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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-cyclopropyl-N-{[6-(2,6-dimethylpyridin-4-yl)-2-fluoro-3-[(2R)-2-(trifluoromethyl)morpholin-4-yl]phenyl]methyl}acetamide 1394908-61-2 C24H27F4N3O2
2-cyclopropyl-N-{[6-(2,6-dimethylpyridin-4-yl)-2-fluoro-3-[(2R)-2-(trifluoromethyl)morpholin-4-yl]phenyl]methyl}acetamide
—— 4-(5-chloro-2,3-dihydrobenzo[d]thiazol-2-yl)-2,6-dimethoxyphenol 1393371-35-1 C15H14ClNO3S
4-(5-chloro-2,3-dihydrobenzo[d]thiazol-2-yl)-2,6-dimethoxyphenol
—— 5-(4-chlorophenyl)-4-methyl-3-(4-(piperidin-1-ylsulfonyl)phenyl)thiophene-2-carboxylic acid 1394375-46-2 C23H22ClNO4S2
5-(4-chlorophenyl)-4-methyl-3-(4-(piperidin-1-ylsulfonyl)phenyl)thiophene-2-carboxylic acid
—— 2-chloro-6-(quinolin-3-yloxy)-benzamide 1314007-22-1 C16H11ClN2O2
2-chloro-6-(quinolin-3-yloxy)-benzamide
—— 2-[2-((S)-2-methyl-2,3-dihydroindol-1-yl)-2-oxoethyl]-6-(2-methylmorpholin-4-yl)-3H-pyrimidin-4-one 1384071-08-2 C20H24N4O3
2-[2-((S)-2-methyl-2,3-dihydroindol-1-yl)-2-oxoethyl]-6-(2-methylmorpholin-4-yl)-3H-pyrimidin-4-one
—— ethyl 1,5,5-trimethyl-7-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxylate 1391938-62-7 C14H19NO3
ethyl 1,5,5-trimethyl-7-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxylate
—— tert-butyl 6-(2-chloro-4-(1-methyl-1H-pyrazol-5-yl)phenylamino)-2-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridine-1-carboxylate 1400285-07-5 C26H26ClN7O2
tert-butyl 6-(2-chloro-4-(1-methyl-1H-pyrazol-5-yl)phenylamino)-2-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridine-1-carboxylate
—— (R)-2-methyl-5-(4-propyl-6-{3-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-ylamino)benzonitrile 1394805-26-5 C25H30N6S
(R)-2-methyl-5-(4-propyl-6-{3-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-ylamino)benzonitrile
—— 2-(2-iodophenyl)-5-methyl-1,3,4-oxadiazole 1092114-30-1 C9H7IN2O
2-(2-iodophenyl)-5-methyl-1,3,4-oxadiazole
—— 2-(dimethylamino)-8-methyl-6,9-dihydro-5H-pyrrolo[3,2-h]quinazoline-7-carboxylic acid 1391938-99-0 C14H16N4O2
2-(dimethylamino)-8-methyl-6,9-dihydro-5H-pyrrolo[3,2-h]quinazoline-7-carboxylic acid
—— N-[(1,3-dimethyl-5-naphthalen-2-yloxypyrazol-4-yl)methylidene]hydroxylamine 143583-33-9 C16H15N3O2
N-[(1,3-dimethyl-5-naphthalen-2-yloxypyrazol-4-yl)methylidene]hydroxylamine
—— N-(4-((4-((5-methyl-1H-pyrazol-3-yl)amino)-6-(4-(piperidin-1-yl)butanamido)pyrrolo[2,1-f][1,2,4]triazin-2-yl)thio)phenyl)cyclopropanecarboxamide 1315588-75-0 C29H35N9O2S
N-(4-((4-((5-methyl-1H-pyrazol-3-yl)amino)-6-(4-(piperidin-1-yl)butanamido)pyrrolo[2,1-f][1,2,4]triazin-2-yl)thio)phenyl)cyclopropanecarboxamide
—— (S)-3-(2-fluoro-phenyl)-3-{[5-methoxy-6-o-tolyl-pyridine-2-carbonyl]amino}propionic acid 1391842-73-1 C23H21FN2O4
(S)-3-(2-fluoro-phenyl)-3-{[5-methoxy-6-o-tolyl-pyridine-2-carbonyl]amino}propionic acid
—— Methyl 1-[2-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]ethyl]cyclobutane-1-carboxylate 1398047-73-8 C19H27NO4
Methyl 1-[2-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]ethyl]cyclobutane-1-carboxylate
—— 4-((4-(1H-indazol-4-yl)-6-morpholino-1,3,5-triazin-2-yl)oxy)-N,N-dimethylbenzamide 1391924-81-4 C23H23N7O3
4-((4-(1H-indazol-4-yl)-6-morpholino-1,3,5-triazin-2-yl)oxy)-N,N-dimethylbenzamide
—— N2-(3-amino-4-methoxyphenyl)-N4,N4-diethyl-6-propylpyrimidine-2,4-diamine 1394851-63-8 C18H27N5O
N2-(3-amino-4-methoxyphenyl)-N4,N4-diethyl-6-propylpyrimidine-2,4-diamine
—— 4-[3-(2-cyclohexylethoxy)benzoyl]-N-(1,2,4-triazol-4-yl)piperazine-1-carboxamide 1008767-58-5 C22H30N6O3
4-[3-(2-cyclohexylethoxy)benzoyl]-N-(1,2,4-triazol-4-yl)piperazine-1-carboxamide
—— 1-[2-fluoro-3-(hydroxymethyl)phenyl]-4-(pyridin-3-yl)piperidin-4-ol 1400758-90-8 C17H19FN2O2
1-[2-fluoro-3-(hydroxymethyl)phenyl]-4-(pyridin-3-yl)piperidin-4-ol
—— 4-(((1R,3R)-3-amino-2,2,3-trimethylcyclopentyl)amino)pyrrolo[1,2-b]pyridazine-3-carboxamide 1400688-98-3 C16H23N5O
4-(((1R,3R)-3-amino-2,2,3-trimethylcyclopentyl)amino)pyrrolo[1,2-b]pyridazine-3-carboxamide
—— 1-(2-bromoethoxy)-3-chloro-5-fluorobenzene 1396723-59-3 C8H7BrClFO
1-(2-bromoethoxy)-3-chloro-5-fluorobenzene
—— N-(5-(4-(4-cyanophenyl)-4-fluoropiperidine-1-carbonyl)-2,4-dimethylphenyl)-6-morpholinonicotinamide 1399176-28-3 C31H32FN5O3
N-(5-(4-(4-cyanophenyl)-4-fluoropiperidine-1-carbonyl)-2,4-dimethylphenyl)-6-morpholinonicotinamide
—— 4-(1-benzylpiperidin-4-yloxy)-7-(2-fluoro-4-methanesulfonylphenyl)thieno[3,2-d]pyrimidine 1384951-34-1 C25H24FN3O3S2
4-(1-benzylpiperidin-4-yloxy)-7-(2-fluoro-4-methanesulfonylphenyl)thieno[3,2-d]pyrimidine
—— (2S,4R)-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-1-[(2S)-3,3-dimethyl-2-(pyrimidin-5-ylamino)butanoyl]-4-[[2-(4-propan-2-yloxyphenyl)-[1]benzothiolo[3,2-d]pyrimidin-4-yl]oxy]pyrrolidine-2-carboxamide 1315324-99-2 C43H48N8O7S2
(2S,4R)-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-1-[(2S)-3,3-dimethyl-2-(pyrimidin-5-ylamino)butanoyl]-4-[[2-(4-propan-2-yloxyphenyl)-[1]benzothiolo[3,2-d]pyrimidin-4-yl]oxy]pyrrolidine-2-carboxamide
—— (2R)-N-{1-[3-bromo-4-methoxy-5-(3-methoxypropoxy)phenyl]ethyl}-N-cyclopropylmorpholin-2-carboxamide 1399846-47-9 C21H31BrN2O5
(2R)-N-{1-[3-bromo-4-methoxy-5-(3-methoxypropoxy)phenyl]ethyl}-N-cyclopropylmorpholin-2-carboxamide
—— 7-(4-morpholin-4-ylsulfonylanilino)-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide 1214931-97-1 C24H25N5O5S
7-(4-morpholin-4-ylsulfonylanilino)-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide
—— ethyl 5-(3,4-difluorophenyl)-4-methyl-3-(4-sulfamoylphenyl)thiophene-2-carboxylate 1394373-42-2 C20H17F2NO4S2
ethyl 5-(3,4-difluorophenyl)-4-methyl-3-(4-sulfamoylphenyl)thiophene-2-carboxylate
—— 4-(2-Aminoethoxy)-N-ethylbenzamide hydrochloride 1392489-13-2 C11H16N2O2*ClH
4-(2-Aminoethoxy)-N-ethylbenzamide hydrochloride
—— 2,2-dimethyl-7-[3-(methylsulfonyl)phenyl]-2,3-dihydro-4H-chromen-4-one 1393844-18-2 C18H18O4S
2,2-dimethyl-7-[3-(methylsulfonyl)phenyl]-2,3-dihydro-4H-chromen-4-one
—— (S)-3-{4-[3-(cyclopropylmethylamino)pyrrolidin-1-yl]-6-propylpyrimidin-2-ylamino}benzonitrile 1394314-92-1 C22H28N6
(S)-3-{4-[3-(cyclopropylmethylamino)pyrrolidin-1-yl]-6-propylpyrimidin-2-ylamino}benzonitrile
—— (S)-3-{[6-(2-chloro-3-methyl-phenyl)-5-methoxy-pyridine-2-carbonyl]-amino}-3-(2-fluoro-phenyl)-propionic acid 1391843-41-6 C23H20ClFN2O4
(S)-3-{[6-(2-chloro-3-methyl-phenyl)-5-methoxy-pyridine-2-carbonyl]-amino}-3-(2-fluoro-phenyl)-propionic acid
—— methyl 3-(4-ethoxy-6-methoxypyrimidin-2-yl)acrylate 1394162-36-7 C11H14N2O4
methyl 3-(4-ethoxy-6-methoxypyrimidin-2-yl)acrylate
—— N4-ethyl-N2-(4-fluorophenyl)-N4-(2-methoxyethyl)-6-propylpyrimidine-2,4-diamine 1394851-71-8 C18H25FN4O
N4-ethyl-N2-(4-fluorophenyl)-N4-(2-methoxyethyl)-6-propylpyrimidine-2,4-diamine
—— (S)-3-{4-butyl-6-[3-(cyclopropylmethylamino)pyrrolidin-1-yl]pyrimidin-2-ylamino}benzonitrile 1394316-74-5 C23H30N6
(S)-3-{4-butyl-6-[3-(cyclopropylmethylamino)pyrrolidin-1-yl]pyrimidin-2-ylamino}benzonitrile
—— 1-benzyl-4-[3-fluoro-1-(propan-2-yl)piperidin-4-yl]-1,4-diazepane 1373272-50-4 C20H32FN3
1-benzyl-4-[3-fluoro-1-(propan-2-yl)piperidin-4-yl]-1,4-diazepane
—— (2S,4R)-1-[(2S)-2-cyclohexyl-2-(4-fluoroanilino)acetyl]-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-4-[[2-(4-propan-2-yloxyphenyl)-[1]benzofuro[3,2-d]pyrimidin-4-yl]oxy]pyrrolidine-2-carboxamide 1315325-22-4 C47H51FN6O8S
(2S,4R)-1-[(2S)-2-cyclohexyl-2-(4-fluoroanilino)acetyl]-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-4-[[2-(4-propan-2-yloxyphenyl)-[1]benzofuro[3,2-d]pyrimidin-4-yl]oxy]pyrrolidine-2-carboxamide
—— 3,5-difluoro-4'-propyl-4-(1,2,2-trifluorovinyl)biphenyl 1313599-39-1 C17H13F5
3,5-difluoro-4'-propyl-4-(1,2,2-trifluorovinyl)biphenyl
—— 2-amino-5-butyl-4-(furan-3-yl)-6-(thiophen-3-yl)pyrimidine 1395343-81-3 C16H17N3OS
2-amino-5-butyl-4-(furan-3-yl)-6-(thiophen-3-yl)pyrimidine
—— (S)-3-amino-1-phenylazocan-2-one 1400677-55-5 C13H18N2O
(S)-3-amino-1-phenylazocan-2-one
—— 2-chloro-4-(1,5-dimethyl-1H-pyrazol-4-yl)aniline 1400287-25-3 C11H12ClN3
2-chloro-4-(1,5-dimethyl-1H-pyrazol-4-yl)aniline
—— dicarbonyl(η5-cyclopentadienyl)(2-norbornen-2-yl)iron 110078-14-3 C14H14FeO2
dicarbonyl(η5-cyclopentadienyl)(2-norbornen-2-yl)iron
—— 4-[(S)-4-carboxy-2-({4-[2-((R)-2-cyano-pyrrolidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073450-99-3 C29H34N6O8
4-[(S)-4-carboxy-2-({4-[2-((R)-2-cyano-pyrrolidin-1-yl)-2-oxo-ethoxy]-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 2-(6-methoxychroman-3-yl)-7-(pyridin-4-yl)quinazolin-4-ol 1227361-45-6 C23H19N3O3
2-(6-methoxychroman-3-yl)-7-(pyridin-4-yl)quinazolin-4-ol
—— N-{(1S,2R)-1-benzyl-3-[(4-fluoro-3-methylbenzyl)amino]-2-hydroxypropyl}-1-ethyl-5-[(2-propylpiperidin-1-yl)carbonyl]-1H-pyrazole-3-carboxamide 1106668-69-2 C33H44FN5O3
N-{(1S,2R)-1-benzyl-3-[(4-fluoro-3-methylbenzyl)amino]-2-hydroxypropyl}-1-ethyl-5-[(2-propylpiperidin-1-yl)carbonyl]-1H-pyrazole-3-carboxamide
—— (3-cyclohexylmethyl-1,4,7-trimethyl-2-oxo-1,2-dihydroquinolin-5-yloxy)acetic acid 1221181-21-0 C21H27NO4
(3-cyclohexylmethyl-1,4,7-trimethyl-2-oxo-1,2-dihydroquinolin-5-yloxy)acetic acid
—— 5-[4-(2-fluoro-phenyl)-but-3-ynyl]-pyrazolo[1,5-a]pyrimidine 1228353-51-2 C16H12FN3
5-[4-(2-fluoro-phenyl)-but-3-ynyl]-pyrazolo[1,5-a]pyrimidine
—— (1R,3R,4R)-3-[4-(1-adamantyl)-2,6-dihydroxyphenyl]-4-isopropenyl-1-(hydroxymethyl)cyclohexane 1605280-75-8 C26H36O3
(1R,3R,4R)-3-[4-(1-adamantyl)-2,6-dihydroxyphenyl]-4-isopropenyl-1-(hydroxymethyl)cyclohexane
—— 4-[(S)-4-ethoxycarbonyl-2-({4-[2-((S)-2-ethylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-6-fluoro-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073449-39-4 C34H45FN6O9
4-[(S)-4-ethoxycarbonyl-2-({4-[2-((S)-2-ethylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-6-fluoro-7-methyl-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester
—— 4-[(4-Fluoro-phenyl)-hydroxy-methyl]-piperidine-4-carbonitrile 1229831-30-4 C13H15FN2O
4-[(4-Fluoro-phenyl)-hydroxy-methyl]-piperidine-4-carbonitrile
—— 3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[[5-(4-methylphenyl)pyridin-2-yl]carbamoylamino]propanoic acid 1323992-06-8 C35H33FN6O6
3-[3-Fluoro-4-[5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-[[5-(4-methylphenyl)pyridin-2-yl]carbamoylamino]propanoic acid
—— 4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclopropylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-5-fluoro-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester 1073448-18-6 C32H39FN6O9
4-[(S)-4-carboxy-2-({4-[2-((S)-2-cyclopropylcarbamoyl-pyrrolidin-1-yl)-2-oxo-ethoxy]-5-fluoro-quinoline-2-carbonyl}-amino)-butyryl]-piperazine-1-carboxylic acid ethyl ester