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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-chloro-2-(3-(2,4-difluorophenoxy)azetidin-1-yl)nicotinic acid 1380753-85-4 C15H11ClF2N2O3
5-chloro-2-(3-(2,4-difluorophenoxy)azetidin-1-yl)nicotinic acid
—— methyl 4-(1-(5-chloro-2-(3-(3-(trifluoromethyl)phenoxy)pyrrolidin-1-yl)nicotinamido)cyclopropyl)benzoate 1380755-42-9 C28H25ClF3N3O4
methyl 4-(1-(5-chloro-2-(3-(3-(trifluoromethyl)phenoxy)pyrrolidin-1-yl)nicotinamido)cyclopropyl)benzoate
—— (S)-2-methyl-1-(4-trifluoromethyl-phenyl)-pyrrolidine-2-carboxylic acid (5-tert-butyl-isoxazol-3-yl)-amide 1234315-85-5 C20H24F3N3O2
(S)-2-methyl-1-(4-trifluoromethyl-phenyl)-pyrrolidine-2-carboxylic acid (5-tert-butyl-isoxazol-3-yl)-amide
—— 5-(4-methylpyridin-3-yl)-2-(phenoxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one 1382782-37-7 C19H18N4O2
5-(4-methylpyridin-3-yl)-2-(phenoxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
—— 2-<Bis(methylthio)methylene>-1,3-benzodithiole 124005-79-4 C10H10S4
2-<Bis(methylthio)methylene>-1,3-benzodithiole
—— 6-<(N-methylamidiniothio)phenyl-λ3-iodanyl>-2,4-dinitrophenolate 100351-30-2 C14H13IN4O5S
6-<(N-methylamidiniothio)phenyl-λ3-iodanyl>-2,4-dinitrophenolate
—— diethyl <3-methyl-5-(5-methyl-2-thienylmethyl)-2-thienyl>-methylphosphonate 141191-55-1 C16H23O3PS2
diethyl <3-methyl-5-(5-methyl-2-thienylmethyl)-2-thienyl>-methylphosphonate
—— tert-butyl (S)-2-(bis(4-(dimethylamino)phenyl)(hydroxy)methyl)pyrrolidine-1-carboxylate 1203648-37-6 C26H37N3O3
tert-butyl (S)-2-(bis(4-(dimethylamino)phenyl)(hydroxy)methyl)pyrrolidine-1-carboxylate
—— 13,18-dihydro-13,18-dibromo-6b,12b<9',10'>anthracenoacenaphth<1,2-a>acenaphtylene 173725-68-3 C36H20Br2
13,18-dihydro-13,18-dibromo-6b,12b<9',10'>anthracenoacenaphth<1,2-a>acenaphtylene
—— N-(((3S,5S)-3-(3-aminopropyl)-2-oxo-1-(2-phenylbutyl)-1,4-diazepan-5-yl)methyl)-2-naphthamide 1185652-32-7 C30H38N4O2
N-(((3S,5S)-3-(3-aminopropyl)-2-oxo-1-(2-phenylbutyl)-1,4-diazepan-5-yl)methyl)-2-naphthamide
—— N-(5-{3-[1-(phenylsulfonyl)-1H-pyrazol-4-yl]-6-quinoxalinyl}-3-pyridinyl)benzenesulfonamide 1083322-76-2 C28H20N6O4S2
N-(5-{3-[1-(phenylsulfonyl)-1H-pyrazol-4-yl]-6-quinoxalinyl}-3-pyridinyl)benzenesulfonamide
—— 1,2-bis(2-neopentoxy-5-phenyl-3-thienyl)perfluorocyclopentene 1385022-38-7 C35H34F6O2S2
1,2-bis(2-neopentoxy-5-phenyl-3-thienyl)perfluorocyclopentene
—— 1-<2-Triaethylsilyl-aethyl>-4-trimethylsilyl-benzol 18547-44-9 C17H32Si2
1-<2-Triaethylsilyl-aethyl>-4-trimethylsilyl-benzol
—— 9,9-Dichlor-nona-2,4,6,8-tetraensaeure-ethylester 18804-15-4 C11H12Cl2O2
9,9-Dichlor-nona-2,4,6,8-tetraensaeure-ethylester
—— Vismodegib (m4) 1370525-65-7 C25H22Cl2N2O10S
Vismodegib (m4)
—— benzyl (2-(((5-((2,4-dioxothiazolidin-5-yl)methyl)-1,3,4-oxadiazol-2-yl)(4-fluoro-6-phenylbenzo[d]thiazol-2-yl)methyl)sulfonyl)ethyl)carbamate 1532558-32-9 C30H24FN5O7S3
benzyl (2-(((5-((2,4-dioxothiazolidin-5-yl)methyl)-1,3,4-oxadiazol-2-yl)(4-fluoro-6-phenylbenzo[d]thiazol-2-yl)methyl)sulfonyl)ethyl)carbamate
—— 1-Fluoro-2-(fluoro-dinitro-methyl)-benzene 136312-33-9 C7H4F2N2O4
1-Fluoro-2-(fluoro-dinitro-methyl)-benzene
—— 3-methoxy-1-methyl-4-oxo-5-(2-oxo-2-phenylethyl)-N-(tetrahydrofuran-2-ylmethyl)-4,5-dihydro-1H-pyrrolo[3,2-c]quinoline-2-carboxamide 1186245-09-9 C27H27N3O5
3-methoxy-1-methyl-4-oxo-5-(2-oxo-2-phenylethyl)-N-(tetrahydrofuran-2-ylmethyl)-4,5-dihydro-1H-pyrrolo[3,2-c]quinoline-2-carboxamide
—— 3-(4-chlorophenyl)-2-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enehydrazide 1346570-39-5 C21H18ClN3O2
3-(4-chlorophenyl)-2-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enehydrazide
—— —— 1239276-40-4 C23H18ClF10N3O3
—— 7-hydroxy-N-(pyrrolidin-3-yl)-2-(thiophen-2-yl)-1H-benzo[d]imidazole-4-carboxamide 1224879-73-5 C16H16N4O2S
7-hydroxy-N-(pyrrolidin-3-yl)-2-(thiophen-2-yl)-1H-benzo[d]imidazole-4-carboxamide
—— 2-(4-chlorobenzyl)-5-[(3-pyridin-3-ylpyrrolidin-1-yl)carbonyl]-1-(2,2,2-trifluoroethyl)-1H-benzimidazole 1225211-97-1 C26H22ClF3N4O
2-(4-chlorobenzyl)-5-[(3-pyridin-3-ylpyrrolidin-1-yl)carbonyl]-1-(2,2,2-trifluoroethyl)-1H-benzimidazole
—— 6-(2-(3-(2-methoxyacetamido)phenylamino)pyrimidin-4-yloxy)-N,2-dimethylbenzofuran-3-carboxamide 1213703-49-1 C24H23N5O5
6-(2-(3-(2-methoxyacetamido)phenylamino)pyrimidin-4-yloxy)-N,2-dimethylbenzofuran-3-carboxamide
—— 2-amino-N-cyclopropyl-4-(2,4-dichloro-6-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]ethoxy}phenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide 1207961-39-4 C23H22Cl2F3N7O2
2-amino-N-cyclopropyl-4-(2,4-dichloro-6-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]ethoxy}phenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
—— 3-(4-((4-methyl-6-(1-methyl-1H-benzo[d]imidazol-2-yl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl)phenyl)propanenitrile 1207604-06-5 C29H29N5
3-(4-((4-methyl-6-(1-methyl-1H-benzo[d]imidazol-2-yl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl)phenyl)propanenitrile
—— US8653087, III-180 1213244-65-5 C30H33N9O
US8653087, III-180
—— 7-Chloro-8,10-dihydroxy-13-oxa-17,18,19-triazatricyclo[15.2.1.06,11]icosa-1(20),6(11),7,9,18-pentaene-4,12-dione 1222967-97-6 C16H16ClN3O5
7-Chloro-8,10-dihydroxy-13-oxa-17,18,19-triazatricyclo[15.2.1.06,11]icosa-1(20),6(11),7,9,18-pentaene-4,12-dione
—— 2-amino-2-(3-(3,4,5-trimethoxyphenethyl)phenethyl)propane-1,3-diol 1221257-97-1 C22H31NO5
2-amino-2-(3-(3,4,5-trimethoxyphenethyl)phenethyl)propane-1,3-diol
—— N-(5-bromopyrazine-2-yl)-4-trifluoromethylbenzamide 1373940-47-6 C12H7BrF3N3O
N-(5-bromopyrazine-2-yl)-4-trifluoromethylbenzamide
—— 1,5-phenyl-3,7-tert-butyl-1,5-diaza-3,7-diphosphacyclooctane 1246735-85-2 C24H36N2P2
1,5-phenyl-3,7-tert-butyl-1,5-diaza-3,7-diphosphacyclooctane
—— 6-(3-(4-acetylpiperazin-1-yl)phenylamino)-4-(1-phenylcyclopropylamino)nicotinamide 1374213-83-8 C27H30N6O2
6-(3-(4-acetylpiperazin-1-yl)phenylamino)-4-(1-phenylcyclopropylamino)nicotinamide
—— —— 1382190-78-4 C31H39MoN3
—— trans-8-chloro-10-hydroxy-10-(1α-methyl-2-oxobutyl)spiro<11H-benzo<a>xanthen-11,2'(1'H)-naphtho<2,1-b>furan>-9(10H)-one 136229-20-4 C33H25ClO5
trans-8-chloro-10-hydroxy-10-(1α-methyl-2-oxobutyl)spiro<11H-benzo<a>xanthen-11,2'(1'H)-naphtho<2,1-b>furan>-9(10H)-one
—— HCDT-6-ol-11-one 169395-05-5 C14H14O2
HCDT-6-ol-11-one
—— 2-<2-<2-(tripropylsilyl)ethylamino>ethylthio>benzoic acid 121405-75-2 C20H35NO2SSi
2-<2-<2-(tripropylsilyl)ethylamino>ethylthio>benzoic acid
—— (S)-N-(benzyloxy)-4-acetoxymethyl-2-azetidinone 121719-63-9 C13H15NO4
(S)-N-(benzyloxy)-4-acetoxymethyl-2-azetidinone
—— (6R,7R)-3-Chloro-7-diacetylamino-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid 121463-86-3 C11H11ClN2O5S
(6R,7R)-3-Chloro-7-diacetylamino-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (2S)-2-[[(2R)-2-acetamido-3-[2-[[(2R,3R,4R,5S,6R)-3-acetamido-4-hydroxy-6-(hydroxymethyl)-5-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]amino]-2-oxoethyl]sulfanylpropanoyl]amino]-6-[[2-[(2R,3S,4R,5R,6R)-5-acetamido-6-azido-4-hydroxy-2-(hydroxymethyl)oxan-3-yl]oxyacetyl]amino]-N-[(2R)-3-[2-[[(2R,3R,4R,5S,6R)-3-acetamido-4-hydroxy-6-(hydroxymethyl)-5-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]amino]-2-oxoethyl]sulfanyl-1-amino-1-oxopropan-2-yl]hexanamide 1000684-35-4 C56H93N13O32S2
(2S)-2-[[(2R)-2-acetamido-3-[2-[[(2R,3R,4R,5S,6R)-3-acetamido-4-hydroxy-6-(hydroxymethyl)-5-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]amino]-2-oxoethyl]sulfanylpropanoyl]amino]-6-[[2-[(2R,3S,4R,5R,6R)-5-acetamido-6-azido-4-hydroxy-2-(hydroxymethyl)oxan-3-yl]oxyacetyl]amino]-N-[(2R)-3-[2-[[(2R,3R,4R,5S,6R)-3-acetamido-4-hydroxy-6-(hydroxymethyl)-5-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]amino]-2-oxoethyl]sulfanyl-1-amino-1-oxopropan-2-yl]hexanamide
—— —— 1312697-33-8 C22H13ClF9N3O2
—— N-(3-fluoro-4-(2-(1-(2-ethoxy-acetyl)-1H-pyrazol-4-yl)pyridin-4-yloxy)phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide 1225278-50-1 C29H25F2N5O5
N-(3-fluoro-4-(2-(1-(2-ethoxy-acetyl)-1H-pyrazol-4-yl)pyridin-4-yloxy)phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— —— 1336886-79-3 C33H44FN7O2Si
—— 4-(7-bromo-1-oxo-1H-6-azaisoquinolin-2-ylmethyl)benzenesulfonamide 1055721-91-9 C15H12BrN3O3S
4-(7-bromo-1-oxo-1H-6-azaisoquinolin-2-ylmethyl)benzenesulfonamide
—— N-(3,5-dichloropyridin-4-yl)-3-[3-[(1S,2R,5R,6S,7S,8R,9R,11R,13R,14R)-2-ethyl-6-[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-8-[(2S,3R,4S,6R)-3-hydroxy-6-methyl-4-(methylamino)oxan-2-yl]oxy-9-methoxy-1,5,7,9,11,13-hexamethyl-4,12,16-trioxo-3,17-dioxa-15-azabicyclo[12.3.0]heptadecan-15-yl]propoxy]-4-methoxybenzamide 1266348-05-3 C54H80Cl2N4O16
N-(3,5-dichloropyridin-4-yl)-3-[3-[(1S,2R,5R,6S,7S,8R,9R,11R,13R,14R)-2-ethyl-6-[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-8-[(2S,3R,4S,6R)-3-hydroxy-6-methyl-4-(methylamino)oxan-2-yl]oxy-9-methoxy-1,5,7,9,11,13-hexamethyl-4,12,16-trioxo-3,17-dioxa-15-azabicyclo[12.3.0]heptadecan-15-yl]propoxy]-4-methoxybenzamide
—— butyric acid (S)-6,7-dimethoxy-9,10,11,12,12a,13-hexahydro-9a-aza-cyclopenta[b]triphenylene-3-yl ester 1223488-16-1 C26H29NO4
butyric acid (S)-6,7-dimethoxy-9,10,11,12,12a,13-hexahydro-9a-aza-cyclopenta[b]triphenylene-3-yl ester
—— 4-((3-(3-amino-1-deutero-1-hydroxypropyl)phenyl)ethynyl)heptan-4-ol 1222168-98-0 C18H27NO2
4-((3-(3-amino-1-deutero-1-hydroxypropyl)phenyl)ethynyl)heptan-4-ol
—— N-benzyl-N-[3-methoxy-4-(4-phenylpiperazin-1-ylcarbonyl)phenyl]benzenesulfonamide 1214150-67-0 C31H31N3O4S
N-benzyl-N-[3-methoxy-4-(4-phenylpiperazin-1-ylcarbonyl)phenyl]benzenesulfonamide
—— N-[4-tert-Butyl-5-methoxy-2-(2-oxo-1,2-dihydro-pyridin-3-yl)-benzyl]-4-chloro-benzenesulfonamide 1224633-46-8 C23H25ClN2O4S
N-[4-tert-Butyl-5-methoxy-2-(2-oxo-1,2-dihydro-pyridin-3-yl)-benzyl]-4-chloro-benzenesulfonamide
—— (2S,4S)-1-(2-(2H-1,2,3-triazol-2-yl)acetyl)-4-((5-chloro-2-thienyl)methyl)-N-(4-(4-fluorophenoxy)phenyl)pyrrolidine-2-carboxamide 1221877-97-9 C26H23ClFN5O3S
(2S,4S)-1-(2-(2H-1,2,3-triazol-2-yl)acetyl)-4-((5-chloro-2-thienyl)methyl)-N-(4-(4-fluorophenoxy)phenyl)pyrrolidine-2-carboxamide
—— bis(2-aminobenzophenone-2-furoylhydrazone)nickel(II) chloride 156124-50-4 C36H30Cl2N6NiO4
bis(2-aminobenzophenone-2-furoylhydrazone)nickel(II) chloride
—— (N-tert-butyl-α-deuterio-o-methylbenzylamine)tricarbonylchromium 155678-03-8 C15H19CrNO3
(N-tert-butyl-α-deuterio-o-methylbenzylamine)tricarbonylchromium