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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-chloro-N-(((3S,5S)-2-oxo-1-((S)-2-phenylbutyl)-3-(3-(piperidin-1-yl)propyl)-1,4-diazepan-5-yl)methyl)-2-naphthamide 1185654-65-2 C35H45ClN4O2
6-chloro-N-(((3S,5S)-2-oxo-1-((S)-2-phenylbutyl)-3-(3-(piperidin-1-yl)propyl)-1,4-diazepan-5-yl)methyl)-2-naphthamide
—— ethyl 2-(3,4-dichlorophenyl)-5-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylate 1226760-83-3 C19H15Cl2NO4
ethyl 2-(3,4-dichlorophenyl)-5-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylate
—— 12-O-deacetyl-12-oxo-18-episcalaradial 104900-66-5 C25H36O3
12-O-deacetyl-12-oxo-18-episcalaradial
—— (1R,2S,5S)-3-[(2S)-2-[[1-(tert-butylsulfonylmethyl)cyclohexyl]carbamoylamino]-3,3-dimethylbutanoyl]-N-[(1S,2R)-1-[2-(cyclopropylamino)-2-oxoacetyl]-2-ethylcyclopropyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide 1101838-22-5 C36H59N5O7S
(1R,2S,5S)-3-[(2S)-2-[[1-(tert-butylsulfonylmethyl)cyclohexyl]carbamoylamino]-3,3-dimethylbutanoyl]-N-[(1S,2R)-1-[2-(cyclopropylamino)-2-oxoacetyl]-2-ethylcyclopropyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide
—— 4-[(4-methyl-1H-indol-5-yl)amino]-5-{(E)-2-[4-(morpholin-4-ylmethyl)phenyl]ethenyl}pyridine-3-carbonitrile 1160919-85-6 C28H27N5O
4-[(4-methyl-1H-indol-5-yl)amino]-5-{(E)-2-[4-(morpholin-4-ylmethyl)phenyl]ethenyl}pyridine-3-carbonitrile
—— N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide 1416309-47-1 C32H43N5O3
N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
—— tert-butyl 4-{2-[4-(trifluoromethyl)phenyl]oxazolo[5,4-b]pyridin-6-yl}piperidine-1-carboxylate 1415992-16-3 C23H24F3N3O3
tert-butyl 4-{2-[4-(trifluoromethyl)phenyl]oxazolo[5,4-b]pyridin-6-yl}piperidine-1-carboxylate
—— 2'-aminomethyl-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carboxylic acid 1-methyl-piperidin-4-yl ester 1333398-88-1 C26H28N4O3
2'-aminomethyl-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carboxylic acid 1-methyl-piperidin-4-yl ester
—— N-[6-amino-5-(2-chlorophenyl)pyridin-2-yl]isoxazole-5-carboxamide 1079400-80-8 C15H11ClN4O2
N-[6-amino-5-(2-chlorophenyl)pyridin-2-yl]isoxazole-5-carboxamide
—— (2S,4R)-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-1-[(2S)-2-(3,4-difluoroanilino)-3,3-dimethylbutanoyl]-4-[[2-(4-propan-2-yloxyphenyl)-[1]benzofuro[3,2-d]pyrimidin-4-yl]oxy]pyrrolidine-2-carboxamide 1315324-59-4 C45H48F2N6O8S
(2S,4R)-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-1-[(2S)-2-(3,4-difluoroanilino)-3,3-dimethylbutanoyl]-4-[[2-(4-propan-2-yloxyphenyl)-[1]benzofuro[3,2-d]pyrimidin-4-yl]oxy]pyrrolidine-2-carboxamide
—— ethyl 4-{[[(3-chloro-1H-indol-6-yl)methyl](4-methylisoquinolin-3-yl)amino]-sulfonyl}benzoate 1400699-80-0 C28H24ClN3O4S
ethyl 4-{[[(3-chloro-1H-indol-6-yl)methyl](4-methylisoquinolin-3-yl)amino]-sulfonyl}benzoate
—— 4-phenyl-1-3-[(E)-3-phenyl-2-propenoyl]phenyl-2,3-dihydro-1H-2-imidazolone 1338086-81-9 C24H18N2O2
4-phenyl-1-3-[(E)-3-phenyl-2-propenoyl]phenyl-2,3-dihydro-1H-2-imidazolone
—— ethyl 3-[2-[(1R)-1-[(2R)-3-[(2R,4R)-2-[(3-fluoro-4-methylphenyl)methyl]-4-hydroxypyrrolidin-1-yl]-2-hydroxypropoxy]ethyl]phenyl]propanoate 1232831-69-4 C28H38FNO5
ethyl 3-[2-[(1R)-1-[(2R)-3-[(2R,4R)-2-[(3-fluoro-4-methylphenyl)methyl]-4-hydroxypyrrolidin-1-yl]-2-hydroxypropoxy]ethyl]phenyl]propanoate
—— 7-[4-(diethylamino)anilino]-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide 1214931-71-1 C24H27N5O2
7-[4-(diethylamino)anilino]-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide
—— 2-{1-[6-ethyl-2-(4-fluorophenylamino)pyrimidin-4-yl]piperidin-2-yl}ethanol 1394804-84-2 C19H25FN4O
2-{1-[6-ethyl-2-(4-fluorophenylamino)pyrimidin-4-yl]piperidin-2-yl}ethanol
—— 3-(2,4-dioxo-1H-thieno[3,4-d]pyrimidin-3-yl)-1-prop-2-enyl-5-(trifluoromethyl)indole-2-carboxylic acid 1154596-77-6 C19H12F3N3O4S
3-(2,4-dioxo-1H-thieno[3,4-d]pyrimidin-3-yl)-1-prop-2-enyl-5-(trifluoromethyl)indole-2-carboxylic acid
—— (3R)-N-(2-{[6-(5-cyclopropyl-4-methyl-1H-imidazol-2-yl)pyridin-2-yl]amino}ethyl)pyrrolidine-3-carboxamide 1373272-94-6 C19H26N6O
(3R)-N-(2-{[6-(5-cyclopropyl-4-methyl-1H-imidazol-2-yl)pyridin-2-yl]amino}ethyl)pyrrolidine-3-carboxamide
—— 2-cyclopropyl-1-[4-[4-[5-[[(2S)-morpholin-2-yl]methylamino]pyrido[3,4-b]pyrazin-7-yl]phenyl]piperazin-1-yl]ethanone 1415792-68-5 C27H33N7O2
2-cyclopropyl-1-[4-[4-[5-[[(2S)-morpholin-2-yl]methylamino]pyrido[3,4-b]pyrazin-7-yl]phenyl]piperazin-1-yl]ethanone
—— (S)-N-[1-(2-{[3-(aminomethyl)phenyl]amino}-6-propylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide 1394316-95-0 C20H28N6O
(S)-N-[1-(2-{[3-(aminomethyl)phenyl]amino}-6-propylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
—— ethyl 5-[2-fluoro-6-[(1R)-1-[(2R)-3-[(2S)-2-[(3-fluoro-4-methylphenyl)methyl]pyrrolidin-1-yl]-2-hydroxypropoxy]ethyl]phenyl]pentanoate 1232831-96-7 C30H41F2NO4
ethyl 5-[2-fluoro-6-[(1R)-1-[(2R)-3-[(2S)-2-[(3-fluoro-4-methylphenyl)methyl]pyrrolidin-1-yl]-2-hydroxypropoxy]ethyl]phenyl]pentanoate
—— 3-amino-6-methoxy-N-(2-methoxyethyl)-N-methyl-2-(3-oxo-4H-quinoxalin-2-yl)-1H-indole-5-carboxamide 1055898-40-2 C22H23N5O4
3-amino-6-methoxy-N-(2-methoxyethyl)-N-methyl-2-(3-oxo-4H-quinoxalin-2-yl)-1H-indole-5-carboxamide
—— 6-[3-(Difluoromethoxy)anilino]-1-[(4-methylphenyl)methyl]-3-propan-2-yl-1,3,5-triazine-2,4-dione 1239686-55-5 C21H22F2N4O3
6-[3-(Difluoromethoxy)anilino]-1-[(4-methylphenyl)methyl]-3-propan-2-yl-1,3,5-triazine-2,4-dione
—— 4-(1-(4-chloro-5-(5-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl)-2-methylbenzoyl)piperidin-4-yl)benzonitrile 1399177-62-8 C25H26ClN5O2
4-(1-(4-chloro-5-(5-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl)-2-methylbenzoyl)piperidin-4-yl)benzonitrile
—— 5-Chloroisoquinoline-4-carboxylic acid 1368270-12-5 C10H6ClNO2
5-Chloroisoquinoline-4-carboxylic acid
—— 4-(3-amino-6-(4-(N-cyclopropyl-N-methylsulfamoyl)phenyl)pyrazin-2-yl)-2-isopropoxybenzamide 1396771-92-8 C24H27N5O4S
4-(3-amino-6-(4-(N-cyclopropyl-N-methylsulfamoyl)phenyl)pyrazin-2-yl)-2-isopropoxybenzamide
—— 2-{1-[2-(3-amino-4-chlorophenylamino)-6-propylpyrimidin-4-yl]piperidin-2-yl}ethanol 1394804-94-4 C20H28ClN5O
2-{1-[2-(3-amino-4-chlorophenylamino)-6-propylpyrimidin-4-yl]piperidin-2-yl}ethanol
—— [5-(tert-butylamino)-2-pyridyl]-[(4R)-6-fluoro-4-isopropoxy-spiro[chromane-2,4'-piperidine]-1'-yl]methanone 1394030-51-3 C26H34FN3O3
[5-(tert-butylamino)-2-pyridyl]-[(4R)-6-fluoro-4-isopropoxy-spiro[chromane-2,4'-piperidine]-1'-yl]methanone
—— N-(2-(4-amino-1H-pyrazol-1-yl)ethyl)-4-fluoropyridin-2-amine 1394162-22-1 C10H12FN5
N-(2-(4-amino-1H-pyrazol-1-yl)ethyl)-4-fluoropyridin-2-amine
—— 4-chloro-N-[1-(4-fluorophenyl)-2-methyl-1-oxopropan-2-yl]-2-pyridin-3-yl-1,3-thiazole-5-carboxamide 1415890-07-1 C19H15ClFN3O2S
4-chloro-N-[1-(4-fluorophenyl)-2-methyl-1-oxopropan-2-yl]-2-pyridin-3-yl-1,3-thiazole-5-carboxamide
—— (6S,14S)-2-hydroxy-3,9,11-trimethoxy-6-methyl-5,8,13,13a-tetrahydro-6H-dibenzo[a,g]quinolizine 1415465-93-8 C21H25NO4
(6S,14S)-2-hydroxy-3,9,11-trimethoxy-6-methyl-5,8,13,13a-tetrahydro-6H-dibenzo[a,g]quinolizine
—— N-(tert-butoxycarbonyl)-S-({6-[4-({[4-(1-ethylpropyl)phenyl](isopropyl)amino}methyl)phenyl]pyridin-2-yl}methyl)-L-cysteine 1013907-90-8 C35H47N3O4S
N-(tert-butoxycarbonyl)-S-({6-[4-({[4-(1-ethylpropyl)phenyl](isopropyl)amino}methyl)phenyl]pyridin-2-yl}methyl)-L-cysteine
—— {[2'-(1-aminoethyl)-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-ylcarbamoyl]-methylsulfanyl}-acetic acid ethyl ester 1333399-94-2 C26H28N4O4S
{[2'-(1-aminoethyl)-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-ylcarbamoyl]-methylsulfanyl}-acetic acid ethyl ester
—— 7-[4-(2-methylmorpholin-4-yl)phenyl]-N-[[(2S)-morpholin-2-yl]methyl]pyrido[3,4-b]pyrazin-5-amine 1415790-07-6 C23H28N6O2
7-[4-(2-methylmorpholin-4-yl)phenyl]-N-[[(2S)-morpholin-2-yl]methyl]pyrido[3,4-b]pyrazin-5-amine
—— 4-[4-(2-cyclohexylethoxy)benzoyl]-N-pyridin-3-ylpiperidine-1-carboxamide 1008765-40-9 C26H33N3O3
4-[4-(2-cyclohexylethoxy)benzoyl]-N-pyridin-3-ylpiperidine-1-carboxamide
—— 5-chloro-N-((2',4'-difluorobiphenyl-4-yl)methyl)-1-(phenylsulfonyl)-1H-indole-2-sulfonamide 1394431-62-9 C27H19ClF2N2O4S2
5-chloro-N-((2',4'-difluorobiphenyl-4-yl)methyl)-1-(phenylsulfonyl)-1H-indole-2-sulfonamide
—— 2-{1-[2-(3-amino-4-fluorophenylamino)-6-propylpyrimidin-4-yl]piperidin-2-yl}ethanol 1394804-93-3 C20H28FN5O
2-{1-[2-(3-amino-4-fluorophenylamino)-6-propylpyrimidin-4-yl]piperidin-2-yl}ethanol
—— 3-({[(1S)-1-(4-fluorophenyl)ethyl](2-naphthoyl)amino}methyl)benzoic acid 1398583-45-3 C27H22FNO3
3-({[(1S)-1-(4-fluorophenyl)ethyl](2-naphthoyl)amino}methyl)benzoic acid
—— N-(6-(4-(4-cyanophenyl)piperidine-1-carbonyl)-3-methylpyridin-2-yl)-6-(isopropylamino)nicotinamide 1399179-39-5 C28H30N6O2
N-(6-(4-(4-cyanophenyl)piperidine-1-carbonyl)-3-methylpyridin-2-yl)-6-(isopropylamino)nicotinamide
—— 1-[(4-Chlorophenyl)methyl]-3-(2-phenylethyl)-6-[3-(trifluoromethyl)anilino]-1,3,5-triazine-2,4-dione 1239686-27-1 C25H20ClF3N4O2
1-[(4-Chlorophenyl)methyl]-3-(2-phenylethyl)-6-[3-(trifluoromethyl)anilino]-1,3,5-triazine-2,4-dione
—— 3-(5-(4-amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)pyridin-2-yloxy)-2,2-dimethylpropanoic acid 1246211-19-7 C17H19N5O5
3-(5-(4-amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)pyridin-2-yloxy)-2,2-dimethylpropanoic acid
—— 3-bromo-8-fluoro-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312455-78-9 C13H12BrFN2O
3-bromo-8-fluoro-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one
—— (3-{3-[(tert-butoxycarbonyl-ethyl-amino)-methyl]-5-methyl-pyridin-2-yl}-4-methoxy-phenyl)-acetic acid ethyl ester 1219696-26-0 C25H34N2O5
(3-{3-[(tert-butoxycarbonyl-ethyl-amino)-methyl]-5-methyl-pyridin-2-yl}-4-methoxy-phenyl)-acetic acid ethyl ester
—— 8-cyclopropyl-2-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-7-naphthalen-1-ylmethyl-5-oxo-5H-thiazolo[3,2-a]pyridine-3-carboxylic acid methyl ester 1235550-98-7 C31H25NO5S
8-cyclopropyl-2-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-7-naphthalen-1-ylmethyl-5-oxo-5H-thiazolo[3,2-a]pyridine-3-carboxylic acid methyl ester
—— 3-(6-iodo-2-methyl-4-oxoquinazolin-3(4H)-yl)benzoic acid 1237744-93-2 C16H11IN2O3
3-(6-iodo-2-methyl-4-oxoquinazolin-3(4H)-yl)benzoic acid
—— N-[[(2S)-morpholin-2-yl]methyl]-7-[4-(4-propan-2-ylsulfonylpiperazin-1-yl)phenyl]pyrido[3,4-b]pyrazin-5-amine 1415792-66-3 C25H33N7O3S
N-[[(2S)-morpholin-2-yl]methyl]-7-[4-(4-propan-2-ylsulfonylpiperazin-1-yl)phenyl]pyrido[3,4-b]pyrazin-5-amine
—— 1-[(6-Chloropyridin-3-yl)methyl]-3-propan-2-yl-6-(3-propan-2-yloxyanilino)-1,3,5-triazine-2,4-dione 1239686-95-3 C21H24ClN5O3
1-[(6-Chloropyridin-3-yl)methyl]-3-propan-2-yl-6-(3-propan-2-yloxyanilino)-1,3,5-triazine-2,4-dione
—— N-{[1-(4-chlorophenyl)cyclopentyl]methyl}-3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzamide 1243203-78-2 C24H26ClN3O2
N-{[1-(4-chlorophenyl)cyclopentyl]methyl}-3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzamide
—— 1-(2-cyano-2-methyl-acetylamino)-cyclopropanecarboxylic acid [5-(4-fluoro-2-trifluoromethyl-phenylamino)-pyridin-2-ylmethyl]-amide 1242453-39-9 C21H19F4N5O2
1-(2-cyano-2-methyl-acetylamino)-cyclopropanecarboxylic acid [5-(4-fluoro-2-trifluoromethyl-phenylamino)-pyridin-2-ylmethyl]-amide
—— N-(((3S,5S)-3-(3-aminopropyl)-2-oxo-1-((1-phenylcyclohexyl)methyl)-1,4-diazepan-5-yl)methyl)-2-naphthamide 1185652-35-0 C33H42N4O2
N-(((3S,5S)-3-(3-aminopropyl)-2-oxo-1-((1-phenylcyclohexyl)methyl)-1,4-diazepan-5-yl)methyl)-2-naphthamide
—— (6aS)-2-methoxy-3-[6-[4-[2-[(3,4,5-trimethoxyphenyl)methylamino]benzoyl]piperazin-1-yl]hexoxy]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-11-one 1235987-91-3 C40H51N5O7
(6aS)-2-methoxy-3-[6-[4-[2-[(3,4,5-trimethoxyphenyl)methylamino]benzoyl]piperazin-1-yl]hexoxy]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-11-one