yl)methyl)picolinamide
—— 3-[4-(3,4-Difluorophenyl)piperidin-1-yl]-1-[4-[3-(2-methylpropoxy)-4-nitroanilino]piperidin-1-yl]propan-1-one 1247034-35-0 C29H38F2N4O4
3-[4-(3,4-Difluorophenyl)piperidin-1-yl]-1-[4-[3-(2-methylpropoxy)-4-nitroanilino]piperidin-1-yl]propan-1-one
—— N-[[1-(4-tert-butylphenyl)piperidin-4-yl]methyl]-N-methyl-4-[4-nitro-3-(trifluoromethyl)anilino]piperidine-1-carboxamide 1247035-75-1 C30H40F3N5O3
N-[[1-(4-tert-butylphenyl)piperidin-4-yl]methyl]-N-methyl-4-[4-nitro-3-(trifluoromethyl)anilino]piperidine-1-carboxamide